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Pilsicainide HCl (Synonyms: SUN 1165)

Name: Pilsicainide HCl
Brand: TargetMol
SKU: T7811
Price: 31 USD
Availability: InStock
Rating: 5 (10 reviews)

Catalog No. T7811 Copy Product Info

Purity: 99.80%

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Pilsicainide HCl (SUN 1165) is a pure sodium channel blocker

Pilsicainide HCl

Copy Product Info

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Catalog No. T7811

Synonyms SUN 1165

Pilsicainide HCl (SUN 1165) is a pure sodium channel blocker

Cas No. 88069-49-2

Pack Size	Price	USA Stock	Global Stock
10 mg	$31	In Stock	In Stock
25 mg	$64	In Stock	In Stock
50 mg	$89	In Stock	In Stock
1 mL x 10 mM (in DMSO)	$39	In Stock	In Stock

For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)

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For research use only—not for human use. No sales to individuals. Use as intended only.

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Batch Information

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Purity:99.80%

Resource Download

COA HNMR HPLC LCMS

Product Introduction

Pilsicainide HCl AI Summary

Pilsicainide HCl has demonstrated a low level of activity in inhibiting cell viability when compared to the arbidol control in Vero E6 cells infected with SARS-CoV-2. The assay results indicate an inhibition index of 0.08672, suggesting that this compound is not highly effective in this specific bioactivity assay..

Note: Summary generated by AI. Data source: ChEMBL

Bioactivity

Description	Pilsicainide HCl (SUN 1165) is a pure sodium channel blocker
Synonyms	SUN 1165

Chemical Properties

Molecular Weight	308.85
Formula	C₁₇H₂₅ClN₂O
Cas No.	88069-49-2
Smiles	Cl.Cc1cccc(C)c1NC(=O)CC12CCCN1CCC2
Relative Density.	no data available

Storage & Solubility Information

Storage

Pure form: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 9 mg/mL (29.14 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.2378 mL	16.1891 mL	32.3782 mL	161.8909 mL
5 mM	0.6476 mL	3.2378 mL	6.4756 mL	32.3782 mL
10 mM	0.3238 mL	1.6189 mL	3.2378 mL	16.1891 mL
20 mM	0.1619 mL	0.8095 mL	1.6189 mL	8.0945 mL

Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc