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PW0464 ((Rac)-Razpipadon) is a non-catechol D1R agonist and potent omplete G protein biased ligand with an EC50 (Gs-cAMP)=5.8 nM for the study of neurological disorders.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $166 | In Stock | |
5 mg | $416 | In Stock | |
10 mg | $695 | In Stock | |
25 mg | $1,330 | In Stock | |
50 mg | $1,980 | In Stock | |
1 mL x 10 mM (in DMSO) | $458 | In Stock |
Description | PW0464 ((Rac)-Razpipadon) is a non-catechol D1R agonist and potent omplete G protein biased ligand with an EC50 (Gs-cAMP)=5.8 nM for the study of neurological disorders. |
Targets&IC50 | cAMP assay (HEK293T cells):5.8 nM (EC₅₀) |
In vitro | PW0464 is a non-catechol selective dopamine D1/D5 receptor agonist. In HEK293T cells overexpressing D1R or D5R, PW0464 activates G-protein signaling (cAMP production) with an EC₅₀ of 5.8 nM, indicating high potency[1]. |
Alias | PW 0464, (Rac)-Razpipadon |
Molecular Weight | 389.35 |
Formula | C19H17F2N3O4 |
Cas No. | 1643462-93-4 |
Smiles | O=C1NC(=O)N(C(C=2C=CC(OC3=NC=CC=C3OC(F)F)=CC2C)=C1C)C |
Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice./Shipping at ambient temperature. | |||||||||||||||||||||||||
Solubility Information | DMSO: 18 mg/mL (46.23 mM), Sonication is recommended. | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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