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Targets

Libraries

PPI Inhibitor Library Covalent Natural Product Library Endoplasmic Reticulum Stress Compound Library Carboxylic Acid Fragment Library With Solubility FDA-Approved Kinase Inhibitor Library Adrenergic Receptor-Targeted Compound Library Ubiquitination Compound Library Rare Natural Compound Library AMPK-Targeted Compound Library Cyclic Peptide Library Tyrosine Kinase Inhibitor Library Kinase Inhibitor Library MAPK Inhibitor Library Anti-COVID-19 Compound Library Neurotransmitter Receptor Compound Library GPCR Compound Library Cuproptosis Compound Library Serotonin Receptor-Targeted Compound Library NO PAINS Compound Library PI3K-AKT-mTOR Compound Library Neural Regeneration Compound Library High Solubility Pharmacophore Fragment Library Cytoskeletal Signaling Pathway Compound Library Transcription Factor-Targeted Compound Library Lipid Metabolism Compound Library Flavonoid Natural Product Library NF-κB Signaling Compound Library Covalent Inhibitor Library Endocrinology-Hormone Compound Library Pre-plated Diversity Sets GPCR Compound Library Plus Macrocyclic Compound Library Cell Cycle Compound Library Calcium Antagonist Library Bioactive Compounds Library Max Methylation Compound Library Neuronal Signaling Compound Library Histamine & Melatonin Receptor-Targeted Compound Library Pyroptosis Compound Library Fluorochemical Library Glutamine Metabolism Compound Library Peptide Compound Library Drug-induced Liver Injury (DILI) Compound Library Exosome Compound Library Chemokine Inhibitor Library Anti-Alzheimer's Disease Compound Library
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Reagents



