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α1 adrenoceptor-MO-1

Name: α1 adrenoceptor-MO-1
Brand: TargetMol
SKU: T10003
Price: 209 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T10003Cas No. 161905-64-2

α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enantiomer.

α1 adrenoceptor-MO-1

🥰Excellent

Purity: 99.89%

Catalog No. T10003Cas No. 161905-64-2

α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enantiomer.

Pack Size	Price	Availability
1 mg	$209	In Stock
5 mg	$413	In Stock
10 mg	$571	In Stock
25 mg	$826	In Stock
50 mg	$1,130	In Stock
100 mg	$1,530	In Stock
200 mg	$2,070	In Stock
1 mL x 10 mM (in DMSO)	$491	In Stock

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Bulk & Custom

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.89%

ee:100%

Resource Download

COA LCMS CSFC HNMR ORP

Product Introduction

Bioactivity

Description	α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enantiomer.
In vitro	The S enantiomer of α1 adrenoceptor-MO-1 exhibits higher activity compared to the R enantiomer[1].

Chemical Properties

Molecular Weight	385.89
Formula	C₂₀H₂₄ClN₅O
Cas No.	161905-64-2
Smiles	O=C1N2C(=NN1CCCN3[C@@H](C)CN(CC3)C4=CC(Cl)=CC=C4)C=CC=C2
Relative Density.	1.31 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (129.57 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.5914 mL	12.9571 mL	25.9141 mL	129.5706 mL
5 mM	0.5183 mL	2.5914 mL	5.1828 mL	25.9141 mL
10 mM	0.2591 mL	1.2957 mL	2.5914 mL	12.9571 mL
20 mM	0.1296 mL	0.6479 mL	1.2957 mL	6.4785 mL
50 mM	0.0518 mL	0.2591 mL	0.5183 mL	2.5914 mL
100 mM	0.0259 mL	0.1296 mL	0.2591 mL	1.2957 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc