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G-6599
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Catalog No. T206987Cas No. 2901806-51-5
G-6599 is a monovalent degrader targeting SMARCA2/A4, with DC50 values of 0.018 nM and 0.056 nM, respectively. It demonstrates degradation activity and antiproliferative effects in AR-dependent prostate cancer cell lines.
G-6599
😃Good
Catalog No. T206987Cas No. 2901806-51-5
G-6599 is a monovalent degrader targeting SMARCA2/A4, with DC50 values of 0.018 nM and 0.056 nM, respectively. It demonstrates degradation activity and antiproliferative effects in AR-dependent prostate cancer cell lines.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 10 mg | Inquiry | 10-14 weeks | |
| 50 mg | Inquiry | 10-14 weeks |
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Product Introduction
Bioactivity
Chemical Properties
| Description | G-6599 is a monovalent degrader targeting SMARCA2/A4, with DC50 values of 0.018 nM and 0.056 nM, respectively. It demonstrates degradation activity and antiproliferative effects in AR-dependent prostate cancer cell lines. |
| Molecular Weight | 523.672 |
| Formula | C31H37N7O |
| Cas No. | 2901806-51-5 |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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