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Enprofylline

Name: Enprofylline
Brand: TargetMol
SKU: T21389
Price: 37 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T21389Cas No. 41078-02-8

Alias Enprofyllinum, Enprofilina, 3-propylxanthine, 3-n-Propylxanthine

Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor. Enprofylline is used in asthma, chronic obstructive pulmonary disease, and in the management of sickle cell disease, diabetic neuropathy, and cerebrovascular insufficiency.

Enprofylline

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Purity: 98.37%

Catalog No. T21389Alias Enprofyllinum, Enprofilina, 3-propylxanthine, 3-n-PropylxanthineCas No. 41078-02-8

Pack Size	Price	USA Warehouse	Global Warehouse
2 mg	$37	In Stock	In Stock
5 mg	$59	In Stock	In Stock
10 mg	$85	In Stock	In Stock
25 mg	$152	In Stock	In Stock
50 mg	$238	In Stock	In Stock
100 mg	$353	In Stock	In Stock
200 mg	$490	-	In Stock
1 mL x 10 mM (in DMSO)	$57	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Batch Information

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Purity:98.37%

Appearance:Solid

Color:White

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor. Enprofylline is used in asthma, chronic obstructive pulmonary disease, and in the management of sickle cell disease, diabetic neuropathy, and cerebrovascular insufficiency.
Targets&IC50	A2B receptor:7 μM (Ki)
Synonyms	Enprofyllinum, Enprofilina, 3-propylxanthine, 3-n-Propylxanthine

Chemical Properties

Molecular Weight	194.19
Formula	C₈H₁₀N₄O₂
Cas No.	41078-02-8
Smiles	CCCn1c2nc[nH]c2c(=O)[nH]c1=O
Relative Density.	1.367 g/cm3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: Insoluble

DMSO: 60 mg/mL (308.98 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	5.1496 mL	25.7480 mL	51.4960 mL	257.4798 mL
5 mM	1.0299 mL	5.1496 mL	10.2992 mL	51.4960 mL
10 mM	0.5150 mL	2.5748 mL	5.1496 mL	25.7480 mL
20 mM	0.2575 mL	1.2874 mL	2.5748 mL	12.8740 mL
50 mM	0.1030 mL	0.5150 mL	1.0299 mL	5.1496 mL
100 mM	0.0515 mL	0.2575 mL	0.5150 mL	2.5748 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc