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TargetMol | Compound Library

Anti-Cancer Active Compound Library

Catalog No. L2160

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 4270 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2160

Anti-Cancer Active Compound Library

sizeIn stock

  • 1 mg
  • 10 µL x 10 mM (in DMSO)
  • 20 µL x 10 mM (in DMSO)
  • 30 µL x 10 mM (in DMSO)
  • 50 µL x 10 mM (in DMSO)
  • 100 µL x 10 mM (in DMSO)
  • 250 µL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 4270 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
PI3K
EGFR
ROS
Ras
VEGFR
Akt
Antibiotic
Microtubule Associated
Parasite
mTOR
Topoisomerase
Epigenetic Reader Domain
Antifungal
Caspase
Reactive Oxygen Species
ERK
Bcl-2 Family
FLT
Dehydrogenase
STAT
Nucleoside Antimetabolite/Analog
COX
PDGFR
HDAC
PARP
p38 MAPK
Histone Methyltransferase
FGFR
c-Met/HGFR
TNF
Estrogen Receptor/ERR
Wnt/beta-catenin
Cytochromes P450
c-Kit
HIV Protease
Ferroptosis
Interleukin
Raf
Src
MDM-2/p53
JAK
Phosphatase
HSP
MMP
Antioxidant
Virus Protease
Influenza Virus
Estrogen/progestogen Receptor
Kras
PKC
AMPK
Bcr-Abl
NO Synthase
ALK
Aurora Kinase
Androgen Receptor
PPAR
E1/E2/E3 Enzyme
JNK
Calcium Channel
Nrf2
MEK
SARS-CoV
P-gp
DUB
HIF/HIF Prolyl-Hydroxylase
GSK-3
FAK
IL Receptor
TLR
PROTACs
MAPK
p53
HSV
IGF-1R
Antiviral
Mitophagy
TGF-beta/Smad
DNA Alkylator/Crosslinker
Mitochondrial Metabolism
c-RET
AChR
Drug Metabolite
Chk
Histone Demethylase
Sirtuin
PDE
ATM/ATR
Gamma-secretase
Potassium Channel
Lipoxygenase
Proteasome
TAM Receptor
Tyrosine Kinases
HER
Trk receptor
c-Fms
Pim
Adrenergic Receptor
Molecular Glues
Histone Acetyltransferase
Sodium Channel
DNA-PK
5-HT Receptor
S6 Kinase
PERK
Cholinesterase (ChE)
Casein Kinase
Mdm2
Retinoid Receptor
Transferase
HIF
ROS Kinase
Hedgehog/Smoothened
PLK
DNA Methyltransferase
PD-1/PD-L1
Integrin
Reductase
Smo
ADC Cytotoxin
Serine Protease
Anti-infection
IAP
Kinesin
YAP
HBV
GABA Receptor
Histamine Receptor
Fatty Acid Synthase
Aryl Hydrocarbon Receptor
CXCR
TRP/TRPV Channel
PKA
DNA Alkylation
HCV Protease
Glutathione Peroxidase
Tyrosinase
Beta Amyloid
PDK
Phospholipase
LPL Receptor
Antifolate
S1P Receptor
IDO
c-Myc
Isocitrate Dehydrogenase (IDH)
Dopamine Receptor
Antifection
Ligands for E3 Ligase
Indoleamine 2,3-Dioxygenase (IDO)
BTK
transporter
Carbonic Anhydrase
DNA
GPCR
IκB/IKK
Serine/threonin kinase
MAO
Aromatase
DHFR
CSF-1R
Prostaglandin Receptor
IKZF
Immunology/Inflammation related
Syk
ROCK
CaMK
ATPase
Adenosine Receptor
DYRK
Rho
NOS
OXPHOS
Cell Cycle Arrest
NADPH
AhR
Monoamine Oxidase
glycosidase
Glutaminase
Survivin
Monocarboxylate transporter
