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LY2452473
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Catalog No. T15804Cas No. 1029692-15-6
Alias OPK-88004, OPK 88004, LY-2452473, LY 2452473
LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.
LY2452473
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Purity: 99.72%
Catalog No. T15804Alias OPK-88004, OPK 88004, LY-2452473, LY 2452473Cas No. 1029692-15-6
LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $30 | In Stock | In Stock | |
| 5 mg | $65 | In Stock | In Stock | |
| 10 mg | $93 | In Stock | In Stock | |
| 25 mg | $143 | In Stock | In Stock | |
| 50 mg | $188 | In Stock | In Stock | |
| 100 mg | $281 | In Stock | In Stock | |
| 200 mg | $429 | - | In Stock | |
| 1 mL x 10 mM (in DMSO) | $70 | In Stock | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.72%
Appearance:Solid
Color:White
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Product Introduction
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Chemical Properties
Storage & Solubility Information
| Description | LY2452473 (OPK 88004) is an orally available and selective androgen receptor modulator with potential anticancer activity for the study of prostate cancer. |
| In vivo | METHODS: The disposition and metabolism of LY2452473 in humans was characterized following a single oral dose of 15 mg (100 μCi) of [¹⁴C]LY2452473 in six healthy male subjects. RESULTS: LY2452473 was rapidly absorbed (time to maximum plasma concentrations of LY2452473 and total radioactivity was 2-3 hours) and slowly eliminated (plasma terminal half-life of 27 hours, duration of LY2452473 and total radioactivity of 51 hours). [1] |
| Synonyms | OPK-88004, OPK 88004, LY-2452473, LY 2452473 |
| Molecular Weight | 374.44 |
| Formula | C22H22N4O2 |
| Cas No. | 1029692-15-6 |
| Smiles | C(N1C2=C(C=3C1=CC=C(C#N)C3)C[C@H](NC(OC(C)C)=O)C2)C4=CC=CC=N4 |
| Relative Density. | 1.28 g/cm3 (Predicted) |
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 60 mg/mL (160.24 mM), Sonication is recommended. | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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