Powder: -20°C for 3 years | In solvent: -80°C for 1 year
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template. It inhibits both G-protein- and β-arrestin-mediated signaling pathways [1].
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Description | D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template. It inhibits both G-protein- and β-arrestin-mediated signaling pathways [1]. |
Targets&IC50 | D 3 Receptor:66 nM (Ki) |
Molecular Weight | 455.59 |
Formula | C27H37NO5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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D3R ligand 1 GPCR/G Protein Neuroscience Dopamine Receptor inhibitor inhibit