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CIA-1 (Free base)

Name: CIA-1 (Free base)
Brand: TargetMol
SKU: T71534L
Price: 52 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T71534LCas No. 452087-38-6

Alias CIA-1(Free base)

CIA-1 (Free base) is a nuclear receptor COUP-TFII inhibitor with IC50 values ranging from 1.2 μM to 7.6 μM in prostate cancer cell lines. CIA-1 (Free base) inhibits tumor growth in a mouse model of prostate cancer xenografts.

CIA-1 (Free base)

🥰Excellent

Purity: 99%

Catalog No. T71534LAlias CIA-1(Free base)Cas No. 452087-38-6

Pack Size	Price	Availability
1 mg	$52	In Stock
5 mg	$123	In Stock
10 mg	$197	In Stock
25 mg	$396	In Stock
50 mg	$619	In Stock
100 mg	$953	In Stock

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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Purity:99%

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COA

Product Introduction

Bioactivity

Description	CIA-1 (Free base) is a nuclear receptor COUP-TFII inhibitor with IC50 values ranging from 1.2 μM to 7.6 μM in prostate cancer cell lines. CIA-1 (Free base) inhibits tumor growth in a mouse model of prostate cancer xenografts.
Synonyms	CIA-1(Free base)

Chemical Properties

Molecular Weight	329.42
Formula	C₁₇H₁₉N₃O₂S
Cas No.	452087-38-6
Smiles	N(CCC1=CC(OC)=C(OC)C=C1)C2=C3C(SC(C)=C3)=NC=N2

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 60 mg/mL (182.14 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.0356 mL	15.1782 mL	30.3564 mL	151.7819 mL
5 mM	0.6071 mL	3.0356 mL	6.0713 mL	30.3564 mL
10 mM	0.3036 mL	1.5178 mL	3.0356 mL	15.1782 mL
20 mM	0.1518 mL	0.7589 mL	1.5178 mL	7.5891 mL
50 mM	0.0607 mL	0.3036 mL	0.6071 mL	3.0356 mL
100 mM	0.0304 mL	0.1518 mL	0.3036 mL	1.5178 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc