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SBI-810 hydrochloride is a functional selective allosteric modulator of the β-arrestin-biased neurotensin receptor 1 (NTSR1). It modulates NTSR1-G protein signaling in a G protein-specific manner in the presence of the endogenous ligand neurotensin (NT). SBI-810 hydrochloride fully antagonizes NT-induced Gq activation, partially antagonizes NT-induced Gi1 activation, while allowing activation of GoA and G12 by NTSR1.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $83 | 7-10 days | |
5 mg | Preferential | 7-10 days |
Description | SBI-810 hydrochloride is a functional selective allosteric modulator of the β-arrestin-biased neurotensin receptor 1 (NTSR1). It modulates NTSR1-G protein signaling in a G protein-specific manner in the presence of the endogenous ligand neurotensin (NT). SBI-810 hydrochloride fully antagonizes NT-induced Gq activation, partially antagonizes NT-induced Gi1 activation, while allowing activation of GoA and G12 by NTSR1. |
Molecular Weight | 483.045 |
Formula | C27H35ClN4O2 |
Cas No. | 2772746-58-2 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice./Shipping at ambient temperature. |
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