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TargetMol | Compound Library

Anti-Cancer Active Compound Library

Catalog No. L2160

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 4270 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2160

Anti-Cancer Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 4270 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
PI3K
EGFR
ROS
Ras
VEGFR
Akt
Antibiotic
Parasite
Microtubule Associated
Topoisomerase
mTOR
Epigenetic Reader Domain
Caspase
Antifungal
Reactive Oxygen Species
Bcl-2 Family
ERK
Dehydrogenase
COX
FLT
Nucleoside Antimetabolite/Analog
STAT
PDGFR
PARP
p38 MAPK
Histone Methyltransferase
HDAC
FGFR
Estrogen Receptor/ERR
TNF
Wnt/beta-catenin
c-Met/HGFR
Cytochromes P450
c-Kit
HIV Protease
Ferroptosis
Src
Raf
Interleukin
MDM-2/p53
JAK
HSP
Phosphatase
Antioxidant
MMP
Virus Protease
Influenza Virus
Estrogen/progestogen Receptor
Kras
PKC
AMPK
NO Synthase
Bcr-Abl
ALK
Aurora Kinase
Androgen Receptor
PPAR
JNK
Nrf2
MEK
Calcium Channel
SARS-CoV
P-gp
E1/E2/E3 Enzyme
DUB
HIF/HIF Prolyl-Hydroxylase
GSK-3
FAK
IL Receptor
MAPK
TLR
p53
PROTACs
Mitophagy
TGF-beta/Smad
DNA Alkylator/Crosslinker
HSV
IGF-1R
Antiviral
Mitochondrial Metabolism
c-RET
AChR
Drug Metabolite
Sirtuin
Chk
PDE
Histone Demethylase
ATM/ATR
Lipoxygenase
Gamma-secretase
Potassium Channel
Proteasome
TAM Receptor
Tyrosine Kinases
HER
Trk receptor
c-Fms
Histone Acetyltransferase
Pim
Molecular Glues
S6 Kinase
DNA-PK
Cholinesterase (ChE)
Sodium Channel
Adrenergic Receptor
5-HT Receptor
Retinoid Receptor
PERK
Casein Kinase
Transferase
Hedgehog/Smoothened
Mdm2
HIF
ROS Kinase
DNA Methyltransferase
PLK
Reductase
Smo
GABA Receptor
PD-1/PD-L1
ADC Cytotoxin
Serine Protease
Integrin
CXCR
Fatty Acid Synthase
Kinesin
IAP
YAP
Anti-infection
Histamine Receptor
Aryl Hydrocarbon Receptor
HBV
TRP/TRPV Channel
PDK
PKA
DNA Alkylation
HCV Protease
Glutathione Peroxidase
Tyrosinase
Beta Amyloid
LPL Receptor
Antifolate
c-Myc
IDO
S1P Receptor
Phospholipase
Serine/threonin kinase
Dopamine Receptor
Antifection
Ligands for E3 Ligase
Indoleamine 2,3-Dioxygenase (IDO)
Isocitrate Dehydrogenase (IDH)
transporter
IκB/IKK
Carbonic Anhydrase
DNA
GPCR
BTK
Aromatase
Immunology/Inflammation related
Syk
DHFR
CSF-1R
Prostaglandin Receptor
MAO
IKZF
NADPH
ROCK
NOS
OXPHOS
ATPase
Adenosine Receptor
DYRK
Rho
CaMK
AhR
Monoamine Oxidase
Cell Cycle Arrest
Monocarboxylate transporter
Cysteine Protease
Glutaminase
Survivin
glycosidase
Photosensitizer
IFNAR
Telomerase
Glucosidase
STING
RIP kinase
BCRP
Progesterone Receptor
Ephrin Receptor
Reverse Transcriptase
RANKL/RANK
Glucocorticoid Receptor
NOD-like Receptor (NLR)
Amino Acids and Derivatives
MNK
Tie-2
Cholecystokinin Receptor
Acyltransferase
Proton pump
Opioid Receptor
GPX
Wee1
Methionine Adenosyltransferase (MAT)
iGluR
CCR
GNRH Receptor
PAK
PAI-1
NOD
IRAK
Bcl-6
Lipid
MicroRNA
Chloride channel
IRE1
Cannabinoid Receptor
P2X Receptor
Somatostatin
Discoidin Domain Receptor (DDR)
ABC Transporter
NAMPT
Necroptosis
PSMA
LPA Receptor
BMI-1
Thrombin
ROR
Ligands for Target Protein for PROTAC
Glucokinase
Angiotensin-converting Enzyme (ACE)
Orphan Receptor
RAAS
Endothelin Receptor
Leukotriene Receptor
Pyroptosis
PKM
PYK2
UGT
HMG-CoA Reductase
p97
ATG
GluR
Liver X Receptor
Galectin
MTH1
NMDAR
Hexokinase
Complement System
Myosin
FOXO
Neurokinin receptor
MALT
PTEN
Aminopeptidase
DAPK
FAAH
p62
Hydroxylase
GTPase
cAMP
MELK
GRK
Bombesin Receptor
ACK1
SGK
Lipase
KLF
TOPK
Serotonin Transporter
Decarboxylase
Adenosine Deaminase
APC/C
MyD88
Arrestin
FXR
Xanthine Oxidase
KSP
Cadherin
MLK
CRM1
MRP
PAD
ASK
Protease-activated Receptor
NEDD8
LTR
NR4A
Porcupine
CD73
ribosome
CRISPR/Cas9
Factor Xa
GST
Platelet aggregation
FOXO3
Hck
Annexin A
Arp2/3 Complex
Stearoyl-CoA Desaturase (SCD)
HuR
PAFR
Haspin Kinase
GPCR19
RSV
Drug-Linker Conjugates for ADC
Protease
PI4K
Thyroid hormone receptor(THR)
FLAP
Beta-Secretase
RAR/RXR
DNA gyrase
Acetyl-CoA Carboxylase
FKBP
MIF
Neurotensin Receptor
Thrombopoietin Receptor
Cuproptosis
Factor VIIa
Vitamin
Adiponectin Receptor
ATP Citrate Lyase
E3 Ligase Ligand-Linker Conjugates
Hippo pathway
Sigma receptor
CFTR
CaSR
Gap Junction Protein
Lysosomal Autophagy
PARG(Poly(ADP-ribose) Glycohydrolase)
Advanced Glycation End Products
NUDIX hydrolase
BACE
OCT
Stemness kinase
Na-K-Cl cotransporter
Neuropeptide Y Receptor
SGLT
TMV
Apelin receptor
CYP19A1
Dynamin
P2Y Receptor
B7
LIM Kinase
DPP-4
HCAR
NEDD4-1
Tight Junction Protein
NPC1L1
Kisspeptin
AAK1
LDLR
SIK
Thioredoxin
Glutathione reductase
Liposome
Melatonin Receptor
Amylase
Prolyl Endopeptidase (PREP)
FABP
LDL
Epoxide Hydrolase
LRRK2
Free radical scavengers
GluCls
RXFP receptor
NADPH-oxidase
Glyoxalase
Adenylyl Cyclase
GlyT
PGE Synthase
Urea Transporter
Aquaporin
CD38
VDA
Target Protein Ligand-Linker Conjugates
LAG-3
Monoamine Transporter
PROTAC Linker
Transketolase
CAT
Y Box Binding Protein 1
Arginase
Na+/Ca2+ Exchanger
gp120/CD4
Vasopressin Receptor
Carboxypeptidase
Melanocortin Receptor
GHSR
Poly(ADP-ribose) Glycohydrolase (PARG)
ADC Linker
Ferroportin

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