Shopping Cart

Your shopping cart is currently empty

AZD1940

Name: AZD1940
Brand: TargetMol
SKU: T30252
Price: 132 USD
Availability: InStock
Rating: 5 (10 reviews)

Copy Product Info

😃Good

Catalog No. T30252Cas No. 881413-29-2

Alias UNII-0J0035E9FT, AZD-1940, AZD 1940

AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.

AZD1940

Copy Product Info

😃Good

Purity: 98.68%

Catalog No. T30252Alias UNII-0J0035E9FT, AZD-1940, AZD 1940Cas No. 881413-29-2

AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$132	In Stock	In Stock
5 mg	$328	In Stock	In Stock
10 mg	$563	In Stock	In Stock
25 mg	$891	In Stock	In Stock
50 mg	$1,230	In Stock	In Stock
100 mg	$1,670	-	In Stock
1 mL x 10 mM (in DMSO)	$363	In Stock	In Stock

Add to Cart

Add to Quotation

In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products.If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

Select Batch

Purity:98.68%

Appearance:Solid

Color:White

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	AZD1940 (UNII-0J0035E9FT) is a high affinity CB(1)/CB(2) receptor agonist of the cannabinoid with oral activity. Application in the study of orofacial pain.
Targets&IC50	CB1 receptor (human):7.93 (pKi), CB2 receptor (human):9.06 (pKi)
In vitro	AZD1940 demonstrates high binding affinity towards the CB1 and CB2 receptors in humans, rats, and mice, exhibiting full agonism at both receptor types across these species[1].
In vivo	After given orally to human, the mean maximum plasma concentration (Cmax) for AZD1940 800 mg was 9.3 nmol/L . The mean concentration over post-dose eight hours for AZD1940 was 236 nmol.h/L[1].
Synonyms	UNII-0J0035E9FT, AZD-1940, AZD 1940

Chemical Properties

Molecular Weight	413.52
Formula	C₂₀H₂₉F₂N₃O₂S
Cas No.	881413-29-2
Smiles	CCS(=O)(=O)Nc1ccc2n(CC3CCC(F)(F)CC3)c(nc2c1)C(C)(C)C
Relative Density.	1.28 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 90 mg/mL (217.64 mM), Sonication is recommended.

In Vivo Formulation

10% DMSO+40% PEG300+5% Tween 80+45% Saline: 3.3 mg/mL (7.98 mM), Sonication is recommended.

Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4183 mL	12.0913 mL	24.1826 mL	120.9131 mL
5 mM	0.4837 mL	2.4183 mL	4.8365 mL	24.1826 mL
10 mM	0.2418 mL	1.2091 mL	2.4183 mL	12.0913 mL
20 mM	0.1209 mL	0.6046 mL	1.2091 mL	6.0457 mL
50 mM	0.0484 mL	0.2418 mL	0.4837 mL	2.4183 mL
100 mM	0.0242 mL	0.1209 mL	0.2418 mL	1.2091 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc