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TargetMol | Compound Library

Anti-Cancer Active Compound Library

Catalog No. L2160

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 4270 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2160

Anti-Cancer Active Compound Library

sizeIn stock

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 4270 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
PI3K
EGFR
ROS
Ras
VEGFR
Akt
Antibiotic
Parasite
Microtubule Associated
mTOR
Topoisomerase
Antifungal
Epigenetic Reader Domain
Caspase
Reactive Oxygen Species
ERK
Bcl-2 Family
FLT
Dehydrogenase
Nucleoside Antimetabolite/Analog
STAT
PDGFR
COX
PARP
Histone Methyltransferase
p38 MAPK
HDAC
FGFR
c-Met/HGFR
Estrogen Receptor/ERR
TNF
Wnt/beta-catenin
Cytochromes P450
HIV Protease
c-Kit
Ferroptosis
Interleukin
Src
Raf
JAK
MDM-2/p53
Phosphatase
HSP
Antioxidant
MMP
Virus Protease
Influenza Virus
Estrogen/progestogen Receptor
KRas
PKC
Bcr-Abl
AMPK
NO Synthase
ALK
Aurora Kinase
Androgen Receptor
PPAR
JNK
Calcium Channel
E1/E2/E3 Enzyme
Nrf2
P-gp
SARS-CoV
MEK
GSK-3
DUB
FAK
HIF/HIF Prolyl-Hydroxylase
IL Receptor
TLR
PROTACs
MAPK
p53
HSV
IGF-1R
DNA Alkylator/Crosslinker
Mitophagy
TGF-beta/Smad
Antiviral
Drug Metabolite
Mitochondrial Metabolism
c-RET
AChR
Histone Demethylase
PDE
Chk
Sirtuin
ATM/ATR
Proteasome
Gamma-secretase
Lipoxygenase
Potassium Channel
TAM Receptor
Tyrosine Kinases
HER
Trk receptor
c-Fms
DNA-PK
Pim
Adrenergic Receptor
Molecular Glues
Cholinesterase (ChE)
Histone Acetyltransferase
Sodium Channel
Mdm2
PERK
Casein Kinase
Retinoid Receptor
5-HT Receptor
S6 Kinase
Transferase
Hedgehog/Smoothened
HIF
ROS Kinase
Integrin
Reductase
Smo
PLK
DNA Methyltransferase
PD-1/PD-L1
ADC Cytotoxin
Serine Protease
IAP
Fatty Acid Synthase
GABA Receptor
Anti-infection
Kinesin
YAP
Histamine Receptor
HBV
Aryl Hydrocarbon Receptor
CXCR
HCV Protease
Glutathione Peroxidase
PKA
TRP/TRPV Channel
DNA Alkylation
Tyrosinase
LPL Receptor
Antifolate
Beta Amyloid
PDK
Phospholipase
Dopamine Receptor
c-Myc
IDO
Antifection
Isocitrate Dehydrogenase (IDH)
Ligands for E3 Ligase
Indoleamine 2,3-Dioxygenase (IDO)
S1P Receptor
BTK
GPCR
Carbonic Anhydrase
Serine/threonin kinase
DNA
transporter
IκB/IKK
Aromatase
DHFR
MAO
CSF-1R
Prostaglandin Receptor
IKZF
ATPase
NOS
Adenosine Receptor
DYRK
Rho
ROCK
Immunology/Inflammation related
CaMK
OXPHOS
Syk
Monocarboxylate transporter
NADPH
Cell Cycle Arrest
Glutaminase
glycosidase
Survivin
AhR
Monoamine Oxidase
IFNAR
Progesterone Receptor
Photosensitizer
Cysteine Protease
RIP kinase
Glucosidase
Telomerase
BCRP
STING
Ephrin Receptor
Reverse Transcriptase
NOD
Proton pump
Amino Acids and Derivatives
Tie-2
GNRH Receptor
Cholecystokinin Receptor
RANKL/RANK
Glucocorticoid Receptor
iGluR
Opioid Receptor
PAK
CCR
Wee1
Acyltransferase
MNK
PAI-1
Methionine Adenosyltransferase (MAT)
GPX
IRAK
NOD-like Receptor (NLR)
Chloride channel
MicroRNA
RAAS
Bcl-6
NAMPT
IRE1
P2X Receptor
ABC Transporter
Somatostatin
Lipid
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
ROR
Ligands for Target Protein for PROTAC
Necroptosis
ATG
Liver X Receptor
Leukotriene Receptor
Glucokinase
PYK2
UGT
Endothelin Receptor
Angiotensin-converting Enzyme (ACE)
GluR
Orphan Receptor
PSMA
Aminopeptidase
Pyroptosis
LPA Receptor
BMI-1
HMG-CoA Reductase
Thrombin
p97
PKM
MALT
GTPase
Galectin
Myosin
MTH1
NMDAR
Hexokinase
FAAH
PTEN
cAMP
MELK
p62
FOXO
Hydroxylase
Complement System
Neurokinin receptor
DAPK
NEDD8
CRM1
MyD88
LTR
Arrestin
Lipase
TOPK
Factor Xa
MRP
Serotonin Transporter
FXR
NR4A
GRK
Bombesin Receptor
ACK1
Xanthine Oxidase
PAD
KSP
Cadherin
Porcupine
CD73
Decarboxylase
ASK
GST
ribosome
KLF
CRISPR/Cas9
Adenosine Deaminase
SGK
Platelet aggregation
APC/C
Protease-activated Receptor
MLK
FOXO3
Thyroid hormone receptor(THR)
RAR/RXR
Factor VIIa
MIF
CaSR
Hck
Neurotensin Receptor
Vitamin
Adenylate cyclase
Annexin A
FLAP
Adiponectin Receptor
PAFR
Haspin Kinase
Arp2/3 Complex
DNA gyrase
Stearoyl-CoA Desaturase (SCD)
Vasopressin Receptor
Thrombopoietin Receptor
ATP Citrate Lyase
GPCR19
E3 Ligase Ligand-Linker Conjugates
HuR
RSV
Drug-Linker Conjugates for ADC
Hippo pathway
Acetyl-CoA Carboxylase
FKBP
Protease
PI4K
Cuproptosis
Gap Junction Protein
Sigma receptor
Lysosomal Autophagy
CFTR
PARG(Poly(ADP-ribose) Glycohydrolase)
Apelin receptor
Advanced Glycation End Products
CAT
NPC1L1
CD38
CYP19A1
NUDIX hydrolase
Dynamin
Y Box Binding Protein 1
Arginase
P2Y Receptor
Na+/Ca2+ Exchanger
gp120/CD4
VDA
Melatonin Receptor
OCT
Kisspeptin
B7
Target Protein Ligand-Linker Conjugates
Stemness kinase
LDLR
Amylase
LAG-3
SIK
Prolyl Endopeptidase (PREP)
FABP
LDL
GlyT
Na-K-Cl cotransporter
PROTAC Linker
DPP-4
Neuropeptide Y Receptor
Thioredoxin
HCAR
Epoxide Hydrolase
Transketolase
SGLT
PGE Synthase
Beta-Secretase
Glutathione reductase
LRRK2
Free radical scavengers
Urea Transporter
GluCls
NEDD4-1
Carboxypeptidase
TMV
Melanocortin Receptor
Oxytocin Receptor
GHSR
Aquaporin
RXFP receptor
NADPH-oxidase
Tight Junction Protein
Liposome
Glyoxalase
Ferroportin
ADC Linker
Poly(ADP-ribose) Glycohydrolase (PARG)

Keywords