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Lu AA33810
🥰Excellent
Catalog No. T22935Cas No. 304008-29-5
Alias LuAA33810, Lu AA-33810
Lu AA33810 is a selective neuropeptide Y5 (NPY5) receptor antagonist with an oral activity and blood-brain barrier permeability advantage, exhibiting anti-anxiety and antidepressant-like effects at a Ki = 1.5 nM for rat receptors.
Lu AA33810
🥰Excellent
Purity: 97.92%
Catalog No. T22935Alias LuAA33810, Lu AA-33810Cas No. 304008-29-5
Lu AA33810 is a selective neuropeptide Y5 (NPY5) receptor antagonist with an oral activity and blood-brain barrier permeability advantage, exhibiting anti-anxiety and antidepressant-like effects at a Ki = 1.5 nM for rat receptors.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $163 | - | In Stock | |
| 5 mg | $408 | - | In Stock | |
| 10 mg | $711 | - | In Stock | |
| 25 mg | $1,080 | - | In Stock | |
| 50 mg | $1,480 | - | In Stock | |
| 100 mg | $1,960 | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:97.92%
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Product Introduction
Bioactivity
Chemical Properties
| Description | Lu AA33810 is a selective neuropeptide Y5 (NPY5) receptor antagonist with an oral activity and blood-brain barrier permeability advantage, exhibiting anti-anxiety and antidepressant-like effects at a Ki = 1.5 nM for rat receptors. |
| Targets&IC50 | Y5 receptor (human):1.5 nM (Ki) |
| In vivo | Lu AA33810 (3-30 mg/kg, oral administration) showed anxiolytic-like effects in SD rats tested with the social interaction test [1]. Lu AA33810 (10 mg/kg/day, intraperitoneal injection) exhibited anxiolytic-like effects in the social interaction test of Flinders Sensitive Line rats and demonstrated antidepressant-like effects in the forced swim test [1]. Lu AA33810 (3 and 10 mg/kg/day, intraperitoneal injection) produced antidepressant-like activity in Wistar rats subjected to chronic mild stress, restoring the stress-induced decrease in sucrose consumption [1]. |
| Synonyms | LuAA33810, Lu AA-33810 |
| Molecular Weight | 423.62 |
| Formula | C19H25N3O2S3 |
| Cas No. | 304008-29-5 |
| Smiles | N(C1=NC=2C=3C(SCCC2S1)=CC=CC3)[C@@H]4CC[C@@H](CNS(C)(=O)=O)CC4 |
| Relative Density. | no data available |
| Color | White |
| Appearance | Solid |
Storage & Solubility Information
| Storage | store at low temperature,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | ||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 32 mg/mL (75.54 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
DMSO
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
Dose Conversion
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Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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