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SCH 221510

Name: SCH 221510
Brand: TargetMol
SKU: T23335
Price: 71 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T23335Cas No. 322473-89-2

Alias SCH-221510, SCH221510

SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used to study neurological disorders.

SCH 221510

🥰Excellent

Purity: 99.54%

Catalog No. T23335Alias SCH-221510, SCH221510Cas No. 322473-89-2

SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used to study neurological disorders.

Pack Size	Price	Availability
1 mg	$71	In Stock
5 mg	$172	In Stock
10 mg	$278	In Stock
25 mg	$562	In Stock
50 mg	$892	In Stock
100 mg	$1,450	In Stock
200 mg	$1,950	In Stock

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Bulk & Custom

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.54%

ee:99.9%

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COA CSFC HNMR LCMS

Product Introduction

Bioactivity

Description	SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used to study neurological disorders.
Targets&IC50	NOP:0.3 nM(Ki ), NOP:12 nM( EC50)
Synonyms	SCH-221510, SCH221510

Chemical Properties

Molecular Weight	397.55
Formula	C₂₈H₃₁NO
Cas No.	322473-89-2
Smiles	C(N1[C@@]2(C[C@@](O)(C[C@]1(CC2)[H])C3=CC=CC=C3)[H])(C4=C(C)C=CC=C4)C5=C(C)C=CC=C5
Relative Density.	1.141 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (125.77 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.5154 mL	12.5770 mL	25.1541 mL	125.7703 mL
5 mM	0.5031 mL	2.5154 mL	5.0308 mL	25.1541 mL
10 mM	0.2515 mL	1.2577 mL	2.5154 mL	12.5770 mL
20 mM	0.1258 mL	0.6289 mL	1.2577 mL	6.2885 mL
50 mM	0.0503 mL	0.2515 mL	0.5031 mL	2.5154 mL
100 mM	0.0252 mL	0.1258 mL	0.2515 mL	1.2577 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc