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EP4 receptor antagonist 2

Name: EP4 receptor antagonist 2
Brand: TargetMol
SKU: T63100
Price: 279 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T63100Cas No. 1965316-82-8

EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor, with an IC50 of 7.8 nM, and exhibits antitumor effects.

EP4 receptor antagonist 2

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Purity: 100%

Catalog No. T63100Cas No. 1965316-82-8

EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor, with an IC50 of 7.8 nM, and exhibits antitumor effects.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$279	-	In Stock
5 mg	$683	-	In Stock
10 mg	$1,090	-	In Stock
25 mg	$1,980	-	In Stock
50 mg	$2,830	-	In Stock
1 mL x 10 mM (in DMSO)	$789	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Purity:100%

ee:99.84%

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Product Introduction

Bioactivity

Description	EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor, with an IC50 of 7.8 nM, and exhibits antitumor effects.
Targets&IC50	EP4:7.8 nM

Chemical Properties

Molecular Weight	475.54
Formula	C₂₇H₂₉N₃O₅
Cas No.	1965316-82-8
Smiles	C(NC1=C(CCCC(O)=O)C=CC(C#N)=C1)(=O)[C@H]2[C@]3(C=4C(=CC=C(C(NC(C)C)=O)C4)OCC3)C2
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

store at low temperature | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline /PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Stock solution preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline /PBS/ddH₂O TargetMol | reagent

mix well and clarify

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