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A2B receptor antagonist 2

Name: A2B receptor antagonist 2
Brand: TargetMol
SKU: T37793
Rating: 4.5 (1 reviews)

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Catalog No. T37793Cas No. 784-90-7

Alias A2B receptor antagonist 2

A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).

A2B receptor antagonist 2

😃Good

Catalog No. T37793Alias A2B receptor antagonist 2Cas No. 784-90-7

A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).

Pack Size	Price	USA Warehouse	Global Warehouse	Quantity
10 mg	$38	1-2 weeks	1-2 weeks

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Product Introduction

Bioactivity

Description	A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
Targets&IC50	A2A (rat):6.8 μM (Ki), A1 (rat):2.30 μM (Ki), A2B (human):3.44 μM (Ki)
Synonyms	A2B receptor antagonist 2

Chemical Properties

Molecular Weight	229.28
Formula	C₁₂H₁₅N₅
Cas No.	784-90-7

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 2 mg/mL (8.72 mM), Sonication and heating to 60℃ are recommended.

Methanol: 5 mg/mL (21.81 mM), Sonication and heating to 60℃ are recommended.

Solution Preparation Table

DMSO/Methanol

	1mg	5mg	10mg	50mg
1 mM	4.3615 mL	21.8074 mL	43.6148 mL	218.0740 mL
5 mM	0.8723 mL	4.3615 mL	8.7230 mL	43.6148 mL

Methanol

	1mg	5mg	10mg	50mg
10 mM	0.4361 mL	2.1807 mL	4.3615 mL	21.8074 mL
20 mM	0.2181 mL	1.0904 mL	2.1807 mL	10.9037 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc