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Autocamtide-2-related inhibitory peptide

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Catalog No. TP2310Cas No. 167114-91-2

Autocamtide-2-related inhibitory peptide is a potent and highly specific inhibitor of CaMKII, with an IC50 of 40 nM.

Autocamtide-2-related inhibitory peptide
Other Forms of Autocamtide-2-related inhibitory peptide:

Autocamtide-2-related inhibitory peptide

🥰Excellent
Catalog No. TP2310Cas No. 167114-91-2
Autocamtide-2-related inhibitory peptide is a potent and highly specific inhibitor of CaMKII, with an IC50 of 40 nM.
Pack SizePriceAvailabilityQuantity
1 mg$56In Stock
5 mg$127In Stock
10 mg$190In Stock
25 mg$313In Stock
50 mg$441In Stock
100 mg$596In Stock
200 mg$791In Stock
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Purity:>99.99%
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Product Introduction

Bioactivity
Description
Autocamtide-2-related inhibitory peptide is a potent and highly specific inhibitor of CaMKII, with an IC50 of 40 nM.
Targets&IC50
CaMK:40 nM
In vitro
Autocamtide-2-related inhibitory peptide (a novel synthetic peptide ATP) is a potent inhibitor of CaM-kinase II with an IC50 of 40 nM, which is active in the presence or absence of Ca2+/calmodulin. It is 50 and 500 times more potent than CaMK-(281-302Ala286) and KN-93,respectively, under the assay condition used[1].
Chemical Properties
Molecular Weight1497.74
FormulaC64H116N22O19
Cas No.167114-91-2
Smiles[C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CCCCN)N)=O)CCCCN)=O)C)=O)CC(C)C)=O)CCCNC(=N)N)=O)(C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H](CC(C)C)C(O)=O)=O)C)=O)CC(O)=O)=O)C(C)C)=O)C)=O)CCC(O)=O)=O)CCC(N)=O)=O)CCCNC(=N)N
Relative Density.no data available
SequenceLys-Lys-Ala-Leu-Arg-Arg-Gln-Glu-Ala-Val-Asp-Ala-Leu
Sequence ShortKKALRRQEAVDAL
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 10 mM, Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM0.6677 mL3.3384 mL6.6767 mL33.3836 mL
5 mM0.1335 mL0.6677 mL1.3353 mL6.6767 mL
10 mM0.0668 mL0.3338 mL0.6677 mL3.3384 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

InhibitorinhibitCaMKIICaMKCalmodulin-dependent protein kinasesCalmodulin-dependent kinasesAutophagyAutocamtide-2-related inhibitory peptideAutocamtide2related inhibitory peptideAutocamtide 2 related inhibitory peptide
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