ito — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T16348	NS5806	NS-5806	Potassium Channel
	NS5806 is an effective potassium current activator. NS5806 slows KV4.3 and KV4.2 current decay in channel complexes containing KChIP2. NS5806 enhances KV4.3/KChIP2 peak current amplitudes (EC50: 5.3 μM).		Potassium Channel
T0866	Propafenone	Rythmol,Propafenonum	Potassium Channel , MRP , Sodium Channel
	Propafenone (Propafenonum) is only found in individuals that have used or taken this drug. It is an antiarrhythmia agent that is particularly effective in ventricular arrhythmias. It also has weak beta-blocking activity....		Potassium Channel , MRP , Sodium Channel
T9845	Thrombin inhibitor 5
	Thrombin inhibitor 5 (compound 385) is a thrombin inhibitor with IC 50s ranging from 0.1 μM to 1 μM. Thrombin inhibitor 5 can be used for venous thromboembolism research[1].
T5915	D-chiro-Inositol	D-(+)-CHIRO-INOSITOL	Endogenous Metabolite
	D-chiro-Inositol (D-(+)-CHIRO-INOSITOL) is an epimer of myo-inositol that is found in certain mammalian glycosylphosphatidylinositol protein anchors and inositol phosphoglycans possessing insulin-like bioactivity.		Endogenous Metabolite
T4950	1,2-Dipalmitoyl-sn-glycerol	(S)-1,2-Dipalmitin	Endogenous Metabolite , PKC
	1,2-Dipalmitoyl-sn-glycerol ((S)-1,2-Dipalmitin) is an analog of the PKC-activating second messenger diacylglycerol (DAG). It weakly activates PKC.		Endogenous Metabolite , PKC
T0299	Lactitol monohydrate	D-Lactitol monohydrate	Others
	Lactitol monohydrate (D-Lactitol monohydrate) is a disaccharide analog of lactulose. It has been widely used to treat constipation and hepatic encephalopathy.		Others
T37422L	Ras Inhibitory Peptide acetate	Ras Inhibitory Peptide acetate(159088-48-9 Free base)	Ras
	Ras Inhibitory Peptide acetate is a peptide involved in the Ras-dependent signaling pathway that plays an important role in human cancers initiated by oncogenic receptors.		Ras
T5817	PKC-theta inhibitor hcl	PKC-theta inhibitor	PKC
	PKC-theta inhibitor hcl is a selective PKC-θinhibitor(IC50:12 nM).		PKC
T7676	LSKL, Inhibitor of Thrombospondin TSP-1 acetate	LSKL, Inhibitor of Thrombospondin TSP-1	TGF-beta/Smad
	LSKL, Inhibitor of Thrombospondin TSP-1 acetate is activation of TGF-β .		TGF-beta/Smad
T10927	Cyt-PTPε Inhibitor-1	Cyt-PTP\|A Inhibitor-1	Phosphatase , Src
	Cyt-PTPε Inhibitor-1 (A Inhibitor-1) is an inhibitor of cytosolic protein tyrosine phosphatase ε. Cyt-PTPε Inhibitor-1 blocks the dephosphorylation of c-Src and exhibits anti-osteoclastic activity.		Phosphatase , Src
T13224	Tubulin inhibitor 6	iHAP1	Microtubule Associated
	Tubulin inhibitor 6 (iHAP1) is an inhibitor of tubulin and a potent inhibitor of multiple cancer cell lines.		Microtubule Associated
TP1216	CaM kinase II inhibitor TFA salt	Autocamtide-2-related inhibitory peptide (TFA)	CaMK
	CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.		CaMK
T4491	LMPTP INHIBITOR 1 hydrochloride	LMPTP INHIBITOR 1 hydrochloride (1908414-82-3(free base))	Phosphatase
	LMPTP INHIBITOR 1 hydrochloride is a selective inhibitor of low molecular weight protein tyrosine phosphatase ( LMPTP ), with an IC 50 of 0.8 μM for LMPTP-A.		Phosphatase
T9892	JAMM protein inhibitor 2	Acetamide, 2-(2-ethylphenoxy)-N-[2-methyl-4-(1-pyrrolidinyl)phenyl]-	Others
	JAMM protein inhibitor 2 (Acetamide, 2-(2-ethylphenoxy)-N-[2-methyl-4-(1-pyrrolidinyl)phenyl]-) is an inhibitor of JAMM protease and can be used for anticancer studies. The IC50s are 10 μM, 46 μM, and 89 μM for thrombin,...		Others
T1529	Miglitol	BAY1099,BAY-m1099	Others
	Miglitol (BAY1099) is an alpha-Glucosidase Inhibitor with antihyperglycemic activity.		Others
T5238	1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine	1,2-Dipalmitoyl-sn-glycero-3-PE,1,2-Dipalmitoyl-sn-glycerol-3-Phosphoethanolamine,1,2-DPPE	Others , Endogenous Metabolite
	1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine (DPPE), a phospholipid member of the glycerophosphonoethanolamine family, is a major component in biological membranes. Studies focused on interactions between DPPE and ch...		Others , Endogenous Metabolite
T4191	Multi-kinase inhibitor 1	Multi-kinase inhibitor I	Others , Bcr-Abl , PDGFR , c-Kit
	Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) is a Multi-kinase inhibitor.		Others , Bcr-Abl , PDGFR , c-Kit
T4466	Pitofenone hydrochloride	Baralgin Ketone Hydrochloride,Pitophenone hydrochloride	AChE
	Pitofenone hydrochloride (Pitophenone hydrochloride), a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively.		AChE
T4656	RAD51 Inhibitor B02	B02	Apoptosis , DNA/RNA Synthesis
	RAD51 Inhibitor B02 (B02) (B02) is an inhibitor of human RAD51 with an IC50 of 27.4 μM.		Apoptosis , DNA/RNA Synthesis
T4338	USP7/USP47 inhibitor	USP7/47 inhibitor-1	DUB
	USP7/USP47 inhibitor (USP7/47 inhibitor-1) is a selective ubiquitin-specific protease 7/47 (USP7/USP47) inhibitor, with EC50s of 0.42 μM and 1.0 μM, respectively.		DUB