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Pulrodemstat benzenesulfonate

Name: Pulrodemstat benzenesulfonate
Brand: TargetMol
SKU: T11882
Price: 55 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T11882Cas No. 2097523-60-7

Alias LSD1-IN-7 benzenesulfonate, CC-90011 benzenesulfonate

Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.

Pulrodemstat benzenesulfonate

🥰Excellent

Purity: 97.67%

Catalog No. T11882Alias LSD1-IN-7 benzenesulfonate, CC-90011 benzenesulfonateCas No. 2097523-60-7

Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.

Pack Size	Price	Availability
1 mg	$55	In Stock
2 mg	$78	In Stock
5 mg	$126	In Stock
10 mg	$198	In Stock
25 mg	$347	In Stock
50 mg	$515	In Stock
100 mg	$747	In Stock
1 mL x 10 mM (in DMSO)	$179	In Stock

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Batch Information

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Purity:97.67%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
Targets&IC50	LSD1:0.25 nM (IC50)
In vivo	LSD1-IN-7 in combination with other LSD1 inhibitor can be treatment of cancer in a mammal, including breast cancer, lung cancer, prostate cancer, glioblastoma, or leukemia.
Synonyms	LSD1-IN-7 benzenesulfonate, CC-90011 benzenesulfonate

Chemical Properties

Molecular Weight	609.64
Formula	C₃₀H₂₉F₂N₅O₅S
Cas No.	2097523-60-7
Smiles	OS(=O)(=O)c1ccccc1.COc1ccc(cc1F)-c1c(nc(N2CCC(N)CC2)n(C)c1=O)-c1ccc(C#N)c(F)c1
Relative Density.	no data available
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 60 mg/mL (98.42 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.6403 mL	8.2016 mL	16.4031 mL	82.0156 mL
5 mM	0.3281 mL	1.6403 mL	3.2806 mL	16.4031 mL
10 mM	0.1640 mL	0.8202 mL	1.6403 mL	8.2016 mL
20 mM	0.0820 mL	0.4101 mL	0.8202 mL	4.1008 mL
50 mM	0.0328 mL	0.1640 mL	0.3281 mL	1.6403 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc