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VPC-13566

Name: VPC-13566
Brand: TargetMol
SKU: T29111
Price: 40 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T29111Cas No. 218464-59-6

VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines and reduces the growth of AR-dependent prostate cancer xenograft tumors in mice.

VPC-13566

🥰Excellent

Purity: 99.55%

Catalog No. T29111Cas No. 218464-59-6

Pack Size	Price	Availability
1 mg	$40	In Stock
5 mg	$98	In Stock
10 mg	$163	In Stock
25 mg	$290	In Stock
50 mg	$466	In Stock
100 mg	$700	In Stock
200 mg	$969	In Stock
1 mL x 10 mM (in DMSO)	$116	In Stock

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Bulk & Custom

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.55%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description

Chemical Properties

Molecular Weight	258.32
Formula	C₁₈H₁₄N₂
Cas No.	218464-59-6
Smiles	CC1=C2C(C(=CN2)C3=NC4=C(C=C3)C=CC=C4)=CC=C1
Relative Density.	1.225 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 65 mg/mL (251.63 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.8712 mL	19.3558 mL	38.7117 mL	193.5584 mL
5 mM	0.7742 mL	3.8712 mL	7.7423 mL	38.7117 mL
10 mM	0.3871 mL	1.9356 mL	3.8712 mL	19.3558 mL
20 mM	0.1936 mL	0.9678 mL	1.9356 mL	9.6779 mL
50 mM	0.0774 mL	0.3871 mL	0.7742 mL	3.8712 mL
100 mM	0.0387 mL	0.1936 mL	0.3871 mL	1.9356 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc