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Ion Channel Inhibitor Library

Catalog No. L2300
  Library Compound List   Excel SDF

Given the central functional role that the ion channel superfamily plays in human physiology, its membrane localization, and the diverse tissue distribution of different members of the family, it represents an attractive potential target class for drug discovery. Ion channelsplay a fundamental role in the way cells communicate. This communication between cells allows for the orchestration of physical and mental activities in humans. A number of diseases occur when ion channels do not function properly. Some examples are diabetes, neuropathic pain, cardiovascular diseases, asthma, epilepsy, and neurodegenerative disease, etc.

The Ion Channel Inhibitor Library by TargetMol, containing 946 compounds targeting ion channels, can be used for research in ion channel, high throughput screening and high content screening for ion channel drug discovery.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Compound Libraries | TargetMol
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 946 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Targets include potassium channel, calcium channel, sodium channel, Proton pump, etc;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L2300)

Publications Cited TargetMol Libraries

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Library Composition

Potassium Channel (170)
Calcium Channel (154)
Sodium Channel (128)
GABA Receptor (106)
TRP/TRPV Channel (99)
Autophagy (81)
iGluR (68)
ATPase (52)
Endogenous Metabolite (52)
AChR (48)
Apoptosis (38)
NMDAR (36)
P-gp (35)
Antibacterial (31)
Parasite (27)
Chloride channel (26)
Proton pump (25)
P2X Receptor (22)
GluR (19)
P450 (19)
5-HT Receptor (18)
Reactive Oxygen Species (17)
COX (16)
NF-κB (16)
CFTR (16)
Adrenergic Receptor (15)
Dopamine Receptor (15)
Antibiotic (12)
HIV Protease (12)
ABC (11)
PPAR (9)
Ferroptosis (9)
Antifungal (9)
transporter (9)
SGLT (8)
Monocarboxylate transporter (8)
CaMK (8)
GPR (8)
Monoamine Transporter (7)
Influenza Virus (7)
TNF (7)
Carbonic Anhydrase (7)
BCRP (7)
HER (7)
Histamine Receptor (7)
MRP (6)
DNA/RNA Synthesis (6)
OAT (6)
Drug Metabolite (6)
Na+/Ca2+ Exchanger (6)
OCT (6)
IL Receptor (6)
EGFR (6)
SARS-CoV (5)
AChE (5)
CRM1 (5)
Phospholipase (5)
Mitochondrial Metabolism (5)
NPC1L1 (5)
Topoisomerase (5)
VDAC (5)
Virus Protease (5)
Antioxidant (5)
PKC (4)
Mitophagy (4)
Cannabinoid Receptor (4)
Myosin (4)
PDE (4)
AMPK (4)
ERK (3)
NO Synthase (3)
Hedgehog/Smoothened (3)
NADPH (3)
TGF-beta/Smad (3)
HDAC (3)
Norepinephrine (3)
CGRP Receptor (3)
Lipoxygenase (3)
mTOR (3)
Caspase (3)
STAT (3)
GluCls (2)
Lipid (2)
Beta Amyloid (2)
MMP (2)
Akt (2)
HSV (2)
Beta-Secretase (2)
Prostaglandin Receptor (2)
GST (2)
Fatty Acid Synthase (2)
Interleukin (2)
IκB/IKK (2)
Aquaporin (2)
RAAS (2)
HBV (2)
PKA (2)
HMG-CoA Reductase (2)
CaSR (2)
Phosphatase (2)
TOPK (2)
Tyrosinase (2)
NOD (2)
AhR (2)
NOD-like Receptor (NLR) (2)
p38 MAPK (2)
Integrin (2)
Src (2)
NOS (2)
Wnt/beta-catenin (2)
DNA Methyltransferase (2)
Serine/threonin kinase (2)
Gamma-secretase (2)
Opioid Receptor (2)
ROS (2)
MEK (2)
GlyT (2)
Na-K-Cl cotransporter (2)
Anti-infection (2)
LDL (2)
Platelet aggregation (2)
Syk (2)
VEGFR (2)
FLT (2)
Gap Junction Protein (1)
S6 Kinase (1)
Sigma receptor (1)
FGFR (1)
Thrombin (1)
HIF/HIF Prolyl-Hydroxylase (1)
HIF (1)
Reverse Transcriptase (1)
Hydroxylase (1)
PKM (1)
CRISPR/Cas9 (1)
Proteasome (1)
HCN Channel (1)
RSV (1)
JNK (1)
Amylase (1)
ROCK (1)
FXR (1)
Cysteine Protease (1)
Serotonin Transporter (1)
PARP (1)
Estrogen Receptor/ERR (1)
N-Acetylglucosaminyltransferase (1)
GSK-3 (1)
Reductase (1)
CSF-1R (1)
Adenosine Receptor (1)
LPL Receptor (1)
PI3K (1)
Dehydrogenase (1)
Estrogen/progestogen Receptor (1)
Piezo Channel (1)
Transferase (1)
Transaminase (1)
Taste receptor (1)
MAO (1)
Glucocorticoid Receptor (1)
Casein Kinase (1)
cAMP (1)
PAI-1 (1)
Nrf2 (1)
Trk receptor (1)
HSP (1)
MAPK (1)
Androgen Receptor (1)
DNA (1)
IGF-1R (1)
Epigenetic Reader Domain (1)
PAK (1)
UGT (1)
PDGFR (1)
BCL (1)
PROTAC Linker (1)
Anion Exchanger (1)
Antifection (1)
BTK (1)
DNA gyrase (1)
MT Receptor (1)
CDK (1)
PAFR (1)
S1P Receptor (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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