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Amauromine

Name: Amauromine
Brand: TargetMol
SKU: T36566
Rating: 4.5 (1 reviews)

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Catalog No. T36566Cas No. 88360-87-6

Amauromine is a peripherally selective and potent cannabinoid receptor type 1 (CB1) receptor antagonist, a novel alkaloid with vasodilatory activity.

Amauromine

😃Good

Catalog No. T36566Cas No. 88360-87-6

Amauromine is a peripherally selective and potent cannabinoid receptor type 1 (CB1) receptor antagonist, a novel alkaloid with vasodilatory activity.

Pack Size	Price	USA Warehouse	Global Warehouse	Quantity
250 μg	$198	35 days	35 days
1 mg	$548	35 days	35 days

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Product Introduction

Bioactivity

Description	Amauromine is a peripherally selective and potent cannabinoid receptor type 1 (CB1) receptor antagonist, a novel alkaloid with vasodilatory activity.
Targets&IC50	CB1:66.6 nM (Kb), CB1:178 nM (Ki)

Chemical Properties

Molecular Weight	508.65
Formula	C₃₂H₃₆N₄O₂
Cas No.	88360-87-6
Smiles	[C@@](C=C)(C)(C)[C@]12[C@](N3[C@@](C1)(C(=O)N4[C@](C3=O)(C[C@]5([C@](C=C)(C)C)[C@]4(NC=6C5=CC=CC6)[H])[H])[H])(NC=7C2=CC=CC7)[H]
Relative Density.	1.28 g/cm3 (Predicted)

Storage & Solubility Information

Storage

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 5.11 mg/mL (10.05 mM), Sonication is recommended.

Ethanol: 5 mg/mL (9.83 mM), Sonication is recommended.

Methanol: 5 mg/mL (9.83 mM), Sonication is recommended.

Solution Preparation Table

Ethanol/Methanol/DMSO

	1mg	5mg	10mg	50mg
1 mM	1.9660 mL	9.8299 mL	19.6599 mL	98.2994 mL
5 mM	0.3932 mL	1.9660 mL	3.9320 mL	19.6599 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc