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CP-409092

Name: CP-409092
Brand: TargetMol
SKU: T10869L
Rating: 4.5 (1 reviews)

😃Good

Catalog No. T10869LCas No. 194098-25-4

CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.

CP-409092

😃Good

Catalog No. T10869LCas No. 194098-25-4

CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.

Pack Size	Price	USA Warehouse	Global Warehouse
25 mg	$1,820	8-10 weeks	8-10 weeks
50 mg	$2,380	8-10 weeks	8-10 weeks
100 mg	$3,100	8-10 weeks	8-10 weeks

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Product Introduction

Bioactivity

Description	CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.
In vivo	[14C]CP-409,092(P.O.; 100 mg/kg; ) treatment, the total recovery is 89.1%+ or -3.2% for male rats and 89.3%+ or -0.58% for female rats. The pharmacokinetics of CP-409,092 (P.O.; 4 and 15 mg/kg;single intravenous) treatment , are characterized by high clearance of 169+ or -18 mL/min/kg, a volume of distribution of 8.99+ or -1.46 L/kg, and an oral bioavailability of 2.9%+ or -3%.

Chemical Properties

Molecular Weight	297.35
Formula	C₁₇H₁₉N₃O₂
Cas No.	194098-25-4
Relative Density.	1.283 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 41.67 mg/mL (140.14 mM), Sonication is recommended.

In Vivo Formulation

10% DMSO+40% PEG300+5% Tween-80+45% Saline: 2 mg/mL (6.73 mM), Sonication is recommeded.

Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.3630 mL	16.8152 mL	33.6304 mL	168.1520 mL
5 mM	0.6726 mL	3.3630 mL	6.7261 mL	33.6304 mL
10 mM	0.3363 mL	1.6815 mL	3.3630 mL	16.8152 mL
20 mM	0.1682 mL	0.8408 mL	1.6815 mL	8.4076 mL
50 mM	0.0673 mL	0.3363 mL	0.6726 mL	3.3630 mL
100 mM	0.0336 mL	0.1682 mL	0.3363 mL	1.6815 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc