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A09-003

Catalog No. T79404 CAS 2911646-14-3

A09-003 is a novel cell cycle protein-dependent kinase-9 CDK-9 inhibitor.A09-003 inhibits the proliferation of a variety of leukemia cell lines and inhibits the increase of leukemia sequence-1 protein in myeloid cells.A09-003 also induces apoptosis, decreases RNA polymerase II activity, and decreases Mcl-1 expression.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

A09-003, CAS 2911646-14-3

Pack Size	Availability	Price/USD
1 mg	In stock	$ 293.00
5 mg	In stock	$ 722.00
10 mg	In stock	$ 987.00
25 mg	In stock	$ 1,520.00
50 mg	In stock	$ 1,980.00
100 mg	In stock	$ 2,500.00

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Purity: 99.84%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Molecular Weight	374.48
Formula	C23H26N4O
CAS No.	2911646-14-3

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Sim KM, et al. A new cyclin-dependent kinase-9 inhibitor A09-003 induces apoptosis in acute myeloid leukemia cells with reduction of myeloid cell leukemia sequence-1 protein. Chem Biol Interact. 2023 Sep 1;382:110554.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

A09-003 2911646-14-3 Apoptosis Cell Cycle/Checkpoint BCL CDK inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.