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AZD1940

Name: AZD1940
Brand: TargetMol
SKU: T30252
Price: 132 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T30252Cas No. 881413-29-2

Alias UNII-0J0035E9FT, AZD-1940, AZD 1940

AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.

AZD1940

🥰Excellent

Purity: 98.68%

Catalog No. T30252Alias UNII-0J0035E9FT, AZD-1940, AZD 1940Cas No. 881413-29-2

AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.

Pack Size	Price	Availability
1 mg	$132	In Stock
5 mg	$328	In Stock
10 mg	$563	In Stock
25 mg	$891	In Stock
50 mg	$1,230	In Stock
100 mg	$1,670	In Stock
1 mL x 10 mM (in DMSO)	$363	In Stock

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Bulk & Custom

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Purity:98.68%

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COA LCMS LCMS HPLC HNMR

Product Introduction

Bioactivity

Description	AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.
Targets&IC50	CB1 receptor (human):7.93 (pKi), CB2 receptor (human):9.06 (pKi)
In vitro	AZD1940 demonstrates high binding affinity towards the CB1 and CB2 receptors in humans, rats, and mice, exhibiting full agonism at both receptor types across these species[1].
In vivo	After given orally to human, the mean maximum plasma concentration (Cmax) for AZD1940 800 mg was 9.3 nmol/L . The mean concentration over post-dose eight hours for AZD1940 was 236 nmol.h/L[1].
Synonyms	UNII-0J0035E9FT, AZD-1940, AZD 1940

Chemical Properties

Molecular Weight	413.52
Formula	C₂₀H₂₉F₂N₃O₂S
Cas No.	881413-29-2
Smiles	CCS(=O)(=O)Nc1ccc2n(CC3CCC(F)(F)CC3)c(nc2c1)C(C)(C)C
Relative Density.	1.28 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 90.0 mg/mL (217.6 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4183 mL	12.0913 mL	24.1826 mL	120.9131 mL
5 mM	0.4837 mL	2.4183 mL	4.8365 mL	24.1826 mL
10 mM	0.2418 mL	1.2091 mL	2.4183 mL	12.0913 mL
20 mM	0.1209 mL	0.6046 mL	1.2091 mL	6.0457 mL
50 mM	0.0484 mL	0.2418 mL	0.4837 mL	2.4183 mL
100 mM	0.0242 mL	0.1209 mL	0.2418 mL	1.2091 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

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