Contact UsQuotation
Shopping Cart
Remove All
  • TargetMol
    Your shopping cart is currently empty
Proceed to checkoutContinue shopping
TOPBioactivityChemical infoStorage&SolubilityCalculator

Perilloxin

😃Good
Catalog No. TN4752Cas No. 263249-77-0

Perilloxin possesses measurable inhibitory activity against cyclooxygenase-1 (COX-1), exhibiting an IC50 value of 23.2 μM, and this biochemical property supports its application as a functional research molecule for studying inflammatory signaling pathways, enzyme inhibition mechanisms, and structure–activity relationships relevant to prostaglandin biosynthesis and inflammation-associated biological processes.

Perilloxin

Perilloxin

😃Good
Catalog No. TN4752Cas No. 263249-77-0
Perilloxin possesses measurable inhibitory activity against cyclooxygenase-1 (COX-1), exhibiting an IC50 value of 23.2 μM, and this biochemical property supports its application as a functional research molecule for studying inflammatory signaling pathways, enzyme inhibition mechanisms, and structure–activity relationships relevant to prostaglandin biosynthesis and inflammation-associated biological processes.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
25 mg$6,970InquiryInquiry
Add to Cart
Add to Quotation
In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Questions
TargetMol
View More

Batch Information

Select Batch
Contact us for more batch information

Resource Download

COA

Product Introduction

Bioactivity
Description
Perilloxin possesses measurable inhibitory activity against cyclooxygenase-1 (COX-1), exhibiting an IC50 value of 23.2 μM, and this biochemical property supports its application as a functional research molecule for studying inflammatory signaling pathways, enzyme inhibition mechanisms, and structure–activity relationships relevant to prostaglandin biosynthesis and inflammation-associated biological processes.
Targets&IC50
COX-1:23.2 μM.
In vitro
Method: Bioassay-guided fractionation of Perilla frutescens stem extracts was performed, and isolated compounds were tested in an in vitro cyclooxygenase-1 inhibition assay.
Result: Perilloxin and dehydroperilloxin inhibited cyclooxygenase-1 with IC50 values of 23.2 μM and 30.4 μM, respectively[1].
Chemical Properties
Molecular Weight274.31
FormulaC16H18O4
Cas No.263249-77-0
SmilesC(C)(C)(O)[C@@H]1OC=2C3=C(C(OC)=CC2C1)C=COC=C3
Relative Density.1.230 g/cm3 (Predicted)
ColorYellow
AppearanceSolid
Storage & Solubility Information
Storagestore at low temperature,keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Stock solution preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (stock solution concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
The above example illustrates how to use "In Vivo Formulation Calculator" and does not represent a recommended formulation for any specific compound. Please select an appropriate dissolution method based on your experimental animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
% Tween 80
% Saline/PBS/ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

PerilloxinCOX-1
Related Tags: buy Perilloxin | purchase Perilloxin | Perilloxin cost | order Perilloxin | Perilloxin chemical structure | Perilloxin in vitro | Perilloxin formula | Perilloxin molecular weight
TargetMol | Logo

Copyright © 2015-2026 TargetMol Chemicals Inc. All Rights Reserved.