Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PW0464, a nanomolar potent complete G protein biased ligand, is a noncatechol D1R agonist, with an EC50 of 5.8 nM (Gs-cAMP)[1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 8-10 weeks | $ 1,530.00 | |
50 mg | 8-10 weeks | $ 1,990.00 | |
100 mg | 8-10 weeks | $ 3,100.00 |
Description | PW0464, a nanomolar potent complete G protein biased ligand, is a noncatechol D1R agonist, with an EC50 of 5.8 nM (Gs-cAMP)[1]. |
In vitro | PW0464 (compound 24) is found to elicit complete G protein bias, showing no activity for D1R-mediated β-arrestin recruitment[1].PW0464 (compound 24), the non-catechol agonist, forms bonds with S1985.42 and S2025.46 via its fluorine atom[2]. |
Synonyms | PW0464 |
Molecular Weight | 389.35 |
Formula | C19H17F2N3O4 |
CAS No. | 1643462-93-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
PW0464 1643462-93-4 PW-0464 PW 0464 inhibitor inhibit