Compounds

Cat No. Product Name
TP1786L Amyloid β-Protein 10-20 acetate Amyloid β-Protein 10-20 acetate(152286-31-2 free base) Beta Amyloid
Amyloid β-Protein 10-20 acetate(152286-31-2 free base) 是 Amyloid-β 肽的片段,可能用于神经系统疾病的研究。Amyloid β 蛋白片段含有 α-分泌酶加工位点(Lys16-L...
T21618L Myelin Basic Protein (87-99) Acetate Myelin Basic Protein (87-99) Acetate (118506-26-6 Free base) Others
Myelin Basic Protein (87-99) Acetate 是一种致脑炎肽,可诱导碱性蛋白特异性 T 细胞增殖。 它导致外周血单核细胞中的 Th1 极化,这与多发性硬化症 (MS) 有牵连。
T4692 Protein kinase inhibitors 1 hydrochlorid Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base)) Others
Protein kinase inhibitors 1 hydrochlorid 是一种新型 HIPK2 抑制剂,IC50 为 74 nM,Kd 为 9.5 nM。
TP1053L Protein Kinase C 19-31 acetate Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate PKC
Protein Kinase C 19-31 acetate(121545-65-1 free base) 是一种蛋白激酶 C (PKC) 的肽抑制剂,源自 PKCa 的假底物调节结构域(残基 19-31),在 25 位用丝氨酸取代野生型丙...
TP1271L Calmodulin-Dependent Protein Kinase II 290-309 acetate Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base) CaMK
Calmodulin-Dependent Protein Kinase II 290-309 acetate 是 Ca2+/calmodulin-dependent protein kinase II 的有效拮抗剂(IC50 = 52 nM...
TP1051L Protein Kinase C Peptide Substrate acetate Protein Kinase C Peptide Substrate acetate(120253-69-2 free base) Others
Protein Kinase C Peptide Substrate acetate(120253-69-2 free base) 以依赖于第二信使和特定衔接蛋白的方式靶向特定细胞间隔物,以响应激活 g 蛋白偶联受体、酪氨酸激酶受体或酪氨酸...
T9892 JAMM protein inhibitor 2  Acetamide, 2-(2-ethylphenoxy)-N-[2-methyl-4-(1-pyrrolidinyl)phenyl]- Others
JAMM protein inhibitor 2 是 JAMM 蛋白酶的抑制剂,可用于抗癌的研究。 对thrombin、Rpn11 和 MMP2 的 IC50 分别为 10 μM、46 μM 和 89 μM。
TP1516L C-Reactive Protein (CRP) 77-82 acetate C-Reactive Protein (CRP) 77-82 acetate(130349-01-8 free base) Others
C-Reactive Protein (CRP) 77-82 acetate(130349-01-8 free base) 是 C-反应蛋白的 77-82 片段。 C-反应蛋白 (CRP) 是炎症的原型标志物,是心血管风险标志物,可能促进动...
TP1270L 2:PN:US20040072744 SEQID:2 claimed protein acetate 2:PN:US20040072744 SEQID:2 claimed protein acetate(389572-87-6 free base) Others
2:PN:US20040072744 SEQID:2 claimed protein acetate(389572-87-6 free base) 是一种合成肽,用于唐氏综合症和精神分裂症的研究。
TP1676L C-Reactive Protein (CRP) 201-206 acetate C-Reactive Protein (CRP) 201-206 acetate(130348-99-1 free base) Others
C-Reactive Protein (CRP) 201-206 acetate(130348-99-1 free base) 是 C-反应蛋白的 201-206 片段。 C-反应蛋白 (CRP) 醋酸盐是炎症的原型标志物,是心血管风险标志...
TP1628L Activated Protein C (390-404), human acetate Activated Protein C (390-404), human acetate(146340-20-7 Free base) APC
Activated Protein C (390-404), human acetate 抑制 APC 抗凝活性。
TP1453 Tau protein (592-597), Human TFA Others
Tau protein (592-597), Human TFA 是人 Tau 蛋白的肽片段。
T9631 IRAK-4 protein kinase inhibitor 2 IRAK
IRAK-4 protein kinase inhibitor 2 是有效的白介素 1 受体相关激酶 4 抑制剂,IC50为 4 μM。它在与炎症和免疫相关的疾病领域有研究价值。
T38919 Protein E7(43-62) Protein E7(43-62)
Protein E7(43-62) is a peptide derived from the E7 protein. The peptide spans the 43rd to 62nd amino acid residues and e...
T40250 SHP2 protein degrader-1 SHP2 protein degrader-1
SHP2 protein degrader-1 is a highly efficient allosteric inhibitor targeting SHP2. It effectively induces degradation of...
T4207 (S,R,S)-AHPC hydrochloride ULM-1,Protein degrader 1 hydrochloride,VHL Ligand 1 hydrochloride Others
(S,R,S)-AHPC hydrochloride 是基于 VH032 的 VHL 配体,可用于募集 von Hippel-Lindau (VHL) 蛋白。它能够利用 linker 与靶蛋白配体连接,得到 PROTAC 分子。
TP1902L1 G-Protein antagonist peptide acetate Adrenergic Receptor
G-Protein antagonist peptide acetate 是一种 substance P 相关肽,可抑制 G 蛋白与其受体的结合。G-Protein antagonist peptide acetate 竞争性和可逆性地抑制...
T60109 Protein kinase inhibitor H-7 蛋白激酶抑制剂H-7,1-(5-Isoquinolinylsulfonyl)-2-methylpiperazine,5-(2-methylpiperazine-1-sulfonyl)isoquinoline PKC
Protein kinase inhibitor H-7 是有效的蛋白激酶 C (PKC) 和环核苷酸依赖性蛋白激酶抑制剂,抑制 PKC 的 Ki 值为 6 μM。
TP1650 Myelin Basic Protein Myelin Basic Protein MBP
Myelin basic protein (MBP) is a protein believed to be important in the process of myelination of nerves in the nervous ...
TP2465 PHYD protein, Arabidopsis Phyd gene product,Phyd protein
PHYD protein, Arabidopsis belongs to the phytochrome apoprotein family in Arabidopsis.
Amyloid β-Protein 10-20 acetate
TP1786L
synonym: Amyloid β-Protein 10-20 acetate(152286-31-2 free base)
Target:
Myelin Basic Protein (87-99) Acetate
T21618L
synonym: Myelin Basic Protein (87-99) Acetate (118506-26-6 Free base)
Target:
Protein kinase inhibitors 1 hydrochlorid
T4692
synonym: Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))
Target:
Protein Kinase C 19-31 acetate
TP1053L
synonym: Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate
Target:
Calmodulin-Dependent Protein Kinase II 290-309 acetate
TP1271L
synonym: Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base)
Target:
Protein Kinase C Peptide Substrate acetate
TP1051L
synonym: Protein Kinase C Peptide Substrate acetate(120253-69-2 free base)
Target:
JAMM protein inhibitor 2 
T9892
synonym: Acetamide, 2-(2-ethylphenoxy)-N-[2-methyl-4-(1-pyrrolidinyl)phenyl]-
Target:
C-Reactive Protein (CRP) 77-82 acetate
TP1516L
synonym: C-Reactive Protein (CRP) 77-82 acetate(130349-01-8 free base)
Target:
2:PN:US20040072744 SEQID:2 claimed protein acetate
TP1270L
synonym: 2:PN:US20040072744 SEQID:2 claimed protein acetate(389572-87-6 free base)
Target:
C-Reactive Protein (CRP) 201-206 acetate
TP1676L
synonym: C-Reactive Protein (CRP) 201-206 acetate(130348-99-1 free base)
Target:
Activated Protein C (390-404), human acetate
TP1628L
synonym: Activated Protein C (390-404), human acetate(146340-20-7 Free base)
Target:
Tau protein (592-597), Human TFA
TP1453
synonym:
Target:
IRAK-4 protein kinase inhibitor 2
T9631
synonym:
Target:
Protein E7(43-62)
T38919
synonym: Protein E7(43-62)
Target:
SHP2 protein degrader-1
T40250
synonym: SHP2 protein degrader-1
Target:
(S,R,S)-AHPC hydrochloride
T4207
synonym: ULM-1,Protein degrader 1 hydrochloride,VHL Ligand 1 hydrochloride
Target:
G-Protein antagonist peptide acetate
TP1902L1
synonym:
Target:
Protein kinase inhibitor H-7
T60109
synonym: 蛋白激酶抑制剂H-7,1-(5-Isoquinolinylsulfonyl)-2-methylpiperazine,5-(2-methylpiperazine-1-sulfonyl)isoquinoline
Target:
Myelin Basic Protein
TP1650
synonym: Myelin Basic Protein MBP
Target:
PHYD protein, Arabidopsis
TP2465
synonym: Phyd gene product,Phyd protein
Target:
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