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α1 adrenoceptor-MO-1

Name: α1 adrenoceptor-MO-1
Brand: TargetMol
SKU: T10003
Price: 209 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T10003Cas No. 161905-64-2

α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enantiomer.

α1 adrenoceptor-MO-1

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Purity: 99.29%

Catalog No. T10003Cas No. 161905-64-2

α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enantiomer.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$209	In Stock	In Stock
5 mg	$413	In Stock	In Stock
10 mg	$571	In Stock	In Stock
25 mg	$826	In Stock	In Stock
50 mg	$1,130	In Stock	In Stock
100 mg	$1,530	In Stock	In Stock
200 mg	$2,070	-	In Stock
1 mL x 10 mM (in DMSO)	$491	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products.If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Batch Information

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Purity:99.29%

ee:100%

Appearance:Solid

Color:White to Yellow

Resource Download

COA ORP HPLC CSFC HNMR

Product Introduction

Bioactivity

Description	α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enantiomer.
In vitro	The S enantiomer of α1 adrenoceptor-MO-1 exhibits higher activity compared to the R enantiomer[1].

Chemical Properties

Molecular Weight	385.89
Formula	C₂₀H₂₄ClN₅O
Cas No.	161905-64-2
Smiles	O=C1N2C(=NN1CCCN3[C@@H](C)CN(CC3)C4=CC(Cl)=CC=C4)C=CC=C2
Relative Density.	1.31 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (129.57 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.5914 mL	12.9571 mL	25.9141 mL	129.5706 mL
5 mM	0.5183 mL	2.5914 mL	5.1828 mL	25.9141 mL
10 mM	0.2591 mL	1.2957 mL	2.5914 mL	12.9571 mL
20 mM	0.1296 mL	0.6479 mL	1.2957 mL	6.4785 mL
50 mM	0.0518 mL	0.2591 mL	0.5183 mL	2.5914 mL
100 mM	0.0259 mL	0.1296 mL	0.2591 mL	1.2957 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc