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Elinafide
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Catalog No. T68061Cas No. 162706-37-8
Elinafide, a dinaphthylimide cytotoxic agent, is a DNA-targeted anticancer agent that has shown antitumor activity in in vitro and in vivo assays.
Elinafide
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Purity: 97.67%
Catalog No. T68061Cas No. 162706-37-8
Elinafide, a dinaphthylimide cytotoxic agent, is a DNA-targeted anticancer agent that has shown antitumor activity in in vitro and in vivo assays.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 5 mg | $41 | In Stock | In Stock | |
| 10 mg | $64 | In Stock | In Stock | |
| 25 mg | $121 | In Stock | In Stock | |
| 50 mg | $167 | In Stock | In Stock | |
| 100 mg | $239 | In Stock | In Stock | |
| 200 mg | $335 | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Batch Information
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Purity:97.67%
Appearance:Solid
Color:Yellow
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Product Introduction
Elinafide AI Summary
Elinafide demonstrates potent bioactivity by inhibiting cell growth in various human cancer cell cultures with low IC50 values. Specifically, it is effective against human colon carcinoma (HT-29) with an IC50 of 14.0 to 38.0 nM, human cervical carcinoma (HeLa) with an IC50 of 70.0 nM, human prostate carcinoma (PC-3) with IC50s ranging from 70.0 to 320.0 nM, and human breast cancer cell line MDA-MB-231 with an IC50 of 60.0 nM. Additionally, Elinafide shows selectivity towards leukemia cell lines and has cytotoxic effects against human NCI-H460 cells with an IC50 of 8.0 nM. In vivo, it has been observed to improve survival times in mouse models with M5076 murine sarcoma cells. These results suggest that Elinafide may hold promise as a potent and selective anticancer agent..
Note: Summary generated by AI. Data source: ChEMBL 
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Elinafide, a dinaphthylimide cytotoxic agent, is a DNA-targeted anticancer agent that has shown antitumor activity in in vitro and in vivo assays. |
| Targets&IC50 | NCI-H460 cells:8 nM, Smooth muscle cells (SMCs):12 nM |
| Molecular Weight | 520.58 |
| Formula | C31H28N4O4 |
| Cas No. | 162706-37-8 |
| Smiles | O=C1C=2C=3C(C(=O)N1CCNCCCNCCN4C(=O)C=5C=6C(C4=O)=CC=CC6C=CC5)=CC=CC3C=CC2 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | ||||||||||
| Solubility Information | DMSO: 1.3 mg/mL (2.5 mM), Sonication is recommended.  | ||||||||||
Solution Preparation Table | |||||||||||
DMSO
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Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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