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Potent Nav1.7 blocker (IC50 = 2.5 nM). Also inhibits Nav1.1, Nav1.2, Nav1.3 and Nav1.6 in the nanomolar range. Exhibits no effects on Cav channels or nAChR at 5 μM. Demonstrates analgesic activity in vivo; antagonizes effects of scorpion-venom toxin OD1 at Nav1.7.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
10 mg | $2,095 | Backorder |
Description | Potent Nav1.7 blocker (IC50 = 2.5 nM). Also inhibits Nav1.1, Nav1.2, Nav1.3 and Nav1.6 in the nanomolar range. Exhibits no effects on Cav channels or nAChR at 5 μM. Demonstrates analgesic activity in vivo; antagonizes effects of scorpion-venom toxin OD1 at Nav1.7. |
Molecular Weight | 3802.41 |
Formula | C162H246N52O43S6 |
Relative Density. | no data available |
Sequence | H-Asp-D-Cys(1)-D-Leu-Lys-D-Phe-Gly-D-Trp-D-Lys-Cys(2)-D-Asn-D-Pro-D-Arg-D-Asn-D-Asp-D-Lys-D-Cys(3)-Cys(1)-D-Ser-Gly-D-Leu-D-Lys-Cys(2)-Gly-D-Ser-D-Asn-His-D-Asn-D-Trp-Cys(3)-D-Lys-D-Leu-D-His-aIle-OH |
Sequence Short | DCLKFGWKCNPRNDKCCSGLKCGSNHNWCKLHX |
Storage | keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
Solubility Information | H2O: 1 mg/mL (0.26 mM), Sonication is recommended. |
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