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CB-5339

Name: CB-5339
Brand: TargetMol
SKU: T60193
Price: 50 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T60193Cas No. 1863952-15-1

p97-IN-1 is a potent inhibitor of p97 with an IC 50 <30 nM [1].

CB-5339

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Purity: 97.66%

Catalog No. T60193Cas No. 1863952-15-1

p97-IN-1 is a potent inhibitor of p97 with an IC 50 <30 nM [1].

Pack Size	Price	Availability
5 mg	$50	In Stock
10 mg	$75	In Stock
25 mg	$128	In Stock
50 mg	$192	In Stock
100 mg	$287	In Stock

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Batch Information

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Purity:97.66%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description

p97-IN-1 is a potent inhibitor of p97 with an IC 50 <30 nM [1].

Chemical Properties

Molecular Weight	412.49
Formula	C₂₄H₂₄N₆O
Cas No.	1863952-15-1
Smiles	CC=1N(C=2C(=C(C(N)=O)C=CC2)C1)C3=NC(NCC4=CC=CC=C4)=C5C(N3)=NCCC5
Relative Density.	1.38 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (121.22 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4243 mL	12.1215 mL	24.2430 mL	121.2151 mL
5 mM	0.4849 mL	2.4243 mL	4.8486 mL	24.2430 mL
10 mM	0.2424 mL	1.2122 mL	2.4243 mL	12.1215 mL
20 mM	0.1212 mL	0.6061 mL	1.2122 mL	6.0608 mL
50 mM	0.0485 mL	0.2424 mL	0.4849 mL	2.4243 mL
100 mM	0.0242 mL	0.1212 mL	0.2424 mL	1.2122 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc