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LPA5 antagonist 1
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Catalog No. T63231 Copy Product Info
Purity: 98.63%
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LPA5 antagonist 1 is a highly potent and selective antagonist of lysophosphatidic acid receptor 5 (LPA5), with an IC₅₀ value of 32 nM. LPA5 antagonist 1 is a small molecule with high brain permeability that significantly alleviates mechanical allodynia in a CFA-induced inflammatory pain model and can be used to study the mechanisms underlying inflammatory and neuropathic pain. LPA5 antagonist 1 is a click chemistry reagent containing an alkyne functional group, capable of undergoing a copper-catalyzed azide-alkyne cycloaddition (CuAAC) reaction with molecules bearing an azide group.
Cas No. 2839471-45-1
| Pack Size | Price | USA Stock | Global Stock | Quantity |
|---|---|---|---|---|
| 25 mg | $1,520 | - | In Stock | |
| 50 mg | $1,980 | - | In Stock | |
| 100 mg | $2,500 | 10-14 weeks | 10-14 weeks |
For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)
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For research use only—not for human use. No sales to individuals. Use as intended only.
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Purity:98.63%
Appearance:Solid
Color:Yellow
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | LPA5 antagonist 1 is a highly potent and selective antagonist of lysophosphatidic acid receptor 5 (LPA5), with an IC₅₀ value of 32 nM. LPA5 antagonist 1 is a small molecule with high brain permeability that significantly alleviates mechanical allodynia in a CFA-induced inflammatory pain model and can be used to study the mechanisms underlying inflammatory and neuropathic pain. LPA5 antagonist 1 is a click chemistry reagent containing an alkyne functional group, capable of undergoing a copper-catalyzed azide-alkyne cycloaddition (CuAAC) reaction with molecules bearing an azide group. |
| Molecular Weight | 486.58 |
| Formula | C28H26N2O4S |
| Cas No. | 2839471-45-1 |
| Smiles | O=C1C=2C=C(OC)C(OC)=CC2C(=CN1C=3C=CC=4SC=C(C4C3)C)C(=O)N5CCC(C#C)CC5 |
| Relative Density. | no data available |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
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Related Tags: LPA5 antagonist 1 chemical structure | LPA5 antagonist 1 formula | LPA5 antagonist 1 molecular weight
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