IFNAR
Telomerase
Progesterone Receptor
Photosensitizer
Ephrin Receptor
Reverse Transcriptase
NOD
Glucosidase
RIP kinase
BCRP
Cysteine Protease
STING
Amino Acids and Derivatives
MNK
RANKL/RANK
Glucocorticoid Receptor
NOD-like Receptor (NLR)
iGluR
CCR
GNRH Receptor
PAK
PAI-1
IRAK
Tie-2
Cholecystokinin Receptor
Acyltransferase
Wee1
Methionine Adenosyltransferase (MAT)
Proton pump
Opioid Receptor
GPX
MicroRNA
Bcl-6
ABC Transporter
NAMPT
RAAS
P2X Receptor
Somatostatin
Discoidin Domain Receptor (DDR)
Chloride channel
IRE1
Cannabinoid Receptor
ROR
Ligands for Target Protein for PROTAC
Glucokinase
Angiotensin-converting Enzyme (ACE)
Orphan Receptor
Necroptosis
Lipid
PSMA
LPA Receptor
BMI-1
Thrombin
ATG
GluR
Liver X Receptor
Endothelin Receptor
PYK2
UGT
Aminopeptidase
HMG-CoA Reductase
p97
Leukotriene Receptor
Pyroptosis
PKM
FOXO
Galectin
MTH1
NMDAR
Hexokinase
Complement System
FAAH
p62
Hydroxylase
GTPase
cAMP
MELK
GST
Myosin
Neurokinin receptor
DAPK
MALT
PTEN
Lipase
KLF
GRK
Bombesin Receptor
ACK1
SGK
NEDD8
LTR
NR4A
Porcupine
CD73
ribosome
CRISPR/Cas9
Factor Xa
Platelet aggregation
TOPK
Serotonin Transporter
Decarboxylase
Adenosine Deaminase
APC/C
CRM1
MRP
PAD
ASK
Protease-activated Receptor
MyD88
Arrestin
FXR
Xanthine Oxidase
KSP
Cadherin
MLK
PAFR
Haspin Kinase
GPCR19
RSV
Drug-Linker Conjugates for ADC
Protease
PI4K
Hck
Annexin A
Arp2/3 Complex
Stearoyl-CoA Desaturase (SCD)
HuR
FOXO3
Factor VIIa
Vitamin
Adiponectin Receptor
ATP Citrate Lyase
E3 Ligase Ligand-Linker Conjugates
Hippo pathway
Sigma receptor
CFTR
CaSR
Vasopressin Receptor
Gap Junction Protein
Lysosomal Autophagy
Thyroid hormone receptor(THR)
FLAP
Beta-Secretase
MIF
Neurotensin Receptor
Adenylate cyclase
Thrombopoietin Receptor
Cuproptosis
RAR/RXR
DNA gyrase
Acetyl-CoA Carboxylase
FKBP
PARG(Poly(ADP-ribose) Glycohydrolase)
Apelin receptor
CYP19A1
Dynamin
P2Y Receptor
B7
DPP-4
HCAR
NEDD4-1
Tight Junction Protein
Advanced Glycation End Products
NUDIX hydrolase
BACE
OCT
Stemness kinase
Na-K-Cl cotransporter
Neuropeptide Y Receptor
SGLT
TMV
CD38
VDA
Target Protein Ligand-Linker Conjugates
LAG-3
PROTAC Linker
Transketolase
CAT
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
Carboxypeptidase
Melanocortin Receptor
Oxytocin Receptor
GHSR
NPC1L1
Kisspeptin
LDLR
SIK
Thioredoxin
Glutathione reductase
Liposome
GlyT
PGE Synthase
Urea Transporter
Aquaporin
Melatonin Receptor
Amylase
Prolyl Endopeptidase (PREP)
FABP
LDL
Epoxide Hydrolase
LRRK2
Free radical scavengers
GluCls
RXFP receptor
NADPH-oxidase
Glyoxalase
Poly(ADP-ribose) Glycohydrolase (PARG)
ADC Linker
Ferroportin

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