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(R)-Indeloxazine benzenesulfonate

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Catalog No. T210304Cas No. 1623762-83-3
Alias AS1069562, (R)-YM-08054 benzenesulfonate

(R)-Indeloxazine benzenesulfonate (AS1069562) is an orally active inhibitor of serotonin (5-HT) and norepinephrine (NE) reuptake, with IC50 values of 0.35 μM and 3.3 μM, respectively. It exhibits analgesic activity and can enhance neurological function by improving neurotrophic support.

(R)-Indeloxazine benzenesulfonate
Other Forms of (R)-Indeloxazine benzenesulfonate:

(R)-Indeloxazine benzenesulfonate

😃Good
Catalog No. T210304Alias AS1069562, (R)-YM-08054 benzenesulfonateCas No. 1623762-83-3
(R)-Indeloxazine benzenesulfonate (AS1069562) is an orally active inhibitor of serotonin (5-HT) and norepinephrine (NE) reuptake, with IC50 values of 0.35 μM and 3.3 μM, respectively. It exhibits analgesic activity and can enhance neurological function by improving neurotrophic support.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
10 mgInquiry10-14 weeks10-14 weeks
50 mgInquiry10-14 weeks10-14 weeks
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction

Bioactivity
Description
(R)-Indeloxazine benzenesulfonate (AS1069562) is an orally active inhibitor of serotonin (5-HT) and norepinephrine (NE) reuptake, with IC50 values of 0.35 μM and 3.3 μM, respectively. It exhibits analgesic activity and can enhance neurological function by improving neurotrophic support.
In vivo
(R)-Indeloxazine benzenesulfonate (AS1069562, STZ-induced diabetic rats, orally, 3, 10, and 30 mg/kg) administered for four weeks exhibits sustained analgesic effects in a rat model of neuropathic pain induced by Streptozotocin (STZ). It also notably restores decreased levels of IGF1 and IGF2 mRNA in the dorsal root ganglia and spinal cord.
SynonymsAS1069562, (R)-YM-08054 benzenesulfonate
Chemical Properties
Molecular Weight389.47
FormulaC20H23NO5S
Cas No.1623762-83-3
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
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