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activity

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    13357
    TargetMol | Inhibitors_Agonists
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    TargetMol | Compound_Libraries
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    662
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    TargetMol | PROTAC
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    TargetMol | Natural_Products
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    TargetMol | Recombinant_Protein
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    TargetMol | Inhibitors_Agonists
clk-in-t3
T149802109805-56-1
CLK-IN-T3 is an inhibitor of CLK1, CLK2, and CLK3 with IC50s of 0.67, 15, and 110 nM. CLK-IN-T3 exhibits anti-cancer activity.
  • $53
In Stock
Size
QTY
SB-334867 free base
SB334867A free base, SB-334867, SB334867, SB 334867
T6140792173-99-0
SB-334867 free base (SB334867A free base) is a selective antagonist of the orexin-1 (OX1) receptor.
  • $35
In Stock
Size
QTY
Pronase E (Activity ≥ 7000 U/g)
Pronase E, Pronase
T138279036-06-0
Pronase E is a mixture of proteolytic enzymes that is obtained from Streptomyces griseus and could digest protein into individual amino acids.
  • $32
In Stock
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STING (WT/R232) activity regulator 126
T60000702662-64-4
STING (WT R232) activity regulator 126 is a STING modulator with antibacterial and antiviral effects.
  • $117
In Stock
Size
QTY
TNFα activity modulator 3
T899322248726-53-4
TNFα Activity Modulator 3 (example 6) is a molecule that regulates TNF activity by inhibiting TNFα-induced NF-κB activation, making it applicable for related research.
  • Inquiry Price
10-14 weeks
Size
QTY
Sorafenib
Bay 43-9006
T0093L284461-73-0
Sorafenib (Bay 43-9006) is a multikinase inhibitor that targets Raf-1, B-Raf, VEGFR2, VEGFR3, VEGFR4, PDGFRβ, FLT3, c-Kit, and others (IC50=6 22 90 15 20 20 57 58 nM) with oral activity. It exhibits antitumor properties and can induce autophagy, apoptosis, and agonistic iron death.
  • $34
In Stock
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QTY
5-Fluorouracil
NSC 19893, Fluorouracil, 5-FU, 5-Fluoracil
T098451-21-8
5-Fluorouracil (5-FU) is a uracil analog and inhibitor of DNA synthesis, exhibiting antitumor activity by affecting pyrimidine synthesis through thymidylate synthase inhibition; it induces apoptosis and autophagy.
  • $30
In Stock
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QTY
Gefitinib
ZD1839
T1181184475-35-2
Gefitinib (ZD1839) is an EGFR first-generation inhibitor with oral activity that inhibits the EGFR 19 Del and L858R mutations. Gefitinib has antitumor activity and is used for the treatment of EGFR-mutated non-small-cell lung cancers. Gefitinib administration RESULTS in the development of the EGFR C797S resistance mutation.
  • $50
In Stock
Size
QTY
TargetMol | Inhibitor Hot
Decitabine
NSC 127716, Dacogen, 5-Aza-CdR, 5-Aza-2'-deoxycytidine
T15082353-33-5
Decitabine (Deoxycytidine) is a deoxycytidine analog, a DNA methyltransferase inhibitor with oral activity. Decitabine has antitumor activity and antimetabolic activity. Decitabine induces cell cycle arrest and apoptosis.
  • $30
In Stock
Size
QTY
IBMX
Methylisobutylxanthine, Isobutylmethylxanthine, 3-Isobutyl-1-methylxanthine, 1-Methyl-3-Isobutylxanthine
T171328822-58-4
IBMX (Methylisobutylxanthine) is a broad-spectrum phosphodiesterase (PDE) inhibitor with inhibitory activity against PDE3, PDE4, and PDE5 (IC50=6.5 26.3 31.7 μM). IBMX enhances the intracellular cAMP level.
  • $33
In Stock
Size
QTY
TargetMol | Inhibitor Hot
Erastin
T1765571203-78-6
Erastin is an iron death activator that acts on the mitochondrial VDAC in a ROS- and iron-dependent manner. Erastin has anti-tumor activity and acts selectively on tumor cells with RAS-carcinogenic mutations.
  • $41
In Stock
Size
QTY
TargetMol | Inhibitor Hot
Ruxolitinib
INCB018424, (R)-Ruxolitinib
T1829941678-49-5
Ruxolitinib (INCB018424) is a JAK1 2 inhibitor (IC50=3.3 2.8 nM) that is potent and selective. Rixolitinib exhibits antitumor activity and induces autophagy and apoptosis.
  • $53
In Stock
Size
QTY
TargetMol | Inhibitor Hot
Trametinib
JTP-74057, GSK1120212
T2125871700-17-3
Trametinib (GSK1120212) is a MEK inhibitor that inhibits MEK1 and MEK2 (IC50=0.7 0.9 nM) with ATP non-competitive and oral activity. Trametinib activates autophagy and induces apoptosis.
  • $31
In Stock
Size
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TargetMol | Inhibitor Hot
Bortezomib
Radiciol, NSC 681239, MG 341, LDP 341, DPBA, Brotezamide
T2399179324-69-7
Bortezomib (LDP 341) is a 20S proteasome inhibitor (Ki=0.6 nM) that is reversible and selective. Bortezomib has antitumor activity and inhibits NF-κB, which can disrupt the cell cycle and induce apoptosis.
  • $48
In Stock
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TargetMol | Inhibitor Hot
ML385
T4360846557-71-9
ML385 is an NRF2 inhibitor (IC50=1.9 μM) with novelty and specificity. ML385 has anti-inflammatory activity by modulating anti-oxidative stress through the inhibition of NRF2. ML385 also exhibits anti-tumor activity.
  • $47
In Stock
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TargetMol | Inhibitor Hot
Staurosporine
CGP 41251, Antibiotic AM-2282, AM-2282
T668062996-74-1
Staurosporine (AM-2282) is a protein kinase inhibitor with ATP-competitive and non-selective inhibitory activity (IC50=6 15 2 3 3000 nM) against PKC, PKA, c-Fgr, phosphorylase kinase and TAOK2. Staurosporine also induces apoptosis.
  • $56
In Stock
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QTY
TargetMol | Inhibitor Hot
BI-2493
T720612937344-16-4In house
BI-2493 is a highly selective pan-KRAS inhibitor and structural analog of BI-2865.BI-2493 exhibits antitumor activity and inhibits tumor cell growth and can be used in the study of cancerous diseases.BI-2493 is a highly selective pan-KRAS inhibitor and structural analog of BI-2865.
  • $629
In Stock
Size
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TargetMol | Inhibitor Hot
RMC-6236
RMC6236
T746982765081-21-6
RMC-6236 is an orally effective and novel triple complex RAS (ON) MULTI inhibitor, which is a potent non covalent inhibitor of multiple RAS variants in GTP binding state. RMC-6236 has anti-tumor activity and can be used in research related to RAS driven tumors. With rich experience in compound synthesis, we can provide fast customized synthesis services for this product according to your research needs.
  • $58
In Stock
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TargetMol | Inhibitor Hot
RMC-7977
T812632765082-12-8
RMC-7977 is a highly selective inhibitor of the active (GTP-bound) forms of KRAS, HRAS, and NRAS with anticancer activity for the study of solid tumors with KRAS G12C mutations.
  • $257
In Stock
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TargetMol | Inhibitor Hot
Insulin (human)
Insulin(human), INSULIN
T822111061-68-0
Insulin (human) is a peptide hormone that promotes glycogen synthesis and regulates glucose levels in the blood. Insulin (human) has hypoglycemic activity and is used clinically to treat hyperglycemia in diabetic patients.
  • $30
In Stock
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TargetMol | Inhibitor Hot
MRTX1133
T93032621928-55-8In house
MRTX1133 is a KRAS G12D inhibitor (KD=0.2 pM) that is potent, selective, and non-covalent. MRTX1133 exhibits inhibitory activity against KRAS G12D-mutated tumors, but not against KRAS wild-type tumors.
  • $197
In Stock
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TargetMol | Inhibitor Hot
Trastuzumab
T9912180288-69-1
Trastuzumab is a humanized monoclonal antibody for patients with invasive breast cancers that overexpress HER2. Trastuzumab has been clinically used to treat HER2 Positive Metastatic Breast Cancer and HER2 Positive Gastric Cancer.
  • $157
In Stock
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TargetMol | Inhibitor Hot
Methicillin sodium salt
Meticillin sodium, Methicillin sodium
T0234132-92-3
Methicillin sodium salt is the sodium salt form of methicillin, a semisynthetic beta-lactam penicillin antibiotic with beta-lactamase resistant activity.
  • $29
In Stock
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TargetMol | Inhibitor Hot
Rosiglitazone
BRL49653
T0334122320-73-4
Rosiglitazone (BRL49653) is a PPARγ agonist, TRPC5 activator, and TRPM3 inhibitor with oral activity. Rosiglitazone is also a hypoglycemic agent and a thiazolidinedione insulin sensitizer.
  • $33
In Stock
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TargetMol | Inhibitor Hot