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LY2452473
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Catalog No. T15804Cas No. 1029692-15-6
Alias OPK-88004, OPK 88004, LY-2452473, LY 2452473
LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.
LY2452473
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Purity: 99.72%
Catalog No. T15804Alias OPK-88004, OPK 88004, LY-2452473, LY 2452473Cas No. 1029692-15-6
LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $30 | In Stock | In Stock | |
| 5 mg | $65 | In Stock | In Stock | |
| 10 mg | $93 | In Stock | In Stock | |
| 25 mg | $143 | In Stock | In Stock | |
| 50 mg | $188 | In Stock | In Stock | |
| 100 mg | $281 | In Stock | In Stock | |
| 200 mg | $429 | - | In Stock | |
| 1 mL x 10 mM (in DMSO) | $70 | In Stock | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.72%
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Product Introduction
Bioactivity
Chemical Properties
| Description | LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer. |
| In vivo | METHODS: The disposition and metabolism of LY2452473 in humans was characterized following a single oral dose of 15 mg (100 μCi) of [¹⁴C]LY2452473 in six healthy male subjects. RESULTS: LY2452473 was rapidly absorbed (time to maximum plasma concentrations of LY2452473 and total radioactivity was 2-3 hours) and slowly eliminated (plasma terminal half-life of 27 hours, duration of LY2452473 and total radioactivity of 51 hours). [1] |
| Synonyms | OPK-88004, OPK 88004, LY-2452473, LY 2452473 |
| Molecular Weight | 374.44 |
| Formula | C22H22N4O2 |
| Cas No. | 1029692-15-6 |
| Smiles | C(N1C2=C(C=3C1=CC=C(C#N)C3)C[C@H](NC(OC(C)C)=O)C2)C4=CC=CC=N4 |
| Relative Density. | 1.28 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 60 mg/mL (160.24 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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