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PG 106 acetate
🥰Excellent
Catalog No. TP1952L
Alias PG 106 acetate(944111-22-2 Free base)
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.
PG 106 acetate
🥰Excellent
Purity: 98.24%
Catalog No. TP1952LAlias PG 106 acetate(944111-22-2 Free base)
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $74 | - | In Stock | |
| 5 mg | $251 | - | In Stock | |
| 10 mg | $358 | - | In Stock | |
| 25 mg | $541 | - | In Stock | |
| 50 mg | $721 | - | In Stock | |
| 100 mg | $987 | - | In Stock | |
| 200 mg | $1,310 | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Batch Information
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Purity:98.24%
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Product Introduction
Bioactivity
Chemical Properties
| Description | PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM. |
| Targets&IC50 | MC3R (human):210 nM |
| Synonyms | PG 106 acetate(944111-22-2 Free base) |
| Molecular Weight | 1068.23 |
| Formula | C53H73N13O11 |
| Smiles | CCCCC(NC(C)=O)C(N[C@H]1CC(NCCCC[C@@H](C(N)=O)NC([C@H](CC2=CNC3=CC=CC=C32)NC([C@H](CCC/N=C(N)\N)NC([C@@H](CC4=CC5=CC=CC=C5C=C4)NC(CCNC1=O)=O)=O)=O)=O)=O)=O.CC(O)=O |
| Color | White |
| Appearance | Solid |
| Sequence | Ac-DL-Nle-Asp(1)-bAla-D-2Nal-Arg-Trp-Lys(1)-NH2 |
| Sequence Short | Ac-{Nle}-D-{Bal}-{D-Nal}-RWK-NH2 (Lactam bridge:Asp2-Lys7) |
Storage & Solubility Information
| Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
Dose Conversion
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Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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