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CCG-100602

Name: CCG-100602
Brand: TargetMol
SKU: T22062
Price: 32 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T22062Cas No. 1207113-88-9

CCG-100602 inhibits RhoA/C-mediated, SRF-driven luciferase expression in PC-3 prostate cancer cells (IC50 :9.8 μM).

CCG-100602

🥰Excellent

Purity: 99.58%

Catalog No. T22062Cas No. 1207113-88-9

CCG-100602 inhibits RhoA/C-mediated, SRF-driven luciferase expression in PC-3 prostate cancer cells (IC50 :9.8 μM).

Pack Size	Price	Availability
5 mg	$32	In Stock
10 mg	$52	In Stock
25 mg	$116	In Stock
50 mg	$198	In Stock
100 mg	$318	In Stock
200 mg	$473	In Stock
1 mL x 10 mM (in DMSO)	$36	In Stock

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Purity:99.58%

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COA HPLC HNMR LCMS

Product Introduction

Bioactivity

Description	CCG-100602 inhibits RhoA/C-mediated, SRF-driven luciferase expression in PC-3 prostate cancer cells (IC50 :9.8 μM).
In vitro	CCG-100602 blocks the expression of MRTF-A/SRF-activated genes. CCG-100602 (3-30?μM) decreases the number of adherent hASC cells[1].

Chemical Properties

Molecular Weight	478.82
Formula	C₂₁H₁₇ClF₆N₂O₂
Cas No.	1207113-88-9
Smiles	FC(F)(F)c1cc(cc(c1)C(F)(F)F)C(=O)N1CCCC(C1)C(=O)Nc1ccc(Cl)cc1
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 100 mg/mL (208.85 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0885 mL	10.4423 mL	20.8847 mL	104.4234 mL
5 mM	0.4177 mL	2.0885 mL	4.1769 mL	20.8847 mL
10 mM	0.2088 mL	1.0442 mL	2.0885 mL	10.4423 mL
20 mM	0.1044 mL	0.5221 mL	1.0442 mL	5.2212 mL
50 mM	0.0418 mL	0.2088 mL	0.4177 mL	2.0885 mL
100 mM	0.0209 mL	0.1044 mL	0.2088 mL	1.0442 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

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