store at low temperature,keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine is an n-alkylated derivative with analgesic activity.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 55.00 | |
5 mg | In stock | $ 128.00 | |
10 mg | In stock | $ 189.00 | |
25 mg | In stock | $ 319.00 | |
50 mg | In stock | $ 478.00 | |
100 mg | In stock | $ 696.00 | |
500 mg | In stock | $ 1,470.00 |
Description | [DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine is an n-alkylated derivative with analgesic activity. |
Targets&IC50 | CHO cells:0.12 nM |
In vitro | Porcine [DPro10] Dynorphin A (1-11) inhibits adenylyl cyclase activity in CHO cells expressing k-opioid receptors, with an IC50 value of 0.12 nM[1]. |
In vivo | Administered intracerebroventricularly (ICV), [DPro10] Dynorphin A (1-11), porcine, exhibits analgesic effects involving thermal cutaneous (tail-flick) and chemical visceral (acetic acid-induced writhing) stimuli, with known differential activation of mu and kappa receptors[2]. |
Synonyms | [DPro10] Dynorphin A (1-11)acetate,porcine(94596-26-6 Free base) |
Molecular Weight | 1422.7 |
Formula | C65H107N21O15 |
store at low temperature,keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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[DPro10] Dynorphin A (1-11)acetate,porcine Endocrinology/Hormones GPCR/G Protein Neuroscience Opioid Receptor [DPro10] Dynorphin A acetate,porcine [DPro10] Dynorphin A (1-11)acetate,porcine(94596-26-6 Free base) inhibitor inhibit