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TargetMol | Compound Library

Anti-Cancer Active Compound Library

Catalog No. L2160

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 4270 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2160

Anti-Cancer Active Compound Library

sizeIn stock

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 4270 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
PI3K
EGFR
ROS
Ras
VEGFR
Akt
Antibiotic
Parasite
Microtubule Associated
Topoisomerase
mTOR
Epigenetic Reader Domain
Caspase
Antifungal
Reactive Oxygen Species
Bcl-2 Family
ERK
FLT
Dehydrogenase
COX
Nucleoside Antimetabolite/Analog
STAT
PDGFR
Histone Methyltransferase
PARP
FGFR
HDAC
p38 MAPK
c-Met/HGFR
TNF
Estrogen Receptor/ERR
Cytochromes P450
Wnt/beta-catenin
c-Kit
HIV Protease
Ferroptosis
Src
Raf
Interleukin
MDM-2/p53
Phosphatase
JAK
HSP
Antioxidant
MMP
Virus Protease
Influenza Virus
Estrogen/progestogen Receptor
Kras
PKC
Bcr-Abl
NO Synthase
AMPK
ALK
Aurora Kinase
Androgen Receptor
PPAR
Nrf2
JNK
MEK
P-gp
E1/E2/E3 Enzyme
Calcium Channel
SARS-CoV
FAK
DUB
HIF/HIF Prolyl-Hydroxylase
GSK-3
TLR
IL Receptor
MAPK
p53
PROTACs
DNA Alkylator/Crosslinker
HSV
IGF-1R
Mitophagy
TGF-beta/Smad
Antiviral
Drug Metabolite
Sirtuin
Mitochondrial Metabolism
c-RET
AChR
PDE
Histone Demethylase
Chk
Lipoxygenase
ATM/ATR
Gamma-secretase
Potassium Channel
Proteasome
TAM Receptor
Tyrosine Kinases
HER
Histone Acetyltransferase
Trk receptor
c-Fms
Pim
Molecular Glues
S6 Kinase
Cholinesterase (ChE)
Sodium Channel
DNA-PK
Adrenergic Receptor
5-HT Receptor
Retinoid Receptor
PERK
Casein Kinase
Transferase
Mdm2
HIF
ROS Kinase
Hedgehog/Smoothened
DNA Methyltransferase
GABA Receptor
PD-1/PD-L1
PLK
Reductase
Smo
ADC Cytotoxin
Anti-infection
Fatty Acid Synthase
Kinesin
CXCR
IAP
Serine Protease
Integrin
YAP
Aryl Hydrocarbon Receptor
HBV
Histamine Receptor
TRP/TRPV Channel
PDK
HCV Protease
Glutathione Peroxidase
Tyrosinase
PKA
DNA Alkylation
LPL Receptor
Antifolate
c-Myc
Phospholipase
IDO
Beta Amyloid
Dopamine Receptor
Antifection
Ligands for E3 Ligase
Indoleamine 2,3-Dioxygenase (IDO)
Serine/threonin kinase
Isocitrate Dehydrogenase (IDH)
S1P Receptor
BTK
transporter
Carbonic Anhydrase
DNA
GPCR
Aromatase
IκB/IKK
Prostaglandin Receptor
MAO
Immunology/Inflammation related
Syk
DHFR
CSF-1R
IKZF
NADPH
ROCK
CaMK
NOS
OXPHOS
ATPase
Adenosine Receptor
DYRK
Rho
AhR
Monoamine Oxidase
Glutaminase
Survivin
Monocarboxylate transporter
Cysteine Protease
glycosidase
Cell Cycle Arrest
IFNAR
Telomerase
RIP kinase
BCRP
STING
Progesterone Receptor
Photosensitizer
Ephrin Receptor
Reverse Transcriptase
Glucosidase
RANKL/RANK
Glucocorticoid Receptor
NOD-like Receptor (NLR)
Wee1
Methionine Adenosyltransferase (MAT)
Proton pump
Opioid Receptor
GPX
iGluR
CCR
PAK
PAI-1
NOD
IRAK
Amino Acids and Derivatives
MNK
Tie-2
Cholecystokinin Receptor
Acyltransferase
Bcl-6
Lipid
P2X Receptor
Somatostatin
Discoidin Domain Receptor (DDR)
Chloride channel
IRE1
Cannabinoid Receptor
ABC Transporter
GNRH Receptor
NAMPT
MicroRNA
Necroptosis
PSMA
LPA Receptor
BMI-1
Thrombin
PYK2
UGT
HMG-CoA Reductase
p97
Leukotriene Receptor
Pyroptosis
PKM
ATG
GluR
Liver X Receptor
ROR
Ligands for Target Protein for PROTAC
Glucokinase
Angiotensin-converting Enzyme (ACE)
Orphan Receptor
RAAS
Endothelin Receptor
Aminopeptidase
DAPK
MALT
PTEN
FAAH
p62
Hydroxylase
GTPase
cAMP
MELK
Galectin
MTH1
NMDAR
Hexokinase
Complement System
Myosin
FOXO
Neurokinin receptor
GRK
Bombesin Receptor
ACK1
SGK
CRM1
MRP
PAD
ASK
Protease-activated Receptor
MyD88
Arrestin
FXR
Xanthine Oxidase
KSP
Cadherin
MLK
NEDD8
LTR
NR4A
Porcupine
CD73
ribosome
CRISPR/Cas9
Factor Xa
GST
Platelet aggregation
Lipase
KLF
TOPK
Serotonin Transporter
Decarboxylase
Adenosine Deaminase
APC/C
FOXO3
Hck
Annexin A
Arp2/3 Complex
Stearoyl-CoA Desaturase (SCD)
HuR
MIF
Neurotensin Receptor
Thrombopoietin Receptor
Cuproptosis
RAR/RXR
DNA gyrase
Acetyl-CoA Carboxylase
FKBP
Factor VIIa
Vitamin
Adiponectin Receptor
ATP Citrate Lyase
E3 Ligase Ligand-Linker Conjugates
Hippo pathway
Sigma receptor
CFTR
CaSR
Gap Junction Protein
Lysosomal Autophagy
PAFR
Haspin Kinase
GPCR19
RSV
Drug-Linker Conjugates for ADC
Protease
PI4K
Thyroid hormone receptor(THR)
FLAP
PARG(Poly(ADP-ribose) Glycohydrolase)
Advanced Glycation End Products
NUDIX hydrolase
OCT
Stemness kinase
Na-K-Cl cotransporter
Neuropeptide Y Receptor
SGLT
TMV
Adenylate cyclase
GlyT
PGE Synthase
Urea Transporter
Aquaporin
Melatonin Receptor
Amylase
Prolyl Endopeptidase (PREP)
FABP
LDL
Epoxide Hydrolase
LRRK2
Free radical scavengers
GluCls
RXFP receptor
NADPH-oxidase
Glyoxalase
CD38
VDA
Target Protein Ligand-Linker Conjugates
LAG-3
PROTAC Linker
Transketolase
CAT
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
Vasopressin Receptor
Carboxypeptidase
Melanocortin Receptor
GHSR
Apelin receptor
CYP19A1
Dynamin
P2Y Receptor
B7
LIM Kinase
DPP-4
HCAR
NEDD4-1
Tight Junction Protein
NPC1L1
Kisspeptin
AAK1
LDLR
SIK
Thioredoxin
Beta-Secretase
Glutathione reductase
Liposome
Poly(ADP-ribose) Glycohydrolase (PARG)
ADC Linker
Ferroportin

Keywords