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Erteberel

Name: Erteberel
Brand: TargetMol
SKU: T6306
Price: 156 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T6306Cas No. 533884-09-2

Alias LY500307

Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.

Erteberel

🥰Excellent

Purity: 99.46%

Catalog No. T6306Alias LY500307Cas No. 533884-09-2

Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.

Pack Size	Price	Availability
1 mg	$156	In Stock
5 mg	$455	In Stock
10 mg	$655	In Stock
25 mg	$987	In Stock
50 mg	$1,360	In Stock
1 mL x 10 mM (in DMSO)	$488	In Stock

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This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.46%

ee:100%

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COA CSFC HNMR LCMS ORP

Product Introduction

Bioactivity

Description	Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.
Targets&IC50	ERβ:1.54 nM (Ki), ERRβ:0.66 nM (EC50), ERβ:3.61 nM (EC50)
Synonyms	LY500307

Chemical Properties

Molecular Weight	282.33
Formula	C₁₈H₁₈O₃
Cas No.	533884-09-2
Smiles	[H][C@]12CCC[C@@]1([H])c1cc(O)ccc1O[C@H]2c1ccc(O)cc1
Relative Density.	1.268 g/cm3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

Ethanol: 57 mg/mL (201.89 mM), Sonication is recommended.

DMSO: 57 mg/mL (201.89 mM), Sonication is recommended.

H2O: <1 mg/mL

Solution Preparation Table

Ethanol/DMSO

	1mg	5mg	10mg	50mg
1 mM	3.5420 mL	17.7098 mL	35.4195 mL	177.0977 mL
5 mM	0.7084 mL	3.5420 mL	7.0839 mL	35.4195 mL
10 mM	0.3542 mL	1.7710 mL	3.5420 mL	17.7098 mL
20 mM	0.1771 mL	0.8855 mL	1.7710 mL	8.8549 mL
50 mM	0.0708 mL	0.3542 mL	0.7084 mL	3.5420 mL
100 mM	0.0354 mL	0.1771 mL	0.3542 mL	1.7710 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc