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Glycylsarcosine
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Catalog No. T8915Cas No. 29816-01-1
Alias GLYCYL-SARCOSINE
Glycylsarcosine (GLYCYL-SARCOSINE) is a dipeptide obtained by formal condensation of the carboxy group of glycine with the amino group of sarcosine
Glycylsarcosine
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Purity: 98.47%
Catalog No. T8915Alias GLYCYL-SARCOSINECas No. 29816-01-1
Glycylsarcosine (GLYCYL-SARCOSINE) is a dipeptide obtained by formal condensation of the carboxy group of glycine with the amino group of sarcosine
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 500 mg | $34 | In Stock | In Stock | |
| 1 g | $52 | In Stock | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:98.47%
Appearance:solid
Color:White
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Product Introduction
Glycylsarcosine AI Summary
Glycylsarcosine exhibits significant bioactivity related to its interactions with various transporter proteins, particularly PEPT1 and PEPT2. It acts as a substrate and modulator of these transporters, demonstrating different affinities across cell types and species. The compound shows complete absorption in the human intestine after oral administration, with varying permeabilities in different membrane models, including higher permeability in the 2/4/A1 cell model. It has a Ki value of 830,000 nM for the inhibition of the human intestinal peptide carrier and an EC50 value of 540,000 nM for activation of the human PEPT1 transporter, with a max activation of 101% relative to Gly-Sar. Additionally, the compound exhibits moderate to high permeability across human Caco-2 cells, evidenced by a Papp value of 1.1 x 10^-5 cm/s. Furthermore, it shows uptake and inhibition activities in PEPT1 and PEPT2-expressing cells with varying Km and Ki values, indicating its role in transporter-mediated drug absorption and potential implications in drug interactions..
Note: Summary generated by AI. Data source: ChEMBL 
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Glycylsarcosine (GLYCYL-SARCOSINE) is a dipeptide obtained by formal condensation of the carboxy group of glycine with the amino group of sarcosine |
| Synonyms | GLYCYL-SARCOSINE |
| Molecular Weight | 146.14 |
| Formula | C5H10N2O3 |
| Cas No. | 29816-01-1 |
| Smiles | CN(CC(O)=O)C(=O)CN |
| Relative Density. | 1.284g/cm3 |
| Sequence | H-Gly-Sar-OH |
| Sequence Short | GG |
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Solubility Information | DMSO: Slightly soluble  |
Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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