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(R)-BAY1238097

🥰Excellent
Catalog No. T13442Cas No. 1564269-85-7

(R)-BAY1238097 represents the R-isomer of BAY1238097, which exhibits relatively lower activity compared to its counterpart. BAY1238097 is a highly potent and selective inhibitor targeting the binding of BET proteins to histones, demonstrating significant anti-proliferative effects in various acute myeloid leukemia (AML) and multiple myeloma (MM) models. The high activity is achieved through the down-regulation of c-Myc levels and the subsequent modulation of its downstream transcriptome.

(R)-BAY1238097
Other Forms of (R)-BAY1238097:

(R)-BAY1238097

🥰Excellent
Purity: 98.77%
Catalog No. T13442Cas No. 1564269-85-7
(R)-BAY1238097 represents the R-isomer of BAY1238097, which exhibits relatively lower activity compared to its counterpart. BAY1238097 is a highly potent and selective inhibitor targeting the binding of BET proteins to histones, demonstrating significant anti-proliferative effects in various acute myeloid leukemia (AML) and multiple myeloma (MM) models. The high activity is achieved through the down-regulation of c-Myc levels and the subsequent modulation of its downstream transcriptome.
Pack SizePriceAvailabilityQuantity
1 mg$48In Stock
5 mg$116In Stock
10 mg$193In Stock
25 mg$426In Stock
50 mg$739In Stock
100 mg$1,190In Stock
200 mg$1,630In Stock
1 mL x 10 mM (in DMSO)$127In Stock
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Purity:98.77%
ee:100%
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Product Introduction

Bioactivity
Description
(R)-BAY1238097 represents the R-isomer of BAY1238097, which exhibits relatively lower activity compared to its counterpart. BAY1238097 is a highly potent and selective inhibitor targeting the binding of BET proteins to histones, demonstrating significant anti-proliferative effects in various acute myeloid leukemia (AML) and multiple myeloma (MM) models. The high activity is achieved through the down-regulation of c-Myc levels and the subsequent modulation of its downstream transcriptome.
Chemical Properties
Molecular Weight451.56
FormulaC25H33N5O3
Cas No.1564269-85-7
SmilesO(C)C=1C=C2C(=NN(C(NC)=O)[C@H](C)CC2=CC1OC)C3=CC=C(C=C3)N4CCN(C)CC4
Relative Density.1.22 g/cm3 (Predicted)
Storage & Solubility Information
Storagestore at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 120 mg/mL (265.75 mM), Sonication is recommended.
H2O: < 0.1(insoluble)
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.2145 mL11.0727 mL22.1455 mL110.7273 mL
5 mM0.4429 mL2.2145 mL4.4291 mL22.1455 mL
10 mM0.2215 mL1.1073 mL2.2145 mL11.0727 mL
20 mM0.1107 mL0.5536 mL1.1073 mL5.5364 mL
50 mM0.0443 mL0.2215 mL0.4429 mL2.2145 mL
100 mM0.0221 mL0.1107 mL0.2215 mL1.1073 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
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Keywords

BETBAY-1238097BAY1238097BAY 1238097(R)-BAY-1238097(R)BAY1238097(R) BAY1238097
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