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PI3Kδ/BET-IN-1

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Catalog No. T204249Cas No. 3054869-10-9

PI3Kδ/BET-IN-1 (compound 10b) exhibits excellent and balanced activity against PI3Kδ (IC50= 112 nM) and BRD4-BD1 (IC50= 19 nM), while also demonstrating strong antiproliferative effects in DLBCL cells.

PI3Kδ/BET-IN-1

PI3Kδ/BET-IN-1

😃Good
Catalog No. T204249Cas No. 3054869-10-9
PI3Kδ/BET-IN-1 (compound 10b) exhibits excellent and balanced activity against PI3Kδ (IC50= 112 nM) and BRD4-BD1 (IC50= 19 nM), while also demonstrating strong antiproliferative effects in DLBCL cells.
Pack SizePriceAvailabilityQuantity
10 mgInquiry10-14 weeks
50 mgInquiry10-14 weeks
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Product Introduction

Bioactivity
Description
PI3Kδ/BET-IN-1 (compound 10b) exhibits excellent and balanced activity against PI3Kδ (IC50= 112 nM) and BRD4-BD1 (IC50= 19 nM), while also demonstrating strong antiproliferative effects in DLBCL cells.
Targets&IC50
BRD4 BD1:19 nM
Chemical Properties
Molecular Weight522.662
FormulaC27H34N6O3S
Cas No.3054869-10-9
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice./Shipping at ambient temperature.

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