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WAY-270250

Name: WAY-270250
Brand: TargetMol
SKU: T77624
Price: 30 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T77624Cas No. 852367-46-5

WAY-270250 is an IGF-1R/SRC inhibitor.

WAY-270250

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Purity: 99.97%

Catalog No. T77624Cas No. 852367-46-5

WAY-270250 is an IGF-1R/SRC inhibitor.

Pack Size	Price	USA Warehouse	Global Warehouse
5 mg	$30	-	In Stock
10 mg	$45	-	In Stock
25 mg	$90	-	In Stock
50 mg	$133	-	In Stock
100 mg	$198	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Batch Information

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Purity:99.97%

Appearance:Solid

Color:Green

Resource Download

COA HNMR LCMS

Product Introduction

WAY-270250 AI Summary

WAY-270250 shows a bioactivity of displacing [3H]flumazenil from benzodiazepine receptors in bovine brain membranes, with a Ki value of 606.0 nM, indicating potential activity in modulating these receptors. Additionally, it exhibits inhibitory activity against c-MET with an IC50 value greater than 100000.0 nM and against IGF-1R with an IC50 value of 63000.0 nM..

Note: Summary generated by AI. Data source: ChEMBL

Bioactivity

Description

WAY-270250 is an IGF-1R/SRC inhibitor.

Chemical Properties

Molecular Weight	292.33
Formula	C₁₈H₁₆N₂O₂
Cas No.	852367-46-5
Smiles	C(C(NCC1=CC=C(C)C=C1)=O)(=O)C=2C=3C(NC2)=CC=CC3
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (171.04 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.4208 mL	17.1040 mL	34.2079 mL	171.0396 mL
5 mM	0.6842 mL	3.4208 mL	6.8416 mL	34.2079 mL
10 mM	0.3421 mL	1.7104 mL	3.4208 mL	17.1040 mL
20 mM	0.1710 mL	0.8552 mL	1.7104 mL	8.5520 mL
50 mM	0.0684 mL	0.3421 mL	0.6842 mL	3.4208 mL
100 mM	0.0342 mL	0.1710 mL	0.3421 mL	1.7104 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc