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MRT-2359

Name: MRT-2359
Brand: TargetMol
SKU: T67934
Price: 48 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T67934Cas No. 2803881-11-8

MRT-2359 is a potent and orally available GSPT1 reducer with antitumour activity.MRT-2359 inhibits the growth of drug-resistant non-small cell lung cancer (NSCLC) and small cell lung cancer (SCLC) cells.MRT-2359 exhibits preferential activity in MYC-driven cell lines.

MRT-2359

🥰Excellent

Purity: 99.39%

Catalog No. T67934Cas No. 2803881-11-8

Pack Size	Price	Availability
1 mg	$48	In Stock
5 mg	$112	In Stock
10 mg	$188	In Stock
25 mg	$378	In Stock
50 mg	$619	In Stock
100 mg	$938	In Stock
200 mg	$1,260	In Stock
1 mL x 10 mM (in DMSO)	$186	In Stock

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Batch Information

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Purity:99.39%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description

Chemical Properties

Molecular Weight	495.38
Formula	C₂₂H₁₇F₄N₃O₆
Cas No.	2803881-11-8
Smiles	O=C1N(CC=2C1=CC(COC(NC3=CC(OC(F)(F)F)=CC=C3F)=O)=CC2)C4C(=O)NC(=O)CC4
Relative Density.	1.548 g/cm3 at 20℃ (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

store at low temperature,keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 25 mg/mL (50.47 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0187 mL	10.0933 mL	20.1865 mL	100.9326 mL
5 mM	0.4037 mL	2.0187 mL	4.0373 mL	20.1865 mL
10 mM	0.2019 mL	1.0093 mL	2.0187 mL	10.0933 mL
20 mM	0.1009 mL	0.5047 mL	1.0093 mL	5.0466 mL
50 mM	0.0404 mL	0.2019 mL	0.4037 mL	2.0187 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc