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Z-HA155

Name: Z-HA155
Brand: TargetMol
SKU: T11533
Price: 30 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T11533Cas No. 1312201-00-5

Alias CS-963

Z-HA155 (CS-963) selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.

Z-HA155

🥰Excellent

Purity: 99.18%

Catalog No. T11533Alias CS-963Cas No. 1312201-00-5

Z-HA155 (CS-963) selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.

Pack Size	Price	Availability
1 mg	$30	In Stock
5 mg	$68	In Stock
10 mg	$108	In Stock
25 mg	$222	In Stock
50 mg	$357	In Stock
100 mg	$528	In Stock
200 mg	$755	In Stock
1 mL x 10 mM (in DMSO)	$70	In Stock

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Batch Information

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Purity:99.18%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	Z-HA155 (CS-963) selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.
Targets&IC50	ATX:5.7 nM
In vitro	HA155 completely attenuates the thrombin-mediated increase in platelet-derived LPA dose-dependently [2].HA155 is an ATX inhibitor by binding to the ATX active site [3].
Synonyms	CS-963

Chemical Properties

Molecular Weight	463.29
Formula	C₂₄H₁₉BFNO₅S
Cas No.	1312201-00-5
Smiles	OB(O)c1ccc(COc2ccc(\C=C3/SC(=O)N(Cc4ccc(F)cc4)C3=O)cc2)cc1
Relative Density.	no data available
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 8 mg/mL (17.27 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.1585 mL	10.7924 mL	21.5848 mL	107.9238 mL
5 mM	0.4317 mL	2.1585 mL	4.3170 mL	21.5848 mL
10 mM	0.2158 mL	1.0792 mL	2.1585 mL	10.7924 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc