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Cat No. product name
Fr12275 7-Methoxy-1-tetralone 7-Methoxy-1-tetralone may have insecticidal activity.
Fr12277 4-Hydroxy-6-methylcoumarin
Fr12290 4-Methoxycoumarine 4-Methoxycoumarin has antitumour effects.
Fr12339 4-(4-Methoxyphenyl)-2-butanone
Fr12596 3-Acetylcoumarin
Fr12662 4-Ethoxycoumarin
Fr13711 Tropinone Tropinone is a decane alkaloid, used as an intermediate in the synthesis of atropine sulfate.
Fr13756 Isonicotinic acid Isonicotinic acid is a metabolite of Isoniazid. Isoniazid is converted to Isonicotinic acid by hydrazinolysis, with the biotransformation also to be catalyzed b...
Fr13883 3-Methoxyphenylacetic acid 3-Methoxyphenylacetic acid belongs to the class of organic compounds known as anisoles. 3-Methoxyphenylacetic acid is slightly soluble (in water) and a weakly a...
Fr14207 Isopulegol
Fr14438 p-Toluic Acid p-Toluic Acid belongs to the class of organic compounds known as benzoic acids. 4-Methylbenzoic acid has been primarily detected in saliva. Within the cell, 4-...
Fr16605 Lupinine
Fr16741 Oxindole Oxindole structure has been used in receptor tyrosine kinases (RTKs) inhibitors such as SU4984 and intedanib, the RTK family represents an important therapeutic...
Fr16745 4-Hydroxyphenylacetonitrile 4-Hydroxyphenylacetonitrile shows strong antioxidative activity.
S00015 Tea polyphenol Tea polyphenol, also called green tea extract, are a mixture of chemical compounds, such as flavanoids and tannins, found naturally in tea. Polyphenols are powe...
T0001 Ferrous fumarate Iron(II) fumarate, also named as ferrous fumarate, is the iron(II) salt of fumaric acid, a reddish-orange powder, applied to supply iron intake.
T0003 Sodium Nitroprusside Sodium Nitroprusside is a potent vasodilator, releasing in blood with no spontaneously.
T0006 Methylene Blue trihydrate Methylene blue is a compound consisting of dark green crystals or crystalline powder, having a bronze-like luster. Solutions in water or alcohol have a deep blu...
T0010 Mercaptopurine Mercaptopurine is an antimetabolite antineoplastic agent with immunosuppressant properties. It interferes with nucleic acid synthesis by inhibiting purine metab...
T0011 Phenethyl alcohol Phenethyl alcohol is an antimicrobial, antiseptic, and disinfectant. It is used also as an aromatic essence and preservative in pharmaceutics and perfumery.
T0013 Mecarbinate Mecarbinate is arbidol hydrochloride's chemical intermediate.
T0014 cis-Anethol Anethole is a type of aromatic compound that exists widely in nature, widely utilized as a seasoning substance.
T0015 Mephenesin Mephenesin is a centrally acting muscle relaxant with a short duration of action.
T0016 Mexenone Mexenone is a benzophenone-derived sun protection.
T0017 Phenolphthalein Phenolphthalein is an acid-base indicator which is colorless in acid solution, but turns pink to red as the solution becomes alkaline. It is used medicinally as...
T0019 Betaine hydrochloride Betaine hydrochloride is an acidic form of betaine, a vitamin-like substance observed in grains and other foods; gains the amplification of DNA by decreasing th...
T0021 Vanatone It is an inhibitor of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1)
T0023 Valethamate bromide Valethamate bromide is an anticholinergic agent.
T0027 Octisalate Ethylhexyl salicylate, or octyl salicylate, is an organic compound used as an ingredient in sunscreens and cosmetics to absorb UVB (ultraviolet) rays from the s...
T0028 4-Amino-3-hydroxybutyric Acid Agent for improving learning or memory [US6803366]Gamma Hydroxybutyric Acid, commonly abbreviated GHB, is an illegal therapeutic drug in multiple countries. In ...
T0032 DL-Xylose Xylose is a sugar first derived from wood. Xylose is classified as a monosaccharide of the aldopentose type.
T0037 Halazone Halazone is fine white powder with an odor of chlorine.
T0043 2-Amino-6-methylheptane Octodrine is a stimulant drug,a platinum complex form of which was also investigated as a possible anti-tumor drug.
T0056 Oxeladin citrate Oxeladin is a highly potent and effective cough suppressant,which can treat all types of cough of various etiologies. It is not related to opium or its derivati...
T0066 Dichlorophen Dichlorophen is a nontoxic laxative vermicide of chlorinated phenol compound. Dichlorophen is used as a veterinary fungicide, anthelmintic, and anti-protozoa...
T0067 Oxiniacic Acid Oxiniacic Acid is a nicotinic acid derivative, used to treat hyperlipoidemia.
T0069 Uracil Uracil is a common naturally occurring pyrimidine found in RNA, it base pairs with adenine and is replaced by thymine in DNA. Methylation of uracil produces thy...
T0071 Homosalate Homosalate is an organic compound used as a chemical UV filter. It is an ester formed from salicylic acid and 3,3,5-trimethylcyclohexanol, a derivative of cyclo...
T0073 Octyl 4-methoxycinnamate Octinoxate is an organic compound that is used is in sunscreens and other cosmetics to absorb UV-B rays from the sun, protecting the skin from damage,primarily ...
T0077 Dantrolene sodium salt Dantrolene is a skeletal muscle relaxant and can interfere with excitation-contraction coupling in the muscle fiber. It is used for the treatment of spasticity ...
T0131 Cepharanthine Cepharanthine, a biscoclaurine alkaloid, suppresses tumor necrosis factor (TNF)-α-mediated NFκB stimulation, plasma membrane lipid peroxidation and platel...
T0144 Ftaxilide Ftaxilide has antibacterial property, used as antiseptic.
T0148L Folinic Acid Calcium Salt Pentahydrate Folinic Acid, a reduced folic acid, is used in combination with other chemotherapeutics.
T0150 Hydroxyhexamide Hydroxyhexamide is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agents.
T0170 Fosfomycin calcium Fosfomycin calcium is an antibiotic, used for the treatment of urinary tract infections and intestinal infections caused by susceptible strains.
T0176 Aloin B It is used as a stimulant-laxative, treating constipation by inducing bowel movements.[2] The compound is present in what is commonly referred to as the aloe la...
T0179 Ticagrelor Ticagrelor is an inhibitor of platelet aggregation. Unlike clopidogrel, ticagrelor is not a prodrug required metabolic activation.
T0183 Pramiracetam Pramiracetam, derived from piracetam, is a more effective nootropic drug . According to reports, Pramiracetam improved cognitive defects related with traumatic...
T0187 Amorolfine hydrochloride Amorolfine Hydrochloride is an antifungal reagent. It exerts the antifungal activity by selectively interrupting two steps in the pathway of ergosterol synthesi...
T0192 Levetiracetam Levetiracetam is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onset seizures. Levet...
T0195 Secnidazole Secnidazole is a second-generation 5-nitroimidazole antimicrobial that is structurally related to other 5-nitroimidazoles including [DB00916] and [DB00911], but...
T0198 Sodium ceftiofur Ceftiofur sodium, an antibiotic of the cephalosporin type (third generation), is used as veterinary medicine.
T0200 Thioctic acid Thioctic acid is an octanoic acid bridged with two sulfurs so that it is sometimes also called a pentanoic acid in some naming schemes. It is biosynthesized by ...
T0224 Meropenem Meropenem is a carbapenem antibiotic with broad spectrum of activity that is administered intravenously and used for severe bacterial infections due to sensitiv...
T0227 Bromisoval Bromisoval is a mild hypnotic and sedative with potential toxicity.
T0233 Ethamivan Etamivan (INN) or ethamivan (USAN), is a respiratory stimulant drug concerned with nikethamide. Its trade name is Analepticon, and no longer used in the US.
T0237 Closantel Closantel, a salicylanilide anthelmintic compound, shows different anthelmintic spectra and obvious toxicity in mammals.
T0238 2-(Acetyloxy)-3-Methylbenzoic Acid 2-(Acetyloxy)-3-Methylbenzoic Acid is used in qHTS Assay for Inhibitors of hydroxysteroid (17-beta) dehydrogenase 4, HSD17B4 with activity value of 19.95 µM
T0239 Lonidamine Lonidamine is an indazole carboxylic acid derivative, principally inhibiting aerobic glycolytic activity, by its effect on mitochondrially-bound hexokinase (HK)...
T0240 Trimetozine Trimetozine is a sedative that has been marketed in Europe since 1959. It has mild tranquilizing effects and has been used to treat anxiety.
T0241 Sulfanilylurea Sulfacarbamide is a blood sugar-lowering agent.
T0243 Vanitiolide A choleretic.
T0244 Tilorone dihydrochloride Tilorone dihydrochloride is an orally active interferon inducer, and has antineoplastic and anti-inflammatory actions.
T0251 GemcitabineHOT Gemcitabine is a DNA synthesis inhibitor that can inhibit the growth of MIAPaCa2, BxPC3 and Capan2 cells (IC50s: 40/18/12 nM). It can also induce autophagy.
T0257 Mepiroxol Mepiroxol, an antihyperlipidemic, is also called 3-PYRIDINEMETHANOL N-OXIDE.
T0258 Carsalame Carsalam is a nonsteroidal anti-inflammatory drug.
T0259 Chromocarbe Chromocarb is a vascular protective agent used to treat venous disorders and microvascular affections.
T0265 Merbromin Merbromin is an organomercuric disodium salt compound and a fluorescein, used as a topical antiseptic for minor cuts and scrapes.
T0271 Iodipamide Iodipamide is a water-soluble radiographic contrast media for intravenous cholangiography and cholecystography.
T0273 Mefexamide hydrochloride Mefexamide hydrochloride is a central stimulant.
T0275 Meticrane Meticrane is a sulphonamide-derivative with thiazide-like diuretic activity.
T0278 Escin Escin is biosynthesized from protoaescigenin and barringtogenol, occurring in the seeds of Aesculus.
T0281 Meclocycline sulfosalicylate salt Meclocycline (INN), a tetracycline antibiotic, is used topically (i.e. for skin infections) as it is totally insoluble in water and may damage kidney and liver ...
T0284 Sulfogaiacol Sulfogaiacol is an antitussive agent, used for acute respiratory tract infections and cough.
T0286 Bephenium Hydroxynaphthoate Bephenium hydroxynaphthoate is a B-type AChR activator, formerly used in the treatment of hookworm infections and ascariasis.
T0288 Procodazole Procodazole is a non-specific active immunoprotective agent against viral and bacterial infections.
T0289 Aminacrine 9-Aminoacridine is a highly fluorescent anti-infective dye used clinically as a topical antiseptic and experimentally as a mutagen, due to its interaction with ...
T0292 Orbifloxacin Orbifloxacin is a broad-spectrum fluoroquinolone antibiotic.
T0293 Metyrapone Metyrapone is an inhibitor of the enzyme STEROID 11-BETA-MONOOXYGENASE. It is used as a test of the feedback hypothalamic-pituitary mechanism in the diagnosis o...
T0296 Pempidine Pempidine is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.
T0299 Lactitol monohydrate Lactitol monohydrate is a disaccharide analog of lactulose. It has been widely used to treat constipation and hepatic encephalopathy.
T0306 Undecenoic acid Undecylenic Acid is a natural or synthetic fungistatic fatty acid, with antifungal activity.
T0307 Tyloxapol Tyloxapol is a non-ionic liquid polymer used as a surfactant.
T0308 Etidronate Etidronic is a diphosphonate which affects calcium metabolism. It inhibits ectopic calcification and slows down bone resorption and bone turnover.
T0310 Actarit Actarit is an anti-inflammatory drug.
T0311 Diathesin Diathesin is an intermediate for medicine, perfume, pesticide.
T0312 Blutene chloride Blutene chloride, a phenothiazine, is used as a biological stain, a hemostatic, and a dye for silk and wool. Blutene chloride is also used as a diagnostic aid f...
T0315 Acedoben Acedoben (4-acetamidobenzoic acid) is the acetyl derivative of para-aminobenzoic acid (PABA).
T0316 Citiolone Citiolone, a drug used in liver treatment, is a derivative of the amino acid cysteine.
T0323 Oxantel Pamoate Oxantel pamoate is used as an Antinematodal agent.
T0325 Diperodon hydrochloride Diperodon is a local anaesthetics.
T0328 Hexetidine Hexetidine is a bactericidal and fungicidal antiseptic. It is used as a 0.1% mouthwash for local infections and oral hygiene.
T0332 D-Sorbitol Sorbitol is a polyhydric alcohol with about half the sweetness of sucrose. Sorbitol occurs naturally and is also produced synthetically from glucose. It was for...
T0336 Benzalkonium chloride Benzalkonium chloride is a cationic surface-acting agent containing the quaternary ammonium group. It has three main categories of use: as a cationic surfactant...
T0339 Resorcin monoacetate Resorcinol monoacetate is an antiseptic and a disinfectant, is a chemical intermediate for the production of many other pharmaceuticals, and can be used to trea...
T0340 Bisoctrizole Bisoctrizole is a benzotriazole-based organic compound that is added to sunscreens to absorb UV rays.
T0341 Dimethyl sulfoxide Dimethyl sulfoxide is a highly polar organic liquid, that is used widely as a chemical solvent. Because of its ability to penetrate biological membranes, it is ...
T0342 Carvedilol phosphate Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intr...
T0344L Miconazole nitrate Miconazole nitrate, an imidazole antifungal agent, selectively affects the integrity of fungal cell membranes, high in ergosterol content and different in compo...
T0346 Camylofin Camylofin is an antimuscarinic, used for relaxing smooth muscle.
T0347 Phenol Red Phenol Red is a pH indicator, red dye, and diagnostic aid for measurement of renal function. It is used also for researches of the gastrointestinal and other sy...
T0352 Dibenzothiophene Dibenzothiophene, a component of petroleum oils, is a sulfur-containing polycyclic aromatic hydrocarbon (PAH) derivate consisting of 3 fused rings with keratoly...
T0355 Valpramide Valpromide is a carboxamide derivative of valproic acid, used in the treatment of epilepsy and some affective disorders.
T0356 Nitromide Nitromide is an anti-parasitic drug.
T0359 2-Aminoheptane 2-Aminoheptane is used for proteomics research.
T0363 Morantel tartrate Morantel tartrate is an antinematodal agent used mainly for livestock.
T0367 Fluocinolone acetonide Fluocinolone acetonide is a glucocorticoid derivative used topically in the treatment of various skin disorders. It is usually employed as a cream, gel, lotion,...
T0368 Cinepazide maleate Cinepazide maleate, a maleate salt form of cinepazide, is a vasodilator.
T0376 Crotamiton Crotamiton is an antipruritic and a scabicidal agent available as a lotion or cream for topical use only. It is a colorless to slightly yellowish oil with a fai...
T0377 Clofazimine Clofazimine is a phenazine dye with anti-mycobacterial and anti-inflammatory activities. Clofazimine has a slow bactericidal effect on Mycobacterium leprae and ...
T0379 Risedronic Acid Risedronic acid (Risedronate ), a pyridinyl biphosphonate, can inhibit osteoclast-mediated bone resorption.
T0382 Eprodisate disodium Eprodisate Disodium is a negatively charged sulfonated inhibitor of fibrillogenesis, that can be used in the treatment of amyloid A (AA) amyloidosis.
T0390 Alkomide Aklomide is used in poultry to treat parasites.
T0392 Artemisinin Artemisinin is an ancient Chinese herbal therapy for malarial fevers which has been recently found to have potent activity against many forms of malarial organi...
T0395 Pyrantel tartrate Pyrantel tartrate is broad spectrum anthelmintic for livestock.
T0396 Pipemidic acid Pipemidic acid, a new antibacterial agent, inhibits the activity of Pseudomonas aeruginosa.
T0398 Carzenide Carzenide is an organic synthesis intermediate.
T0399 Methyl salicylate Methyl salicylate (oil of wintergreen or wintergreen oil) is an organic ester naturally produced by many species of plants, particularly wintergreens. For acute...
T0400 Nitroxoline Nitroxoline is a urinary antibacterial agent active against susceptible gram-positive and gram-negative organisms commonly found in urinary tract infections.
T0402 Octocrilene Octocrylene is used as an ingredient in sunscreens and cosmetics. This organic compound can penetrate into the skin where it acts as a photosensitizer. This res...
T0404 Hydroxyquinoline Oxyquinoline is a heterocyclic phenol and derivative of quinoline with antiseptic, disinfectant, and pesticide properties. It is used as a stabilizer for hydrog...
T0408 Dehydrocholic acid Dehydrocholic acid is a synthetic bile acid, produced by the oxidation of cholic acid.
T0409 Phthalylsulfacetamide Phthalylsulfacetamide is a sulfonamide antibiotic used for topical application to the skin and the conjunctiva.
T0411 Calcium gluconate Calcium gluconate is the calcium salt of gluconic acid, used as a calcium replenisher in hypocalcemic states.
T0413 Cinromide Cinromide is used as a novel anticonvulsant agent.
T0415 Guanidine hydrochloride Guanidine hydrochloride is a strong organic base existing primarily as guanidium ions at physiological pH. It is found in the urine as a normal product of prote...
T0416 Sodium gluconate Sodium Gluconate is the sodium salt of gluconic acid with a chelating property.
T0420 Pentetic Acid Pentetic Acid is an edetate and a chelating agent used in preparing radiopharmaceuticals.
T0422 Talc Talc is a mineral composed of hydrated magnesium silicate.
T0423 Edetate Trisodium Edetate Trisodiumis used to bind metal ions in the chelation therapy.
T0429 Glucosamine Glucosamine is an amino sugar and a prominent precursor in the biochemical synthesis of glycosylated proteins and lipids. Supplemental glucosamine may help to r...
T0430 Imidazolidinyl urea Imidazolidinyl urea is an antimicrobial preservative used in cosmetics.
T0432 Diclofenac diethylamine Diclofenac Diethylamine, a non-selective COX inhibitor, is utilized as a nonsteroidal anti-inflammatory drug (NSAID).
T0434 Dicurone Glucuronolactone is a naturally occurring chemical that is an important structural component of nearly all connective tissues. Glucuronolactone is also found in...
T0435 Sulfinpyrazone Sulfinpyrazone is a uricosuric drug that is used to reduce the serum urate levels in gout therapy. It lacks anti-inflammatory, analgesic, and diuretic propertie...
T0438 Proflavine Hemisulfate Proflavine Hemisulfate is the hemisulfate salt form of proflavine, an acridine-derived fluorescent contrast and disinfectant agent that can potentially be used ...
T0442 Bucetin Bucetin is a pharmaceutical drug that acts as an analgesic and antipyretic. Bucetin was withdrawn from use in 1986 due to renal toxicity.
T0447 Carvedilol Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intr...
T0452 Dropropizine Dropropizine, a racemic non-opiate antitussive agent, is served as a cough suppressant.
T0454 Florfenicol Florfenicol is a fluorinated synthetic analog of thiamphenicol. In the United States, florfenicol is currently used to treat bovine respiratory disease (BRD) as...
T0454L Florfenicol Florfenicol, a fluorinated synthetic analog of thiamphenicol, is currently indicated for the therapy of bovine respiratory disease (BRD) associated with Mannhei...
T0461 Berberine hydrochloride Berberine hydrochloride is an alkaloid from Hydrastis canadensis L., Berberidaceae and also found in many other plants. It is relatively toxic to parenterally b...
T0464 Carbetapentane citrate Pentoxyverine Citrate, an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.
T0471 Decoquinate Decoquinate is a coccidiostat for poultry.
T0491 Ethyl vanillin Ethylvanillin is a flavorant used in the production of chocolate. It is about three times as potent as vanillin.
T0492 Dimethyl fumarate Dimethyl fumarate, a fumarate derivative, is used as antiinflammatory and immunomodulatory agent.
T0495 Aminothiazole Aminothiazole, a thyroid inhibitor,displays antibacterial activity.
T0496 Creatinine Creatinine is the breakdown product of creatine, a constituent of muscle tissue, that is excreted by the kidney and whose serum level is used to evaluate kidney...
T0497 Lauroseptol Cetrimonium Bromide is is a mixture of different quaternary ammonium salts, which is a known component of the broad-spectrum antiseptic cetrimide.
T0499 Oxybenzone Oxybenzone is an organic compound used in sunscreens. It is a derivative of benzophenone.
T0500 Capitrol Capitrol is a synthetic quinoline derivative with antibacterial activity. Although the mechanism of action is not fully understood, topical administration of ch...
T0501 Leucobasal Leucobasal is a synthetic derivate of hydroquinone and depigmenting agent. Although the exact mechanism of the depigmenting effects of mequinol remains unclear,...
T0503 Meglumine Meglumine, a derivative of sorbitol, is used in conjunction with iodinated organic compounds as contrast medium.
T0507 L-Pyroglutamic acid L-Pyroglutamic acid, a cyclized derivative of the L-GLUTAMIC ACID, can elevate blood levels. This function may be associated with problems of GLUTATHIONE or GLU...
T0509 Dermofongin Cloxyquin is a monohalogenated 8-hydroxyquinoline with activity against bacteria, fungi, and protozoa.
T0513 Iodoquinol Diiodohydroxyquinoline, a topical therapeutic agent, has satisfactory antibacterial properties.
T0517 Pancreatin Pancreatin is a mixture of several digestive enzymes secreted by the exocrine cells of the pancreas. It is composed of amylase, lipase and protease.
T0519 Euquinine Euquinine generally is served as the febrifuge, antimalarial, and tonic.
T0526 2-Amino-5-nitrobenzophenone 2-Amino-5-nitrobenzophenone is used as industrial and organic intermediate.
T0527 2,3,4-Trimethoxybenzaldehyde 2,3,4-Trimethoxybenzaldehyde is used as medicine intermediate.
T0528 4-Fluoroanisole 4-Fluoroanisole is a intermediates in medicine, pesticide, liquid crystal materials.
T0529 Dulcitol Dulcitol is a sugar alcohol that is a metabolic breakdown product of galactose.
T0530 Flavanone Flavanones from citrus fruits have also been shown to exert beneficial effects on human vascular function. In particular, chronic interventions with orange juic...
T0531 Intermediate of Pregabalin Intermediate of Pregabalin.
T0533 N-Aminopiperidine hydrochloride 1-Aminopiperidine is a metabolite (M1) of the canabinoid receptor 1 antagonist Rimonabant, an antiobesity agent.
T0534 Bis(4-cyanophenyl)methanol Bis(4-cyanophenyl)methanol is a metabolite of Letrozole.
T0535 Memantine Related Compound B Memantine impurity B is an impurity of Memantine.
T0536 Cyclopropanecarbonitrile Cyclopropyl cyanide is the minimum carbon ring molecule with a cyanide group attached. It has mainly used in experiments with microwave spectroscopy, photodisso...
T0537 Desbenzyl Donepezil Hydrochloride Desbenzyl Donepezil Hydrochloride is an impurity of Donepezil.
T0538 3-Methyloxindole 3-Methyl-2-oxindole is a reactant for O-acetylation reactions, enantioselective α-amination reactions and for aldol reactions with glyoxal derivatives and more...
T0539 Hydrocaffeic acid Dihydrocaffeic Acid is a natural product containing a catechol group with an α,β-unsaturated carboxylic acid chain. Dihydrocaffeic Acid has been shown to have...
T0540 Dibenzosuberol Dibenzosuberol, an organic compound, is used as a Pharmaceutical intermediate.
T0541 Fluoronaphthalene Fluoronaphthalene is incompatible with strong oxidizing agents.
T0542 Homoisovanillic acid Homoisovanillic acid is used as pharmaceutical intermediates.
T0544 Dichlorodiphenylmethane Dichlorodiphenylmethane is used as pharmaceutical intermediates.
T0545 1-(2-Hydroxyethyl)imidazolidine-2-thione 1-(2-Hydroxyethyl)imidazolidine-2-thione is used as pharmaceutical intermediates.
T0546 Trimethylacetic anhydride Trimethylacetic anhydride is used as medical intermediate
T0547 FlutaMide Related CoMpound B FlutaMide Related CoMpound B is used as pharmaceutical intermediates.
T0548 Methyl 5-methylnicotinate Methyl 5-methylnicotinate is used as pharmaceutical intermediates.
T0549 4'-tert-Butylacetophenone 4'-tert-Butylacetophenone is used as medical intermediate
T0550 Domperidone EP Impurity A Domperidone EP Impurity A is used as pharmaceutical intermediates.
T0551 D-Ornithine monohydrochloride D-Ornithine monohydrochloride is used as pharmaceutical intermediates.
T0552 Isonicotinamide Isonicotinamide is used as pharmaceutical intermediate to synthesis Cefalonium, etc.
T0553 4-Hydroxyisophthalic acid 4-Hydroxyisophthalic acid is used as medical intermediate
T0554 Dibutylurea Dibutylurea is used as pharmaceutical intermediates.
T0555 4-Diethylamino-2-butyn-1-ol 4-Diethylamino-2-butyn-1-ol is used as pharmaceutical intermediates.
T0556 6-Methoxy-2-naphthoic acid 6-Methoxy-2-naphthoic acid is an modulator of NMDAR.
T0557 3-(Methylamino)toluene 3-(Methylamino)toluene is used as dye intermediates
T0558 Hydroferulic acid Hydroferulic acid is used as the intermediates of perfume and essence.
T0559 Dibenzosuberone Dibenzosuberone, pharmaceutical intermediates, is used for the synthesis of drug amitriptyline.
T0560 3,3-Diphenylpropylamine 3,3-Diphenylpropylamine is used for synthetic drugs Mepramidil
T0561 2-Methoxy-5-sulfamoylbenzoic acid 2-Methoxy-5-sulfamoylbenzoic Acid is a metabolite of the antipsychotic drug, Sulpiride.
T0562 Protocatechuic acid Protocatechuic acid (3, 4-dihydroxybenzoic acid) is a natural phenolic compound found in many edible and medicinal plants. Recent studies indicate that it could...
T0563 Homoveratronitrile Homoveratronitrile is an impurity of Verapamil. It is also an intermediate in the preparation of the muscle relaxant Papverine.
T0564 1-Indanone 1-Indanone is the intermediate od Indinavir.
T0565 Bis(2-chloroethyl)amine hydrochloride Bis(2-chloroethyl)amine hydrochloride is used as pharmaceutical intermediate.
T0566 2-Methylbenzhydrol 2-Methylbenzhydrol is used as pharmaceutical intermediates.
T0567 2-Amino-5-chlorobenzoic acid 5-Chloroanthranilic Acid is a metabolite of the pesticide Chlordimeform. It can be used in the preparation of disease-modifying antirheumatic drugs (DMARDs).
T0568 Homoveratrumic acid Homoveratrumic acid is the papaverine intermediate, used to synthesis cardiovascular drugs.
T0569 Pyrazinoic acid Pyrazinoic acid is the intermediate of pyrazole thiamethoxam sulfur.
T0570 3,5-Dihydroxybenzoic acid 3,5-Dihydroxybenzoic Acid is a metabolite of alkylresorcinol in human urine and plasma. It is also used as a biomarker of whole grain wheat and rye.
T0571 2-Methylbenzene-1-sulfonamide 2-Methylbenzene-1-sulfonamide is used for saccharin, pharmaceutical intermediates, etc.
T0572 Methyl EudesMate Methyl EudesMate is the intermediate of antibacterial efficiency medicine trimethoprim.
T0573 2-Methoxynaphthalene 2-Methoxynaphthalene is served as Odor agents.
T0574 Diphenyl sulfide Diphenyl sulfide is used as pesticide, medicine, dye intermediates.
T0575 1-Methylimidazole 1-Methylimidazole is a metabolite of 1-methyl-2-thioimidazole (methimazole) which inhibits bone resorption.
T0576 Diethylaminoethoxyethanol Diethylaminoethoxyethanol is served in the production of cough medicine Toclase and so on.
T0577 Chlorobenzothiazolinone Chlorobenzothiazolinone inhibits recombinant human chymase using bis(succinoyl-L-alanyl-L-prolyl-L-phenylalanylamide) as substrate after 1 hr by fluorescence as...
T0578 Erythrosin B Iodeosin, a tetraiodofluorescein, is used as a red coloring in some foods (cherries, fish), as a stain of some cell types, and as a disclosure of DENTAL PLAQUE....
T0580 4-Pentynoic acid 4-Pentynoic acid has been used in reactions with 1-bromo-1-alkynes in the presence of a Pd catalyst yields biologically active ynenol lactones. It also is used ...
T0581 Isomaltose Isomaltose is a reducing disaccharide, similar to maltose, but with an α-(1-6)-linkage instead of the α-(1-4)-linkage.
T0582 Fructooligosaccharides Fructooligosaccharides is a levorotatory monosaccharide and an isomer of glucose.
T0583 Erythritol Erythritol is a four-carbon sugar that is found in algae, fungi, and lichens. It is twice as sweet as sucrose and can be used as a coronary vasodilator.
T0584 Maltose Maltose is a dextrodisaccharide from malt and starch. It is used as a sweetening agent and fermentable intermediate in brewing.
T0584L D-(+)-Maltose monohydrate D-(+)-Maltose monohydrate, a dextrodisaccharide from starch and malt, is used as a fermentable intermediate and sweetening agent in brewing.
T0585 Maltitol Maltitol is a sugar alcohol (polyol) used as a sugar substitute.
T0586 Lactose Lactose is a disaccharide derived from galactose and glucose that is found in milk.
T0587 L(+)-Arabinose Arabinose is an aldopentose, including an aldehyde (CHO) functional group.
T0589 Xylitol Xylitol is a five-carbon sugar alcohol derived from XYLOSE by reduction of the carbonyl group. It is as sweet as sucrose and used as a noncariogenic sweetener.
T0591 Alpha-D-galactose D-Galactose is an aldohexose that exists naturally in the D-form in lactose, cerebrosides, gangliosides, and mucoproteins and is converted enzymatically into D-...
T0592 Mannose Mannose is a hexose or fermentable monosaccharide and isomer of glucose from manna, the ash Fraxinus ornus and related plants.
T0596 Phenylhydantoin 5-Phenylhydantoin is a metabolite of Mephenytoin. 5-Phenylhydantoin has been shown to bind to voltage-dependent sodium channels (NVSC) and has anti-epileptic pr...
T0598 Iminostilbene Iminostilbene (Dibenzazepine) is a chemical precursor of carbamazepine which is used primarily in the treatment of epilepsy and neuropathic pain.
T0599 N-Methyl-N-(trimethylsilyl)trifluoroacetamide N-Methyl-N-(trimethylsilyl)trifluoroacetamide is a metabolite of Famprofazone in humans.
T0600 10,11-Dihydrocarbamazepine 10,11-Dihydrocarbamazepine is used as pharmaceutical intermediates.
T0601 Phthalic Acid Monobenzyl Ester Monobenzyl Phthalate is Phthalate metabolite.
T0604 Desalkylterbuthylazine Desalkylterbuthylazine is used as pharmaceutical intermediates.
T0606 Monobutyl Phthalate Monobutyl Phthalate is a di-n-Butylphthalate (DBP) metabolite.
T0607 Dihydroartemisinin Dihydroartemisinin is a metabolite of artemisinin.
T0608 Heptachlor-endo-epoxide Heptachlor-endo-epoxide is a degradation product of heptachlor that occurs in soil and in or on crops when treatments with heptachlor, an insecticide, have been...
T0609 Azobenzene Azobenzene is a compound constituted of two phenyl rings linked by an N=N double bond. Azobenzene is the simplest example of an aryl azo chemical compound. The ...
T0611 4-Hydroxy-3-methoxymandelic acid 4-Hydroxy-3-methoxymandelic acid is a chemical intermediate.
T0612 DL-6-Methoxy-Alpha-Methyl-2-Naphthalenemethanol DL-6-Methoxy-Alpha-Methyl-2-Naphthalenemethanol is used as pharmaceutical intermediates.
T0613 Beta-Hydroxyisovaleric acid Used as medical intermediates
T0614 4-Amino-5-Chloro-2-Methoxybenzoic Acid 4-Amino-5-chloro-2-methoxybenzoic Acid (Metoclopramide EP Impurity C) is a Metoclopramide metabolite.
T0615 1-(3-Chlorophenyl)piperazine hydrochloride 1-(3-Chlorophenyl)piperazine hydrochloride is used for the synthesis of trazodone, Etoperidone, Nefazodone, etc.
T0621 Diphenyl oxide Diphenyl oxide is used in the manufacture of spices and dyes.
T0622 2-Chlorophenothiazine 2-Chlorophenothiazine is used as the intermediate of Chlorpromazine hydrochloride.
T0623 Diphenylacetonitrile Diphenylacetonitrile is used as herbicide and industrial intermediate.
T0624 4-Hydroxybenzophenone 4-Hydroxybenzophenone is used as an intermediate of infertility drugs Clomifene.
T0628 Iminodibenzyl Iminodibenzyl is used for the intermediates of antiepileptic drug carbamazepine.
T0629 Atropic acid Atropic acid (Ipratropium EP Impurity D) is an impurity of Ipratropium bromide and Atropine Sulfate.
T0630 Ethyleneurea Ethyleneurea is used as a formaldehyde scavenger and intermediate.
T0631 2-Phenylbutyric acid 2-Phenylbutyric Acid is used as an industrial intermediate.
T0632 Gallic acid trimethyl ether Gallic acid trimethyl ether are potent antioxidants and inhibitor of cytokine production. It can ameliorate chronic stress-induced various behavioral and bioche...
T0633 (2-Chlorophenyl)phenyl-methanone (2-Chlorophenyl)phenyl-methanone is used as pharmaceutical intermediate.
T0634 2-Acetyl-4-butyramidophenol 2-Acetyl-4-butyramidophenol is gray crystalline powder.
T0635 p-(2-Methoxyethyl) phenol p-(2-Methoxyethyl) phenol, an important kind of pharmaceutical intermediates, is primarily used in the synthesis of metoprolol which is effective drugs in the t...
T0636 4-Methylmorpholine N-oxide 4-Methylmorpholine N-oxideis an organic compound, used in organic chemistry as a co-oxidant and sacrificial catalyst in oxidation reactions.
T0637 2-Acetyl-6-methoxynaphthalene 2-Acetyl-6-methoxynaphthalene, the key intermediate of naphthalene tome and naproxen, is used in synthetic non-steroidal anti-inflammatory analgesic medicine an...
T0638 2-Methyl-4-nitroimidazole 2-Methyl-5-nitroimidazole is a kind of small molecular compounds.
T0640 Butyl benzyl phthalate Butyl benzyl phthalate is used as a plasticizer for PVC.
T0643 Diclofenac Amide Diclofenac Amide is used as a intermediates of Diclofenac.
T0644 3-Amino-5-methylisoxazole 3-Amino-5-methylisoxazole is pharmaceutical intermediates, used in the production of sulfonamide drugs.
T0645 N-(1-Adamantyl)acetamide N-(1-Adamantyl)acetamide is used as intermediates for synthesis of amantadine hydrochloride.
T0650 Phenyl acetate Phenyl acetate, the ester of a phenol and acetic acid, can be produced by reacting acetic anhydride with phenol. Another way is produced by decarboxylation of a...
T0653 Tris(2-chloroethyl) phosphate Tris(2-chloroethyl) phosphate is served as flame retardants.
T0657 3,4-Dimethoxybenzyl alcohol 3,4-Dimethoxybenzyl Alcohol is an organic compound.
T0658 2-(2-Hydroxyethyl)pyridine 2-Pyridineethanol is used as an industrial chemistry intermediate.
T0659 Bispyrazolone Bispyrazolone is light yellow or white crystalline powder.
T0661 Dimethylsulfamoyl chloride Dimethylsulfamoyl Chloride is a kind of small molecular compound.
T0662 2-Hydroxybenzimidazole 2-Hydroxybenzimidazole is used as an intermediate in industry.
T0664 Nicotinic acid hydrazide Nicotinic acid hydrazide is a small molecular compound.
T0665 2,6-Dihydroxypurine Xanthine is a product on the pathway of purine degradation. Xanthine is subsequently converted to uric acid by the action of the Xanthine oxidase enzyme. Xanthi...
T0666 4-Chlorosalicylic acid 4-Chlorosalicylic acid is antimicrobial compositions comprising a metal salt and a benzoic acid analog.
T0667 Flecainide Impurity D Flecainide Impurity D is used as an intermediate in industry.
T0668 1-Aminohydantoin hydrochloride 1-Aminohydantoin hydrochloride is an organic compound.
T0669 Chloramine-T Chloramine-T is a N-chlorinated, and N-deprotonated sulfonamide, used as a biocide and a mild disinfectant.
T0671 2-Naphthol 2-Naphthol is an isomer of 1-naphthol, differing by the location of the hydroxyl group on the naphthalene ring.
T0686 Orlistat Orlistat is an Intestinal Lipase Inhibitor. The mechanism of action of orlistat is as a Lipase Inhibitor.
T0690 Quinine Quinine is a natural cinchona alkaloid that has been used for centuries in the prevention and therapy of malaria. Quinine is also used for idiopathic muscle cra...
T0691 Sulisobenzone Sulisobenzone (benzophenone-4), an ingredient in certain sunblocks, protects the skin against damage by short-wave UVA ultraviolet light and UVB.
T0693 Niflumic acid Niflumic acid is a Ca2+-activated Cl- channel blocker and an analgesic and anti-inflammatory agent used in the therapy of rheumatoid arthritis.
T0694 Pranlukast Pranlukast is a cysteinyl leukotriene receptor-1 antagonist. It antagonizes or reduces bronchospasm caused, principally in asthmatics, by an allergic reaction t...
T0695 Avobenzone Avobenzone, an oil-soluble ingredient, is a dibenzoylmethane derivative used in sunscreen products to absorb the full spectrum of UVA rays.
T0697 Aspartame Aspartame, an artificial, non-carbohydrate sweetener, is aspartyl-phenylalanine-1-methyl ester.
T0698 Dioxybenzone Dioxybenzone (benzophenone-8) is a derivative of benzophenone, used in sunscreen to block UVB and short-wave UVA (ultraviolet) rays.
T0699 Sulfamonomethoxine Sulfamonomethoxine is a long-acting sulfonamide antibacterial agent, blocks the synthesis of folic acid by inhibiting synthetase of dihydropteroate.
T0701 Broxyquinoline Broxyquinoline is an antiprotozoal agent, and it can release oxygen free radicals from the water in mucous membranes.
T0710 L-Cycloserine L-cycloserine irreversibly inhibits GABA pyridoxal 5′-phosphate-dependent aminotransferase in E. coli, as well in the brains of various animals, results in in...
T0715 Chlormezanone Chlormezanone is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.
T0719 Tetrabenazine Tetrabenazine is a drug formerly used as an antipsychotic and treatment of various movement disorders. Tetrabenazine blocks neurotransmitter uptake into adrener...
T0721 Piroctone olamine Piroctone olamine is a compound sometimes used in the treatment of fungal infections. Piroctone olamine is the ethanolamine salt of the hydroxamic acid derivati...
T0722 Ursolic acid Ursolic acid(Bungeolic acid), a natural pentacyclic triterpenoid carboxylic acid, shows anti-tumor effects.
T0724 Formononetin Formononetin is an O-methylated isoflavone and a phytoestrogen from the root of Astragalus membranaceus.
T0727 Piperonyl butoxide Piperonyl butoxide is an insecticide synergist, particularly for rotenone and pyrethroids.
T0729 Benzyl benzoate Benzyl benzoate is one of the older preparations used for the therapy of scabies. Scabies is a skin infection caused by the Sarcoptes scabiei. Its symptoms are ...
T0730 Triacetin Triacetin is a triglyceride that is used as an antifungal agent.
T0738 Urea Urea is formed in the liver from ammonia produced by the deamination of amino acids. It is the principal end metabolite of protein catabolism and accounts for a...
T0739 Guaifenesin Guaifenesin is an expectorant that also has some muscle relaxing action. It is used in many cough preparations.
T0741 Sulfamethazine Sulfamethazine is a sulfanilamide anti-infective agent. It has a spectrum of antimicrobial action similar to other sulfonamides.
T0743 DL-Carnitine DL-Carnitine is the constituent of liver and striated muscle. In therapeutically It is used to stimulate pancreatic and gastric secretions and to treat hyperlip...
T0744 Zinc undecylenate 10-Undecenoic acid zinc salt, a synthetic or natural fungistatic fatty acid, is used topically in creams against eczemas, fungal infections, ringworm, and other...
T0755 Carbaglu Carglumic acid is an orphan drug used to treat hyperammonemia in patients with N-acetyl glutamate synthase absence. This rare hereditary disease results in elev...
T0756 Ethoxyquin Ethoxyquin is an antioxidant used in animal feeds.
T0762 Trans-Anethole Anethole (anise camphor), an organic compound, is widely served as a condiment substance. It is a derivative of phenylpropene, a type of aromatic compound that ...
T0763 Diolane Diolane, colorless liquid, is a chiral diol. It is an industrial compound produced from diacetone alcohol by hydrogenation.
T0768 Oxolamine citrate Oxolamine is a cough suppressant that is able to be used as a generic drug in many jurisdictions.
T0770 Carbadox Carbadox is an antibacterial agent that has been used in veterinary practice for treating swine dysentery and enteritis and for promoting growth. However, its u...
T0771 Casanthranol Casanthranol is a concentrated mixture of anthranol glycosides from cascara sagrada (dried bark of Rhamnus p.) and used as a laxative in constipation and variou...
T0772 Troxerutin Troxerutin, a natural bioflavonoid, is isolated from Sophora japonica. It has many benefits and medicinal properties.
T0777 Tilmicosin Tilmicosin is a macrolide antibiotic. It is used in veterinary medicine for the treatment of bovine respiratory disease and ovine respiratory disease associated...
T0781 Dithiopropanol An anti-gas warfare agent that is effective against Lewisite (dichloro(2-chlorovinyl)arsine) and formerly known as British Anti-Lewisite or BAL. It acts as a ch...
T0787 Butylated hydroxyanisole Butylated hydroxyanisole (BHA) is an antioxidant consisting of a mixture of two isomeric organic compounds, 2-tert-butyl-4-hydroxyanisole and 3-tert-butyl-4-hyd...
T0791 Reserpine Reserpine is an alkaloid found in the roots of Rauwolfia serpentina and R. vomitoria. Reserpine inhibits the uptake of norepinephrine into storage vesicles resu...
T0799 Lactulose Lactulose ,a synthetic disaccharide ,is used in the treatment of constipation and hepatic encephalopathy.
T0801 Tannic acid Tannic acid is a novel hERG channel blocker.
T0803 Acetrizoic acid Acetrizoic acid is the first monomeric ionic compound used as an X-ray contrast agent.
T0807 Basibrol 2,2,2-Tribromoethanol is an organic compound used to anesthetize mice.
T0819 Spiramycin Spiramycin is a macrolide antibiotic produced by Streptomyces ambofaciens. The drug is effective against gram-positive aerobic pathogens, N. gonorrhoeae, and st...
T0823 Thioctamide Lipoamide is a trivial name for 6,8-dithiooctanoic amide. It is 6,8-dithiooctanoic acid's functional form where the carboxyl group is attached to protein (or an...
T0827 Cefsulodine sodium Cefsulodin sodium salt hydrate is a β lactam antibiotic.
T0828 Bromhexine hydrochloride Bromhexine hydrochloride is a mucolytic agent used in the treatment of respiratory disorders associated with viscid or excessive mucus. 
T0829 Etofylline Etofylline is used for difficulty in breathing, asthma, breathing difficulty and other conditions.
T0833 Benzoic acid Benzoic acid is a fungistatic compound that is widely used as a food preservative. It is conjugated to GLYCINE in the liver and excreted as hippuric acid.
T0834 Ethylparaben Ethylparaben is a Standardized Chemical Allergen. The physiologic effect of ethylparaben is by means of Increased Histamine Release, and Cell-mediated Immunity.
T0844 Sulfamethoxypyridazine Sulfamethoxypyridazine is a sulfanilamide antibacterial agent.
T0845 Cyromazine Cyromazine is an ectoparasiticide. Insect growth regulator. Specific activity against dipterous larvae. Cyromazine is a fda approved for use in livestock.
T0850 Primaquine diphosphate Primaquine Phosphate is the phosphate salt form of primaquine, a synthetic, 8-aminoquinoline derivative with antimalarial properties. Although its mechanism...
T0852 Carbazochrome sodium sulfonate Carbazochrome sodium sulfonate (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.
T0860 Mefloquine hydrochloride Mefloquine is a quinoline derivative used for the prevention and therapy of P. falciparum malaria.
T0861 Tylosin tartrate Tylosin tartrate, a macrolide antibiotic, is approved for the control of mycoplasmosis in poultry.
T0872L Amprolium Hydrochloride Amprolium is a coccidiostat that interferes with thiamine metabolism.
T0873 Dinitolmide Dinitolmide, a poultry feed additive, is a coccidiostat for poultry.
T0874 Dimetridazole Dimetridazole is a drug that combats protozoan infections. It is a nitroimidazole class drug. It has been banned by the Canadian government as a livestock feed ...
T0875 Acetylcysteine Acetylcysteine is the N-acetyl derivative of CYSTEINE. It is used as a mucolytic agent to reduce the viscosity of mucous secretions. It has also been shown to h...
T0876 Clioquinol Clioquinol is an orally bioavailable, lipophilic, copper-binding, halogenated 8-hydroxyquinoline with antifungal, antiparasitic and potential antitumor activiti...
T0877 Gallic acid Ursolic acid (UA), a pentacyclic triterpene acid, is used in anticancer chemotherapies.
T0881 6-Aminocaproic acid Aminocaproic acid is an antifibrinolytic agent that acts by inhibiting plasminogen activators which have fibrinolytic properties.
T0885 Sulfamethoxazole Sulfamethoxazole is a Sulfonamide Antimicrobial. The mechanism of action of sulfamethoxazole is as a Cytochrome P450 2C9 Inhibitor. The chemical classification ...
T0887 D(+)-Glucose D(+)-Glucose is a primary source of energy for living organisms. It is naturally occurring and is found in fruits and other parts of plants in its free state. I...
T0889 Saccharin Flavoring agent and non-nutritive sweetener.
T0891 Sulphadione 4,4'-Diaminodiphenylsulfone has activity against a wide range of bacteria but mainly employed for its actions against mycobacterium leprae.
T0896 Furaltadone hydrochloride Furaltadone hydrochloride is an antibacterial and shows distinct curative effect in the treatment of coccidiosis.
T0898 Chloroxylenol Chloroxylenol (4-chloro-3,5-dimethylphenol), a broad spectrum antimicrobial chemical compound, is used to control virus, bacteria, fungi, and algae. It is used ...
T0899 Dehydroacetic acid Dehydroacetic acid, a pyrone derivative, is served frequently as a fungicide and bactericide.
T0900 Cetylpyridinium chloride monohydrate Cetylpyridinium chloride (CPC), a cationic quaternary ammonium compound, is used in certain classes of throat sprays, mouthwashes, lozenges, toothpaste, nasal s...
T0901 Chlorobutanol Chlorobutanol is a chemical preservative, sedative hypnotic and weak local anaesthetic similar in nature to chloral hydrate. It has antibacterial and antifungal...
T0908 Chloquinan Chlorquinaldol is a Standardized Chemical Allergen. The physiologic effect of chlorquinaldol is by means of Increased Histamine Release, and Cell-mediated Immun...
T0910 Terpin Monohydrate Terpin hydrate, a cis-form hydrate, is derived from sources such as oil of turpentine, oregano, thyme, and eucalyptus. It is used as an insect repellent and exp...
T0912L Tetracycline Tetracycline is a naphthacene antibiotic that inhibits AMINO ACYL TRNA binding during protein synthesis.
T0914 Metacetamol METACETAMOL is an organic compound.
T0917 Sulfaquinoxaline sodium Sulfa drugs, used in the treatment of avian coccidiosis.
T0919 Benfluorex hydrochloride Tamoxifen is an antineoplastic nonsteroidal selective estrogen receptor modulator (SERM).
T0921 Sulfabenzamide Sulfabenzamide is a sulfonamide antibacterial agent used alone or with sulfathiazole and sulfacetamide as a topical, intravaginal antibacterial preparation...
T0922 Zoxazolamine Zoxazolamine is a uricosuric and muscle relaxant. Zoxazolamine acts centrally as a muscle relaxant, but the mechanism of its action is not understood.
T0924 Benzocaine Benzocaine is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.
T0925 Allantoin Allantoin, a urea hydantoin found in urine and plants, is used in dermatological preparations.
T0926 Azelaic acid Azelaic acid is bactericidal against Propionibacterium acnes and Staphylococcus epidermidis due to its inhibitory effect on the synthesis of microbial cellular ...
T0927 Butylparaben Butylparaben is a standardized chemical allergen, increasing histamine release, and cell-mediated immunity.
T0933 Delta-Gluconolactone Gluconolactone is a naturally-occurring food additive used as a sequestrant, an acidifier, or a curing, pickling, or leavening agent. It is a cyclic ester of D-...
T0940 Acesulfame Potassium Acesulfame potassium is a non-nutritive sweetener.
T0941 Cyclamic acid Cyclamic acid is an artificial sweetening agent, usually employed as Na or Ca salt (cyclamate). Use suspended in some countries, including USA, because of possi...
T0949 Amstat Tranexamic acid is an Antifibrinolytic Agent. The physiologic effect of tranexamic acid is by means of Decreased Fibrinolysis.
T0953 Cefazolin sodium salt Cefazolin binds to and inactivates penicillin-binding proteins (PBP) located on the inner membrane of the bacterial cell wall. Cefazolin Sodium is the sodium sa...
T0955 Oxyclozanide Oxyclozanide is a salicylanilide anthelmintic used in grazing animals for fasciola and cestode infestations.
T0956 Abamectin Avermectin B1 (Abamectin) is served as anthelmintic and insecticide.
T0959 Ethopabate Ethopabate is an inhibitor of folate metabolism, used as a coccidiostat in poultry.
T0960 Iopanoic acid Iopanoic acid is an iodine-containing radiocontrast medium used in cholecystography.
T0961 Trometamol Trometamol is a proton acceptor used to treat acidemia. It inhibits both isoforms of cyclooxygenases (COX1 and COX2), thereby blocking the conversion of arachid...
T0967 Teicoplanin Teicoplanin is a semisynthetic glycopeptide antibiotic, used to treat Gram-positive bacteria.
T0969 Doramectin Doramectin is an antiparasitic agent.
T0977 Medrysone Medrysone is a topical, synthetic glucocorticoid with metabolic, anti-inflammatory and anti-allergic properties. Medrysone exerts its effect by interacting with...
T0982 (+)-Emetine dihydrochloride hydrate Emetine is a drug used as both an anti-protozoal and to induce vomiting. It is produced from the ipecac root.
T0983 Artamine Artamine, possessing antineoplastic properties, induces apoptosis by a p53-mediated mechanism and inhibits angiogenesis by chelating with copper, a cofactor for...
T0983L DL-Penicillamine DL-Penicillamine is a chelating agent recommended for the removal of excess copper in patients with Wilson's disease. DL-Penicillamine is only found in individu...
T0985 Oxacillin sodium Oxacillin sodium is an antibiotic similar to FLUCLOXACILLIN used in resistant staphylococci infections.
T0989 7-Aminocephalosporanic acid 7-Aminocephalosporanic acid is used for synthesis of cephalosporin antibiotics and intermediates.
T10001 (E)-Alprenoxime (E)-Alprenoxime is the isomer of the Alprenoxime which is a site-activated ocular β-blocker.
T10002 (E)-Crotylbarbital (E)-Crotylbarbital is the isomer of Crotylbarbital. Crotylbarbital has sedative and hypnotic effects and can be used for the treatment of insomnia.
T10003 α1 adrenoceptor-MO-1 α1 adrenoceptor-MO-1 (S enantiomer) has affinity at alpha 1 adrenergic receptor with alphalytic activity and analgesic action. It has more active than R enanti...
T10004 Palmitodiolein Palmitodiolein is a triacylglycerol existed in vegetable oils.
T10005 1,2-Dipalmitoyl-sn-glycerol 3-phosphate 1,2-Dipalmitoyl-sn-glycerol 3-phosphate, a phosphatidic acid, is a human endogenous metabolite.
T10005L 1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium 1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium, a phosphatidic acid, is a human endogenous metabolite.
T10008 BTM-1086 BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.
T1001 Dicloxacillin sodium Dicloxacillin NaOH is a narrow-spectrum β-Lactam antibiotic of the penicillin class, used to treat infections caused by susceptible Gram-positive bacteria.
T10010 1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol 1-(2-Quinoxalinyl)-1,2,3,4-butanetetrol is an endogenous metabolite.
T10011 1,3,5-Tricaffeoylquinic acid 1,3,5-Tricaffeoylquinic acid is a tricaffeoylquinic acid derivative isolated from Helichrysum populifolium with anti-HIV effect.
T10012 P7C3-OMe P7C3-OMe, a pro-neurogenic agent, has therapeutic benefits in neurodegenerative diseases. The R-enantiomer of P7C3-OMe is far more active than the S-enantiomer.
T10013 1-Acetyl-3-o-toluyl-5-fluorouracil 1-Acetyl-3-o-toluyl-5-fluorouracil is a potent antineoplastic agent.
T10014 (1α,1'S,4β)-Lanabecestat (1α,1'S,4β)-Lanabecestat is a Beta site APP Cleaving Enzymel (BACE1) inhibitor, and has IC50s of 2.2 nM (TR-FRET assay) and 0.28 nM (sAPPp release assay), res...
T10015 1-Deazaadenosine 1-Deazaadenosine is a potent Adenosine deaminase inhibitor (Ki: 0.66 μM). It exhibits anti-cancer activities in vitro and has the potential to be a chemotherap...
T10016 Hydrocarbon chain derivative 1 Hydrocarbon chain derivative 1 has inhibitory activities against lipid synthesis.
T10017 1-Linoleoyl Glycerol 1-Linoleoyl Glycerol is a fatty acid glycerol that has been isolated from Saururus chinensis roots.
T10018 1-Methyladenine 1-Methyladenine is a product of alkylation damage in DNA which can be repaired by damage reversal by oxidative demethylation.
T10019 1-Methylcytosine 1-Methylcytosine is a methylated form of cytosine. It is used as a nucleobase of hachimoji DNA, in which it pairs with Isoguanine.
T10020 1-Methyluric acid 1-Methyluric acid acts on the urinary bladder mucosa and increases blood glucose, triglyceride, insulin, and cholesterol levels.
T10021 1-Methylxanthine 1-Methylxanthine is an essential human urinary metabolite of caffeine and theophylline. 1-Methylxanthine enhances the radiosensitivity of tumor cells.
T10022 1-Myristoyl-2-stearoyl-sn-glycero-3-phosphocholine 1-Myristoyl-2-stearoyl-sn-glycero-3-phosphocholine is an endogenous metabolite.
T10023 1-Naphthol 1-naphthol is an excited state proton transfer (ESPT) fluorescent molecular probe.
T10024 1-Octanol 1-Octanol (Octanol), a saturated fatty alcohol, is a T-type calcium channels (T-channels) inhibitor with an IC50 of 4 μM for native T-currents[1]. 1-Octanol is...
T10025 1-PeCSO 1-PeCSO is isolated from onion or garlic bulbs. It acts as a key compound in garlic greening and reacts with lachrymatory factor synthase.
T10026 Tachykinin antagonist 1 Tachykinin antagonist 1 is an antagonist of neurokinin receptors extracted from patent US5968923 (example 32).
T10027 Anticonvulsant agent 1 Anticonvulsant agent 1 is an anticonvulsant compound extracted from patent WO2001062726A2 (Compound 156).
T10028 PDE4 inhibitor intermediate 1 PDE4 inhibitor intermediate 1 is a PDE4 inhibitor synthesis intermediate.
T10029 1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine 1-Stearoyl-2-arachidonoyl-sn-glycero-3-phosphocholine is an endogenous metabolite.
T1003 Tylosin Tylosin is a macrolide antibiotic obtained from cultures of Streptomyces fradiae. The drug is effective against many microorganisms in animals but not in humans...
T10030 1-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine 1-Stearoyl-2-linoleoyl-sn-glycero-3-phosphocholine is an endogenous metabolite.
T10031 EP1-antanoist-1 EP1-antagonist-1 is an EP1 antagonist (pKi: 7.54; pIC50: 8.5).
T10034 10,11-Dehydrocurvularin 10,11-Dehydrocurvularin is an antibiotic and a strong activator of the heat shock response. It inhibits the TGF-β signaling pathway and has anti-tumorous activ...
T10035 10,12-Tricosadiynoic acid 10,12-Tricosadiynoic acid is a highly selective and orally active inhibitor of acyl-CoA oxidase-1 (ACOX1). It can treat the high-fat diet- or obesity-induced me...
T10036 10β,17β-dihydroxyestra-1,4-dien-3-one 10β,17β-dihydroxyestra-1,4-dien-3-one is a brain-targeting bioprecursor prodrug of the main human estrogen, 17β-estradiol. It alleviates hot flushes in rat m...
T10037 10-​Isobutyryloxy-​8,​9-​epoxythymol isobutyrate 10-Isobutyryloxy-8,9-epoxythymol isobutyrate is a major constituent of Inula helenium and Inula royleana root cultures.
T10038 11-cis-Vaccenyl acetate 11-cis-Vaccenyl acetate is a male-specific lipid that mediates aggregation behavior in both male and female flies, which activates olfactory neurons located in ...
T10039 11-Deoxymogroside IIE 11-Deoxymogroside IIE is a cucurbitane glycoside, isolated from Siraitia grosvenorii fruits.
T1004 Benzyladenine 6-Benzylaminopurine, benzyl adenine or BAP is a first-generation synthetic cytokinin that elicits plant growth and development responses, setting blossoms and s...
T10040 11-Deoxymogroside IIIE 11-Deoxymogroside IIIE is a natural compound isolated from Siraitia grosvenorii.
T10041 11-Ketodihydrotestosterone 11-Ketodihydrotestosterone is a metabolite of 11β-Hydroxyandrostenedione. It is an active androgen and is also a potent androgen receptor (AR) agonist (Ki: 20....
T10042 11-Oxomogroside IIa 11-Oxomogroside IIa is a cucurbitane glycoside extracted from the fruits of Siraitia grosVenorii. It has inhibitory effects against the EBV-EA activation induce...
T10043 11-Oxomogroside IIe 11-Oxomogroside IIe is a triterpene glycoside isolated from Siraitia grosvenori[1].
T10045 15-Acetyl-deoxynivalenol 15-Acetyl-deoxynivalenol is a highly toxic trichothecene found in cereals and exhibits toxicity to HepG2 cells.
T10047 16-Methoxystrychnine 16-Methoxystrychnine is a alkaloid[1].
T10048 17a-Hydroxypregnenolone 17a-Hydroxypregnenolone is a pregnane steroid. It is a prohormone in the formation of dehydroepiandrosterone (DHEA).
T10049 1alpha, 25-Dihydroxy VD2-D6 1alpha, 25-Dihydroxy VD2-D6 is a deuterated form of vitamin D.
T1005 Amoxicillin Amoxicillin binds to and inactivates penicillin-binding proteins (PBPs) located on the inner membrane of the bacterial cell wall. Amoxicillin Anhydrous is the a...
T10050 1alpha-Hydroxy VD4 1alpha-Hydroxy VD4 can effectively induce the differentiation of monoblastic leukaemia U937, P39/TSU, and P31/FUJ cells.
T10051 5-HT3 antagonist 1 5-HT3 antagonist 1 is a potent and selective antagonist of 5-HT3 receptor.
T10052 AR-08 AR-​08 is an α2-adrenergic receptor agonist, used for the treatment of attention-deficit hyperactivity disorder (ADHD).
T10054 CI-949 CI-949 is an allergic mediator release inhibitor, which inhibits leukotriene C4/D4 (LTC4/LTD4), histamine, and thromboxane B2 (TXB2) release (IC50s: 0.5 μM, 11...
T10055 CHEMBL333994 CHEMBL333994 is a potent and orally effective antagonist of Cholecystokinin A (CCK-A; IC50: 0.67 nM).
T10056 Neurokinin antagonist 1 Neurokinin antagonist 1 is an antagonist of Neurokinin extracted from patent WO1998045262A1.
T10057 LTD4 antagonist 1 LTD4 antagonist 1 is a potent and orally active antagonist of leukotriene D4 (LTD4; Ki: 0.57 nM).
T10059 Neuromuscular Disorder-Targeting Compound 1 Neuromuscular Disorder-Targeting Compound 1 is a compound used in the research of neuromuscular disorders, for example, symptoms of chronic fatigue syndrome and...
T10060 (1S,2S,3R)-DT-061 (1S,2S,3R)-DT-061 is an enantiomer of DT-061 which is an orally bioavailable activator of PP2A.
T10062 (-)-GSK598809 (-)-GSK598809 is an isomer of GSK598809 that is a potent and selective antagonist of dopamine D3 Receptor.
T10063 LDL-IN-3 LDL-IN-3 is an anti-atherosclerotic agent extracted from patent WO/2005/039596A1 (example C25).
T10064 LH secretion antagonist 1 LH secretion antagonist 1 is an antagonist of luteinizing hormone secretion with analgesic activity.
T10065 2',3'-cGAMP 2',3'-cGAMP is an endogenous cGAMP in mammalian cells. It binds to STING with a high affinity and is a potent inducer of IFN-β.
T10065L 2',3'-cGAMP sodium 2',3'-cGAMP sodium is an endogenous cGAMP in mammalian cells. It binds to STING with a high affinity and is a potent inducer of IFN-β.
T10066 2',5'-Dideoxyadenosine 2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 µM).
T10068 2'-Azido-2'-deoxyuridine 2'-Azido-2'-deoxyuridine (N3dUrd) is a ribonucleotide reductase inhibitor with anti-cancer activity.
T10069 AMPK activator 1 AMPK activator 1 is an AMPK activator extracted from patent WO2013116491A1 (compound No.1-75, EC50: <0.1μM).
T1007 Lupetidin Lupetidin is a neuropathic blocker, with antihypertensive effect.
T10071 Itch-Targeting Compound 1 Itch-Targeting Compound 1 is an anti-itching compound.
T10072 2-Hydroxy Ibuprofen 2-Hydroxy Ibuprofen is a metabolite of Ibuprofen. Ibuprofen is an anti-inflammatory inhibitor targeting COX-1/COX-2 (IC50s: 13 μM/370 μM).
T10073 2-Iodomelatonin 2-Iodomelatonin is a potent agonist of melatonin receptor 1 (MT1, Ki: 28 pM), it is more 5-fold selective for MT1 over MT2.
T10074 2-Keto-D-Glucose 2-Keto-D-Glucose (D-Glucosone) is a key intermediate in a secondary metabolic pathway leading to the antibiotic Cortalcerone. It is found in various natural sou...
T10076 2-Methylcitric acid 2-Methylcitric acid (Methylcitric acid) is an endogenous metabolite in the 2-methylcitric acid cycle. It accumulates in methylmalonic and propionic acidemias.
T10076L 2-Methylcitric acid trisodium 2-Methylcitric acid trisodium (Methylcitric acid) is an endogenous metabolite in the 2-methylcitric acid cycle. It accumulates in methylmalonic and propionic ac...
T10077 2-O-β-D-Glucopyranosyl-L-ascorbic acid 2-O-β-D-Glucopyranosyl-L-ascorbic acid (AA-2βG) is isolated from Lycium Fruit. It is a stable vitamin C analog with anti-tumor activity.
T10078 2-PCCA hydrochloride 2-PCCA hydrochloride is an agonist of GPR88 receptor. It inhibits GPR88-mediated cAMP production (EC50: 116 nM in HEK293 cells).
T10080 PF-592379 PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).
T10082 DPP-IV-IN-1 DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).
T10083 Desethyl KBT-3022 Desethyl KBT-3022 is an active metabolite of the antiplatelet compound KBT-3022.
T10085 20(S)-Hydroxycholesterol 20(S)-hydroxyCholesterol is an allosteric activator of the oncoprotein smoothened (Smo) that activates the hedgehog signaling pathway with an EC50 of 3 μM in N...
T10086 24-Hydroxycholesterol 24-Hydroxycholesterol is a natural sterol, which serves as a positive allosteric modulator of NMDA receptors, and a potent activator of the transcription factor...
T10087 24-Norursodeoxycholic acid 24-norursodeoxycholic acid is a side chain-shortened C23 homolog of UDCA. It has shown potent anti-inflammatory, anti-cholestatic, and anti-fibrotic properties.
T10088 24R-Calcipotriol 24R-Calcipotriol(PRI 2202) is an impurity of Calcipotriol which is a ligand of VDR-like receptors.
T10089 2614W94 2614W94 is a selective, competitive, and reversible inhibitor of monoamine oxidase-A with IC50 of 5 nM and Ki of 1.6 nM with serotonin as a substrate.
T10090 264W94 264W94 is a potent ileal bile acid transporter (IBAT) inhibitor and a new cholesterol-lowering agent. 264W94 has CYP7A1 induction and antilipemic action.
T10091 Anti-inflammatory agent 1 Anti-inflammatory agent 1 is an anti-inflammatory compound extracted from patent WO 2009003229 A1 (example 36).
T10092 PSN-GK1 PSN-GK1 is a potent activator of glucokinase (EC50: 0.13 μM).
T10093 (2R,3R)-E1R (2R,3R)-E1R is an enantiomer of E1R. (2R,3R)-E1R is a sigma-1 receptor positive allosteric modulator for the treatment of cognition/memory disorders.
T10093L E1R E1R is a positive sigma-1 receptor (Sig1R PAM) allosteric modulator. It has a cognition-enhancing activity.
T10094 (2R,3S)-E1R (2R,3S)-E1R (Compound 2c) is an enantiomer of E1R. (2R,3R)-E1R is a sigma-1 receptor positive allosteric modulator for the treatment of cognition/memory disorde...
T10095 (2R,4R)-APDC (2R,4R)-APDC is a selective group II metabotropic glutamate receptors (mGluRs) agonist. It has anticonvulsant and neuroprotective effects.
T10096L Voruciclib Voruciclib is an orally active and selective CDK inhibitor (Ki: 0.626 nM-9.1 nM). Voruciclib represses the expression of MCL-1 in multiple models of diffuse lar...
T10096L2 (2S,3R)-Voruciclib hydrochloride (2S,3R)-Voruciclib hydrochloride is the (2S,3R)-enantiomer of Voruciclib. It is an orally active CDK inhibitor.
T10097 (2S,3S)-E1R (2S,3S)-E1R (Compound 2d) is an enantiomer of E1R. (2R,3R)-E1R is a sigma-1 receptor positive allosteric modulator for the treatment of cognition/memory disorde...
T10099 2'-Deoxypseudoisocytidine 2'-Deoxypseudoisocytidine is a nucleoside analogue.
T10100 QF0301B QF0301B is an antagonist of the α1 adrenergic receptor. It also is a low α2 adrenoceptor, 5-HT2A, and histamine H1 receptor blocker.
T10101 Calcium channel-modulator-1 Calcium channel-modulator-1 is a modulator of calcium channel and blocks aortic contraction (IC50: 0.8 μM).
T10102 3,6-DMAD hydrochloride 3,6-DMAD hydrochloride is an inhibitor of the IRE1α-XBP1 pathway of the unfolded protein response.
T10103 3,3'-Diiodo-L-thyronine 3,3'-Diiodo-L-thyronine (3,3'-T2) is an endogenous metabolite of thyroid hormone. It significantly enhances COX activity.
T10104 3,4-Dihydroxybenzylamine hydrobromide 3,4-Dihydroxybenzylamine hydrobromide (NSC 263475 hydrobromide) is a dopamine analog with cytotoxic and inhibits DNA polymerase activity in melanoma cells.
T10106 3-arylisoquinolinamine derivative 3-arylisoquinolinamine derivative is a compound with antitumor activity.
T10108 3-Bromocytisine 3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, (IC50s: 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh).
T10109 3-Carene 3-Carene is a bicyclic monoterpene in essential oils extracted from pine trees.
T10110 3-CPs 3-CPs (3-Carbethoxypsoralen) is a serotype capsular polysaccharide which can interfere with antibody-mediated bacterial killing.
T10112 3-Hydroxy-4-methoxyacetophenone 3-Hydroxy-4-methoxyacetophenone(Acetoisovanillone) is an active compound isolated from Pycnocycla spinosa. It possesses anti-inflammatory activity and prevents ...
T10115 3-Nitrocoumarin 3-Nitrocoumarin (3-NC) is a potent and selective Phospholipase C-γ (PLCγ) inhibitor.
T10116 3-O-Acetylbufotalin 3-O-Acetylbufotalin is a derivate of bufadienolide with anti-cancer activity.
T10117 3'-​O-​Acetylhamaudol 3'-O-Acetylhamaudol, isolated from the roots of Angelica japonica, exhibits anti-tumor activity through dual actions, anti-angiogenesis and intestinal intraepit...
T10120 3-Oxo Atorvastatin 3-Oxo Atorvastatin is an impurity of Atorvastatin. Atorvastatin is an HMG-CoA reductase inhibitor and has the ability to effectively decrease blood lipids.
T10121 Substance P Receptor Antagonist 1 Substance P Receptor Antagonist 1 has the potential function in gastrointestinal disorders, inflammatory diseases, respiratory, and central nervous system disor...
T10122 Anti-neurodegeneration agent 1 Anti-neurodegeneration agent 1 a neurodegeneration-targeting agent extracted from patent WO2008039514A1 (Compound I).
T10124 Antiulcer Agent 1 Antiulcer Agent 1 is a 2-(3,4-dimethoxyphenyl)ethylamine derivative for oral administration.
T10125 (3R,4R)-A2-32-01 (3R,4R)-A2-32-01 (compound 2) is a specific caseinolytic protein proteases (ClpP) inhibitor (EC50: 4.5 μM).
T10126 (3R,5R)-Rosuvastatin (3R,5R)-Rosuvastatin is the (3R,5R)-enantiomer of Rosuvastatin. Rosuvastatin is a competitive HMG-CoA reductase inhibitor (IC50: 11 nM).
T10127 (3R,5S)-Atorvastatin sodium (3R,5S)-Atorvastatin sodium is an impurity of Atorvastatin. Atorvastatin is an HMG-CoA reductase inhibitor and has the ability to effectively decrease blood lip...
T10128 (3S,5R)-Fluvastatin D6 sodium (3S,5R)-Fluvastatin D6 sodium is the deuterium-labeled (3S,5R)-Fluvastatin sodium. Fluvastatin is a first fully synthetic, competitive HMG-CoA reductase inhibit...
T10129 (3S,5R)-Fluvastatin sodium (3S,5R)-Fluvastatin sodium is the (3S,5R)-enantiomer of Fluvastatin. Fluvastatin is a first fully synthetic, competitive HMG-CoA reductase inhibitor (IC50: 8 nM...
T10130 (3S,5R)-Pitavastatin calcium (3S,5R)-Pitavastatin calcium is the enantiomer of Pitavastatin which is a potent HMG-CoA reductase inhibitor.
T10131 (3S,5R)-Rosuvastatin (3S,5R)-Rosuvastatin is the (3R,5R)-enantiomer of Rosuvastatin. Rosuvastatin is a competitive HMG-CoA reductase inhibitor (IC50: 11 nM).
T10132 (3S,5S)-Pitavastatin calcium (3S,5S)-Pitavastatin calcium is the 3-epimer of Pitavastatin which is a potent HMG-CoA reductase inhibitor.
T10133 3'-Azido-3'-deoxy-5-methylcytidine 3'-Azido-3'-deoxy-5-methylcytidine (CS-92) is a potent xenotropic murine leukemia-related retrovirus (XMRV) inhibitor (CC50: 43.5 μM) in MCF-7 cells. It also i...
T10134 4,7,10,13,16-Docosapentaenoic acid 4,7,10,13,16-Docosapentaenoic acid is an endogenous metabolite.
T10135 4-Acetamidophenyl acetate 4-Acetamidophenyl acetate is an impurity of Acetaminophen. Acetaminophen is a selective COX-2 inhibitor (IC50: 25.8 μM) and is a potent hepatic N-acetyltransfe...
T10136 4-Acetylsimvastatin 4-Acetylsimvastatin is acetylated simvastatin. Simvastatin is a competitive inhibitor of HMG-CoA reductase (Ki: 0.2 nM).
T10137 4-​Bromo A23187 4-Bromo A23187 is a halogenated analog of the calcium ionophore A-23187. 4-Bromo A23187 is a calcium modulator and induces apoptosis in different cells.
T10138 4-Desmethoxy Omeprazole 4-Desmethoxy Omeprazole is the active metabolite of Omeprazole. Omeprazole is a proton pump inhibitor (PPI). Omeprazole shows competitive inhibition of CYP2C19 ...
T10139 4-Desmethyl Istradefylline 4-Desmethyl Istradefylline is a Istradefylline metabolite. Istradefylline is a very potent, selective, and orally active adenosine A2A receptor antagonist with ...
T10140 4-Diethylaminobenzaldehyde 4-Diethylaminobenzaldehyde is a reversible aldehyde dehydrogenase (ALDH) inhibitor (Ki: 4 nM for ALDH1). It displays a potent anti-androgenic effect (IC50: 1.71...
T10141 4'-Ethynyl-2'-deoxyadenosine 4'-Ethynyl-2'-deoxyadenosine (4'-E-dA) is a nucleoside reverse transcriptase (RT) inhibitor. It is potent against drug-resistant HIV variants (EC50: 98 nM in MT...
T10142 4-Ethynyl-L-phenylalanine 4-Ethynyl-L-phenylalanine is a selective, reversible and competitive inhibitor of tryptophan hydroxylase (TPH). 4-Ethynyl-L-phenylalanine is a competitive inhib...
T10143 4-Hydroxyacetophenone oxime 4-Hydroxyacetophenone oxime is an impurity of Acetaminophen (Paracetamol). Acetaminophen is a potent COX-2 and hepatic NAT2 inhibitor and used antipyretic and a...
T10144 4-Hydroxyatomoxetine D3 4-Hydroxyatomoxetine D3 is a deuterium labeled 4-Hydroxyatomoxetine. 4-Hydroxyatomoxetine is an active metabolite of Atomoxetine. 4-Hydroxyatomoxetine is metabo...
T10145 4-Hydroxyatomoxetine 4-Hydroxyatomoxetine is an active metabolite of Atomoxetine. 4-Hydroxyatomoxetine is metabolized by CYP2D6. Atomoxetine is a noradrenaline reuptake inhibitor.
T10147 4-Hydroxymephenytoin 4-Hydroxymephenytoin is the metabolism of an antiepileptic drug mephenytoin. Mephenytoin is used as a CYP2C19 substrate.
T10148 4-Hydroxynonenal 4-Hydroxynonenal (4-HNE) is an oxidative/nitrosative stress biomarker. It is a substrate and an inhibitor of acetaldehyde dehydrogenase 2 (ALDH2).
T10149 4-Hydroxypropranolol D7 hydrochloride 4-Hydroxypropranolol D7 hydrochloride is deuterium-labeled 4-Hydroxypropranolol hydrochloride. 4-Hydroxypropranolol hydrochloride is an active metabolite of Pro...
T10150 4-Hydroxypropranolol hydrochloride 4-Hydroxypropranolol hydrochloride is an active metabolite of Propranolol, with a potency comparable to Propranolol. It inhibits β1- and β2-adrenergic recepto...
T10153 4-O-Methyl honokiol 4-O-Methyl honokiol, a natural neolignan isolated from Magnolia officinalis, acts as a PPARγ agonist and inhibits NF-κB activity, used for cancer and inflamma...
T10154 MAO-B-IN-1 MAO-B-IN-1 is a monoamine oxidase B inhibitor and can be used for the research of neurological diseases.
T10155 4'-Raloxifene-β-D-glucopyranoside 4'-Raloxifene-β-D-glucopyranoside is a metabolite of Raloxifene. 4'-Raloxifene-β-D-glucopyranoside is a selective and orally active estrogen receptor antagoni...
T10157 Regorafénib N-oxyde (M2) Regorafénib N-oxyde M2 is an active metabolite of Regorafenib. Regorafenib is a multi-target inhibitor for VEGFR1/2/3, PDGFRβ, RET, Kit, and Raf-1 (IC50s: 13/...
T10158 42-(2-Tetrazolyl)rapamycin 42-(2-Tetrazolyl)rapamycin is a prodrug compound of a rapamycin analog extracted from patent US 20080171763 A1, Example 1.
T10159 48740 RP 48740 RP (RP-55778) is a platelet-activating factor (PAF) antagonist.
T10161 Antiasthmatic Compound 1 Antiasthmatic Compound 1 is an antiasthmatic agent.
T10163 4'-Methylchrysoeriol 4'-Methylchrysoeriol is a potent inhibitor of cytochrome P450 enzymes (IC50: 19 nM for human P450 1B1-dependent EROD).
T10164 5,6-Dihydroxyindole 5,6-Dihydroxyindole is a melanin precursor and has a broad-spectrum antibacterial, antiviral, antifungal, antiparasitic activity. It has cytotoxic effects and i...
T10165 5-A-RU 5-A-RU (5-Amino-6-(D-ribitylamino)uracil), a precursor of bacterial Riboflavin, is a mucosal-associated invariant T (MAIT) cells activator. 5-A-RU forms potent ...
T10165L 5-A-RU hydrochloride 5-Amino-6-(D-ribitylamino)uracil hydrochloride, a precursor of bacterial Riboflavin, is a mucosal-associated invariant T (MAIT) cells activator. 5-A-RU forms po...
T10166 Lipid peroxidation inhibitor 1 Lipid peroxidation inhibitor 1 is an inhibitor of lipid peroxidation (IC50: 0.07 μM).
T10167 5-Dehydroepisterol 5-Dehydroepisterol is an episterol derivative with anti-fungal activities. It can be formed by C-5 sterol desaturase and converted into 24-methylenecholesterol ...
T1017 Fluoroethyl Flurothyl is a convulsant used in experimental animals.
T10171 5-Hydroxypyrazine-2-Carboxylic Acid 5-Hydroxypyrazine-2-Carboxylic Acid is a metabolite of anti-tuberculosis drug pyrazinamide.
T10172 5-Iodo-indirubin-3'-monoxime 5-Iodo-indirubin-3'-monoxime is a potent GSK-3β, CDK5/P25 and CDK1/cyclin B inhibitor, competing with ATP for binding to the catalytic site of the kinase (IC50...
T10173 MCHR1 antagonist 1 MCHR1 antagonist 1 is a selective antagonist of melanin-concentrating hormone-1 (MCH1) receptor (Kb: 1 nM, Ki: 4 nM at human MCH1).
T10174 5-R-Rivaroxaban 5-R-Rivaroxaban is (R)-enantiomer of Rivaroxaban. Rivaroxaban (BAY 59-7939) is a highly potent and selective, direct Factor Xa (FXa) inhibitor (IC50 0.7 nM; Ki ...
T10175 (5E,9E,13E)-Teprenone (5E,9E,13E)-Teprenone is an isomer of Teprenone with antiulcer activity. It induces transcriptional activation of HSP genes that may increase gastric mucosal de...
T10176 TRPV antagonist 1 TRPV antagonist 1 is an antagonist of transient receptor potential vanilloid (TRPV; IC50 < 250 nM).
T10177 (5Z,2E)-CU-3 (5Z,2E)-CU-3 is a selective inhibitor against the α-isozyme of DGK (IC50: 0.6 μM), competitively inhibits the affinity of DGKα for ATP (Km: 0.48 mM).
T10178 Guanosine 5'-triphosphate trisodium salt hydrate 5'-GTP trisodium salt hydrate, an activator of the signal-transducing G proteins, serves as a precursor of mononucleotide units in the enzymatic biosynthesis of...
T10179 5β-​Dutasteride 5β-Dutasteride is the S configuration of Dutasteride. It is a potent inhibitor of both 5 alpha-reductase isozymes.
T10180 6-Alpha Naloxol 6-Alpha Naloxol(Alpha-Naloxol) is an opioid antagonist and is a human metabolite of naloxone.
T10181 6-beta-Naloxol D5 hydrochloride 6-beta-Naloxol D5 hydrochloride is the deuterium-labeled 6-beta-Naloxol, which is an opioid antagonist closely related to naloxone.
T10182 6-Hydroxybenzbromarone 6-Hydroxybenzbromarone is the major metabolite of Benzbromarone. 6-Hydroxybenzbromarone is a protein Eyes Absent 3 (EYA3) inhibitor (IC50: 21.5 μM). It is an a...
T10183 6-Methoxytricin 6-Methoxytricin is a flavonoid isolated from Artemisia iwayomogi. It is an inhibitor on aldose reductase (AR) and advanced glycation endproduct (AGE) formation ...
T10184 6-Methyl-5-azacytidine 6-Methyl-5-azacytidine is a potent DNMT inhibitor.
T10185 6-Phosphogluconic acid 6-Phosphogluconic acid is a potent and competitive phosphoglucose isomerase (PGI) inhibitor (Kis: 48 μM for glucose 6-phosphate and 42 μM for fructose 6-phosp...
T10186 6-Quinoxalinecarboxylic acid, 2,3-bis(bromomethyl)- 6-Quinoxalinecarboxylic acid, 2,3-bis(bromomethyl)-, derived from 2,3-Bis(bromomethyl)quinoxaline, shows antibacterial activity.
T10187 6-Raloxifene-β-D-glucopyranoside 6-Raloxifene-β-D-glucopyranoside is a benzothiophene glucuronidated at the 6' position. It is a selective and orally active estrogen receptor antagonist. 6-Ral...
T10188 6RK73 6RK73 is a covalent irreversible and specific UCHL1 inhibitor (IC50: 0.23 µM). 6RK73 shows almost no inhibition of UCHL3 (IC50: 236 µM).
T10189 7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene 7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene is a liver receptor homolog-1 (LRH-1) antagonist (IC50: 3.1 μM).
T10190 7-BIA 7-BIA is a receptor-type protein tyrosine phosphatase D (PTPRD) inhibitor (IC50: 1-3 μM).
T10191 7-Chlorokynurenic acid sodium salt 7-Chlorokynurenic acid sodium salt (7-CKA sodium salt) is a potent and selective antagonist of the glycine B coagonist site of the NMDA receptor (IC50: 0.56 μM...
T10191L 7-Chlorokynurenic acid 7-Chlorokynurenic acid (7-CKA) is a potent and selective antagonist of the glycine B coagonist site of the N-methyl-D-aspartate (NMDA) receptor (IC50=0.56 μM)....
T10193 7-Desmethyl-agomelatine 7-Desmethyl-agomelatine is a metabolite of Agomelatine and has less activity than Agomelatine. Agomelatine is a melatonergic (MT1 and MT2) agonist and 5-HT2C an...
T10194 7-Methylguanine 7-Methylguanine is a metabolite of DNA methylation. It can be generated by methylating agents and used as a probe of DNA–protein interactions and a key compon...
T10195 7-O-Geranylscopoletin 7-O-Geranylscopoletin is a natural coumarin from the root of Atalantia monophylla. Various parts of this plant have been used for folk medicine for several purp...
T10196 7α-Hydroxy-4-cholesten-3-one 7α-Hydroxy-4-cholesten-3-one is an intermediate in the synthesis of bile acids from cholesterol. It is a PXR agonist. 7α-Hydroxy-cholest-4-en-3-one is a bioma...
T10197 8,​9-​Epoxy-​3-​isobutyryloxy-​10-​(2-​methylbutanoyl)​thymol 8,9-Epoxy-3-isobutyryloxy-10-(2-methylbutanoyl)thymol is a chemical composition of essential oils from Telekia speciosa. It also shows marked antipro-liferative...
T10198 8-M-PDOT 8-M-PDOT (AH-002) is a selective melatonin MT2 receptor agonist. It is 5.2-fold selective for MT2 over MT1 receptors. 8-M-PDOT binds human recombinant MT2 and M...
T10199 GNF-PF-3777 GNF-PF-3777 (8-Nitrotryptanthrin) is a potent inhibitor of human indoleamine 2,3-dioxygenase 2 (hIDO2; Ki: 0.97 μM).
T10200 9-Hydroxyellipticine hydrochloride 9-Hydroxyellipticine hydrochloride is a inhibitor of Topo II and RyR. It exhibits antitumor, antioxidant and catecholamine-releasing activities. 9-Hydroxyellipt...
T10201 PDE IV-IN-1 PDE IV-IN-1 is a phosphodiesterase IV inhibitor used for the research of COPD, asthma, or other inflammatory diseases.
T10203 A 1120 A 1120 is a nonretinoid retinol-binding protein 4 (RBP4) antagonist (Ki: 8.3 nM), which disrupts the interaction between RBP4 and its binding partner transthyre...
T10204 A-317491 sodium salt hydrate A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors.
T10205 A-395 A-395 is an antagonist of polycomb repressive complex 2 (PRC2) protein-protein interactions that potently inhibits the trimeric PRC2 complex (EZH2-EED-SUZ12, IC...
T10209 A-887826 A-887826 is a selective, orally bioavailable, and voltage-dependent Na(v1.8) channel blocker (IC50: 11 nM). It attenuates neuropathic tactile allodynia in vivo.
T10211 Aβ42-IN-1 Aβ42-IN-1 is a novel and orally active γ-secretase modulator (GSM). Aβ42-IN-1 potently reduced Aβ42 levels (IC50: 0.091 µM) without CYP3A4 inhibition.
T10212 A2AR-agonist-1 A2AR-agonist-1 is a potent A2AR and ENT1 agonist (Ki: 4.39 and 3.47 for A2AR and ENT1. It targets the Adenosine A2A Receptor and Adenosine Transporter for Neuro...
T10215 AAPK-25 AAPK-25 is a potent and selective Aurora/PLK dual inhibitor with anti-tumor activity, which can cause mitotic delay and arrest cells in prometaphase, followed b...
T10216 AB-680 AB-680 is a highly potent, reversible, and selective inhibitor of CD73 (an ectonucleotidase, Ki: 4.9 pM for hCD73) with anti-tumor activity, displays >10,000-fo...
T10217 Abarelix Acetate Abarelix (PPI 149; R 3827) Acetate is a potent gonadotrophin-releasing hormone (GnRH) antagonist, used for prostate cancer research.
T10217L Abarelix Abarelix (R3827; PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.
T10218 Abatacept Abatacept (CTLA4lg) is a soluble fusion protein consisting of the extracellular domain of human CTLA4 and a fragment of the Fc portion of human IgG1 (hinge and ...
T10219 ABBV-4083 ABBV-4083 is a Tylosin A analog that has potent anti-Wolbachia and anti-filarial activity.
T10221 Abeprazan hydrochloride Abeprazan (DWP14012) hydrochloride is a potassium-competitive acid blocker. It inhibits H+, K+- ATPase by reversible potassium-competitive ionic binding with no...
T10221L Abeprazan Abeprazan (DWP14012) is a potassium-competitive acid blocker and it is developed as a potential alternative to proton pump inhibitor for the treatment of acid-r...
T10222 ABMA ABMA is a broad-spectrum inhibitor of intracellular toxins and pathogens. ABMA efficiently protects cells against various pathogens including viruses, intracell...
T10223 ABT-100 ABT-100 is a potent, highly selective, and orally active farnesyl transferase inhibitor with broad-spectrum antitumor activity.
T10224 ABT-418 hydrochloride ABT-418 hydrochloride is a selective agonist of nAChRs with cognitive enhancing and anxiolytic activities. It activates cholinergic channel and can be used for ...
T10225 ABT-546 ABT-546 (A-216546) is a potent, highly selective, and active endothelin ETA receptor antagonist with a Ki of 0.46 nM for [125I]endothelin-1 binding to cloned hu...
T10226 Sofiniclin Sofiniclin (ABT 894) is an agonist of nicotinic acetylcholine receptor (nAChR). It is used for the research for attention-deficit/hyperactivity disorder (ADHD).
T10227 Ac-Gly-BoroPro Ac-Gly-BoroPro is a selective FAP inhibitor (Ki: 23 nM).
T10229 Acebutolol D7 Acebutolol D7 is a deuterium-labeled Acebutolol. Acebutolol is a selective antagonist of the β1 adrenergic receptor used in the treatment of angina pectoris, h...
T1023 Cefoxitin sodium Cefoxitin sodium is a semisynthetic cephamycin antibiotic resistant to beta-lactamase.
T10230 MC-4R Agonist 1 MC-4R Agonist 1 is an agonist of human melanocortin-4 receptor (MC-4R) and can be used in the research of sexual dysfunction, obesity, and diabetes.
T10231 Acetazolamide D3 Acetazolamide D3 is a deuterium-labeled Acetazolamide. Acetazolamide is a potent carbonic anhydrase inhibitor.
T10232 Acetophenazine dimaleate Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression.
T10233 Acetylarenobufagin Acetylarenobufagin is a steroidal hypoxia-inducible factor-1 (HIF-1) modulator.
T10235 Acetyllovastatin Acetyllovastatin (acetate of Lovastatin) presents a moderate inhibitory effect against the acetylcholinesterase (IC50: 79 μg/mL). Lovastatin displays antifunga...
T10236 ACHN-975 TFA ACHN-975 TFA is a selective LpxC inhibitor with a subnanomolar inhibitory. It is against a wide range of gram-negative bacterias with low MIC values (≤1 μg/m...
T10236L ACHN-975 ACHN-975 is against a wide range of gram-negative bacterias with low MIC values (≤1 μg/mL)[1]. ACHN-975 is a selective LpxC inhibitor and exhibits a subnanom...
T10237 ACHP Hydrochloride ACHP Hydrochloride (IKK-2 Inhibitor VIII) is a highly potent and selective IKK-β inhibitor (IC50: 8.5 nM).
T10239 Acolbifene Acolbifene (EM-652; SCH 57068) is a fourth-generation selective estrogen receptor antagonist (LC50: 22 nM).
T10241 Acrivastine D7 Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.
T10242 ACT-389949 ACT-389949 is a potent and selective agonist of formyl peptide receptor type 2 (FPR2)/Lipoxin A4 receptor (ALX), with an EC50 of 3 nM for FPR2/ALX internalizati...
T10243 ACX-362E ACX-362E is an orally available DNA polymerase IIIC (pol IIIC) inhibitor, acts as an antimicrobial agent to treat Gram-positive infections (MIC50: 2 μg/mL for ...
T10246 Adapalene sodium salt Adapalene (CD 271; Differin) sodium salt is a synthetic retinoid and a Retinoic acid receptor agonist.
T10248 Adenosine antagonist-1 Adenosine antagonist-1 is an adenosine A3 receptor (AA3R) antagonist.
T10249 Adoprazine Adoprazine is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.
T10250 ADRA1D receptor agonist 1 ADRA1D receptor agonist 1 is a potent, selective, and orally active α1D adrenoceptor antagonist (Ki: 1.6 nM).
T10251 Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA Adrenocorticotropic Hormone (ACTH) (1-39), rat (TFA) is a potent melanocortin 2 receptor (MC2) agonist.
T10252 ADU-S100 disodium salt ADU-S100 (MIW815) disodium salt is an activator of stimulator of interferon genes (STING).
T10252L ADU-S100 enantiomer ammonium salt ADU-S100 (MIW815) enantiomer ammonium salt is the less active enantiomer of ADU-S100. ADU-S100 is an activator of the stimulator of interferon genes (STING).
T10252L2 ADU-S100 ammonium salt ADU-S100 ammonium salt is an stimulator of interferon genes (STING) activator.
T10252L3 ADU-S100 ADU-S100 is an activator of stimulator of interferon genes (STING).
T10253 AD 0261 AD 0261 is a radical scavenger. It has a strong inhibitory action on the generation of lipid peroxides and superoxide anions.
T10257 Afatinib N-Oxide Afatinib N-Oxide is an impurity of Afatinib in oxidative degradation. Afatinib is an irreversible EGFR family inhibitor.
T10259 AGI-25696 AGI-25696 is a methionine adenosyltransferase 2A (MATA2 ) inhibitors useful for the treatment of cancer. It blocks the growth of MTAP-deleted tumors in vivo.
T10260 Aglafoline Aglafoline inhibits in a concentration-dependent manner the aggregation and ATP release reaction induced in washed rabbit platelets by PAF (platelet-activating ...
T10261 AGN 196996 AGN 196996 is a potent and selective RARα antagonist (Ki: 2 nM) and little binding affinity for RARβ (Ki: 1087 nM) and RARγ (Ki: 8523 nM).
T10262 AGN 205327 AGN 205327 is a potent synthetic RARs agonist (EC50s: 3766/734/32 nM for RARα/β/γ) and has no inhibition on RXR.
T10263 AGN 205728 AGN 205728 is a potent and selective RARγ antagonist (Ki: 3 nM; IC95: 0.6 nM) and has no inhibition on RARα and RARβ.
T10264 AGN 192836 AGN 192836 is a potent and selective α2 adrenergic agonist (EC50s: 8.7, 41 and 6.6 nM for α2A, α2B and α2C receptor).
T10265 AGN 194078 AGN 194078 is a selective RARα agonist (Kd: 3 nM; EC50: 112 nM).
T10266 Agomelatine D6 Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.
T10268 AGX51 AGX51 is a first-in-class pan-Id (inhibitors of DNA-binding/differentiation proteins) antagonist and degrader.
T10269 AHR antagonist 2 AHR antagonist 2 is a potent aryl hydrocarbon receptor (AHR) antagonist, extracted from patent WO2019101641A1, compound example 1 (IC50s: 0.885 and 2.03 nM for ...
T10270 BAY 2416964 BAY 2416964 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1 (example 192, IC50: 341 nM). It has th...
T10271 AHR antagonist 4 AHR antagonist 4 is a potent aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018146010A1 (example 293; IC50: 82.2 nM). It has anti-cancer ef...
T10272 AHR antagonist 5 AHR antagonist 5 is a potent and orally active aryl hydrocarbon receptor (AHR) antagonist extracted from patent WO2018195397 (example 39; IC50 < 0.5 µΜ). It s...
T10273 AhR modulator-1 AhR modulator-1 is a selective and orally active aryl hydrocarbon receptor (AhR) modulator. It inhibits metastasis, in part, by inhibiting prostatic VEGF produc...
T10278 Alamethicin Alamethicin is isolated from Trichoderma viride. It is a channel-forming peptide antibiotic and induces voltage-gated conductance in model and cell membranes.
T10279 Alfacalcidol-D6 Alfacalcidol-D6 is a deuterated Alfacalcidol. Alfacalcidol is a non-selective VDR activator medication.
T1028 Moxonidine Moxonidine is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.
T10280 Alimemazine D6 Alimemazine D6 is a deuterium-labeled Alimemazine. Alimemazine is an antihistamine.
T10281 Alimemazine Alimemazine (Trimeprazine) is generally used as an antipruritic agent and also a hemagglutinin (HA)-receptor antagonist. Alimemazine also acts as a partial agon...
T10282 Aliskiren D6 Hydrochloride Aliskiren (CGP 60536) D6 Hydrochloride is a deuterium-labeled Aliskiren. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM).
T10284 ALK-IN-6 ALK-IN-6 is an orally bioavailable inhibitor of anaplastic lymphoma kinase (ALK, IC50s: 71 nM, 18.72 nM, and 36.81 nM for ALK wild, ALK F1196M and ALK F1174L).
T10285 ALK inhibitor 1 ALK inhibitor 1 is a selective ALK kinase inhibitor.
T10286 ALK/ROS1-IN-1 ALK/ROS1-IN-1 is a potent and selective anti-crizotinib-resistant ALK/ROS1 dual inhibitor (IC50s: 0.530 μM and 0.174 μM for ROS1 and ALK enzyme).
T10288 Alogliptin (13CD3) Alogliptin (SYR-322) 13CD3 is the deuterium-labeled Alogliptin. Alogliptin is a selective inhibitor of DPP-4.
T10289 Alosetron ((Z)-2-butenedioate) Alosetron (GR 68755) (Z)-2-butenedioate is a Serotonin 5HT3-receptor antagonist that is used in the treatment of irritable bowel syndrome.
T10290 Alpertine Alpertine is an antipsychotic agent extracted from patent US 5955459 A.
T10291 α-Truxillic acid α-Truxillic acid is formed by the dimerization of two molecules of α-trans-cinnamic acid with anti-inflammatory activities.
T10295 Amantanium bromide Amantanium bromide is a quaternary ammonium compound used as an antiseptic/disinfectant for therapeutic function.
T10297 AMG 487 (S-enantiomer) AMG 487 S-enantiomer is the S enantiomer of AMG 487. AMG 487 is an CXCR3 antagonist.
T10297L AMG 487 AMG 487 is an orally active and selective antagonist of CXC chemokine receptor 3 (CXCR3). It inhibits the binding of CXCL10 and CXCL11 to CXCR3 with IC50s of 8....
T10301 AMG8380 AMG8380 is an orally active and less active enantiomer of AMG8379 served as a negative control. AMG8380 inhibits human and mouse voltage-gated sodium channel Na...
T10301L AMG8379 AMG8379 potently and reversibly blocks endogenous Tetrodotoxin (TTX)-sensitive sodium channels in dorsal root ganglia (DRG) neurons with an IC50 of 3.1 nM[1]. A...
T10302 Amibegron hydrochloride Amibegron hydrochloride is a selective β3-adrenoceptor agonist (EC50: 3.5 nM for β-adrenoceptor in rat colon). It has anxiolytic and antidepressant activity.
T10303 Aminoacyl tRNA synthetase-IN-1 Aminoacyl tRNA synthetase-IN-1 is an inhibitor of bacterial aminoacyl tRNA synthetase (aaRS).
T10304 Aminochlorthenoxazin Aminochlorthenoxazin is an antipyretic and analgesic agent.
T10305 Amiselimod hydrochloride Amiselimod hydrochloride is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.
T10306 Amoxicillin D4 Amoxicillin D4 (Amoxycillin D4) is a deuterium-labeled Amoxicillin. Amoxicillin is an antibiotic with broad-spectrum antimicrobial activity.
T10307 AMPA receptor modulator-1 AMPA receptor modulator-1 is an orally active, and selective AMPAR regulatory protein TARP γ-8 negative modulator (pIC50: 9.7), more selective over GluA1/γ-2 ...
T10308 AMPD2 inhibitor 1 AMPD2 inhibitor 1 is an inhibitor of adenosine monophosphate deaminase 2 (AMPD2), used in the research of salt craving, sugar craving, umami craving, and addict...
T10309 Amphethinile Amphethinile is an anti-tubulin agent. The Ka of Amphethinile with tubulin is 1.3 μM.
T1031 Cloxacillin sodium monohydrate Cloxacillin Sodium is the sodium salt of cloxaclliin, a semisynthetic beta-lactamase resistant penicillin antibiotic with antibacterial activity.
T10310 Amphotericin B methyl ester Amphotericin B methyl ester is the derivative of the antibiotic Amphotericin B. Amphotericin B methyl ester is the cholesterol-binding compound that possesses s...
T10311 Amphotericin X1 Amphotericin X1 is a derivative of Amphotericin B with good antifungal activity. Amphotericin X1 inhibits Candida albicans 33/079, Cryptococcus neoformans 451, ...
T10313 AMXT-1501 tetrahydrochloride AMXT-1501 tetrahydrochloride is an inhibitor of polyamine transport. It blocks tumor growth in immunocompetent mice but not in athymic nude mice lacking T cells...
T10314 AM 103 AM 103 is a potent and selective FLAP inhibitor (IC50: 4.2 nM).
T10315 AN-3485 AN-3485 is a Toll-Like Receptor(TLR) inhibitor (IC50s: 18 to 580 nM).
T10316 AN3199 AN3199 is a PDE4 inhibitor (IC50: 94.5 nM).
T10319 Anamorelin Anamorelin is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
T10319L Anamorelin Fumarate Anamorelin Fumarate is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
T10320 Androgen receptor antagonist 1 Androgen receptor antagonist 1 is an orally available full androgen receptor antagonist (IC50: 59 nM). It can be used in the synthesis of PROTAC AR degraders, w...
T10322 Angiotensin III Angiotensin III is an agonist of angiotensin 1 (AT1) and AT2 receptor.
T10322L Angiotensin III TFA Angiotensin III TFA is an agonist of angiotensin 1 (AT1) and AT2 receptor.
T10324 Anhydrosimvastatin Anhydrosimvastatin is an impurity of Simvastatin. Simvastatin is an HMG-CoA reductase inhibitor.
T10326 Aniline-MPB-amino-C3-PBD Aniline-MPB-amino-C3-PBD is a cytotoxic agent comprised of the non-alkylating group. It is a sequence-selective DNA minor-groove binding agent.
T10328 Anti-parasitic agent 3 Anti-parasitic agent 3 is an anti-parasitic agent.
T10329 anti-TB agent 1 anti-TB agent 1 is a potent and orally active anti-tuberculosis agent (MICs: < 2 nM against the Mtb strains H37Rv, rRMP and rINH).
T1033 Monensin sodium salt Monensin sodium is an antiprotozoal agent produced by Streptomyces cinnamonensis.Monensin sodium salt causes a marked enlargement of the MVBs and regulates exos...
T10331 Anticancer agent 3 Anticancer agent 3 (Compound 4) is a anti-cancer agent.
T10332 Antidepressant agent 1 Antidepressant agent 1 is a pyrazidole-halogeno-derivative with antidepressant effects. It also can be used to increase body temperature.
T10333 Antifungal agent 1 Antifungal agent 1 is an effective antifungal agent.
T10334 Antifungal agent 2 Antifungal agent 2 is a broad-spectrum fungal inhibitor that inhibits the growth of pertinent species of Cryptococcus, Candida, and Aspergillus at a concentrati...
T10336 Antimalarial agent 1 Antimalarial agent 1 is an effective antimalarial agent.
T10338 Antisauvagine-30 TFA Antisauvagine-30 TFA (aSvg-30 TFA) is a highly selective and competitive antagonist of CRF2 receptor peptidic. It shows a Kd of 1.4 nM and 150 nM for mCRFR2β a...
T1034 DocetaxelHOT Docetaxel is a microtubule inhibitor that inhibits microtubule disassembly (IC50: 0.2 μM).
T10340 Antitrypanosomal agent 2 Antitrypanosomal agent 2 is a potent and selective inhibitor of trypanosoma brucei.
T10341 Antitumor agent-19 Antitumor agent-19 is an antitumor agent targeting tumor-associated macrophages (TAMs) to serve as an effective TAMs modulator (EC50s: 17.18 μM and 18.87 μM i...
T10342 Antitumor agent-2 Antitumor agent-2 has antitumor action and anti-inflammatory action. It is sourced from patent CN102250203 (compound 6a-r).
T10343 AOH1160 AOH1160 is a potent orally available small molecule proliferating cell nuclear antigen (PCNA) inhibitor. It interferes with DNA replication, blocks homologous r...
T10345 Apcin-A Apcin-A is an anaphase-promoting complex (APC) inhibitor. It interacts strongly with Cdc20 and inhibits the ubiquitination of Cdc20 substrates. Apcin-A can be u...
T10346 Apelin agonist 1 Apelin agonist 1 is an oral selective apelin agonist AM-2995, an agonist of the APJ (APLNR, angiotensin receptor like-1) receptor. It may be used in the treatme...
T10348 Apigenin-7-diglucuronide Apigenin-7-diglucuronide is a flavonoid glycoside that exists in an assortment of medicinal plants with anti-inflammatory or ant-oxidant activities. It protects...
T10349 Apixaban 13CD3 Apixaban 13CD3 (BMS-562247-01 13CD3) is a deuterium-labeled Apixaban. Apixaban is a reversible inhibitor of Factor Xa (Ki: 0.08 nM and 0.17 nM in human and rabb...
T1035 Hesperidin Hesperidin is a flavanone glycoside found in citrus fruits with antioxidant, anti-inflammatory, anti-carcinogenic, and antihypertensive and lipid-lowering activ...
T10351 Aprocitentan D4 Aprocitentan D4 (ACT-132577 D4) is a deuterium-labeled Aprocitentan. Aprocitentan is a major and pharmacologically active metabolite of Macitentan. Aprocitentan...
T10355 Apyramide Apyramide is an anti-inflammatory compound.
T10356 AQ-13 dihydrochloride AQ-13 dihydrochloride is an antimalarial drug. It is effective against drug-resistant strains of Plasmodium falciparum.
T10357 AR-13324 analog mesylate AR-13324 analog mesylate is an inhibitor of Rho-kinase and a norepinephrine transporter and reduces intraocular pressure in normotensive monkey eyes.
T10358L AR-13324 M1 metabolite AR-13324 M1 metabolite is a hydrolysis metabolite of AR-13324 mesylate.
T10358L2 Netarsudil mesylate Netarsudil mesylate is an inhibitor of Rho-associated protein kinase (ROCK) and norepinephrine transporter (NET) with effective in intraocular pressure (IOP) re...
T10359 AR antagonist 1 AR antagonist 1 is a potent antagonist of the androgen receptor. It binds to E3 ligase ligands with weak binding affinities to VHL protein in the synthesis of P...
T1036 Netilmicin sulfate Netilmicin Sulfate is an aminoglycoside antibiotic.
T10360 AR-A 2 AR-A 2 is a selective 5-HT1B receptor antagonist, with a high affinity to guinea pig cortex 5HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki: 0.24 and 0...
T10361 AR-C102222 hydrochloride AR-C102222 hydrochloride is a competitive, orally active, and highly selective inducible nitric oxide synthase (iNOS) inhibitor (IC50: 37 nM). It has antinocice...
T10362 AR453588 AR453588 is an orally bioavailable anti-diabetic glucokinase activator (EC50: 42 nM) with anti-hyperglycemic activity.
T10362L AR453588 hydrochloride AR453588 hydrochloride is an orally bioavailable anti-diabetic glucokinase activator (EC50: 42 nM) with anti-hyperglycemic activity.
T10363 Arazine Arazine (N-Acetyl-S-farnesyl-L-cysteine) is a cell-permeable modulator of G protein and GPCR signaling. Arazine can be a substrate for isoprenylcysteine methylt...
T10365 Arg-AMS Arg-AMS is a potent arginyl tRNA synthetase inhibitor that displays tightly bound inhibitory characteristics for the A-domains in non-ribosomal peptide syntheta...
T10366 Arg-Gly-Asp-Ser Arg-Gly-Asp-Ser is an integrin-binding sequence that inhibits integrin receptor function. It decreases systemic inflammation via inhibition of collagen-triggere...
T10367 Arginase inhibitor 1 Arginase inhibitor 1 is a potent inhibitor of human arginases I and II (IC50s: 223 and 509 nM).
T10368 Aripiprazole (D8) Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).
T10369 Aristeromycin Aristeromycin is an adenosine analog and an antibiotic and. It is a potent S-adenosylhomocysteine hydrolase (AHCY) inhibitor.
T1037 Doripenem Hydrate Doripenem Hydrate is a broad-spectrum injectable antibiotic, used for Gram-positive, Gram-negative and anaerobic pathogens.
T10370 ARN 077 ARN 077 is a selective N-acylethanolamine acid amidase (NAAA) inhibitor (IC50: 7 nM for human NAAA). ARN 077 significantly increases palmitoyl ethanolamine (PEA...
T10372 ARQ 069 ARQ 069 (3.8-60 μM; for 2 hours) reduces the degree of phosphorylation of FGFR (predominantly FGFR2) in a concentration-dependent manner, without decreasing β...
T10373 (R)-Filanesib (R)-Filanesib is the R-enantiomer of ARRY-520. (R)-Filanesib is a synthetic kinesin spindle protein (KSP) inhibitor (IC50: 6 nM).
T10377 Artefenomel Artefenomel (OZ439) is a synthetic antimalarial agent with the artemisinin pharmacophore.
T10378 Artelinic acid Artelinic acid, a derivative of Artemisinin, is an antimalarial drug for the treatment of multidrug-resistant strains of Plasmodium falciparum.
T10379 Arzoxifene hydrochloride Arzoxifene hydrochloride is a selective estrogen receptor modulator that is a potent estrogen antagonist in mammary and uterine tissue.
T10381 AS2717638 AS2717638 is an orally active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist (IC50: 38 nM for hLPA5). It also significantly improves PGF2α-, ...
T10386 Asp-AMS Asp-AMS is a strong competitive inhibitor of the mitochondrial enzyme and also an aspartyl-tRNA synthetase inhibitor.
T10387 ASP1126 ASP1126 is a selective and orally active sphingosine-1-phosphate (S1P) agonist (EC50s: 7.12 nM, 517 nM for hS1P1 and hS1P3).
T10388 Asparagusic acid Asparagusic acid is unique to asparagus. It is responsible for the odorous urine excreted after eating asparagus. Its derivatives ihydroasparagusic acid have an...
T10389 Aspartyl-alanyl-diketopiperazine Aspartyl-alanyl-diketopiperazine (DA-DKP) is an immunomodulatory molecule generated by cleavage and cyclization from the N-terminus of human albumin.
T10390 Asperphenamate Asperphenamate is a fungal metabolite of Aspergillus flatiipes with anti-cancer effect (IC50s: 92.3 μM, 96.5 μM, and 97.9 μM in T47D, MDA-MB-231, and HL-60 c...
T10391 Aspirin Aluminum Aspirin Aluminum is an intermolecular compound that can inhibit gastrointestinal mucosal disorders induced by NSAIDs extracted from patent WO 2010064441 A1.
T10392 Aspoxicillin Aspoxicillin is a broad-spectrum antimicrobial agent against 68 isolates of Actinobacillus pleuropneumoniae (MIC90 <= 0.05 μg/ml). Aspoxicillin has a long half...
T10394 ATB107 ATB107 is a potent and novel inhibitor of indole-3-glycerol phosphate synthase (IGPS, KD: 3 μM).
T10395 ATM-3507 trihydrochloride ATM-3507 trihydrochloride is a potent tropomyosin inhibitor (IC50s: 3.83-6.84 μM in human melanoma cell lines).
T10395L ATM-3507 ATM-3507 is an inhibitor of tropomyosin. In human melanoma cell lines, the IC50s are from 3.83-6.84 μM.
T10397 ATN-161 trifluoroacetate salt ATN-161 trifluoroacetate salt is a novel integrin α5β1 antagonist that inhibits angiogenesis and growth of liver metastases in a murine model.
T10398 ATN-161 ATN-161 is a novel integrin α5β1 antagonist that inhibits angiogenesis and growth of liver metastases in a murine model.
T10399 Atorvastatin 3-Deoxyhept-2E-Enoic Acid Atorvastatin 3-Deoxyhept-2E-Enoic Acid is an impurity of Atorvastatin. Atorvastatin is an HMG-CoA reductase inhibitor and has the ability to effectively decreas...
T10400 Atorvastatin acetonide tert-butyl ester Atorvastatin acetonide tert-butyl ester is a useful pharmaceutical intermediate in the preparation of Atorvastatin salts. Atorvastatin is an HMG-CoA reductase i...
T10401 Atorvastatin acetonide Atorvastatin acetonide is an impurity of Atorvastatin and extracted from patent WO2011131605A1 (Compound 4). Atorvastatin is an HMG-CoA reductase inhibitor and ...
T10402 Atorvastatin Epoxy Tetrahydrofuran Impurity Atorvastatin Epoxy Tetrahydrofuran Impurity is an impurity isolated oxidative degradation products of Atorvastatin. Atorvastatin is an orally active HMG-CoA red...
T10403 Atorvastatin ethyl ester Atorvastatin ethyl ester is a derivative of Atorvastatin. It displays strong inhibition of the 9-cis-RA-induced Gal4 reporter activity.
T10404 ATP synthase inhibitor 1 ATP synthase inhibitor 1 is an inhibitor of the c subunit of the F1/FO-ATP synthase complex. It inhibits mitochondrial permeability transition pore (mPTP) openi...
T10405 ATPA ATPA is a selective glutamate receptor GluR5 activator (EC50s: 0.66, 1.4, 9.5, 23, 32, 18, and 14 μM for GluR5wt, GluR5(S721T), GluR5(S741M), GluR5(S721T, S741...
T10406 ATR inhibitor 1 ATR inhibitor 1 is an ATR inhibitor extracted from patent WO2015187451A1 (compound I-l, Ki< 1 µΜ).
T10408 ATWLPPR Peptide TFA ATWLPPR Peptide TFA is a selective neuropilin-1 inhibitor and inhibits VEGF165 binding to NRP-1. It has the potential in reducing the early retinal damage cause...
T1041 Risedronate Sodium Risedronate sodium is an aminobisphosphonate derivative of etidronic acid and CALCIUM CHANNEL BLOCKER that inhibits BONE RESORPTION and is used for the treatmen...
T10410 ATX inhibitor 1 ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, bis-pNPP).
T10411 AU1235 AU1235 is a Mycobacterium tuberculosis inhibitor.
T10413 Autogramin-1 Autogramin-1 potently inhibits autophagy induced by either mTORC1 inhibition (Rapamycin; IC50: 0.44 μM) or starvation (IC50: 0.17 μM).
T10414 Autogramin-2 Autogramin-2 potently inhibits autophagy induced by either mTORC1 inhibition (Rapamycin; IC50: 0.14 μM) or starvation (IC50: 0.27 μM).
T10420 Avarofloxacin Avarofloxacin (JNJ-Q2) is a broad-spectrum fluoroquinolone antibacterial drug being developed for the treatment of acute bacterial skin and community-acquired p...
T10421 AVE5688 AVE5688 is an inhibitor of glycogen phosphorylase (GP, IC50s: 430 nM and 915 nM; Kds: 170 nM and 530 nM for rmGPb and rmGPa). It can be used for the research of...
T10423 AWZ1066S AWZ1066S is a highly specific anti-Wolbachia drug candidate for the short-course treatment of filariasis (EC50: 2.5 nM in cell assay).
T1043 Salifungin Detail unknown.
T10430 AZD 2066 AZD 2066 is a selective, orally active, and brain-penetrant mGluR5 antagonist with analgesic activity.
T10432 AZD-8529 AZD-8529 is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: 285 nM). It shows no positive allosteric modulator respon...
T10432L AZD-8529 mesylate AZD-8529 mesylate is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: 285 nM). It shows no positive allosteric modulat...
T10435 Linaprazan Linaprazan inhibits gastric H+, K+-ATPase by K+-competitive binding (IC50: 1.0 μM). It is an acid-suppressing compound with a rapid onset of action and potent ...
T10439 Azelnidipine D7 Azelnidipine D7 is a deuterium-labeled Azelnidipine. Azelnidipine is an L-type calcium channel blocker.
T1044 Clopidol Clopidol is a very effective anticoccidial agent used in poultry.
T10440 Azilsartan D5 Azilsartan (TAK-536) D5 is the deuterium-labeled Azilsartan. Azilsartan is a specific antagonist of the angiotensin II type 1 receptor.
T10441 Azosemide Azosemide is a potent NKCC1 inhibitor (IC50s: 0.246 µM and 0.197 µM for hNKCC1A and NKCC1B).
T10443 Aβ42-IN-1 free base Aβ42-IN-1 free base is an orally active, high brain exposure γ-secretase modulator. It potently reduces Aβ42 levels (IC50: 0.091 µM), and significantly redu...
T10444 TAK1/MAP4K2 inhibitor 1 TAK1/MAP4K2 inhibitor 1 is a potent dual inhibitor of TGFβ-activated kinase 1 (TAK1) and MAP4K2 (IC50s: 41.1 nM and 18.2 nM).
T10446 BA-53038B BA-53038B is an HBV core protein allosteric modulator (CpAM), binding to the HAP pocket and modulating HBV capsid assembly in a distinct manner (EC50: 3.32 μM)...
T10447 BAA473 BAA473, a bile acid analog, is a potent activator of the pyrin inflammasome. It induces the secretion of IL-18 through activation of the inflammasome in both my...
T10448 Bacampicillin Bacampicillin is an improved oral bioavailability penicillin antibiotic which is a prodrug of ampicillin.
T10448L Bacampicillin hydrochloride Bacampicillin hydrochloride is an improved oral bioavailability penicillin antibiotic which is a prodrug of ampicillin.
T10449 BACE-1 inhibitor 1 BACE-1 inhibitor 1 (Compound 8a) is an effective BACE-1 inhibitor (IC50: 56 nM).
T10455 Bafilomycin B1 Bafilomycin B1, a macrolide antibiotic isolated from Streptomyces sp, acts as an inhibitor of K+-dependent ATPase of E. coli. It also inhibits Gram-positive bac...
T10457 BAN ORL 24 BAN ORL 24 is a potent and selective NOP receptor antagonist (IC50s: 0.27, 2500, 6700 and > 10000 nM for NOP, κ-, μ- and δ-receptors).
T10458 Banoxantrone D12 Banoxantrone D12 (AQ4N D12) is the deuterium-labeled Banoxantrone. Banoxantrone is a bioreductive agent that can be reduced to a stable, DNA-affinity compound A...
T10459 Banoxantrone dihydrochloride Banoxantrone dihydrochloride (AQ4N dihydrochloride) is a bioreductive agent that can be reduced to a stable, DNA-affinity compound AQ4, which is a topoisomerase...
T10460 Batabulin Batabulin is an antitumor compound, which binds covalently and selectively to a subset of the β-tubulin isotypes, thereby disrupting microtubule polymerization...
T10462 Bavisant dihydrochloride Bavisant (JNJ-310010740) dihydrochloride is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, involving wa...
T10462L Bavisant dihydrochloride hydrate Bavisant dihydrochloride hydrate (JNJ31001074AAC) is a highly selective, orally active antagonist of the human H3 receptor with a novel mechanism of action, inv...
T10467 BAY-1816032 BAY-1816032 is a potent and orally available inhibitor of bidding uninhibited by benzimidazoles 1 ( BUB1) kinase (IC50: 7 nM).
T10469 BAY-298 BAY-298 is an orally active and selective luteinizing hormone receptor (LH-R) antagonist (IC50s: 96 nM, 23 nM, and 78 nM for hLH (human LH) and rLH (rat LH) and...
T10471 BAY 60-2770 BAY 60-2770 is a selective and orally active soluble guanylyl cyclase (sGC) activator with antifibrotic effect. It increases the activity of sGC in a nitric oxi...
T10472 Bay 65-1942 R form Bay 65-1942 R form is the less active R-form of Bay 65-1942. Bay 65-1942 is a selective and ATP-competitive IKKβ inhibitor.
T10473 BAY-678 BAY-678 is an orally bioavailable, selective and cell-permeable inhibitor of human neutrophil elastase (HNE; IC50: 20 nM).
T10473L BAY-677 BAY-677 is an inactive control for BAY-678. BAY-678 is an orally bioavailable, highly potent, selective and cell-permeable inhibitor of human neutrophil elastas...
T10474 BAY-7598 BAY-7598 is a potent, selective, and orally bioavailable MMP12 inhibitor (IC50s: 0.085, 0.67, and 1.1 nM for human/murine/rat MMP12).
T10475 BAY-784 BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).
T10476 BAY-899 BAY-899 is an orally active and selective of antagonist luteinizing hormone receptor (LH-R; IC50s: 185 nM and 46nM for human LH and rat LH). It can reduce sex h...
T10478 BAY-Y 3118 BAY-Y 3118, a new chlorofluoroquinolone, has antimicrobial activity.
T10481 BAY 73-6691 racemate BAY 73-6691 racemate is a phosphodiesterase 9 inhibitor sourced from patent WO 2017070293 A1.
T10482 BB-Cl-Amidine BB-Cl-Amidine is an inhibitor peptidyl arginine deminase (PAD).
T10482L BB-Cl-Amidine hydrochloride BB-Cl-Amidine hydrochloride is an inhibitor peptidyl arginine deminase (PAD).
T10484 BCL2-IN-1 BCL2-IN-1 is a potent Bcl-2 inhibitor (Ki <0.01 nM).
T10486 BCI BCI is an allosteric inhibitor of dual-specificity phosphatase (DUSP; EC50s: 13.3 and 8.0 μM for DUSP6 and DUSP1 in cells) and does not inhibit DUSP5.
T10486L BCI hydrochloride BCI hydrochloride specifically inhibits DUSP6 and DUSP1 with EC50s of 13.3 and 8.0 μM in cells, respectively. BCI hydrochloride does not inhibit DUSP5. BCI h...
T10487 BCL6-IN-3 BCL6-IN-3 is a BCL6 inhibitor with anti-tumor activity, extracted from patent WO2018215801A1 (example 20a). It exhibits a GI50 of 70 nM in SU-DHL4 cells.
T10489 BCR-ABL-IN-2 BCR-ABL-IN-2 is a BCR-ABL1 tyrosine kinase inhibitor (IC50s: 57 nM, 773 nM for ABL1 native and ABL1 T315I).
T10490 (S)-ML753286 (S)-ML753286 is a breast cancer resistance protein (BCRP) inhibitor (IC50: 0.6 μM on BCRP efflux transporter).
T10491 Galidesivir Galidesivir is an inhibitor of viral RNA-dependent RNA polymerase (RdRp). It inhibits SARS-CoV-2 by tightly binding to its RdRp.
T10491L Galidesivir hydrochloride Galidesivir hydrochloride is an inhibitor of viral RNA-dependent RNA polymerase (RdRp). It inhibits SARS-CoV-2 by tightly binding to its RdRp.
T10492 BD-AcAc 2 BD-AcAc 2 (Ketone Ester), added in diet, could elevate mean blood ketone bodies of 3.5 mm and lowered plasma glucose, insulin, and leptin in animals.
T10493 Beclabuvir Beclabuvir is an allosteric inhibitor that binds to thumb site 1 of the HCV NS5B RNA-dependent RNA polymerase. It inhibits recombinant NS5B proteins from HCV ge...
T10494 Beclomethasone 17-propionate Beclomethasone 17-propionate is an active metabolite of Beclomethasone dipropionate and an agonist of the glucocorticoid receptor (GR). It exhibits greater affi...
T10495L Befiradol Befiradol (NLX-112) is an agonist of 5-HT1A receptor.
T10496 Bencianol Bencianol is a semisynthetic flavonoid with anti-spasmogenic activities.
T10499 H3 receptor-MO-1 H3 receptor-MO-1 is a histamine H3 receptor modulator.
T10501 YM158 free base YM158 free base is a potent and selective antagonist of TXA2 and LTD4 receptor (pA2s: about 8.81 and 8.87).
T10502 Benzcyclane Benzcyclane (Bencyclane) is an inhibitor of platelet aggregation and a vasodilator effective in a variety of peripheral circulation disorders.
T10504 Implitapide Racemate Implitapide Racemate is the racemate of Implitapide. Implitapide is an inhibitor of microsomal triglyceride transfer protein (MTP).
T10508 Asthma relating compound 1 Asthma relating compound 1 is an anti-asthmatic compound extracted from patent EP0295656A1.
T10509 Xanthine oxidase-IN-1 Xanthine oxidase-IN-1 is an inhibitor of xanthine oxidase (IC50: 6.5 nM) extracted from patent WO2008126898A1 (example 3).
T10511 Anti-hypertensive sulfonanilide 1 Anti-hypertensive sulfonanilide 1 is an antihypertensive compound extracted from patent EP0338793A2 (compound XVIIIa,b*).
T10512 Prenyl-IN-1 Prenyl-IN-1 is an inhibitor of protein prenylation, especially a farnesyltransferase (FT) or a geranylgeranyltransferase (GGT) inhibitor. It shows potent activi...
T10513 Benzothiohydrazide Benzothiohydrazide is an analog of Isoniazid. Benzothiohydrazide exhibits antitubercular activity (MICs: 132 μM and 264 μM for M. tuberculosis wild type (H37R...
T10514 FR252384 FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).
T10515 Anti-Heart Failure Agent 1 Anti-Heart Failure Agent 1 is an orally available compound suitable for the treatment of heart failure without inducing vomiting, nausea, and restlessness.
T10516 Beperidium iodide Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).
T10517 BET-BAY 002 (S enantiomer) BET-BAY 002 S enantiomer is an enantiomer of BET-BAY 002 which is a BET inhibitor.
T10518 BET-BAY 002 BET-BAY 002 is an effective BET inhibitor and exhibits efficacy in a multiple myeloma model.
T10519 BET-IN-1 BET-IN-1 is a bromodomain inhibitor extracted from patent WO/2013024104A1 (example 2, plC50: 6.0 - 7.0).
T10523 β3-AR agonist 1 β3-AR agonist 1 is a highly selective, and orally available agonist of β3-adrenergic receptor (EC50: 18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β...
T10524 β-Cryptoxanthin β-Cryptoxanthin is isolated from Satsuma mandarin orange with an anti-stress effect. It is an oxygenated carotenoid and an antioxidant.
T10526 β-NF-JQ1 β-NF-JQ1 is a PROTAC that recruits AhR E3 ligase to target proteins. β-NF-JQ1 is directed against BRD proteins using β-NF as an AhR ligand, induces the inter...
T10527 Betrixaban D6 Betrixaban D6 is a deuterium-labeled Betrixaban. Betrixaban is a selective and orally efficacious FXa inhibitor.
T10528 Bexarotene D4 Bexarotene D4 is a deuterium-labeled Bexarotene (LGD1069). Bexarotene is a selective RXR agonist used in the treatment of cutaneous T-cell lymphoma.
T10529 BF-168 BF-168 is a candidate probe for PET and specifically recognizes both neuritic and diffuse plaques (Ki: 6.4 nM for Aβ1-42).
T1053 Mebeverine hydrochloride Mebeverine hydrochloride, a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gut.
T10530 BF 227 BF 227 is a candidate for an amyloid imaging probe for PET (Ki: 4.3 nM for Aβ1-42 fibrils).
T10532 BI-1408 BI-1408 is a modulator potent of γ secretase (IC50: 0.04 μM for Aβ42).
T10536 BI 703704 BI 703704 is a potent activator of soluble guanylate cyclase (sGC). It inhibits the progression of diabetic nephropathy in the ZSF1 rat.
T10537 BI-749327 BI-749327 is a high selectivity and orally bioavailable antagonist of TRPC6 (IC50s: 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6).
T10538 BI-9321 BI-9321 is a selective and cellular active nuclear receptor-binding SET domain 3 (NSD3)-PWWP1 domain antagonist (Kd: 166 nM). BI-9321 is inactive against NSD2-P...
T10538L BI-9321 trihydrochloride BI-9321 trihydrochloride is a selective and cellular active nuclear receptor-binding SET domain 3 (NSD3)-PWWP1 domain antagonist (Kd: 166 nM). BI-9321 is inacti...
T10539 BIBO3304 TFA BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 recep...
T10540 BIBP3226 TFA BIBP3226 TFA is an effective and selective antagonist of neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor (Kis: 1.1, 79, and 108 nM for rNPY Y1, h...
T10541 Bicyclomycin benzoate Bicyclomycin benzoate, an antibiotic, exhibits activity against a broad spectrum of Gram-negative/Gram-positive bacteria.
T10542 Bifeprunox Bifeprunox is a potent partial agonist of dopamine D2-like and 5-HT1A receptor (pEC50: 6.37 for hippocampus 5-HT1A; pKis: 7.19 and 8.83 for cortex 5-HT1A and st...
T10543 BIIL-260 hydrochloride BIIL-260 hydrochloride is a potent and long-acting orally active antagonist of leukotriene B4 (LTB4) receptor with anti-inflammatory activity. It has a high aff...
T10544 Bimatoprost D5 Bimatoprost (AGN 192024) D5 is a deuterium-labeled Bimatoprost. Bimatoprost is a topical hypotensive agent frequently used for treating glaucoma and ocular hype...
T10545 BIO-32546 BIO-32546 is a modulator of autotaxin (ATX) extracted from the patent US20170158687A1 (example 12b, S-isomer).
T10547 BioE-1115 BioE-1115 is a highly selective PAS kinase (PASK) inhibitor (IC50: ~4 nM). It is also a potent inhibitor of casein kinase 2α (IC50: ~10 μM).
T10551 Bithionol sulfoxide Bithionol sulfoxide is a clinically approved antiparasitic drug with the inhibitory against solid tumor growth in several preclinical cancer models.
T10553 BIX-01338 hydrate BIX-01338 hydrate is an inhibitor of histone lysine methyltransferase.
T10554 Bixin Bixin is isolated from the seeds of Bixa orellana and possesses anti-tumor, anti-inflammatory, and antioxidant activities. Bixin treatment ameliorated cardiac d...
T10557 BLM-IN-1 BLM-IN-1 is an effective Bloom syndrome protein (BLM) inhibitor (KD: 1.81 μM; IC50: 0.95 μM). It induces DNA damage response, apoptosis and proliferation arre...
T10558 Blonanserin D5 Blonanserin D5 is a deuterium-labeled Blonanserin. Blonanserin (AD-5423) is a dopamine D2/5-HT2 receptor antagonist with an atypical antipsychotic effect.
T10559 Blonanserin D8 Blonanserin D8 is a deuterium-labeled Blonanserin. Blonanserin (AD-5423) is a dopamine D2/5-HT2 receptor antagonist with an atypical antipsychotic effect.
T10561 BM-131246 BM-131246 is an oral antidiabetic compound.
T10562 (4-Acetamidocyclohexyl) nitrate (4-Acetamidocyclohexyl) nitrate (BM121307) is an activator of guanylate cyclase.
T10563 BM635 BM635 is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).
T10563L BM635 hydrochloride BM635 hydrochloride is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).
T10563L2 BM635 mesylate BM635 mesylate is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).
T10564 (8R,9S)-Talazoparib (8R,9S)-Talazoparib is Talazoparib enantiomer , less active than Talazoparib on the inhibition of PARP1 (IC50: 144 nM).
T10565 BMS-1001 hydrochloride BMS-1001 hydrochloride is an orally active inhibitor of human PD-L1/PD-1 immune checkpoint with low-toxicity in cells.
T10566 BMS-191095 BMS-191095 is mitochondrial ATP-sensitive potassium (mitoKATP) channel activator.
T10568 BMS-470539 dihydrochloride BMS-470539 dihydrochloride is a highly potent and selective agonist of the melanocortin-1 receptor (MC-1R; IC50: 120 nM; EC50: 28 nM) with anti-inflammatory pro...
T10569 BMS-654457 BMS-654457 is a small-molecule, reversible inhibitor of factor XIa (FXIa; Kis: 0.2 and 0.42 nM for human and rabbit FXIa).
T10571 BMS-901715 BMS-901715 is an effective and selective inhibitor of adapter protein-2 associated kinase 1 (AAK1; IC50: 3.3 nM).
T10572 BMT-124110 BMT-124110 is an effectivet, selective AAK1 inhibitor (IC50: 0.9 nM) with antinociceptive activity. BMT-090605 inhibits BMP-2-inducible protein kinase (BIKE; IC...
T10576 BMY-43748 BMY-43748 is an antibacterial compound with great in vitro and in vivo antibacterial activity.
T10579 BO3482 BO3482 is an antimicrobial compound and can inhibit the growth of methicillin-resistant Staphylococci (MIC90: 6.25 mg/mL).
T10581 Boc-MLF TFA Boc-MLF (TFA) is a specific antagonist of formyl peptide receptor (FPR) and also inhibits signaling through FPRL1 at higher concentrations.
T10582 Borrelidin Borrelidin (Treponemycin) is a bacterial and eukaryal threonyl-tRNA synthetase inhibitor. It is a macrolide antibiotic isolated from Streptomyces rochei.
T10584 Bovinic acid Bovinic acid is a conjugated linoleic acid with anti-atherogenic and anticarcinogenic activities.
T10585 Bozitinib Bozitinib (PLB-1001) is a highly selective inhibitor of the c-MET kinase with blood-brain barrier permeability. Bozitinib binds to the conventional ATP-binding ...
T10586 BPH-1358 free base BPH-1358 (NSC50460) free base is a potent human undecaprenyl diphosphate synthase (UPPS) and farnesyl diphosphate synthase (FPPS) inhibitor (IC50s: 110 nM and 1...
T10586L BPH-1358 BPH-1358 (NSC50460) is a potent human farnesyl diphosphate synthase (FPPS) and undecaprenyl diphosphate synthase (UPPS) inhibitor. With IC50s of 1.8 μM and 110...
T10587 BPH-652 BPH-652 is an S. aureus dehydrosqualene synthase (CrtM) inhibitor (Ki: 1.5 nM; IC50: 100-300 nM for S. aureus pigment formation).
T10588 BPI-9016M BPI-9016M is an effective, orally active, and selective dual inhibitor of c-Met and AXL tyrosine kinases. It suppresses tumor cell growth, invasion, and migrati...
T10589 BPN-15606 besylate BPN-15606 besylate is a highly potent, orally active γ-secretase modulator, attenuates the production of Aβ40 and Aβ42 by SHSY5Y neuroblastoma cells (IC50s: ...
T10589L BPN-15606 BPN-15606 is a highly potent, orally active γ-secretase modulator (GSM), attenuates the production of Aβ42 and Aβ40 by SHSY5Y neuroblastoma cells with IC50 v...
T1059 Retinol palmitate Vitamin A Palmitate is a naturally-occurring phenyl analogue of retinol, with potential antineoplastic and chemopreventive activities.
T10590 BPN14770 BPN14770 is an allosteric inhibitor of selective phosphodiesterase 4D (PDE4D; IC50s: 7.8 nM and 7.4 nM for PDE4D7 and PDE4D3).
T10591 BPO-27 (racemate) BPO-27 racemate is an effective inhibitor of CFTR (IC50: 8 nM).
T10591L (R)-BPO-27 (R)-BPO-27 is an effective inhibitor of the CFTR (IC50: 4 nM).
T10593 BPR1M97 BPR1M97 is a dual-acting mu-opioid receptor (MOP) and nociceptin-orphanin FQ peptide (NOP) receptor agonist (Kis: 1.8 and 4.2 nM) with blood-brain barrier penet...
T10595 BQ-788 BQ-788 is a potent, selective antagonist of ETB receptor (IC50: 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells), poorly inhibiting the bindi...
T10595L BQ-788 sodium salt BQ-788 sodium salt is a potent and selective antagonist of ETB receptor(ETB receptors with an IC50 of 1.2 nM in human Girrardi heart cells).
T10596 BR102375 BR102375 is a non-TZD PPAR γ full agonist (EC50: 0.28 μM) for the treatment of type 2 diabetes.
T10598 BR351 precursor BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).
T10600 BRCA1-IN-1 BRCA1-IN-1 is a novel small-molecule-like inhibitor of BRCA1 (IC50: 0.53 μM; Ki: 0.71 μM).
T10601 BRCA1-IN-2 BRCA1-IN-2 is a cell-permeable protein-protein interaction (PPI) inhibitor for BRCA1 (IC50: 0.31 μM; Kd: 0.3 μM). It has antitumor activities via the disrupti...
T10604 BRD-IN-3 BRD-IN-3 is a highly potent PCAF bromodomain (BRD) inhibitor (IC50: 7 nM). It also exhibits activity against GCN5 and FALZ.
T10605 BRD-K98645985 BRD-K98645985 is a BAF transcriptional repression inhibitor (EC50: ~2.37 µM). It binds ARID1A-specific BAF complexes, potently reverses HIV-1 latency and preve...
T10606 BRD0705 BRD0705 is a potent, paralog selective and orally active GSK3α inhibitor (IC50: 66 nM; Kd: 4.8 μM). BRD0705 displays increased selectivity for GSK3α (8-fold)...
T10608 BRD5648 BRD5648 ((R)-BRD0705) is an inactive (R)-enantiomer of BRD0705. BRD0705 is a GSK3α inhibitor (IC50: 66 nM; Kd: 4.8 μM).
T10609 Brevetoxin-3 Brevetoxin-3 (PbTx-3) is a potent allosteric voltage-gated Na+ channel activator. Brevetoxin-3 has a high affinity to site 5 of the voltage-sensitive Na+ channe...
T1061 Toltrazuril Toltrazuril, an antiprotozoal agent, has effect on Coccidia parasites.
T10610 Brexpiprazole D8 Brexpiprazole D8 (OPC-34712 D8) is a deuterium-labeled Brexpiprazole. Brexpiprazole is a partial agonist of human 5-HT1A and dopamine receptors (Ki: 0.12 nM and...
T10613 BRL 37344 sodium BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.
T10614 BRL-42715 BRL-42715 is an effective inhibitor of bacterial beta-lactamases.
T10616 BRM/BRG1 ATP Inhibitor-1 BRM/BRG1 ATP Inhibitor-1 is an allosteric dual Brahma homolog (BRM)/SWI/SNF related matrix-associated actin-dependent regulator of chromatin subfamily A member ...
T10618 Broflanilide Broflanilide is metabolized to desmethyl-broflanilide, which is a potent antagonist at the insect resistant-to-dieldrin GABA receptor and inhibits S. litura RDL...
T10619 Bromelain Bromelain is an anti-inflammatory drug derived from pineapple stem. It acts through down-regulation of plasma kininogen, degradation of advanced glycation end-p...
T10620 Bromodomain IN-1 Bromodomain IN-1 is an inhibitor of Bromodomain extracted from patent WO2016069578A1 (compound 4).
T10621 Bromodomain inhibitor-8 Bromodomain inhibitor-8 is an inhibitor of BET bromodomain used to treat autoimmune and inflammatory diseases.
T10622 BSc5371 BSc5371 is a potent and irreversible FLT3 inhibitor (Kds: 1.3, 0.83, 1.5, 5.8, and 2.3 nM for mutant FLT3 D835H, FLT3 ITD/D835V, FLT3 ITD/F691L, FLT3-ITD, and w...
T10623 BSH-IN-1 BSH-IN-1 is a potent and covalent inhibitor of gut bacterial recombinant bile salt hydrolases (BSHs; IC50s: 108 nM and 427 nM for B. longum BSH and B. theta BSH...
T10624 BT-13 BT-13 is a selective agonist of glial cell line-derived neurotrophic factor (GDNF) receptor RET independently of GFLs. BT-13 promotes neurite growth from sensor...
T10625 IBT6A IBT6A is an impurity of Ibrutinib. Ibrutinib is a Btk inhibitor (IC50: 0.5 nM). IBT6A can be used in the synthesis of IBT6A Ibrutinib dimer and IBT6A adduct.
T10625L (Rac)-IBT6A hydrochloride (Rac)-IBT6A hydrochloride is a racemate of IBT6A. IBT6A is an impurity of Ibrutinib. IBT6A can be used in the synthesis of IBT6A Ibrutinib dimer and IBT6A adduc...
T10625L2 IBT6A hydrochloride IBT6A hydrochloride is an impurity of Ibrutinib. Ibrutinib is a Btk inhibitor (IC50: 0.5 nM). IBT6A can be used in the synthesis of IBT6A Ibrutinib dimer and IB...
T10626 (Rac)-IBT6A (Rac)-IBT6A is a racemate of IBT6A. IBT6A is an impurity of Ibrutinib. IBT6A can be used in the synthesis of IBT6A Ibrutinib dimer and IBT6A adduct. Ibrutinib i...
T10627 BTK inhibitor 10 BTK inhibitor 10 is a potent and orally active BTK inhibitor extracted from patent WO2018145525 (example 33). It has the potential for rheumatoid arthritis trea...
T10628 BTK inhibitor 13 BTK inhibitor 13 (compound 8) is an effective and selective BTK inhibitor(IC50: 1.2 nM).
T1063 Ticarcillin disodium Ticarcillin Disodium is the disodium salt form of ticarcillin, a broad-spectrum, semi-synthetic penicillin antibiotic with bactericidal and beta-lactamase resis...
T10630 BuChE-IN-TM-10 BuChE-IN-TM-10 (TM-10) is a potent inhibitor of butyrylcholinesterase (BuChE; IC50: 8.9 nM) with the potential to treat Alzheimer’s disease.
T10631 Bucindolol Bucindolol is a blocker of the β1-adrenergic receptor and has intrinsic sympathomimetic activity used in the research of heart failure.
T10632 Bucolome Bucolome is a CYP2C9 inhibitor used as an anti-inflammatory agent or uricosuric agent.
T10633 Bumetanide D5 Bumetanide D5 is a deuterium-labeled Bumetanide. Bumetanide is a Na+-K+-Cl- (NKCC1) inhibitor (IC50s: 0.68 and 4.0 μM for hNKCC1A and hNKCC2A).
T10634 Bunaftide Bunaftide (Bunaftine) is an antiarrhythmic compound.
T10636 5α-reductase-IN-1 5α-reductase-IN-1 is an inhibitor of 5α-reductase, used for the research of patterned alopecia in combination with minoxidil.
T10637 Butin Butin, a major biologically active flavonoid isolated from the Dalbergia odorifera, has strong antioxidant, anti-inflammatory and antiplatelet activities.
T10638 BY27 BY27 is a potent and selective BET BD2 inhibitor (Ki: 3.1 nM) with anti-cancer activity and shows 38, 5, 7, and 21-fold BD1/BD2 selectivity for BRD2, BRD3, BRD4...
T10639 C-021 dihydrochloride C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse (IC50s: 140 nM and 39 nM).
T10640 C-11 C-11 is a tubulin inhibitor and acts as an ADC cytotoxin with cytotoxicity for carcinoma cell lines.
T10642 c-di-AMP c-di-AMP (Cyclic diadenylate) is a STING agonist. It binds to the transmembrane protein STING thereby activating the TBK3-IRF3 signaling pathway.
T10643 c-Fms-IN-1 c-Fms-IN-1 is an inhibitor of FMS kinase (IC50: 0.0008 μM).
T10644 c-Fms-IN-10 c-Fms-IN-10 is the derivative of thieno [3,2-d] pyrimidine, a kinase inhibitor of FMS (Colony-stimulating factor-1 receptor, CSF-1R; IC50: 2 nM) with anti-tumor...
T10646 c-Fms-IN-7 c-Fms-IN-7 is a cFMS inhibitor (IC50: 18.5 nM) extracted from patent WO2011079076A1 (example159).
T10649 c-Fms-IN-3 c-Fms-IN-3 is a novel inhibitor of the c-Fms kinase with potential as an antirheumatic agent and anti-inflammatory agent.
T10651 c-Kit-IN-3 c-Kit-IN-3 is a potent and selective c-KIT kinase inhibitor (IC50s: 4 nM, 8 nM for c-KIT wt, and c-KIT T670I).
T10652 DCC-3014 DCC-3014 is a c-FMS (CSF-IR) and c-Kit dual inhibitor (IC50s: <0.01 μM and 0.1-1 μM) extracted from the patent WO2014145025A2 (Example 10).
T10655 c-Met inhibitor 1 c-Met inhibitor 1 is a c-Met receptor signaling pathway inhibitor, used for the treatment of cancer including glioblastoma, gastric, and pancreatic cancer.
T10656 trans-C75 trans-C75 is an enantiomer of C75. C75 is an inhibitor of fatty acid synthase (FASN).
T10657 C75 C75 is an inhibitor synthetic fatty-acid synthase (FASN) and inhibits prostate cancer cells PC3 (IC50: 35 μM).
T10659 Ca2+ channel agonist 1 Ca2+ channel agonist 1 is an agonist of N-type Ca2+ channel and an inhibitor of Cdk2 (EC50s: 14.23 μM and 3.34 μM) and is used as a potential treatment for mo...
T10661 Calcifediol-D6 Calcifediol-D6 is the deuterated form of Calcifediol, which is a prehormone that is produced in the liver by hydroxylation of vitamin D3 by the enzyme cholecalc...
T10662 Calcimycin hemicalcium salt Calcimycin (A-23187) hemicalcium salt is an antibiotic and a unique divalent cation ionophore (like calcium and magnesium). It induces Ca2+-dependent cell death...
T10662L Calcimycin Calcimycin (A-23187) is an antibiotic and a unique divalent cation ionophore and induces Ca2+-dependent cell death by increasing intracellular calcium concentra...
T10663 Calcitriol D6 Calcitriol D6 is the deuterated form of Calcitriol, which is the hormonally active form of vitamin D. Calcitriol is the active metabolite of vitamin D3 that act...
T10664 Calcium 2-oxoglutarate Calcium 2-oxoglutarate is an intermediate in the production of GTP or ATP in the Krebs cycle. It is a reversible inhibitor of tyrosinase (IC50: 15 mM).
T10665 Calcium-Sensing Receptor Antagonists I Calcium-Sensing Receptor Antagonists I is an antagonist of calcium-sensing parathyroid hormone receptors.
T10667 Calmidazolium chloride Calmidazolium chloride (R 24571) is a calmodulin (CaMK) antagonist (Kd: 3 nM), antagonizing CaM-dependent phosphodiesterase and calmodulin-induced activation of...
T10668 Camalexin Camalexin is a phytoalexin isolated from Camelina sativa. It has antifungal, antibacterial, antiproliferative, and anticancer activities. Camalexin can induce R...
T10669 Canagliflozin D4 Canagliflozin D4 is a deuterium-labeled Canagliflozin. Canagliflozin is an SGLT2 inhibitor.
T1067 Amphotericin B Amphotericin B is an antifungal agent with a broad spectrum of activity against many fungal species.
T10670 Candesartan D4 Candesartan D4 is the deuterium labeled Candesartan. Candesartan is an antagonist of angiotensin II receptor.
T10671 Candoxatril Candoxatril is an inhibitor neutral endopeptidase (NEP).
T10672 Capzimin Capzimin is an effective and moderately specific inhibitor of proteasome isopeptidase Rpn11.
T10673 Carbacyclin Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.
T10674 Potassium Channel Activator 1 Potassium Channel Activator 1 is a compound for treating one or more disorders or conditions wherein the dopaminergic system is disrupted.
T10676 Carbodenafil Carbodenafil is a Sildenafil related compound found in healthy foods. Sildenafil is a PDE5 inhibitor (IC50: 5.22 nM).
T10677 Carbodine Carbodine (Carbocyclic cytidine) is a broad-spectrum antiviral agent and targets CTP synthetase that converts UTP to CTP. It possesses significant antiviral act...
T10678 Carboxypeptidase G2 (CPG2) Inhibitor Carboxypeptidase G2 (CPG2) Inhibitor is a new CPG2 Inhibitor with antitumor activity.
T10679 Carcainium chloride Carcainium chloride (QX 572) is a derivative of Lidocaine with antitussive effect.
T1068 Anthralin Anthralin is an anthracene derivative that disrupts MITOCHONDRIA function and structure and is used for the treatment of DERMATOSES, especially PSORIASIS. It ma...
T10682 CARM1-IN-1 hydrochloride CARM1-IN-1 shows high and selective CARM1 inhibition, with lower or no activity against a panel of different PRMTs or HKMTs. In human LNCaP cells, CARM1-IN-1 do...
T10682L CARM1-IN-1 CARM1-IN-1 is a potent and specific inhibitor of Coactivator-associated arginine methyltransferase 1(CARM1; IC50: 8.6 μM). It shows very low activity against P...
T10684 Carnostatine Carnostatine (SAN9812) is a potent and selective carnosinase 1 (CN1) inhibitor (Ki: 11 nM for recombinant hCN1) and can be used for the treatment of diabetic ne...
T10684L Carnostatine hydrochloride Carnostatine (SAN9812) hydrochloride is a potent and selective carnosinase 1 (CN1) inhibitor (Ki: 11 nM for recombinant hCN1) and can be used for the treatment ...
T10685 Carpaine Carpaine, an alkaloid isolated from Carica papaya Linn, has anti-thrombocytopenic activity. It has the anti-plasmodial activity to prevent malaria.
T10685L Carpaine hydrochloride Carpaine hydrochloride, an alkaloid isolated from Carica papaya Linn, has anti-thrombocytopenic activity. It has the anti-plasmodial activity to prevent malaria...
T10686 Carvedilol metabolite 4-Hydroxyphenyl Carvedilol 4-Hydroxyphenyl Carvedilol is a metabolite of Carvedilol. Carvedilol is a beta-blocker/alpha-1 blocker.
T10687 Casein Kinase II Inhibitor IV Casein Kinase II Inhibitor IV is an inducer of epidermal keratinocyte differentiation.
T10687L Casein Kinase II Inhibitor IV Hydrochloride Casein Kinase II Inhibitor IV Hydrochloride is an inducer of epidermal keratinocyte differentiation.
T10689 Cauloside D Cauloside D, a triterpene glycoside isolated from Caulophyllum robustum Max, inhibits the expression of iNOS and proinflammatory cytokines with anti-inflammato...
T10690 Cav 2.2 blocker 1 Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.
T10692 CB-1158 dihydrochloride CB-1158 dihydrochloride is an effective and orally active inhibitor of arginase (IC50s: 86 nM and 296 nM for recombinant human arginase 1 and 2).
T10692L CB-1158 CB-1158 is a potent and orally bioavailable inhibitor of arginase (IC50s: 86 and 296 nM for recombinant human arginase 1 and 2).
T10693 CB-6644 CB-6644 is a selective inhibitor of the RUVBL1/2 complex and blocks the ATPase activity of RUVBL1/2 (IC50: 15 nM).
T10695 CB1151 CB1151 is a 20-epi analogue of 1,25 dihydroxyvitamin D3 with anti-tumor effects. It inhibits MCF-7 cell growth (IC50: 0.82 nM).
T10696 CB2 modulator 1 CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.
T10697 CB2R-IN-1 CB2R-IN-1 is a potent inverse agonist of the cannabinoid CB2 receptor (Ki: 0.9 nM).
T10698 CBB1003 CBB1003 is a new inhibitor of histone demethylase LSD1 (IC50: 10.54 μM).
T10698L CBB1003 hydrochloride CBB1003 hydrochloride is a new inhibitor of histone demethylase LSD1 (IC50: 10.54 μM).
T10699 CBB1007 hydrochloride CBB1007 Hcl is a selective, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1).
T10699L CBB1007 CBB1007 is a potent, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1).
T10699L2 CBB1007 trihydrochloride CBB1007 trihydrochloride is a selective, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1).
T1070 Cefmetazole sodium Cefmetazole sodium is a semisynthetic cephamycin antibiotic with a broad spectrum of activity against both gram-positive and gram-negative microorganisms. It ha...
T10700 (+)-CBI-CDPI1 (+)-CBI-CDPI1 is an enhanced functional analog of CC-1065. It is a DNA alkylating agent and an antibody-drug conjugates (ADCs) toxin.
T10701 (+)-CBI-CDPI2 (+)-CBI-CDPI2 is an enhanced functional analog of CC-1065.
T10704 CCB02 CCB02 is a selective CPAP-tubulin interaction inhibitor (IC50: 689 nM) with anti-tumor activity. CCB02 shows no inhibition on the cell cycle- and centrosome-rel...
T10706 CCI-006 CCI-006 is a selective inhibitor and chemosensitizer of MLL-rearranged leukemia cells. It inhibits mitochondrial respiration resulting in insurmountable mitocho...
T10707 CCK-B Receptor Antagonist 2 CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).
T10715 CCR6 inhibitor 1 CCR6 inhibitor 1 is a potent and selective CCR6 inhibitor (IC50s: 0.45 and 6 nM for monkey and human CCR6), much more selective at CCR6 over human CCR1 (IC50, >...
T10716 CCR7 Ligand 1 CCR7 Ligand 1 (CCR7-Cmp2105) is an allosteric Ligand and antagonist for human CC chemokine receptor 7 (CCR7) with a Kd of 3 nM. CCR7 Ligand 1, thiadiazole-dioxi...
T10720 CD235 CD235 is a structurally similar analog of CD161. CD161 is an orally bioavailable inhibitor of BET bromodomain.
T10721 CD73-IN-1 CD73-IN-1 is an inhibitor of CD73 with anticancer activity extracted from patent WO 2017153952 A1 (example 80).
T10722 CD80-IN-3 CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).
T10723 CDC25B-IN-1 CDC25B-IN-1 is a potent inhibitor of cell division cycle 25B (CDC25B) phosphatase (Ki: 8.5 μM). It potently inhibits cell proliferation and colony formation.
T10725 Cdc7-IN-3 Cdc7-IN-3 is a potent inhibitor of Cdc7 kinase extracted from patent WO2019165473A1 (compound I-A).
T10726 Cdc7-IN-4 Cdc7-IN-4 is a potent inhibitor of Cdc7 kinase extracted from patent WO2019165473A1 (compound I-C).
T10727 Cdc7-IN-5 Cdc7-IN-5 is a potent inhibitor of Cdc7 kinase extracted from patent WO2019165473A1 (compound I-B).
T10728 Cdc7-IN-6 Cdc7-IN-6 is a potent Cdc7 kinase inhibitor (IC50=4 nM) extracted from patent WO2019165473A1(compound I- D) with anti-tumor activity.
T10729 Cdc7-IN-7 Cdc7-IN-7 is a potent inhibitor of Cdc7 kinase extracted from patent WO2019165473A1 (compound I-E).
T10732 Tematropium Tematropium (CDDD3602) is an anticholinergic.
T10734 CDK ligand for PROTAC CDK ligand for PROTAC is a CDK inhibitor with antitumor activity. It has been used to design PROTAC CDK4/6 degraders.
T10734L CDK ligand for PROTAC hydrochloride CDK ligand for PROTAC hydrochloride is a CDK inhibitor with antitumor activity. It has been used to design PROTAC CDK4/6 degraders.
T10748 CE(20:5(5Z,8Z,11Z,14Z,17Z) CE(20:5(5Z,8Z,11Z,14Z,17Z) is an endogenous metabolite.
T10749 Cebranopadol ((1α,4α)stereoisomer) Cebranopadol ((1α,4α)stereoisomer) is a stereoisomer of cebranopadol which is a potent ORL-1 agonist.
T1075 Vitamin K1 Vitamin K1 a fat-soluble, naturally occurring vitamin with antihemorrhagic and prothrombogenic activity.
T10750 Cecropin A TFA Cecropin A TFA is an antimicrobial polypeptide isolated from Hyalaphora cecropia pupae with anti-inflammatory, anti-bacterial, and anti-cancer activity.
T10752 Ceftezole Ceftezole is an alpha-glucosidase inhibitor with in vivo anti-diabetic activity. It is a broad-spectrum cephem antibiotic against many species of gram-positive ...
T10753 Ceftibuten Ceftibuten is a third-generation cephalosporin antibiotic.
T10754 Ceftriaxone sodium salt Ceftriaxone sodium salt is an antibiotic useful for the treatment of a number of bacterial infections.
T10755 Celgosivir hydrochloride Celgosivir hydrochloride (MBI 3253 hydrochloride) is an α-glucosidase I inhibitor and inhibits bovine viral diarrhoea virus (BVDV) (IC50: 1.27 μM).
T10755L Celgosivir Celgosivir (MBI 3253; MDL 28574) is an inhibitor of α-glucosidase I. In vitro assay, it inhibits bovine viral diarrhoea virus (BVDV) ( IC50: 1.27 μM).
T10757 Cenobamate S-Entiomer Cenobamate S-Enantiomer is a Cenobamate's S-enantiomer.
T10758 Centafadine Centanafadine is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 83 nM for human...
T10758L Centafadine hydrochloride Centanafadine hydrochloride is a dual inhibitor of norepinephrine (NE)/dopamine (DA) transporter, also inhibits serotonin transporter (IC50s: 6 nM, 38 nM, and 8...
T10759 CEP-28122 mesylate salt CEP-28122 mesylate salt is a highly selective orally active ALK inhibitor (IC50: 1.9 nM in an enzyme-based TRF assay).
T10760 Ceramides Mixture Ceramides Mixture, an endogenous ceramide, consists of hydroxy and non-hydroxy fatty acid-containing ceramides. It is involved in the regulation of cell cycle a...
T10761 Ceranib-2 Ceranib-2 is a potent and nonlipid ceramidase inhibitor that inhibits cellular ceramidase activity (IC50: 28 μM in SKOV3 cells). It induces the accumulation of...
T10762 Ceranib1 Ceranib1 is an inhibitor of ceramidase. It inhibits the proliferation of ovarian cancer cells. Ceranib1 inhibits ceramidase activity toward an exogenous ceramid...
T10763 Ceratamine A Ceratamine A is an antimitotic heterocyclic alkaloid isolated from the marine sponge Pseudoceratina sp., acts as a microtubule-stabilizing agent with cytotoxici...
T10764 Cercosporamide Cercosporamide is a ATP-competitive Pkc1 kinase inhibitor (IC50 <50 nM; Ki <7 nM). It also is a unique Mnk inhibitor.
T10765 Cereblon modulator 1 Cereblon modulator 1 is a cereblon (CRBN) E3 ligase modulator. It specifically binds to CRBN, thereby affecting the activity of the ubiquitin E3 ligase complex.
T10766 Ceritinib D7 Ceritinib D7 (LDK378 D7) is a deuterium-labeled Ceritinib. Ceritinib is an ATP-competitive inhibitor of ALK tyrosine kinase.
T10768 Cetilistat impurity 1 Cetilistat impurity 1 is an impurity of Cetilistat. Cetilistat is an inhibitor of pancreatic lipase. Cetilistat inhibits rat and human pancreatic lipase activit...
T10771 CETP-IN-3 CETP-IN-3 is an inhibitor of the plasma glycoprotein cholesterol ester transfer protein (CETP), elevating HDL-C through inhibition of CETP.
T10772 Cevipabulin Cevipabulin (TTI-237) is a microtubule-active antitumor compound and inhibits the binding of [3H] vinblastine to tubulin (IC50: 18-40 nM in the human tumor cell...
T10772L Cevipabulin fumarate Cevipabulin (TTI-237) fumarate is a microtubule-active antitumor compound and inhibits the binding of [3H] vinblastine to tubulin (IC50: 18-40 nM in the human t...
T10774 CFM-2 CFM-2 is a selective non-competitive AMPAR antagonist.
T10776 CFTR corrector 4 CFTR corrector 4 is a highly potent and orally active corrector of cystic fibrosis transmembrane conductance regulator (CFTR). It can increase CFTR levels at th...
T10779 CGP 25454A CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.
T1078 Sulfadimethoxine Sulfadimethoxine is a sulfanilamide that is used as an anti-infective agent.
T10780 CGP-53153 CGP-53153 is a steroidal inhibitor of 5 alpha-reductase (IC50s: 36 and 262 nM in rat and human prostatic tissue).
T10781 CGP 78608 hydrochloride CGP 78608 hydrochloride is a highly selective antagonist at the glycine binding site of the NMDA receptor (IC50: 6 nM). CGP 78608 acts as a potentiator of GluN1...
T10782 CGP52411 CGP52411 (DAPH) is a highly selective, orally active, and ATP-competitive EGFR inhibitor (IC50: 0.3 μM). It blocks the toxic influx of Ca2+ ions into neuronal ...
T10783 CGS 15435 CGS 15435 is a potent inhibitor of thromboxane (TxA2) synthetase (IC50: 1 nM). It has a selectivity for Tx synthetase 100000-fold greater than that for PGI2 syn...
T10785 Chalcone 4 (hydrate) Chalcone 4 hydrate, an anti-parasite compound, inhibits the growth of Theileria and Babesia.
T10787 Chitise-IN-1 Chitinase-IN-1 is an insect chitinase and N- acetyl hexosaminidase inhibitor and pesticide.
T10788 Chitise-IN-2 Chitinase-IN-2 is an insect chitinase and N- acetyl hexosaminidase inhibitor and pesticide.
T10788L Chitise-IN-2 hydrochloride Chitinase-IN-2 hydrochloride is an insect chitinase and N- acetyl hexosaminidase inhibitor and pesticide.
T10795 Chlordantoin Chlordantoin is an antifungal agent with the potential for vaginal candidiasis treatment.
T10796 Chlormethiazole hydrochloride Clomethiazole hydrochloride is an anticonvulsant and sedative. It is neuroprotective and prevents the degeneration of serotonergic nerve terminals induced by 3,...
T10797 Chlormidazole hydrochloride Chlormidazole hydrochloride has inhibitory activity against many fungi and some gram-positive cocci. It can be applied in fungal and bacterial infections of ski...
T10798 Chlorpromazine D6 hydrochloride Chlorpromazine D6 hydrochloride is the deuterium-labeled Chlorpromazine. Chlorpromazine is an inhibitor of dopamine receptors, potassium channels, 5-HT receptor...
T1080 2-Aminoethanethiol Cysteamine is a Cystine Depleting Agent. The mechanism of action of cysteamine is as a Cystine Disulfide Reduction.
T10803 CHMFL-KIT-033 CHMFL-KIT-033 is a potent and selective inhibitor of the c-KIT T670I mutant (IC50: 0.045 μM) for gastrointestinal stromal tumors (GISTs).
T10805 Cholesterol glucuronide Cholesterol glucuronide is an endogenous metabolite of lipid generated by UDP glucuonyltransferase in the liver.
T10806 Cholesteryl arachidote Cholesteryl arachidonate is a human endogenous metabolite.
T10807 Cholesteryl Linolete Cholesteryl Linolenate is a human endogenous metabolite.
T10808 CHPG sodium salt CHPG sodium salt is a selective agonist of mGluR5. In BV2 microglial cells, it attenuates SO2-induced oxidative stress and inflammation through the TSG-6/NF-κB...
T10809 CHPG CHPG is a selective agonist of mGluR5. In BV2 microglial cells, it attenuates SO2-induced oxidative stress and inflammation through the TSG-6/NF-κB pathway.
T10810 Chromomycin A3 Chromomycin A3 is an aureolic acid-type antitumor antibiotic. Chromomycin A3 has a variety of utilities as a staining agent for human sperm chromatin, autophagy...
T10811 Chymase-IN-1 Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).
T10812 Cicloprolol hydrochloride Cicloprolol is a partial agonist of β 1-adrenoceptor.
T10813 Cilobradine hydrochloride Cilobradine is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels.
T10814 Cicalcet metabolite M4 Cinacalcet metabolite M4 is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.
T10815 Cinmoylglycine Cinnamoylglycine is a glycine conjugate of cinnamic acid and a urinary metabolite in humans. It is used as a potential urinary biomarker.
T10816 Cinrizine D8 Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.
T10817 Cipemastat Cipemastat is a competitive inhibitor of human collagenases 1, 2, and 3 (Kis: 3.0, 4.4, and 3.4 nM).
T10818 Ciprofibrate D6 Ciprofibrate D6 is a deuterium-labeled Ciprofibrate. Ciprofibrate is an agonist of peroxisome proliferator-activated receptor.
T10819 Cipropride S entiomer Cipropride S enantiomer is the S enantiomer of cipropride which is an antiemetic drug.
T1082 Benzyl isothiocyanate Benzyl isothiocyanate (BITC) is an isothiocyanate originally found in cruciferous vegetables. It shows immunomodulatory, anti-parasitic, antibiotic, antioxidati...
T10820 Ciraparantag Ciraparantag is an inhibitor of thrombin and factor Xa. Ciraparantag is a broad-spectrum reversal agent for anticoagulants, including unfractionated heparin, lo...
T10820L Ciraparantag TFA Ciraparantag TFA is an inhibitor of thrombin and factor Xa. Ciraparantag is a broad-spectrum reversal agent for anticoagulants, including unfractionated heparin...
T10822 Cirsimarin Cirsimarin is a flavonoid isolated from Microtea debilis. It shows a potent antilipogenic effect and decreases adipose tissue deposition in mice. Cirsimarin has...
T10825 Citrinin Citrinin is a mycotoxin that causes contamination in the food and is associated with different toxic effects. Citrinin also possesses a broad spectrum of bioact...
T10826 CK-666 CK-666 is a cell-permeable inhibitor of actin-related protein Arp2/3 complex. It binds to the Arp2/3 complex, stabilizes the inactive state of the complex, bloc...
T10828 CK2/PIM1-IN-1 CK2/PIM1-IN-1 is an inhibitor of CK2 and PIM1 (IC50s: 3.787 μM and 4.327 μM). It is developed for the research of proliferative disorders such as cancer, as w...
T10830 CL 316243 CL316243 is a highly potent selective agonist of β3-adrenoceptor (EC50: 3 nM) but is an extremely poor to β1/2- receptors. CL316243 is an effective stimulant ...
T10831 Cl-amidine Cl-amidine is an orally active inhibitor of peptidyl arginine deminase (PAD) (IC50s: 0.8 μM, 6.2 μM, and 5.9 μM for PAD1, PAD3, and PAD4). Cl-amidine induces...
T10831L Cl-amidine hydrochloride Cl-amidine hydrochloride is an orally active peptidyl arginine deaminase (PAD) inhibitor (IC50: 5.9 μM for PAD4). It induces apoptosis in cancer cells and it a...
T10831L2 Cl-amidine TFA Cl-amidine TFA is an orally active inhibitor of peptidyl arginine deminase (PAD) (IC50s: 0.8 μM, 6.2 μM, and 5.9 μM for PAD1, PAD3, and PAD4). Cl-amidine ind...
T10832 CL2-SN-38 CL2-SN-38, a part of the antibody-drug conjugate (ADC), can conjugate with the anti-Trop-2-humanized antibody hRS7. SN-38 is an inhibitor of DNA topoisomerase I...
T10834 CL656 CL656 is a stimulator of interferon genes (STING) activator.
T10835 Cletoquine Cletoquine (Desethylhydroxychloroquine) is a major active metabolite of Hydroxychloroquine. Cletoquine has the ability to against the chikungunya virus (CHIKV)....
T10835L Cletoquine oxalate Cletoquine oxalate (Desethylhydroxychloroquine oxalate) is a major active metabolite of Hydroxychloroquine. Cletoquine has the ability to against the chikunguny...
T10837 Clocapramine hydrochloride hydrate Clocapramine hydrochloride hydrate is an antagonist of the 5-HT2A and D2 receptors.
T10839 Clozic Clozic is a potential anti-arthritic compound.
T10842 Clomipramine D3 Clomipramine D3 is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.1...
T10842L Clomipramine D3 hydrochloride Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter bl...
T10843 CMF019 CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and 8.71 for the human, rat, and mouse).
T10844 CMI-392 CMI-392 is a dual 5-lipoxygenase inhibitor and platelet-activating factor (PAF) receptor antagonist (IC50s: 100 and 10 nM).
T10845 CMK CMK, an RSK2 kinase inhibitor, shows similar potency but less chemical stability compared with FMK.
T10846 CMLD010509 CMLD010509 (SDS-1-021) is a highly selective inhibitor of the oncogenic translation program supporting multiple myeloma (MM)-including key oncoproteins such as ...
T10847 CMLD012072 CMLD012072 is a potent eukaryotic initiation factor 4A (eIF4A) inhibitor with potent anti-neoplastic activity. It can induce RNA clamping of eIF4A1 and eIF4A2.
T10848 CMLD012073 CMLD012073 is a potent eukaryotic initiation factor 4A (eIF4A) inhibitor. It inhibits NIH/3T3 cells (IC50: 10 nM). CMLD012073 inhibits eukaryotic translation in...
T10849 CMLD012612 CMLD012612 is a potent eukaryotic initiation factor 4A (eIF4A) inhibitor. It inhibits cell translation and is cytotoxic to NIH/3T3 cells (IC50: 2 nM).
T10850 CMP-5 CMP-5 is a potent and selective PRMT5 inhibitor, while displays no activity against PRMT1/4/7 enzymes. It selectively blocks S2Me-H4R3 by inhibiting PRMT5 methy...
T10851 CMP-Sialic acid sodium salt CMP-Sialic acid sodium salt is an allosteric inhibitor of UDP-GlcNAc 2-epimerase. It provides a substrate for Golgi sialyltransferases. UDP-GlcNAc 2-epimerase i...
T10852 CNS-5161 hydrochloride CNS-5161 hydrochloride is a new antagonist of NMDA ion-channel. It interacts with the NMDA receptor/ion channel site to produce a noncompetitive blockade of the...
T10853 CNT2 inhibitor-1 CNT2 inhibitor-1 is a potent inhibitor of concentrative nucleoside transporter 2 (CNT2; IC50: 640 nM for hCNT2).
T10854 CNX-500 CNX-500 is a probe consisting of a covalent Btk inhibitor chemically linked to biotin. CNX-500 has inhibitory activity against Btk (IC50: 0.5 nM) and the abilit...
T10856 Cobimetinib R-enantiomer Cobimetinib R-enantiomer is the less active R-enantiomer of Cobimetinib which is a selective MEK inhibitor.
T10857 Coenzyme A Coenzyme A is an obligatory cofactor in all living cells synthesized from pantothenate (Vitamin B5), adenosine triphosphate (ATP), and cysteine.
T10858 COH34 analog 1 COH34 analog 1 is an oxidized analog of COH34. COH34 is a potent inhibitor of poly(ADP-ribose) glycohydrolase (PARG).
T10859 COH34 COH34 is a potent and specific inhibitor of poly(ADP-ribose) glycohydrolase (PARG; IC50: 0.37 nM). COH34 binds to the catalytic domain of PARG (Kd: 0.547 μM), ...
T10860 Col003 Col003 is a selective and potent inhibitor of Hsp47 and competitively binds to the collagen-binding site on Hsp47 (IC50: 1.8 μM). It can be used for the invest...
T10861 Collagen proline hydroxylase inhibitor-1 Collagen proline hydroxylase inhibitor-1 is an antifibroproliferative compound.
T10862 Collagen proline hydroxylase inhibitor Collagen proline hydroxylase inhibitor is an inhibitor collagen proline hydroxylase and useful for antifibrotic proliferative agents.
T10863 Complement C5-IN-1 Complement C5-IN-1 is a small-molecule inhibitor of complement component 5 protein (C5).
T10865 Cot inhibitor-1 Cot inhibitor-1 is an inhibitor of COT/Tpl2.
T10866 Cot inhibitor-2 Cot inhibitor-2 is an inhibitor of COT/Tpl2.
T10868 CP-28888 CP-28888 is an interferon inducer, more potent in mice but less active in man and devoid of antirhinovirus effects.
T10869 CP-409092 hydrochloride CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.
T10871 CP-809101 hydrochloride CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).
T10872 CP-96021 hydrochloride CP-96021 hydrochloride is a potent and orally active antagonist of leukotriene D4 (LTD4)/platelet activating factor receptor (Kis: 34 nM and 37 nM).
T10873 CP-96486 CP-96486 is a potent and orally active antagonist of leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor (Kis: 20 and 24 nM).
T10874 CP-060 CP-​060 is a potent Ca2+ antagonist and inhibits Ca2+ overload with antioxidant and cardioprotective activities.
T10875 CP5V CP5V, a PROTAC, induces mitotic inhibition, and suppresses cancer cell proliferation. It specifically degrades Cdc20 by linking Cdc20 to the VHL/VBC complex for...
T10876 CPA inhibitor CPA inhibitor is a potent carboxypeptidase A (CPA) inhibitor.
T10877 CPDA CPDA is a new potent inhibitor of SH2 domain-containing inositol phosphatase 2 (SHIP2).
T10878 CPFX2090 CPFX2090, a cephalosporin antibacterial compound, is extracted from patent WO2013052568A1 (Example 16g).
T10880 CPPG CPPG is a potent antagonist of group II/III mGlu receptors. CPPG exhibits some selectivity (approximately 20 fold) for group III (IC50: 2.2 nM) over group II (I...
T10881 CPPHA CPPHA is a selective positive allosteric modulator of the mGluR5 receptor.
T10884 CRAC intermediate 1 CRAC intermediate 1 is a key intermediate in the chemical synthesis of a series of CRAC channel inhibitors.
T10885 CRAC intermediate 2 CRAC intermediate 2 is an intermediate for CRAC inhibitor synthesis extracted from patent WO 2013059666A1.
T10886 Crocetine dimethyl ester Crocetine dimethyl ester (Dimethylcrocetin) is found in the stigmas of saffron (Crocus sativus L.) with antioxidant activity.
T10890 CRTh2 antagonist 3 CRTh2 antagonist 3 is a powerful chemokine receptor homologous molecule expressed on Th2 cell (CRTh2) antagonists. CRTh2 antagonist 3 enhanced the activity of P...
T10893 CS-722 Free base CS-722 free base is a synthetic central muscle relaxant with muscle relaxant activity and inhibitory effect on spinal reflex. CS-722 free base may inhibit spont...
T10895 CSN5i-3 CSN5i-3 is an effective, selective, oral CSN5 inhibitor that can inhibit CSN-catalyzed Cul1 adenylation with IC50 value of 5.8 nM.
T10896 CSRM617 CSRM617 is a selective small molecule inhibitor of the transcription factor ONECUT2 (OC2, the main regulator of androgen receptor). The Kd in SPR analysis is 7....
T10897 CT-721 CT-721 is a potent and time-dependent Bcr-Abl kinase inhibitor with an IC50 of 21.3 nM against wild-type Bcr-Abl kinase and has anti-chronic myeloid leukemia (C...
T10900 CUDA CUDA is an effective soluble cyclohydrolase inhibitor with IC50 of 11.1 nM and 112 nM for mouse sEH and human sEH, respectively. CUDA selectively increases the ...
T10901 Curcumin D6 Curcumin D6 (difluoroformylmethane D6) is deuterium-labeled curcumin (Turmeric yellow). Curcumin (Turmeric yellow) is a natural phenolic compound with various p...
T10902 CWHM-1008 CWHM-1008 is an effective oral antimalarial drug. The EC50 values of the drug-sensitive Plasmodium falciparum 3D7 and drug-resistant Dd2 strains are 46 and 21 n...
T10903 CWHM-1552 CWHM-1552 is an effective oral inhibitor of Plasmodium falciparum. For the 3D7 and Dd2 strains, the IC50 is 51 nM and 53 nM, respectively.
T10906 CXCR7 modulator 1 CXCR7 modulator 1 is an effective and orally bioavailable peptoid hybrid CXCR7 modulator with Ki of 9 nM.
T10907 CXCR7 modulator 2 CXCR7 modulator 2 is a 7-type C-X-C chemokine receptor (CXCR7) modulator with a Ki of 13 nM.
T10909 Cyclic-di-GMP Cyclic-di-GMP is a STING agonist and ubiquitous second messenger, which regulates the formation, motility and virulence of biofilms in various bacterial species...
T1091 Chlortalidone Chlorthalidone is a benzenesulfonamide-phthalimidine that tautomerizes to a BENZOPHENONES form. It is considered a thiazide-like diuretic.
T10910 Cycloartenol Cyclopentanol is a plant sterol compound and one of the key precursors for biosynthesis of various sterol compounds. Cycloartenol inhibits the migration of glio...
T10912 S1PR1-MO-1 S1PR-MO-1 is a modulator of sphingosine-1-phosphate receptor and is used to study hyperproliferative inflammatory diseases.
T10913 Cyclobuxine D Cyclobuxine D is a steroidal alkaloid extracted from Buxus microphylla. Cyclostatin D has obvious bradycardia effect on rat heart, and inhibits acetylcholine an...
T10915 Cycloguanil D6 Nitrate Cycloguanil D6 Nitrate is a dihydrofolate reductase inhibitor, deuterium-labeled Cycloguanil.
T10916 Cycloguanil D6 Cycloguanil D6 is a dihydrofolate reductase inhibitor, deuterium-labeled Cycloguanil.
T10918 NEP-In-1 NEP-IN-1 is a neutral endopeptidase (NEP) inhibitor with IC50 of 2 nM for dNEP.
T10919 Cyclophilin inhibitor 1 Cyclophilin inhibitor 1 is an effective and orally bioavailable cyclophilin A inhibitor with a Kd of 5 nM, showing potent anti-HCV activity, and an EC50 for HCV...
T10920 Cyclo(Arg-Gly-Asp-D-Phe-Val) TFA Arg-Gly-Asp-D-Phe-Val (TFA) has anti-tumor activity and is an inhibitor of integrin αvβ3.
T10921 CYM 9484 CYM 9484 is a selective and potent neuropeptide Y (NPY) Y2 receptor antagonist with IC50 value of 19 nM.
T10922 CYP11B2-IN-1 CYP11B2-IN-1 is a CYP11B2 inhibitor with IC50 of 2.3 nM. CYP11B2-IN-1 inhibits CYP11B1 with IC50 of 142 nM.
T10925 Cysteine Protease inhibitor Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine Protease
T10925L Cysteine Protease inhibitor hydrochloride Cysteine protease inhibitor hydrochloride is an inhibitor of cysteine protease. Target: Cysteine Protease
T10926 CYT-1010 CYT-1010 is an mu-opioid receptor agonist extracted from patent WO2013173730A2. The EC50 for the inhibition of β-arrestin recruitment and cAMP production is 13...
T10926L CYT-1010 hydrochloride CYT-1010 hydrochloride is an mu-opioid receptor agonist extracted from patent WO2013173730A2. The EC50 for β-arrestin recruitment and cAMP production inhibitio...
T10927 cyt-PTPε Inhibitor-1 cyt-PTPε inhibitor 1 is a potent cytosolic protein tyrosine phosphatase epsilon (cyt-PTPε) inhibitor, which binds to the catalytic domain of cyt-PTPε and blo...
T10929 D-3263 D-3263 is an agonist of transient receptor potential melatonin member 8 (TRPM8) with potential antitumor activity.
T10929L D-3263 hydrochloride D-3263 hydrochloride is enteric-coated, orally bioavailable (transient receptor potential melatonin member 8) TRPM8 agonist.
T10930 D-AP5 D-AP5 is a NMDA receptor antagonist.
T10931 d-Atabrine dihydrochloride d-Atabrine hydrochloride is the active enantiomer of quinacrine and has anti-pr virus activity.
T10932 D-Cl-amidine D-Cl-amidine is an effective and highly selective PAD1 inhibitor. D-Cl-amidine has a good correlation and no obvious toxicity.
T10933 D-Cysteine D-cysteine is the D-isomer of cysteine and a powerful inhibitor of the growth of E. coli. D-cysteine is mediated by D-amino acid oxidase to produce H2S, and is ...
T10934 D-Gluconic acid D-gluconic acid is a carboxylic acid that has antiseptic and chelating properties through oxidation.
T10935 D-Glutamic acid D-glutamic acid, the enantiomer of L-glutamic acid, is widely used in medicine and food.
T10936 D-I03 D-I03 is a selective RAD52 inhibitor with a Kd of 25.8 µM. D-I03 specifically inhibits RAD52-dependent single-chain annealing (SSA) and D-loop formation, with ...
T10938 D-Kynurenine D-kynurenine is a metabolite of D-tryptophan, which can be used as a biological precursor of KYNA and 3-hydroxykynurenine. D-Kynurenine is an agonist of G prote...
T10939 D,L-Cystathionine dihydrochloride D,L-Cystathionine dihydrochloride is an intermediate in the synthesis of cysteine, which acts from the isotype of cysteine-β-synthase (CBS) produced by leucine...
T10939L L-Cystathionine L-Cystathionine is a key nonprotein amino acid. Which is related to metabolic conditions.
T10940 D-Mannoheptulose D-mannoheptose is the main non-structural carbohydrate in avocado. D-mannoheptose is a specific inhibitor of D-glucose phosphorylation. D-mannoheptose can preve...
T10941 D-Ribonolactone D-ribolactone is a sugar lactone, an inhibitor of E. coli β-galactosidase, and Ki is 26 mM.
T10942 D-Threitol D-threitol is used as an antifreeze.
T10943 D-(-)-Lactic acid D-(-)-lactic acid is a normal intermediate in sugar fermentation (oxidation, metabolism). D-(-)-lactic acid is identified as a competitive inhibitor of ProDH (p...
T10944 D13-9001 The KD values of D13-9001 in Escherichia coli and Pseudomonas aeruginosa were 1.15μM and 3.57μM, respectively. D13-9001 has antibiotic activity. It is an effe...
T10945 D18024 D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.
T10947 D8-MMAD D8-MMAD is a deuterated form of MMAD, which is a microtubule destroyer.
T10948 D8-MMAE D8-MMAE (D8-Monomethyl auristatin E) is an effective mitotic inhibitor and tubulin inhibitor, deuterated MMAE.
T10949 D8-MMAF D8-MMAF is a microtubule destroyer, deuterated form of MMAF.
T10950 Dabigatran D4 hydrochloride Dabigatran D4 hydrochloride is deuterium-labeled dabigatran, which is a reversible and selective direct thrombin inhibitor (DTI) with a Ki value of 4.5 nM.
T10951 Dabigatran ethyl ester hydrochloride Dabigatran ethyl ester hydrochloride is an effective inhibitor of ribosyl dihydronicotinic acid amide dehydrogenase (NQO2) with an IC50 value of 0.8 μM and is ...
T10952 Dabuzalgron Dabuzalgron (Ro 115-1240) is an orally active selective alpha-1A adrenergic receptor agonist used to treat urinary incontinence. Dabuzaron prevents cardiotoxici...
T10953 Dafadine-A Dafadine-A is an analog of dafadine and a novel inhibitor of DAF-9 cytochrome P450 in the nematode Caenorhabditis elegans. Mammalian orthologs that also inhibit...
T10954 DAGLβ-IN-1 DAGLβ-IN-1 is a universal intermediate for designing DAGL tailored activity-based probes, and is an inhibitor of diacylglycerol lipase-β (DAGLβ).
T10956 Dansyl glutathione Dansyl glutathione is a capture agent used for quantitative assessment and identification of reactive metabolites.
T10957 Dapagliflozin impurity Dapagliflozin impurity is the enantiomer of Dapagliflozin, Dapagliflozin is a sodium glucose transporter 2 inhibitor.
T10958 Dapagliflozin D5 Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.
T10959 Daphnin Daphnin is one of the main coumarin bioactive ingredients with antibacterial activity. Daphnine is isolated from the entire Daphne fragrance, which is a folk me...
T10960 Darbufelone Darbufelone is a dual inhibitor of cellular PGF2α and LTB4 production. Dabfilon effectively inhibited PGHS-2 (IC50 = 0.19 μM), but had a much smaller effect o...
T10960L Darbufelone mesylate Darbufelone mesylate (CI-1004 mesylate) is a dual inhibitor of cellular PGF2α and LTB4 production. Dabfilon effectively inhibited PGHS-2 (IC50 = 0.19 μM), but...
T10961 Darenzepine Darenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1.
T10962 Dasatinib D8 Dasatinib D8 is deuterium-labeled dasatinib. Dasatinib is a dual Bcr-Abl and Src family tyrosine kinase inhibitor.
T10963 Dazopride Dazopride is an antiemetic agent.
T10964 DB1976 DB1976 is a selenium-thiophene analogue of DB270, a potent, cell-permeable and highly effective transcription factor PU.1 inhibitor. DB1976 strongly inhibits PU...
T10964L DB1976 hydrochloride DB1976 hydrochloride is a selenium selenium analogue of DB270, a potent and permeable cell transcription factor PU.1 inhibitor. In vitro, DB1976 hydrochloride e...
T10966 DC-5163 DC-5163 is a potent inhibitor of glyceraldehyde 3-phosphate dehydrogenase (GAPDH) with IC50 of 176.3 nM and Kd of 3.192 μM. DC-5163 selectively inhibits cancer...
T10967 DC_C66 DC_C66 DC_C66 has good selectivity for CARM1, PRMT1 (IC50 = 21μM), PRMT6 (IC50 = 47μM) and PRMT5. It is a cell-permeable, selective co-activator related argin...
T10968 DC0-NH2 The cytotoxicity of DC0-NH2 is 1000 times that of commonly used anti-cancer drugs (such as doxorubicin). It is the effect part of ADC. It is a simplified simula...
T10969 DC1SMe DC1 is an ADC cytotoxin, similar to the small groove-binding DNA alkylating agent CC-1065. DC1 can be used to synthesize antibody-drug conjugates targeted to th...
T10970 DC1 DC1 can be used to synthesize antibody-drug conjugates targeted to the treatment of cancer, is an ADC cytotoxin, similar to the small groove-binding DNA alkylat...
T10971 DC10SMe DC10SMe is a DNA alkylating agent that can be used in the synthesis of antibody-drug conjugates (ADC). The IC50 of DC10SMe for Ramos, Namalwa and HL60 / s cance...
T10972 DC4 DC4 can be used to synthesize antibody-drug conjugate (ADC), which is an ADC cytotoxin. DC4 can be used for targeted therapy of tumors.
T10973 DC41SMe DC41SMe is a DC1 derivative that is cytotoxic to Ramos, Namalwa and HL60 / s with IC50s ranging from 18-25 pM. DC1 is a simplified analogue of CC-1065, an antib...
T10974 DC41 DC41 is a derivative of DC1. DC1 is a simplified analogue of CC-1065, an antibody conjugate of cytotoxic DNA alkylating agents, used for targeted treatment of c...
T10975 DC44SMe The IC50 of DC44SMe for Ramos, Namalwa and HL60 / s cancer cells was 2.0 nM, 2.8 nM and 1.9 nM, respectively. DC44SMe can be used for targeted treatment of canc...
T10976 DC4SMe The IC50s of DC4SMe on Ramos, Namalwa and HL60 / s cancer cells were 1.9 nM, 2.9 nM and 1.8 nM, respectively. DC4SMe can be used for targeted therapy of tumors....
T10977 DCEBIO DCEBIO stimulates the secretion of Cl- through the activation of the hIK1 K + channel and the activation of the apical Cl- conductance. DCEBIO is a derivative o...
T10978 DCG-IV DCG-IV is an effective agonist of class II mGluR. DCG-IV has anticonvulsant and neuroprotective effects. The EC50 of mGlu2R and mGlu3R are 0.35 and 0.09 μM, re...
T10979 DCPIB DCPIB is a selective, reversible and effective volume-regulated anion channel (VRAC) inhibitor that voltage-dependently activates potassium channels TREK1 and T...
T1098 Denatonium benzoate Denatonium, a quaternary ammonium cation, is a compound of a salt with an inert anion like saccharide or benzoate. Its structure is involved in the local anesth...
T10982 ddATP ddATP is a dideoxynucleotide, used as a chain extension inhibitor for DNA polymerase, and used for DNA sequencing by the Sanger method.
T10983 DDP-38003 trihydrochloride DDP-38003 trihydrochloride is a novel, orally available histone lysine specific demethylase 1A (KDM1A / LSD1) inhibitor with IC50 of 84 nM.
T10983L DDP-38003 dihydrochloride DDP-38003 dihydrochloride is an orally available histone lysine-specific demethylase 1A (KDM1A/LSD1) inhibitor (IC50: 84 nM).
T10984 DDR-TRK-1 DDR-TRK-1 is a selective discoid domain receptor 1 (DDR1) inhibitor with IC50 value of 9.4 nM. DDR-TRK-1 also inhibits the TRK family.
T10985 DDR Inhibitor DDR inhibitor is a potent discidin domain receptor (DDR) inhibitor. The IC50 of DDR2 is 3.3 nM, and DDR1 has 53% inhibition at 1.5 nM.
T10986 DDX3-IN-1 DDX3-IN-1 is a DEAD-box polypeptide 3 (DDX3) inhibitor with CC50 of 50 and 36 μM for HIV and HCV, respectively. Antiviral activity.
T10987 Decarboxy Moxifloxacin Decarboxy Moxifloxacin is a decarboxylated compound of moxifloxacin. Moxifloxacin is an oral active 8-methoxyquinolone antibiotic used in acute bacterial sinusi...
T10992 Delamanid D4 Delamanid D4 is deuterium-labeled Delamanid. Delamanid is a newer mycobacterial cell wall synthesis inhibitor that inhibits the synthesis of mucus acid.
T10993 δ-Amyrenone Delta-Amyrenone (Delta-Amyrone) has anti-inflammatory effects and is a pentacyclic triterpenoid compound of linear streptomyces.
T10997 Derazantinib Racemate Derazantinib Racemate is the racemate of Derazantinib; is a potent inhibitor of FGFR1-3.
T10998 Deriglidole Deriglidole is a peripheral adrenoceptor antagonist with high affinity for α2-adrenoceptor.
T10999 Desbutyl Lumefantrine Desbutyl Lumefantrine is a metabolite of lumefantrine with antimalarial activity.
T1100 Polymyxin B sulfate Polymyxin B sulphate is a mixture of polymyxins B1 and B2, obtained from Bacillus polymyxa strains. They are basic polypeptides of about eight amino acids and h...
T11000 Descarbamoyl cefuroxime Descarbamoyl cefuroxime is also an intermediate in the synthesis of cephalosporin antibiotics. Decarbamyl cefuroxime is a degradation product of cefuroxime.
T11001 Desethyl chloroquine Desethyl chloroquine is the main deethyl metabolite of chloroquine. Chloroquine diphosphate is an inhibitor of autophagy and toll-like receptors (TLRs). Deethyl...
T11001L Desethyl chloroquine diphosphate Desethyl chloroquine diphosphate is the main deethyl metabolite of chloroquine. Chloroquine diphosphate is an inhibitor of autophagy and toll-like receptors (TL...
T11002 Desethylamiodarone hydrochloride Desethylamiodarone hydrochloride (N-desethylamiodarone hydrochloride) is formed by the CYP3A isozyme. Amiodarone is an antiarrhythmic drug that inhibits ATP-sen...
T11003 Desfluoro-ezetimibe Desfluoro-ezetimibe is the defluorinated impurity of ezetimibe. Ezetimibe is an effective, metabolically stable cholesterol absorption inhibitor. Ezetimibe is a...
T11006 Desmethyl ferroquine Desmethyl ferroquine is the active and major metabolite of Ferroquine.Desmethyl ferroquine shows significant activity against Chloroquine-susceptible and resist...
T11007 Desmethyl Levofloxacin Desmethyl Levofloxacin is a metabolite of levofloxacin. Levofloxacin is a synthetic fluoroquinolone drug, an antibacterial agent that can inhibit the super-coil...
T11008 Desmethylnortriptyline Desmethylnortriptyline is a metabolite of nortriptyline. Nortriptyline is a tricyclic antidepressant. It is the main active metabolite of amitriptyline and is u...
T11009 Destruxin B Destruxin B is a cyclic peptide with insecticidal and anticancer activity isolated from the insect pathogenic fungus Metarhizium isopliae. Destruxin B induces a...
T1101 Minocycline hydrochloride Minocycline is a tetracycline antibiotic with excellent absorption and tissue penetration that is used for several bacterial infections as well as treatment of ...
T11011 Dexpramipexole dihydrochloride Dexpramipexole dihydrochloride ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine agonist.
T11012 Dextran Dextran (Dextran 40) has an inhibitory effect on platelet aggregation and coagulation factors, and is used as an agent for increasing plasma volume.
T11013 Dextrorotation nimorazole phosphate ester Dextrorotation nimorazole phosphate ester is an anti-anaerobic and anti-parasitic agent. D-morpholine ornidazole organic phosphate is a newly developed, highly ...
T11014 DFP00173 DFP00173 is a potent and selective aquaporin 3 (AQP3) inhibitor. DFP00173 inhibits mouse and human AQP3 with IC50 of ~0.1-0.4 μM. Compared with the homologous ...
T11016 DGAT-1 inhibitor 2 DGAT-1 inhibitor 2 is an effective DGAT-1 inhibitor; anti-obesity drug. Objective: DGAT-1 acyl-CoA: diacylglycerol acyltransferase 1 (DGAT1) is one of two known...
T11017 DGN462 DGN462 is an effective DNA alkylating agent with anti-tumor activity, as in acute myeloid leukemia (AML). DGN462 can be used as a cytotoxic component of antibod...
T11018L (-)-DHMEQ (–)-DHMEQ is an effective inhibitor of NF-κB.
T11020 DHODH-IN-11 DHODH-IN-11 is a leflunomide derivative and weak dihydroorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.03.
T11021 DHODH-IN-12 DHODH-in -12 (Compound 12b) is a leflunomide derivative and a weak dihydrorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.07.
T11025 DHODH-IN-2 DHODH-IN-2 is an inhibitor of human dihydroorotate dehydrogenase (HsDHODH), which can inhibit measles virus replication, with a pMIC50 value of 8.6.
T11026 DHODH-IN-3 DHODH-IN-3 is an effective inhibitor of human dihydroorotate dehydrogenase (HsDHODH) with IC50 value of 261 nM. DHODH-IN-3 binds to the ubiquinone binding cavit...
T11027 DHODH-IN-4 DHODH-IN-4 is a human and Plasmodium falciparum dihydroorotate dehydrogenase (DHODH) inhibitor. The IC50 values of PfDHODH and HsDHODH are 4 μM and 0.18 μM, r...
T11028 DHODH-IN-5 DHODH-in -5 is a potent inhibitor of human dihydrogen dehydrogenase (DHODH). For human recombinant DHODH, its pIC50 is 7.8. DHODH-IN-5 inhibits measles virus re...
T11029 DHODH-IN-7 DHODH-IN-7 is a human dihydroorotate dehydrogenase (DHODH) inhibitor with IC50 of 0.91 μM. DHODH-IN-7 induces the differentiation of acute myeloid leukemia.
T11033 DI-591 DI-591 is an effective, high-affinity and cell-permeability inhibitor for DCN1-UBC12 interaction. DI-591 binds to DCN1 and DCN2 with Ki values of 12 and nM and ...
T11035 diABZI STING agonist-1 (Tautomerism) diABZI STING agonist-1 Tautomerism is a selective stimulator of interferon gene (STING) receptor agonists, with EC50 of 130 and 186 nM for humans and mice, resp...
T11037 Diacylglycerol acyltransferase inhibitor-1 Diacylglycerol acyltransferase inhibitor-1 is a diacylglycerol acyltransferase (DGAT1) inhibitor.
T11038 Dibutyryl-cGMP sodium Dibutyryl-cGMP sodium (Bt2cGMP sodium) is a cell-permeable cGMP analog. Dibutyryl-cGMP sodium preferentially activates cGMP-dependent protein kinase (PKG). Dibu...
T11039 Didesethyl chloroquine Didesethyl chloroquine is an effective myocardial inhibitor. Diethylchloroquine (Bisdesethylchloroquine) is the main metabolite of the antimalarial drug chloroq...
T11040 Dihydro Dutasteride Dihydro Dutasteride is a metabolite of Dutasteride. Dutasteride is an effective inhibitor of five α-reductase isozymes.
T11041 Dihydro-β-erythroidine hydrobromide Dihydro-β-erythroidine hydrobromide(DHβE) is a potent, oral active and competitive antagonist of neuronal nicotinic acetylcholine receptors (nAChRs). Dihydro-...
T11042 Dihydrocytochalasin B Dihydrocytochalasin B (H2CB) is a cell division inhibitor that changes the morphology of cells, similar to cytochalasin B. Does not inhibit glucose transport. D...
T11043 Dihydroergocristine mesylate Dihydroergocristine mesylate (DHEC mesylate) is an inhibitor of γ-secretase (GSI), which can reduce the production of Alzheimer's disease amyloid beta peptide,...
T11045 Dimethyl fumarate D6 Dimethyl fumarate D6 is a deuterium labeled Dimethyl fumarate. can induces upregulation of antioxidant gene expression.
T11046 Dimethyl-SGD-1882 Dimethyl-SGD-1882 (Dimethyl-PBD dimer) is a highly efficient DNA alkylating agent used as antibody-drug conjugate (ADC) cytotoxin. PBD Dimer is a DNA alkylating...
T11047 DiosMetin 7-O-β-D-Glucuronide DiosMetin 7-O-β-D-Glucuronide is an antioxidant constituent in the fruits of Luffa cylindrical[1].
T11048 DIPQUO DIPQUO is an activator of bone marker alkaline phosphatase (ALP). DIPQUO promotes the differentiation of mouse and human osteoblasts by activating p38MAPK-β. T...
T11049 Diprotin A TFA Diprotin A (TFA) is an inhibitor of dipeptidyl peptidase IV (DPP-IV).
T11050 Dipyrocetyl Dipyrocetyl is extracted from patent WO 2011132171 A1 and has anti-inflammatory and analgesic effects.
T11051 DIQ3 DIQ3 is non-toxic to normal human cell lines and is an effective anti-cancer agent.
T11052 Disitertide Disitertide (P144) is an inhibitor of TGF-β1.
T11053 DJ001 DJ001 is a highly specific, selective and non-competitive protein tyrosine phosphatase σ (PTPσ) inhibitor with IC50 of 1.43 μM. DJ001 promotes the regenerati...
T11054 DL-Norvaline DL-Norvaline is a non-competitive inhibitor of arginase. Derivatives of L-norvaline.
T11057 DM3-SMe DM3-SMe is a maytansine derivative and tubulin inhibitor. It is a cytotoxic part of antibody-drug conjugates (ADCs) and can bind to antibodies via disulfide bon...
T11058 DM3 DM3 (Maytansinoid DM3) is a maytansine mimic containing disulfide or thiol groups and a tubulin inhibitor. It is the cytotoxic part of antibody-drug conjugates ...
T11059 DM4-SMe DM4-SMe is a cytotoxic part of antibody-drug conjugates (ADCs) and a metabolite of antibody-maytansin conjugates (AMCs) and tubulin inhibitors, which can also b...
T11062 dmDNA31 dmDNA31 is a rifamycin antibiotic that can inhibit the DNA-dependent RNA polymerase of bacteria and has strong bactericidal activity against Staphylococcus aure...
T11063 DMT1 blocker 1 DMT1 blocker 1 is a blocker of divalent metal transporter 1 (DMT1) with IC50 of 0.64 μM, which is expected to block the absorption of iron by intestinal cells ...
T11064 DMT1 blocker 2 DMT1 blocker 2, compound 12f, is a direct inhibitor of divalent metal transporter 1 (DMT1) with an IC50 hydrogen peroxide value of 0.83, which is expected to bl...
T11067 VX-984 VX-984 is a potent DNA-PK inhibitor.
T11068 DNA31 DNA31 is a potent RNA polymerase inhibitor.
T11069 DO-264 DO-264 is a selective active inhibitor containing a dehydrogenase domain of 12 (ABHD12) with IC50 of 11 nM.
T1107 Sarafloxacin hydrochloride Sarafloxacin hydrochloride, a quinolone antibiotic drug, is a hydrochloride salt form of sarafloxacin.
T11070 DO34 analog DO34 analog is a triazole DAGL(α) inhibitor extracted from patent WO2017096315 A1, compound 100.
T11070L DO34 DO34 is a highly potent and centrally active inhibitor of diacylglycerol lipase (IC50: 6 nM for DAGLα conversion of SAG to 2-AG).
T11071 Dofequidar fumarate Dofequidar fumarate(MS-209 fumarate), an orally active quinoline compound, has been reported to overcome MDR by inhibiting ABCB1/P-gp, ABCC1/MDR-associated prot...
T11072 Dofetilide D4 Dofetilide D4 (UK 68789 D4) is a deuterium-labeled Dofetilide. Dofetilide is a class III antiarrhythmic drug.
T11073 Dofetilide N-oxide Dofetilide N-oxide (UK-116856) is a metabolite of dofetilide. Dofetilide can block potassium channels and is a tertiary antiarrhythmic drug.
T11074 Dolutegravir intermediate-1 Dolutegravir intermediate-1 is a new synthetic Dolutegravir intermediate extracted from patent WO 2016125192 A2. Dolutegravir is an integrase inhibitor develope...
T11076 Dooku1 Dooku1 is an analog of Yoda1 and a selective antagonist of endogenous Piezo1 channels. Dooku1 inhibits Ca2+ entry induced by 2μMYoda1 with IC50 values of 1.3μ...
T11077 Dopamine D2 receptor antagonist-1 Dopamine D2 receptor antagonist 1 is a negative allosteric modulator (NAM) of dopamine D2 receptor (D2R), with sub-mM affinity.
T11079 NMI 8739 NMI 8739 is a dopamine D2 autoreceptor agonist, which is an amine conjugate of the DHA carrier and the neurotransmitter dopamine.
T1108 Nithiamide Nithiamide is an orally available antiprotozoan agent used in the treatment of vaginal trichomoniasis.
T11085 Dot1L-IN-6 Dot1L-IN-6 is a potent disruptor of telomeric silencing 1-like protein (DOT1L) inhibitor with an IC50 SPA DOT1L of 0.19 nM.
T11086 DOTAP chloride DOTAP chloride is a useful and effective cationic lipid transfection DNA(plasmids, BacMIDs) and modified nucleic acids (antisense oligonucleotides) without the ...
T11087 DOV-216,303 Free Base Dov-216,303 (free base) is an effective trihydroxytryptamine, norepinephrine and dopamine reuptake inhibitor with IC50 values of 14 nM, 20 nM and 78 nM for hSER...
T11089 Doxercalciferol-D3 Doxercalciferol-d3 is the deuterated form of Doxercalciferol and ACTS as vitamin D receptor activator (VDRA), which is a vitamin D2 analogue.
T1109 Zucapsaicin Zucapsaicin is a medication used to treat osteoarthritis of the knee and Others neuropathic pain.Zucapsaicin is a synthetic cis isomer of natural capsaicin that...
T11090 MC-DOXHZN Mc-doxhzn is a protein-binding prodrug of DOXUbicin (DNA topoisomerase II inhibitor) with acid sensitivity.
T11091 Doxylamine D5 succinate Doxylamine D5 succinate first generation antihistamine, deuterium-labeled Doxylamine,
T11093 DPPH The odd electrons of nitrogen atoms in DPPH are reduced by receiving a hydrogen atom from the antioxidant to the corresponding hydrazine.DPPH method can be used...
T11094 DRAK2-IN-1 Drak2-in-1, a potent, selective and ATP-competitive DRAK2 inhibitor, has an IC50 and KIvalue of 3 nM and 0.26 nM, respectively.Drak2-in-1 also had an effect on ...
T11095 DREADD agonist 21 dihydrochloride DREADD agonist 21 dihydrochloride is an effective human toadine acetylcholine M3 receptor (hM3Dq) agonist (EC50=1.7 nM).
T11095L DREADD agonist 21 In addition to being inactive at hM3, DREADD agonist 21, a potent full agonist of hM3Dq (EC50: 1.7 nM), is only 3.5-fold selective for hM3Dq over H1, 40-fold se...
T11096 DRI-C21045 Dri-c21045 showed concentration-dependent inhibition of NF- B activation and all CD40L induced by B cell proliferation. IC50 was 17.1 M and 4.5 M, respectively....
T11097 Drobuline hydrochloride Drobuline hydrochloride has the action of cardiac inhibitor, often used for anti-arrhythmia.
T11098 Droloxifene Droloxifene, a tamoxifen derivative, is an oral active and selective estrogen receptor modulator.Droloxifene induced p53 expression and apoptosis in McF-7 cells...
T11099 Droxicainide Droxicainide is an antiarrhythmic agent.
T11100 DS-1040 Tosylate DS-1040 Tosylate is an oral active, selective thrombolytic inhibitor with IC50s of 5.92 nM and 8.01 nM for human and rat TAFIa, is an orally active, selective i...
T11101 DS08210767 DS08210767 is a highly potent, orally bioavailable antagonist of PTHR1(IC50 : 90 nM).
T11103 DS18561882 DS18561882 also inhibited MTHFD1 (IC50=0.57).DS18561882 had good oral drug kinetics.DS18561882 is a potent isozyme-selective methylene tetrahydrofolate dehydrog...
T11104 DS21360717 DS21360717 is an effective oral tyrosine kinase inhibitor with anticancer activity and IC50 of 0.49 nM.
T11105 DS88790512 DS88790512, IC50 at 11 nM, is an effective, selective, oral bioeffective TRPC6 inhibitor.
T11106 DSP-0565 DSP-0565 shows anti-convulsant activity in various models (scPTZ, MES, 6 Hz and amygdala kindling) with good safety margin. DSP-0565 (compound 17a) is a strong,...
T11107 DSP-1053 Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.
T11108 DSR-6434 DSR-6434 has a strong antitumor effect. DSR-6434 is a potent and selective Toll-like receptor 7 (TLR7) agonist, with EC50s of 7.2 nM and 4.6 nM for human and mi...
T11109 DU717 DU-717 is an antihypertensive agent.
T11113 Duloxetine D3 hydrochloride Duloxetine D3 hydrochloride is a serotonin-norepinephrine reuptake inhibitor (SNRI) with a Ki of 4.6 nM, used for treatment of major depressive disorder and gen...
T11114 Duloxetine metabolite Para-Naphthol Duloxetine Para-Naphthol Duloxetine is a serotonin-norepinephrine reuptake inhibitor (SNRI),is a metabolite of Duloxetine.
T11115 Duocarmycin GA Duocarmycin GA can be used against multi-drug resistant cell lines. Duocarmycin GA is an antibody drug conjugates (ADCs) toxin. Duocarmycin is a DNA alkylating ...
T11116 Duocarmycin MA Duocarmycin MA can be used against multi-drug resistant cell lines.Duocarmycin MA is an antibody drug conjugates (ADCs) toxin. Duocarmycin is a DNA alkylating a...
T11117 Duocarmycin MB Duocarmycin MB can be used against multi-drug resistant cell lines. Duocarmycin MB is an antibody drug conjugates (ADCs) toxin. Duocarmycin is a DNA alkylating...
T11118 Duocarmycin SA Duocarmycin SA is an extremely potent cytotoxic agent capable of inducing a sequence-selective alkylation of duplex DNA.Duocarmycin SA is a potent antitumor ant...
T11119 Duocarmycin Duocarmycin is a DNA minor groove binding alkylating agent and explored as drug–antibody conjugates (ADCs) . Duocarmycin is based on its characteristic curved...
T11120 Duocarmycin TM Duocarmycin TM is a DNA alkylator. Duocarmycin TM is an exceptionally potent antitumor antibiotic.
T11121 Duoperone Duoperone is a neuroleptic agent and also a antiemetic agent in animal models.
T11122 DUPA(OtBu)-OH DUPA(OtBu)-OH is a DUPA precursor. DUPA is used as the targeting moiety to actively deliver Docetaxel (DTX) for treatment of Prostate-Specific Membrane Antigen ...
T11123 DuP 105 DuP 105 is an orally active oxazolidinone, a new class of synthetic antimicrobial agent with activity against gram-positive bacteria.
T11124 Duramycin Duramycin  is a cyclic peptide lantibiotic derived from Streptomyces cinnamoneuma. Duramycin interacts with phosphatidylethanolamine (PE) and has antibacteria...
T11125 Durlobactam sodium salt For the treatment of drug-resistant Gram-negative bacteria including Acinetobacter baumannii. Durlobactam sodium salt is a broad-spectrum β-lactamase inhibitor...
T11126 Durvalumab Durvalumab is an anti-PD-L1 monoclonal antibody, humanized.Durvalumab completely blocked the binding of PD-L1 to PD-1 and CD80, and the IC50s were 0.1 and 0.04 ...
T11127 Dutogliptin tartrate Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.
T11128 Dutogliptin Dutogliptin (PHX-1149 free base) is an oral, effective and selective dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.
T1113 Imazalil Enilconazole is an Agricultural fungicide Enilconazole is a fungicide widely used in agriculture, particularly in the growing of citrus fruits. It is also calle...
T11130 DVD-445 Dvd-445 has good anti-cancer effect.Dvd-445 is an effective peptide covalent thioredoxin reductase 1 (TrxR1) inhibitor with IC50 value of 0.60 mol/L M.
T11134 DZ2002 DZ2002 is a potent and reversible S-Adenosyl-L-homocysteine Hydrolase(SAHH; AdoHcy Hydrolase) inhibitor with Ki of 17.9 nM. IC50 value: 17.9 nM(Ki).
T11135 (E)-10-Hydroxy Nortriptyline maleate (E)-10-Hydroxy Nortriptyline maleate is a metabolite of Nortriptyline. Nortriptyline is a tricyclic antidepressant and the main active metabolite of Amitriptyli...
T11138 (E)-LHF-535 (E)-LHF-535 is the E-isomer of LHF-535. LHF-535 is an antiviral , has EC50s of <1 μM, <1 μM, <1 μM, and 1-10 μM for Lassa, Machupo, Junin, and VSVg virus, ...
T11138L LHF-535 LHF-535 is an antiviral compound. It has EC50s of <1 μM, <1 μM, <1 μM, and 1-10 μM for Lassa, Machupo, Junin, and VSVg virus, respectively.
T11139 (E/Z)-BCI (E/Z)-BCI attenuates LPS-induced inflammatory mediators and ROS production in macrophage cells via activating the Nrf2 signaling axis and inhibiting the NF-κB ...
T1114 Ciclopirox ethanolamine Ciclopirox Olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.
T11141 E64FC26 E64FC26 shows anti-myeloma activity.E64FC26 is a potent pan-inhibitor of the protein disulfide isomerase (PDI) family, with IC50s of 1.9, 20.9, 25.9, 16.3, and ...
T11143 EB-47 EB-47 mimics the substrate NAD+ and extends from the nicotinamide to the adenosine subsite.EB-47, a potent and selective PARP-1/ARTD-1 inhibitor with an IC50 v...
T11144 EC0488 EC0488 was used to synthesize EC0531, which has folic acid receptor specificity and anti-tumor activity.
T11145 EC1454 EC1454 is an anti-tumor compound.
T11146 EC359 EC359Kd, 10.2 nM, interacts directly with LIFR and effectively blocks LIF/LIFR interaction. It is a potent, selective, highly affinity, and oral active leukemia...
T11147 EC5026 EC5026 has the potential to relieve pain by stabilizing natural analgesic and anti-inflammatory mediators. EC5026 (BPN-19186) is a first-in-class, potent and or...
T11148 Ecastolol Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.
T11150 Ecteinascidin 770 Ecteinascidin 770 (ET-770) inhibits U373MG cells and is a 1,2,3, 4-tetrahydroisoquinoline alkaloid with strong anticancer activity.IC50 is 4.83 nM.
T11151 Ecteinascidin-Analog-1 Ecteinascidins is a family of tetrahydroisoquinoline alkaloids with wide range of antitumor and antimicrobial activities. Ecteinascidin-Analog-1 is a useful int...
T11152 Edaravone D5 Edaravone is a strong novel free radical scavenger, and inhibits MMP-9-related brain hemorrhage in rats treated with tissue plasminogen activator. Edaravone D5 ...
T11153 EG00229 EG00229 selectively inhibits VEGF-A binding to NRP1 b1 domain with an IC50 of 3 μM, but has no effect on VEGFA binding to VEGFR-1 and VEGFR-2. EG00229 is a neu...
T11154 EG01377 EG01377 has antiangiogenic, antimigratory, and antitumor effects.EG01377 is a neuropilin-1 (NRP1) antagonist, with a Kd of 1.32 μM for NRP1-b1, and IC50s of bo...
T11156 Nazartinib S-enantiomer Nazartinib is an EGFR inhibitor. Nazartinib S-enantiomer is the less active S-enantiomer of Nazartinib.
T11156L Nazartinib mesylate Nazartinib mesylate is a novel, covalent mutant-selective inhibitor of EGFR (Ki and Kinact: 31 nM and 0.222/min on EGFR(L858R/790M) mutant).
T11165 EGLU EGLU interacts with (lS,3S)-ACPD-sensitive site with a Kd value of 66 μM. EGLU is an antidepressant agent.EGLU ((2S)-α-Ethylglutamic acid; (2S)-α-EGLU) is a...
T11166 EHMT2-IN-1 EHMT2-IN-1 is a potent EHMT inhibitor, . Used in the research of blood disorder or cancer.with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellul...
T11167 EHMT2-IN-2 EHMT2-IN-2 Used in the research of blood disease or cancer. EHMT2-IN-2 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide an...
T11168 EHNA hydrochloride EHNA hydrochloride play roles in mediating diverse pharmacological responses, including antiviral, antitumour and antiarrhythmic effects. EHNA hydrochloride is...
T11170 eIF4A3-IN-1 eIF4A3-IN-1  is a selective eukaryotic initiation factor 4A3 (eIF4A3) inhibitor (IC50=0.26 μM; Kd=0.043 μM), which binds to a non-ATP binding site of eIF4A3...
T11171 eIF4A3-IN-2 eIF4A3-IN-2 is a highly selective and noncompetitive eukaryotic initiation factor 4A-3 inhibitor with an IC50 of 110 nM.
T11173 Elacestrant S enantiomer Elacestrant S enantiomer is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively.
T11173L Elacestrant S enantiomer dihydrochloride  Elacestrant (RAD1901) dihydrochloride is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ...
T11174 (R)-Elagolix Elagolix is a selective, highly potent, short-duration, orally-active, non-peptidethe gonadotropin-releasing hormone receptor (GnRHR) antagonist with KD of 54 p...
T11175 Elenbecestat Elenbecestat is an effective oral bioutilization and CNS penetrating ACE-1 inhibitor for the treatment of Alzheimer's disease.
T11176 Eliglustat hemitartrate Eliglustat Hemitartrate, with an IC50 of 24 nM, is a specific, potent, oral active glucocerebral glycosidase inhibitor.
T11178 ELN 318463 ELN 318463 shows differential inhibition of presenilin (PS1)- and PS2-comprised γ-secretase with EC50s of 12 nM and 656 nM for PS1 and PS2, respectively. ELN ...
T11178L ELN 318463 racemate ELN 318463 shows differential inhibition of presenilin (PS1)- and PS2-comprised γ-secretase with EC50s of 12nM and 656 nM for PS1and PS2, respectively. ELN3184...
T11180 Embramine Embramine, used as an antihistamine and anticholinergic, is a monoethanolamine.
T11182 EMD638683 S-Form  EMD638683 is a highly selective SGK1 inhibitor with IC50 of 3 μM. EMD638683 S-Form is the S-form of EMD638683.
T11184 EML4-​ALK kinase inhibitor 1 EML4-ALK kinase inhibitor 1 is a potent oral active inhibitor of echinoderm microtubule-associated protein-like 4-anaplastic lymphoma kinase (EML4-ALK), with an...
T11187 EMT inhibitor-2  EMT inhibitor-2 inhibits CYP3A4 testosteron and CYP2C9 with IC50s of 49.72 and 5.54 μM, respectively. EMT inhibitor-2  inhibits epithelial-mesenchymal tran...
T11188 Emixustat Emixustat, is an inhibitor of the visual cycle isomerase with an IC50 value of 4.4 nM in vitro. a novel visual cycle modulator.
T11188L Emixustat hydrochloride
T11191 EN6 EN6-mediated ATP6V1A modification decouples the v-ATPase from the Rags, leading to inhibition of mTORC1 signaling, increased lysosomal acidification and activat...
T11192 Enalapril D5 maleate Enalapril D5 maleate is deuterium labeled Enalapril, which is an angiotensin converting enzyme (ACE) inhibitor.
T11193 Enalaprilat D5 Sodium Salt Enalaprilat D5 Sodium Salt is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor.
T11194 Enalaprilat D5 Enalaprilat D5 is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor.
T11195 Enantiomer of Sofosbuvir Enantiomer of Sofosbuvir is an enantiomer of Sofosbuvir, a prescription medicine for the treatment of patients with chronic hepatitis C.
T11197 Enclomiphene D4 hydrochloride Enclomiphene D4 hydrochloride ((E)-Clomiphene D4 hydrochloride; trans-Clomiphene D4 hydrochloride; Enclomifene D4 hydrochloride)  is a potent and orally acti...
T11200 Endoxifen E-isomer (Z)-Endoxifen is an active metabolite generated via actions of CYP3A4/5 and CYP2D6, is a more potent selective estrogen receptor modulator (SERM) than Tamoxifen...
T11202 Enniatin complex  Enniatin complex inhibits enzymes like acyl-CoA: cholesterol acyl transferase and induces apoptosis in several cancer lines . Enniatin complex is a mixture o...
T11203 Enocyanin  Enocyanin shows inhibitory effect on the leucine aminopeptidase, acid phosphatase, γ-glutamyl transpeptidase and esterase activity. Enocyanin is an anthocya...
T11204 ENS-163 phosphate Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.
T11205 ent-Ezetimibe Ezetimibe is a Niemann-Pick C1-like1 (NPC1L1) inhibitor, and is a potent Nrf2 activator.ent-Ezetimibe (ent-SCH 58235) is the RRS-enantiomer of Ezetimibe. Ezetim...
T11207 Entacapone sodium salt Entacapone sodium salt inhibits catechol-O-methyltransferase(COMT) with similar IC50 in different tissues including live, duodenum, kidney and lung, but entacap...
T11208 Enzalutamide D3 Enzalutamide D3 is a deuterium labeled Enzalutamide . Enzalutamide is an androgen receptor (AR) antagonist with an IC50 of 36 nM in LNCaP prostate cells. 
T11212 EPAC 5376753 EPAC 5376753 has an inhibitory effect on Epac1 in Swiss 3T3 cells with IC50 of 4.EPAC 5376753 is an allosteric inhibitor of EPAC,
T11214 EPI-589  EPI-589 has the potential for the treatment of amyotrophic lateral sclerosis (ALS). EPI-589, a quinone derivative, is a safe and well tolerated oxidoreductas...
T11215 Episilvestrol Episilvestrol is a specific eIF4A-targeting translation inhibitor, with antitumor activity. Episilvestrol is a derivative of silvestrol, isolated from the fru...
T11218 ε-​Viniferin  ε-Viniferin possesses potent antioxidant capacity. ε-Viniferin, the dimer of Resveratrol and isolated from Vitis vinifera, displays a potent inhibitory for...
T11219 Equisetin Equisetin is a Quorum-sensing inhibitor (QSI) that attenuates QS-regulated virulence phenotypes in P. aeruginosa without affecting the growth of bacterias, serv...
T11220 ER21355 ER21355 used for treatment of prostatic diseases. ER21355 is an inhibitor of phosphodiesterase 5 (PDE5).
T11221 ERAP1-IN-1  ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates.ERAP1-IN-1 is an endoplasmic reticulum a...
T11223 Eriosematin Eriosematin has anti-proliferative and apoptosis-inducing properties and is a compound extracted from the root of Flemingia philippinensis in the Philippines.
T11227L Eravacycline dihydrochloride Eravacycline dihydrochloride  is a potent and broad-spectrum antibacterial agent. 
T11229 Erlotinib D6
T11232 Erysotrine Erysotrine, shows antibacterial activities,isolated from seed pods of Erythrina latissima.
T11235 Estradiol 3-sulfamate .Estradiol 3-sulfamate inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. Estradiol 3-sulfamate  is a potent, long-acting, and orally activ...
T11236 Estrogen receptor antagonist 1 Estrogen receptor antagonist 1 is a potent estrogen receptor (ER) antagonist.
T11237 Estrogen receptor antagonist 2 Estrogen receptor antagonist 2 is used for the study of breast cancer.Estrogen receptor antagonist 2 is a potent and orally active estrogen receptor (ER) antago...
T11239 Ethacizine hydrochloride Ethacizine hydrochloride  inhibits the depolarizing current responsible for the intraatrial and His-Purkinje-ventricular conduction. Ethacizine hydrochloride...
T11240 Ethacrynic acid D5  Ethacrynic acid also inhibits L-type voltage-dependent and store-operated calcium channel, leading to relaxation of airway smooth muscle (ASM) cells. Ethacry...
T11241 p38 MAPK-IN-2 p38 MAPK-IN-2 is an inhibitor of p38 kinase.
T11242 Ethyl glucuronide Ethyl glucuronide is an endogenous metabolite.
T11243 Ethyl tosylcarbamate Gliclazide is a whole-cell beta-cell ATP-sensitive potassium currents blocker with an IC50 of 184 nM. Ethyl tosylcarbamate is an intermediate in the synthesis ...
T11244 Etimizol Etimizol was shown to relieve amnesia effectively in the origin of which there is the hypoxic component (hypobaric hypoxia, actinomycin D, mechanical injury of...
T11245 Etiracetam Etiracetam  is an acetylcholine agonist and a nootropic drug of the racetam family. Less active than its S-enantiomer Levetiracetam. 
T11246 Etoricoxib D4 Etoricoxib D4 is a non steroidal anti-inflammatory agent, acting as a selective and orally active COX-2 inhibitor, with IC50s of 1.1 μM and 116 μM for COX-2 a...
T11247 Etravirine D4  Etravirine is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used for the treatment of HIV. Etravirine D4 is the deuterium labeled Etravirine.
T11249 Exatecan Exatecan can be used in cancer research.Exatecan is a DNA topoisomerase I inhibitor, with an IC50 of 2.2 μM (0.975 μg/mL)..
T11250 Ezetimibe D4 Ezetimibe D4  is the deuterium labeled Ezetimibe. Ezetimibe is a Niemann-Pick C1-like1 (NPC1L1) inhibitor, and is a potent Nrf2 activator. 
T11252 Ezetimibe phenoxy glucuronide-D4 Ezetimibe phenoxy glucuronide-D4 (Ezetimibe glucuronide-D4) is the deuterium labeled Ezetimibe phenoxy glucuronide.
T11253 Ezetimibe phenoxy glucuronide Ezetimibe phenoxy glucuronide (Ezetimibe glucuronide) is the active metabolite of Ezetimibe. Antihyperlipoproteinemic activity.
T11254 F-1  F-1 is IC50s of 2.1 nM, 2.3 nM, 1.3 nM and 3.9 nM for ALKWT, ROS1WT, ALKL1196M and ALKG1202R, respectively. F-1 is a potent ALK and ROS1 dual inhibitor, supp...
T11256 FAAH inhibitor 1 FAAH inhibitor 1 is a potent fatty acid amide hydrolase (FAAH) inhibitor with an IC50 of 18±8 nM.
T11259 FadD32 Inhibitor-1 FadD32 inhibitor -1 has anti-tuberculosis activity and is an effective FadD32 inhibitor.
T1126 Penicillin V potassium salt Penicillin V potassium is a broad-spectrum penicillin antibiotic used orally in the treatment of mild to moderate infections by susceptible gram-positive organi...
T11261 FAK inhibitor 5 FAK inhibitor 5 is a novel allosteric FAK inhibitor, with IC50 values in the low micromolar range. 
T11262 Falintolol, (Z)- Falintolol, (Z)-, a new β-adrenergic antagonist, is characterized by the presence of an oxime function. 
T11263 FAPI-2 Fapi-2 is a fibroblast activated protein (FAP) inhibitor used in cancer research.
T11264 FAPI-4 Api-4 is a fibroblast activated protein (FAP) inhibitor used in cancer research. 
T11265 Faropenem daloxate Antibacterial Faropenem daloxate is useful for penem and antibiotics. Faropenem medoxomil has excellent in vitro activity against Streptococcus pneumoniae, Hae...
T11266 FAS-IN-1 FAS-IN-1 is a potent inhibitor of Fatty acid synthase (FAS) wtih IC50 of 10 nM.
T11267 FASN-IN-1 FASN-IN-1 is a fatty acid synthase (FASN) inhibitor .
T11268 FD 12-9 FD 12-9, Anti-glioblastoma activity.  is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively. 
T11269 FD-IN-1 FD-IN-1  is a factor D (FD) inhibitor with an IC50  of 12 nM.FD-IN-1 also inhibits factor XIa (FXIa) and Tryptase β2 with IC50s of 7.7 and 6.5µM, respective...
T11270 Febuxostat D9 Febuxostat D9 is deuterium labeled Febuxostat, which is a selective xanthine oxidase inhibitor with Ki of 0.6 nM. 
T11271 Fenclozine Fenclozine is a non-steroidal antiinflammatory drug.
T11272 Fenmetozole Tosylate Fenmetozole Tosylate , acts as an antidepressant drug.  is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor, 
T11273 Fenpiverinium D3 bromide Fenpiverinium bromide has anti-cholinergic and anti-spasmodic effects.Fenpiverinium D3 bromide is a deuterium labeled Fenpiverinium bromide.
T11274 Ferulenol  Ferulenol shows good antimycobacterial activity and haemorrhagic action. Ferulenol, a sesquiterpene prenylated coumarin derivative, specifically inhibits suc...
T11275 Fesoterodine L-mandelate Fesoterodine L-mandelate is a efficacious antimuscarinic agent for the overactive bladder (OAB). 
T11276 Fexofenadine D6 Fexofenadine D6  is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.
T11278 FG8119 FG8119 is a novel benzodiazepine agonist.
T11281 FGI-106 FGI-106 is active against Ebola, Rift Valley and Dengue Fever viruses with EC50s of 100 nM, 800 nM and 400-900 nM, respectively. FGI-106 also inhibits non-hemo...
T11281L FGI-106 tetrahydrochloride  FGI-106 tetrahydrochloride is active against Ebola, Rift Valley and Dengue Fever viruses with EC50s of 100 nM, 800 nM and 400-900 nM, respectively. FGI-106 t...
T11282 FGTI-2734  FGTI-2734 can prevent membrane localization of KRAS, hence solving KRAS resistance problem and thwarting mutant KRAS patient-derived pancreatic tumors. FGTI-...
T11282L FGTI-2734 mesylate  FGTI-2734 mesylate can prevent membrane localization of KRAS, hence solving KRAS resistance problem and thwarting mutant KRAS patient-derived pancreatic tumor...
T11283 Fibracillin Fibracillin is a penicillin antibiotic.
T11284 FIDAS-3  FIDAS-3 effectively competes against S-adenosylmethionine (SAM) for MAT2A binding. FIDAS-3 has anticancer activities. FIDAS-3 is a stilbene derivative and i...
T11285 FIDAS-5  FIDAS-5 effectively competes against S-adenosylmethionine (SAM) for MAT2A binding. FIDAS-5 has anticancer activities. FIDAS-5 is a potent and orally active ...
T11287 Filipin complex Filipin interacts with membrane sterols causing the alteration of membrane structure. Filipin III is the major component of Filipin. Filipin, produced as a mi...
T11288 Filipin III  Filipin interacts with membrane sterols causing the alteration of membrane structure. Filipin III is the major component of Filipin, a 28-membered ring penta...
T11289 Finafloxacin  Finafloxacin exhibits optimal efficacy in slightly acidic environments (pH 5.0-6.0), under which other fluoroquinolones lose activity. Finafloxacin is highly...
T1129 Benfotiamine Benfotiamine is a synthetic S-acyl derivative of thiamine (vitamin B1), used as an antioxidant dietary supplement.
T11290 FK-448 Free base FK-448 Free base is an effective and specific inhibitor of chymotrypsin, with an IC50 of 720 nM. 
T11294 Flavanone hydrazone Flavanone hydrazine effectively inhibits lens protein-induced ocular inflammation.Flavanone hydrazine is a potent non-steroidal anti-inflammatory agent. 
T11295 Flibanserin D4 Flibanserin is a full agonist of the serotonin 5-HT1A receptor (Ki=1 nM) and an antagonist of 5-HT2A (49 nM). Flibanserin D4 is a deuterium labeled Flibanserin...
T11297 FF-10101 succinate FF-10101 succinate is a potent FLT3 inhibitor.
T11297L FF-10101 FF-10101 is a potent inhibitor of FLT3.
T11299 FLT3-IN-4 FLT3-IN-4 is a potent and orally effective Fms-like tyrosine receptor kinase 3 (FLT3; IC50=7 nM) inhibitor ,for treating acute myelogenous leukemia.
T11300 FLT3-IN-6 FLT3-IN-6 is a potent and selective inhibitor of FLT3-ITD (FLT3 mutation) with an IC50 of 1.336 nM. 
T11301 Flomoxef Flomoxef is an antibiotic in oxacephem group and has excellent activity against various gram-positive bacteria.
T11301L Flomoxef sodium Flomoxef sodium is a oxacephem group antibiotic, with excellent activity against various Gram-positive bacteria. 
T11303 Fluorobexarotene Fluorobexarotene possesses an apparent RXR binding affinity that is 75% greater than Bexarotene. Fluorobexarotene  is a potent retinoid-X-receptor (RXR) agoni...
T11304 Fluphenazine enanthate Fluphenazine enanthate is the first long-acting injectable (LAI) antipsychotic for the treatment of schizophrenia. 
T11305 Flurofamide Flurofamide is an effective bacterial urease inhibitor and has potential in the treatment of infected urinary calculi.
T11306 Fluvastatin D6 sodium  Fluvastatin sodium is a first fully synthetic, competitive HMG-CoA reductase inhibitor with an IC50 of 8 nM.Fluvastatin D6 sodium  is deuterium labeled Fluva...
T11307 Fluxametamide Fluxametamide is an insecticide with wide spectrum, acts as an antagonist of GABA- and glutamate-gated chloride channels, with IC50 of 1.95 nM and 225 nM for M....
T11310 FMK-MEA FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor. 
T11311 Foliglurax monohydrochloride Foliglurax monohydrochloride  Antiparkinsonian effect.  is a highly selective and potent, brain-penetrant metabotropic glutamate receptor 4 positive allosteri...
T11312 Formycin A  Formycin A shows antitumor and antiviral activities. Formycin A , a purine nucleoside antibiotic, is a potent human immunodeficiency virus type 1 (HIV-1) inh...
T11313 Forodesine hydrochloride Forodesine hydrochloride is a potent human lymphocyte proliferation inhibitor. Forodesine hydrochloride could induce apoptosis in leukemic cells by increasing t...
T11314 Fosmanogepix  Fosmanogepix (APX001) is an N-phosphonooxymethyl prodrug which is rapidly and completely metabolized by systemic alkaline phosphatases to the active moiety, A...
T11315 Fosmidomycin sodium salt Fosmidomycin sodium salt is active against both Gram-negative and Gram-positive bacteria. Fosmidomycin sodium salt is a phosphonic acid antibiotic and a antima...
T11316 FOY 251 free base FOY 251 free base acts as a proteinase inhibitor. FOY 251 free base is an anti-proteolytic active metabolite camostate.
T11317 FPA-124 FPA-124 interacts with both the pleckstrin homology (PH) and the kinase domains of Akt. FPA-124 induces apoptosis. FPA-124, a cell-permeable copper complex, i...
T11318 Dopexamine hydrochloride Dopexamine hydrochloride is a β2 adrenergic receptor agonist.
T11319 FR183998 free base FR183998 free base is a potent Na+/H+-exchange inhibitor, with IC50s of 0.3 nM, 3.1 nM and 6.5 nM by measurement of pHi change in rat lymphocytes, rat and human...
T11322 Fradafiban Fradafiban binds to the human platelet GP IIb/IIIa complex with a Kd value of 148 nM. Fradafiban is a non-polypeptide platelet glycoprotein IIb/IIIa antagonist.
T11323 Frakefamide TFA  Frakefamide is unable to penetrate the blood-brain-barrier and enter the central nervous system. Frakefamide TFA is a potent analgesic that acts as a periphe...
T11323L Frakefamide Frakefamide is a potent analgesic. It acts as a peripheral active μ-selective receptor agonist. Frakefamide is unable to penetrate the blood-brain-barrier and ...
T11325 Frondoside A possesses anticancer, anti-invasive, anti-metastasis, anti-angiogenic and pro-apoptosis properties with high safety.Frondoside A, a natural glycoside extracted ...
T11327L FR 167653 free base FR 167653 free base is an orally active p38 MAPK inhibitor and is effective in treating inflammation, relieving trauma, and ischemia-reperfusion injury in vivo....
T11330 FTI-2148 diTFA FTI-2148 diTFA is a RAS C-terminal mimetic dual farnesyl transferase (FT-1) and geranylgeranyl transferase-1 (GGT-1) inhibitor with IC50s of 1.4 nM and 1.7 μM,...
T11330L FTI-2148 FTI-2148 is an inhibitor of RAS C-terminal mimetic dual farnesyl transferase (FT-1) and geranylgeranyl transferase-1 (GGT-1)  (IC50s: 1.4 nM and 1.7 μM, re...
T11331 FTI 276 TFA FTI 276 TFA is effective against plasmodium falciparum and humans.It is a protein-based nikyltransferase (PFT) inhibitor with an IC50s of 0.9 nM and 0.5 nM, res...
T11331L FTI 276 FTI-276 is an inhibitor of protein farnesyltransferase (PFT) (IC50s: 0.9 and 0.5 nM for Plasmodium falciparum and human).
T11332 FUBP1–IN-1 FUBP1 - in-1, with an IC50 value of 11.0 M, is an effective FUSE binding protein 1 (FUBP1) inhibitor that can interfere with the binding of FUBP1 to its SINGLE-...
T11333 Fulvene-5  Fulvene-5 has antitumor activity.Fulvene-5 is a potent NADPH oxidase 4 (NOX4) inhibitor with antioxidant properties. Fulvene-5 is a reactive oxygen species (R...
T11334 Fulvestrant R enantiomer Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.
T11335 Fulvestrant S enantiomer Fulvestrant S enantiomer is the less active S enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.
T11336 Fumarate hydratase-IN-2 sodium salt Fumarate hydratase-IN-2 sodium salt is a cell-permeable and competitive fumarate hydratase inhibitor (Ki=4.5 μM) with nutrient-dependent cytotoxicity .
T11337 Fumarate hydratase-IN-1 Fumarate hydratase-IN-1 has antiproliferative activity against several cancer cell lines with a mean IC50 of 2.2 μM. Fumarate hydratase-IN-1 is a cell-permeab...
T11338 Furamidine Furamidine is also a selective and cell-permeable protein arginine methyltransferase 1 (PRMT1) inhibitor with an IC50 of 9.4 μM. Furamidine is selective for P...
T11339 Furegrelate sodium Furegrelate Sodium inhibits human platelet microsomal thromboxane A2 (TxA2) synthase with an IC50 of 15 nM. Furegrelate Sodium is being developed as an antiplat...
T1134 Clofoctol Clofoctol is a bacteriostatic antibiotic with activity against Gram-positive bacteria,used in the treatment of upper and lower respiratory tract infections.
T11341 FXIa-IN-1 FXIa-IN-1  is a potent β-lactam covalent heparin-derived factor XIa (fXIa) inhibitor. 
T11343 G0507 G0507 is a inhibitor of Escherichia coli growth and induces the extracytoplasmic σE stress response. G0507 acts as a chemical probe to dissect lipoprotein tra...
T11344 G150 G150 inhibited interferon expression triggered by DSDNA with IC50 of 10.2 nM.G150 is an effective and highly selective inhibitor of human cyclic GMP-AMP synthas...
T11346 G3-C12 G3-C12 shows anticancer activity. is a galectin-3 binding peptide, with Kd of 88 nM. 
T11347 G6PD activator AG1 G6PD activator AG1 is a glucose-6-phosphate dehydrogenase (G6PD) activator with an EC50 of 3 µΜ.
T11348 G907 G907 traps MsbA in an inward-facing, lipopolysaccharide-bound conformation by wedging into an architecturally conserved transmembrane pocket. Bactericidal acti...
T11349 GABAA receptor agent 1 GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.
T11351 Galanthamine N-Oxide Galanthamine N-Oxide inhibits electric eel acetylcholinesterase (AChE) with an EC50 of 26.2 μM. Galanthamine N-Oxide is a prominent inhibitor of substrate acc...
T11352 Galidesivir triphosphate Galidesivir triphosphate is a substrate for viral RNA-dependent RNA polymerase (RDRP), resulting in termination of viral RNA replication and thus serves as an a...
T11354 Gambogellic acid Gambogellic acid antitumor activity.  is an xanthone isolated from the processed gamboge.
T11358 gamma-secretase modulator 1 γ-secretase inhibitior-1 is useful for Alzheimer's disease. γ-secretase inhibitior-1 is a gamma-secretase modulator.
T11358L gamma-secretase modulator 1 hydrochloride gamma-secretase inhibitior-1 is a gamma-secretase modulator, γ-secretase inhibitior-1 is useful for Alzheimer's disease.
T11359 gamma-secretase modulator 2 gamma-secretase modulator 2 is a potent and selective γ-secretase modulator for treatment of Alzheimer's disease .γ-secretase modulator is modulation of the a...
T1136 Diastase Diastase is any one of a group of enzymes which catalyses the breakdown of starch into maltose.
T11360 gamma-secretase modulator 3 gamma-secretase modulator 3 is a gamma-secretase modulator.
T11361 γ-Secretase modulator 4 γ-Secretase modulator 4 is a potent γ-secretase modulator, reduces the Aβ42 level with IC50s of 0.017 μM and 0.014 μM in mouse and human, respectively. 
T11362 gamma-Secretase Modulators gamma-Secretase Modulators is useful for Alzheimer's disease. IC50 value: Target: γ-secretase modulator.gamma-Secretase Modulators (Amyloid-β production inhib...
T11363 Ganoderic acid F Ganoderic acid F exhibits antitumor and antimetastatic activities through inhibition of angiogenesis and alteration of proteins involving cell proliferation and...
T11364 Ganoderic acid TR Ganoderic acid TR is a broad-spectrum inhibitor against influenza neuraminidases (NAs), particularly H1N1 and H5N1 neuraminidases. The IC50 values of 4.6 and 1...
T11365 Ganodermanontriol Ganodermanontriol exhibits hepatoprotective activity. Ganodermanontriol, a sterol isolated from Ganoderma lucidum, induces anti-inflammatory activity in tert-b...
T11367 Gastrofensin AN 5 free base Gastrofensin AN 5 free base, is an antiulcer agent. a 4-phenyl-tetrahydroisoquinoline derivative.
T11368 GATA4-NKX2-5-IN-1  GATA4-NKX2-5-IN-1 exhibits no activity on the protein kinases involved in the regulation of GATA4 phosphorylation, and it modulates the hypertrophic agonist-i...
T11369 GB-110 GB-110 selectively induces PAR2-mediated intracellular Ca2+ release in HT29 cells with an EC50 of 0.28 μM. GB-110 is a potent, orally active, and nonpeptidic ...
T11369L GB-110 hydrochloride GB-110 hydrochloride selectively induces PAR2-mediated intracellular Ca2+ release in HT29 cells with an EC50 of 0.28 μM. GB-110 hydrochloride is a potent, ora...
T1137 Clorsulon Clorsulon is utilized for the treatment of Fasciola hepatica infections in calves and sheep.
T11370 GB-88 GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 µM. 
T11371 GBR 12783  GBR 12783 can improve memory performance and increase hippocampal acetylcholine release in rats. GBR 12783 is a specific, potent and selective dopamine uptak...
T11373 GCN2-IN-1 GCN2-IN-1 (A-92) is a potent general control nonderepressible 2 kinase (GCN2) inhibitor with an IC50 of 0.3-3 μM in the cell assay and an IC50 of <0.3 μM in t...
T11374 GCN2-IN-6 GCN2-IN-6 is also a eIF2α kinase PERK inhibitor with an IC50 of 0.26 nM (in enzymatic assay) and 230 nM (in cells). GCN2-IN-6  is a potent, and orally availa...
T11375 GCN2iB GCN2iB is an ATP-competitive inhibitor of a serine/threonine-protein kinase general control nonderepressible 2 (GCN2), with an IC50 of 2.4 nM. 
T11376 GC 14 GC 14 is a selective thyroid hormone receptor antagonist, with IC50 values of 200 nM and 35 nM for hTRα and hTRβ, respectively. 
T11377 GDC-0276
T11378 GDC-0834 S-enantiomer  GDC-0834 is a potent and selective BTK inhibitor.GDC-0834 (S-enantiomer) is the S-enantiomer of GDC-0834.
T11378L GDC-0834 Racemate GDC-0834 Racemate is the racemate form of GDC-0834, which is an effective and selective BTK inhibitor
T1138 Taurocholic acid sodium salt hydrate Taurocholic acid sodium salt hydrate is the product of conjugation of taurine with cholic acid. The sodium salt, the main ingredient of the bile of carnivorous ...
T11380 GDC-0927 GDC-0927 is a novel,non-steroidal,  potent, orally bioavailable, selective estrogen receptor antagonist. 
T11382 GDP-​α-D-​mannose disodium
T11384 Gefitinib D8 Gefitinib is an EGFR tyrosine kinase inhibitor, with IC50 of 2-37 nM in NR6wtEGFR cells. Gefitinib D8  is a deuterium labeled Gefitinib. 
T11385 Gefitinib N-oxide  Gefitinib is an EGFR tyrosine kinase inhibitor, with IC50 of 2-37 nM in NR6wtEGFR cells. Gefitinib N-oxide is the N-oxide derivative of Gefitinib.
T11386 Gemcabene calcium Gemcabene calcium , a first-in-class lipid-lowering agent, lowers low-density lipoprotein cholesterol (LDL-C), decreases triglycerides, and raises high-density ...
T11386L Gemcabene Gemcabene is a first-in-class lipid-lowering agent. It shows lowers low-density lipoprotein cholesterol (LDL-C) and decreases triglycerides. It also raises HDL-...
T11387 Gemfibrozil 1-O-β-glucuronide Gemfibrozil 1-O-β-Glucuronide, a metabolite of Gemfibrozil , is a potent and competitive P450 (CYP) isoform CYP2C8 inhibitor with an IC50 of 4.07 μM. 
T11388 Gemilukast Gemilukast is an orally active and potent dual cysteinyl leukotriene 1 and 2 receptors (CysLT1 and CysLT2) antagonist, with IC50s of 1.7, 25 nM for human CysLT1...
T11389 Genz-123346  Genz-123346 blocks the conversion of ceramide to glucosylceramide (GL1) and inhibits GM1 with an IC50 value of 14 nM. Genz-123346 is a potent, orally availab...
T11391 Gepotidacin S enantiomer Gepotidacin S enantiomer is an S enantionmer of gepotidacin.
T11391L Gepotidacin Gepotidacin is a novel triazaacenaphthylene inhibitor of bacterial type II topoisomerase.
T11393 GET73  GET73 significantly affects glutamate transmission in the hippocampus.GET73 is a γ-hydroxybutyric acid (GHB) analog, a naturally occurring neurotransmitter. ...
T11394 GFB-8438 GFB-8438 shows excellent selectivity against TRPC6, other TRP family members, NaV 1.5, as well as limited activity against the hERG channel. GFB-8438 protects m...
T11395 GF 15 GF 15 is a potent inhibitor of centrosomal clustering in tumor cells.
T11397 GGTI298 GGTI298 is a CAAZ peptidomimetic geranylgeranyltransferase I (GGTase I) inhibitor, strongly inhibiting the processing of geranylgeranylated Rap1A with little ef...
T11398 Ginsenoside Ra3 Ginsenoside Ra3, isolated from Panax ginseng, possesses anti-cancer activity. 
T11400 Gisadenafil besylate Gisadenafil besylate (UK 369003-26) is a specific, orally active phosphodiesterase 5 (PDE5) inhibitor ,prevents degradation of cyclic guanosine monophosphate (c...
T11401 GKA50  GKA50 stimulates insulin release from mouse islets of Langerhans and MIN6 cells. GKA50 shows significant glucose lowering in high fat fed female rats. GKA50 ...
T11402 GKI-1 GKI-1 robustly inhibits ROCK1 with an IC50 of 11 µM, but only weakly affected PKA. GKI-1 is a Greatwall (GWL) kinase inhibitor with IC50s of 4.9 and 2.5 µM a...
T11403 Gln-AMS Gln-AMS is an aminoacyl-tRNA synthetases (AARS) inhibitor, which binds the A-domain within the NRPS enzymes. 
T11403L Gln-AMS TFA  Gln-AMS(TFA) inhibits glutaminyl-tRNA synthetase (GlnRS) with a Ki of 1.32 µM. Gln-AMS (TFA) is a type Ia aminoacyl-tRNA synthetase (AARS) inhibitor.
T11404 GLP-1 receptor agonist 3 GLP-1 receptor agonist 3 is a GLP-1 receptor agonist,Example 4A-1, has EC50s of 1.1 nM and 13 nM in Clone H6 and Clone C6 cell lines assay, respectively.
T11405 GLP-1 receptor agonist 4 GLP-1 receptor agonist 4 is a glucagon-like peptide-1 receptor (GLP-1R) agonist , has an EC50 of 64.5 nM. GLP-1 receptor agonist 4 can be used in the research ...
T11406 TT-OAD2 free base TT-OAD2 free base has the potential for diabetes treatment. TT-OAD2 free base is a non-peptide glucagon-like peptide-1 (GLP-1) receptor agonist with an EC50 of...
T11407 GLP-1 receptor agonist 2 GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist.
T11409 GLP-26  GLP-26 disrupts the encapsidation of pre-genomic RNA, causes nucleocapsid disassembly and reduces cccDNA pools. GLP-26 is a HBV capsid assembly modulators (C...
T1141 Fenbendazole Fenbendazole is an antinematodal benzimidazole used in veterinary medicine.
T11410 GLPG0492 R enantiomer GLPG0492 R enantiomer is the R enantiomer of GLPG-0492, which is a novel selective androgen receptor modulator. 
T11410L GLPG0492 GLPG0492 is a novel selective androgen receptor modulator. After oral dosing, it showed anabolic activity on muscle, strongly dissociated from the androgenic ac...
T11411 GLPG1205 GLPG1205 is potent, selective and orally active GPR84 (a G-protein-coupled receptor) antagonist with a favorable PK/PD profile. GLPG1205 has anti-inflammatory ...
T11412 GLS1-IN-1 GLS1-IN-1 is used in the research of GLS1 mediated diseases, such as cancer.GLS1-IN-1 is a GLS1 (the kidney –type glutaminase) inhibitor.
T11413 Glucagon receptor antagonists-1 Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.
T11414 Glucagon receptor antagonists-2 Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist.
T11415 Glucagon receptor antagonists-3 Glucagon receptor antagonist -3 is a highly effective glucagon receptor antagonist.
T11416 Glucagon receptor antagonists-5 Glucagon receptor antagonists-5 has potential for the treatment of type 2 diabetes mellitus (T2DM).Glucagon receptor antagonists-5  is a potent and orally bioa...
T11417 Glucocorticoid receptor agonist Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.
T11418 Glucokise activator 1 Glucokinase activator 1 is a liver-directed glucokinase activator with an EC50 of 34 nM.
T11419 O6BTG-octylglucoside O6BTG-octylglucoside is a potent O6-methylguanine-DNAmethyl-transferase (MGMT) inhibitor, with IC50s of 10 nM in HeLa S3 cells and 32 nM in vitro (cell extract...
T11420 GLUT4 activator 1 GLUT4 activator 1  is a potent glucose transporter type 4 (GLUT4) translocation activator with an EC50 of 0.14 μM.
T11421 Glutamise-IN-1 Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity. Glutaminase-IN-1 , a CB839 derivative, is an allosteric inhibitor of...
T11422 Glutaminyl Cyclase Inhibitor 3 Glutaminyl Cyclase Inhibitor 3 significantly reduced the brain concentrations of pyroform Aβ and total Aβ and restored cognitive functions.Glutaminyl Cyclase ...
T11423 Glutaminyl Cyclase Inhibitor 4  Glutaminyl Cyclase Inhibitor 4 is a potent anti-Alzheimer’s agent. Glutaminyl Cyclase Inhibitor 4 is a potent, selective glutaminyl cyclase (QC) inhibitor ...
T11424 Glutaminyl Cyclase Inhibitor 1 Glutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor with an IC50 of 0.5 μM. 
T11425 Glutaminyl Cyclase Inhibitor 2 Glutaminyl Cyclase Inhibitor 2 is a glutaminyl cyclase inhibitor with an IC50 of 1.23 μM.
T11428 Glyco-Obeticholic acid Glyco-obeticholic acid is an active metabolite of Obeticholic acid. Obeticholic acid is a farnesoid X receptor (FXR) agonist. 
T11429 Glycolic acid oxidase inhibitor 1 Glycolic acid oxidase inhibitor 1 is a glycolate oxidase inhibitor.
T11430 Glycosidase-IN-1 Glycosidase-IN-1 be used to synthesize some immunosuppressive agents and β-glucosidase inhibitors. Glycosidase-IN-1 has hypoglycemic activity.Glycosidase-IN-1...
T11431 Glycosidase-IN-2  Glycosidase-IN-2 has hypoglycemic activity. Glycosidase-IN-2  is an azasugar class of glycosidase inhibitor.
T11432 Glyoxalase I inhibitor free base Glyoxalase I inhibitor (free base) , candidate for anticancer agents. Glyoxalase I inhibitor (free base) is a potent Glyoxalase I (GLO1) inhibitor.
T11433 Glyoxalase I inhibitor Glyoxalase I inhibitor is , candidate for anticancer agents.Glyoxalase I inhibitor is a potent Glyoxalase I inhibitor.
T11434 GlyRS-IN-1  GlyRS-IN-1 can inhibit the growth of bacteria. is a glycyl-tRNA synthase (GlyRS) inhibitor .
T11435 GlyT1 Inhibitor 1 GlyT1 Inhibitor 1,Antipsychotic activity.  is a potent and selective GlyT1 inhibitor with an IC50 of 38 nM for rGlyT1. 
T11437 GNE-0439  GNE-0439 inhibits mutant N1742K channels (IC50=0.37 uM) in membrane potential assays. GNE-0439 possesses a carboxylic acid group, binds outside of the channe...
T11438 GNE-1858 GNE-1858 is a potent and ATP-competitive hematopoietic progenitor kinase-1 (HPK1) inhibitor, with IC50s of 1.9 nM, 1.9 nM, and 4.5 nM for wild-type and the acti...
T11439 GNE-616 GNE-616 shows >1000 nM Kd and >2500-fold selectivity over hNav1.1, hNav1.3, hNav1.4, and hNav1.5. Selectivity over hNav1.2 and hNav1.6 is more modest at 31- an...
T11443 GNE 220 GNE-220 is a potent and selective inhibitor of MAP4K4 with an IC50 of 7 nM.
T11443L GNE 220 Hydrochloride GNE 220 is a potent and selective inhibitor of MAP4K4, with an IC50 of 7 nM. 
T11444 GNF-6231 GNF-6231 shows IC50s of greater than 10 μM on all CYP isoforms tested . GNF-6231 have favorable potency and a PK profile across preclinical species upon oral ...
T11445 GNF179 Metabolite GNF179 metabolite is the metabolite of GNF179, which is an optimized 8,8-dimethyl IP analog that exhibited the potency(4.8 nM against the multidrug resistant st...
T11446 GNF362 GNF362 also inhibits Itpka and Itpkc with IC50 values of 20 nM and 19 nM, respectively. Inositol trisphosphate 3’ kinase B (Itpkb) is a Ca2+-dependent kinase...
T11448 GOAT-IN-1 GOAT-IN-1 is an inhibitor of ghrelin O-acyltransferase (GOAT), which could be useful for the prophylaxis or treatment of obesity, diabetes, hyperlipidemia, meta...
T1145 Diminazene Aceturate Diminazene is a trypanocidal agent.
T11450 Gosogliptin Gosogliptin is a potent and selective inhibitor of dipeptidyl peptidase-IV (DPP-IV). 
T11451 GPI-1046 GPI-1046 is an analog of FK506, which is an immunophilin ligand that has been shown neuroprotective effects in neurodegenerative disease models. GPI-1046 readil...
T11453 GPR120 modulator 1 GPR120 modulator 1 is useful for modulating G protein-coupled receptor 120 (GPR120). 
T11454 GPR120 modulator 2 GPR120 modulator 2 regulates g-protein-coupled receptor 120 (GPR120).
T11455 GPR35 agonist 1 GPR35 agonist 1 showed good potency.It is a highly effective and specific G-protein-coupled receptor-35 (GPR35)/CXCR8 agonist with an EC50 of 5.8 nM.
T11456 GPR40 Activator 1 GPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes. 
T11457 GPR40 Activator 2 GPR40 Activator 2 is a potent GPR40 .
T11459 GPR40 agonist 1 GPR40 agonist 1 is an effective new GPR40 agonist with EC50 of 17 nM for rGPR40 and 2 nM for hGPR40.
T11461 NE 52-QQ57 NE 52-QQ57 has anti-inflammatory activity. NE 52-QQ57 is a selective, and orally available GPR4 antagonist with an IC50 of 70 nM. 
T11464 GRL0617 GRL0617 is a selective and competitive SARS-CoVPLpro and deubiquitinase noncovalent inhibitor(IC50 : 0.6 μM, Ki : 0.49 μM).
T11465 GS-6207 GS-6207 displays a mean EC50 of 50 pM (20-160 pM) against 23 HIV-1 clinical isolates from different subtypes in peripheral blood mononuclear cells (PBMCs). GS-6...
T11466 GSK-2793660 GSK-2793660 can be used for the reaearch of bronchiectasis. GSK-2793660 is an oral, irreversible inhibitor of Cathepsin C (CTSC). 
T11472 GSK 525768A GSK 525768A has no activity towards BET. GSK 525768A is the inactive enantiomer of GSK525762A.
T11473 GSK-5498A GSK-5498A is a selective small molecule blocker of CARC (IC50, 1 μM); pro-inflammatory cytokine release from T-cells in a variety of species , and inhibits me...
T11476 GSK-J2 GSK-J1 is a potent inhibitor of H3K27me3/me2-demethylases JMJD3/KDM6B and UTX/KDM6A. GSK-J2 is an isomer of GSK-J1 that does not have any specific activity. 
T11477 GSK1059865 GSK1059865 is a potent orexin 1 receptor antagonist.
T1148 Menbutone Menbutone is a derivative of oxobutyric acid, and is a choleretic. Menbutone shows a rapid onset of action, reaching its maximum plasma level within 1 hour and ...
T11480 GSK205 GSK205 is a potent, selective TRPV4 antagonist with an IC50 of 4.19  μM for inhibiting TRPV4-mediated Ca2+ influx. 
T11481 GSK2239633A GSK2239633A inhibits the binding of [125I]-TARC to human CCR4 with a pIC50 of 7.96 ± 0.11. GSK2239633A is a CC-chemokine receptor 4 (CCR4) antagonist.
T11482 GSK2245035 GSK2245035 has pEC50s of 9.3 and 6.5 for IFNα and TFNα. GSK2245035 effectively suppresses allergen-induced Th2 cytokine production in human peripheral blood c...
T11485 GSK2643943A GSK2643943A is a deubiquitylating enzyme (DUB) inhibitor, with an IC50 of 160 nM for USP20/Ub-Rho. 
T11488 GSK2850163 GSK2850163 is a novel inhibitor of inositol-requiring enzyme-1 alpha (IRE1α) which can inhibit  RNase activity and IRE1α kinase activity with IC50s of 200 an...
T11488L GSK2850163 hydrochloride GSK2850163 hydrochloride can inhibit IRE1α kinase activity and RNase activity with IC50s of 20 and 200 nM, respectively. GSK2850163 hydrochloride is a novel i...
T11489 GSK2850163 S entiomer GSK2850163 is an inositol-requiring enzyme-1 alpha (IRE1a) inhibitor. GSK2850163 S enantiomer is the inactive enantiomer of GSK2850163.
T11490 GSK2945
T11490L GSK2945 hydrochloride GSK2945 hydrochloride enhances cholesterol 7α-hydroxylase (CYP7A1) level and cholesterol metabolism. GSK2945 hydrochloride is a class of tertiary amine, and i...
T11492 GSK2983559 free acid GSK2983559 free acid has excellent activity in blocking many proinflammatory cytokine responses in vivo and in human inflammatory bowel disease explant samples....
T11493 GSK3004774 GSK3004774 shows an EC50 of 50 nM for human CaSR. GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and ...
T11494 GSK3532795 GSK3532795  is a potent, orally active, second-generation HIV-1 maturation inhibitor, with EC50s of 10.2, 1.9, 2.7 and 13 nM for HIV-1 WT(human serum), HIV-1 W...
T11495 GSK4028 GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe,in a time-resolved fluorescence resonance energy transf...
T11495L GSK 4027 GSK 4027 is a PCAF/GCN5 bromodomain chemical probe. In a time-resolved fluorescence resonance energy transfer (TR-FRET) assay, it has a pIC50 of 7.4±0.11 for P...
T11496 GSK598809 GSK598809 is a selective and potent dopamine D3 Receptor (DRD3) antagonist, with a pKi of 8.9.
T11497 GSK656 GSK656 acting as an inhibitor of Mycobacterium tuberculosis (Mtb) leucyl-tRNA synthetase (LeuRS), is a potent antitubercular agent, with an IC50 of 0.2 μM. 
T11498 GSK682753A GSK682753A is a selective and highly potent inverse agonist of the epstein-barr virus-induced receptor 2 (EBI2) with an IC50 of 53.6 nM. 
T11499 GSK726701A GSK726701A is a new type of prostaglandin E2 receptor 4 (EP4) partial agonist with a pEC50 of 7.4.
T11502 Epelsiban Epelsiban is a selective, potent and orally bioavailable oxytocin receptor antagonist, with a pKi of 9.9 for human oxytocin receptor.
T11504 GSTO-IN-2 GSTO-IN-2 is a glutathione S-transferase inhibitor with IC50s of 1.4, 16.3, and 3.6 μM for GSTP1-1, GSTM1, and GSTA2. 
T11505 GSTO1-IN-1 GSTO1-IN-1 is a potent glutathione S-transferase omega 1 (GSTO1) inhibitor with an IC50 of 31 nM.
T11506 Guaiapate Guaiapate is a cough suppressant.
T11507 Guancydine Guancydine  is an antihypertensive agent. 
T11508 Camicil Camicinal is a small molecule, selective motilin receptor agonist with pEC50 of 7.9.
T11508L Camicil hydrochloride Camicinal hydrochloride  is a small molecule, selective motilin receptor agonist with pEC50 of 7.9. 
T11509 Guanfu base H
T11510 Guanfu base I Guanfu base I has a potent anti-arrhythmic effect.Guanfu base I  is an active metabolite of Guanfu base A, isolated from Aconitum coreanum.
T11511 Guanosine-5'-triphosphate disodium salt Guanosine-5'-triphosphate disodium salt  is an activator of the signal transducing G proteins and also serves as an energy-rich precursor of mononucleotide uni...
T11512 Guanoxabenz Guanoxabenz is an α2 adrenergic receptor agonist. 
T11513 Gum arabic Gum Arabic is an anti-oxidant, and can protect against experimental hepatic-, renal- and cardiac toxicities. Gum Arabic also can be used in immunohistochemistr...
T11514 Gusperimus trihydrochloride Gusperimus trihydrochloride  is a derivative of the antitumor antibiotic spergualin with immunosuppressant activity. 
T11515 Gut restricted-7 Gut restricted-7 decreases gut bacterial BSHs and decreases deconjugated bile acid levels in feces of mice. Gut restricted-7 (GR-7) is a potent, covalent and o...
T11516 GV-196771A GV-196771A  is an NMDA receptor antagonist. and is the sodium salt form of GV196771.
T11517 GV-58 GV-58 is a potent, selective N- and P/Q-type Ca2+ channels agonist with EC50 of 7.21/8.81 uM for N-type/P-Q-type Ca2+ channel; 20-fold less potent CDK inhibitor...
T11519 GW768505A free base GW768505A free base has anti-angiogenic activity.GW768505A free base is a potent dual inhibitor of VEGFR2 (KDR) and Tie-2, with a pIC50 of 7.81 for VEGFR2. 
T11520 GW806742X GW806742X has activity against VEGFR2. GW806742X is a Mixed Lineage Kinase Domain-Like protein (MLKL) inhibitor which binds the MLKL pseudokinase domain with a...
T11522 GYKI 52466 dihydrochloride GYKI 52466 dihydrochloride is inactive against N-methyl-D-aspartate (NMDA) or γ-aminobutyric acid responses. GYKI 52466 dihydrochloride ia a muscle relaxant an...
T11524 H-89 H-89 has weak inhibition on PKG, PKC, Casein Kinase, and others kinases. H-89 is a potent and selective inhibitor of cyclic AMP-dependent protein kinase (prot...
T11525 GW311616 GW-311616 is a orally bioavailable,potent , long duration and selective human neutrophil elastase (HNE) inhibitor with IC50 value of 22 nM and Ki value of 0.31 ...
T11525L GW311616 hydrochloride GW-311616 is a potent, long duration,orally bioavailable and selective human neutrophil elastase (HNE) inhibitor with IC50 value of 22 nM and Ki value of 0.31 n...
T11526 DPP-IV-IN-2 DPP-IV-IN-2 is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (DPIV)  with IC50s of 0.1 and 0.95 μM, respectively.
T11527 H-Ser-His-OH H-Ser-His-OH, an endogenous metabolite,is a short peptide with hydrolysis cleavage activity.
T11528 H100 H100 is a Cl- transport inhibitor,  no effect against KCl cotransporter, in human erythrocytes.  with partial effects against both the NaK2Cl cotransporter a...
T11529 H3B-120 H3B-120 has anti-cancer activity. H3B-120 is a highly selective, competitive and allosteric carbamoyl phosphate synthetase 1 (CPS1) inhibitor with an IC50 of 1...
T11530 H3B-6545 Hydrochloride H3B-6545 Hydrochloride is an  selective, oral estrogen receptor covalent antagonist (SERCA). 
T11530L H3B-6545 H3B-6545 is an oral and selective antagonist of estrogen receptor covalent (SERCA).
T11533 HA155 HA-155 is a selective and potent autotaxin (ATX) inhibitor with an IC50 of 5.7 nM.
T11534 Haemanthamine Haemanthamine has pro-apoptotic, antioxidant, antiviral, antimalarial and anticonvulsant activities. Haemanthamine is a crinine-type alkaloid isolated from the...
T11534L Haemanthamine hydrochloride Haemanthamine hydrochloride targets ribosomal that inhibits protein biosynthesis during the elongation stage of translation. Haemanthamine hydrochloride has pro...
T11535 Haloperidol D4 Haloperidol D4 is deuterium labeled haloperidol.
T11536 Haloperidol D4' Haloperidol D4' is deuterium labeled haloperidol.
T11537 HAT-IN-1 HAT-IN-1 used in the research of cancer. is an inhibitor of HAT.
T11538 Hck-IN-1 Hck-IN-1 is a direct and wide HIV-1 Nef antagonists with an IC50 of 100-300 nM for wild-type HIV-1 replication. Hck-IN-1 binds pocket residue Asn126 and has ant...
T11539 HCV-IN-29 HCV-IN-29 is a hepatitis C virus (HCV) inhibitor .
T11540 HCV-IN-3 HCV-IN-3 is a hepatitis C virus (HCV) NS3/4a protein inhibitor, with an IC50 of 20 μM, a Kd of 29 μM.
T11541 HCV-IN-30 HCV-IN-30  is a HCV NS5A replication complex inhibitor, with IC50s of 901 and 102 nM for genotypes 1a and 1b replicons, respectively.
T11545 hDDAH-1-IN-2 hDDAH-1-IN-2 reveals an excellent profile regarding cell toxicity/viability. hDDAH-1-IN-2 is a selective, orally active human dimethylarginine dimethylaminohyd...
T11545L hDDAH-1-IN-2 sulfate hDDAH-1-IN-2 reveals an excellent profile regarding cell toxicity/viability. hDDAH-1-IN-2 is a selective, orally active human dimethylarginine dimethylaminohyd...
T11546 hDHODH-IN-1 hDHODH-IN-1 has anti-inflammatory effect. hDHODH-IN-1 is a human dihydroorotate dehydrogenase (hDHODH) inhibitor. 
T11547 hDHODH-IN-2 hDHODH-IN-1 has anti-inflammatory activity.hDHODH-IN-2 is an analogue of the active metabolite of Leflunomide. hDHODH-IN-2 is a human dihydroorotate dehydrogena...
T11548 HCV-IN-7 HCV-IN-7 shows a superior pan-genotypic profile and a good pharmacokinetic profile coupled with a favorable liver uptake. HCV-IN-7 has anti-viral activity. HCV...
T11548L HCV-IN-7 hydrochloride HCV-IN-7 hydrochloride shows a superior pan-genotypic profile and a good pharmacokinetic profile coupled with a favorable liver uptake. HCV-IN-7 hydrochloride h...
T11549 Helioxanthin 8-1 Helioxanthin 8-1 is an analogue of helioxanthin, exhibites significant in vitro anti-HBV/HCV/HSV-1/HIV activity with EC50 of >5/10/1.4/15 uM. IC50 value: >5/10/...
T11550 Helioxanthin derivative 5-4-2 Helioxanthin derivative 5-4-2 is an analogue of helioxanthin, exhibites significant in vitro anti-HBV activity with EC50 of 0.08 uM in HepG2.2.15 cells. Anti-H...
T11551 Helvolic acid Helvolic acid  is an antibiotic isolated from Xylaria sp, active against the Gram-positive bacteria. 
T11552 hDDAH-1-IN-1 hDDAH-1-IN-1 TFA potently inhibits hDDAH-1 (Ki = 18 µM) without significantly affecting NOSs and arginase.
T11552L hDDAH-1-IN-1 TFA hDDAH-1-IN-1 TFA  is a potent and selective non-amino acid catalytic site inhibitor of human dimethylarginine dimethylaminohydrolase-1 (hDDAH-1), with a Ki of ...
T11553L Heptamidine Heptamidine is a useful tool for the investigation of Myotonic dystrophy (DM). Heptamidine is an effective Pentamidine-related inhibitor of the calcium-binding ...
T11555 Heptasaccharide Glc4Xyl3 Heptasaccharide Glc4Xyl3, is used for the identification and analysis of diverse xyloglucan-active enzymes in nature.  a covalent inhibitor of endo-xyloglucan...
T11556 HET0016 HET0016 also is a selective CYP450 inhibitor, which has been shown to inhibit angiogenesis and tumor growth. HET0016 is a potent and selective 20-hydroxyeicosa...
T11557 FASN-IN-3 FASN-IN-3 is a fatty acid synthase (FASN) inhibitor.
T11558 Hexyl gallate Hexylgallate , a alkyl ester derivative of gallic acid, exhibits potent antimalarial activity against Plasmodium falciparum, with IC50 of 0.11 mM. 
T11559 HG-12-6 HG-12-6 can modulate IRAK4 activity in autoimmunity and inflammation. HG-12-6 is a type II inhibitor of IRAK4. HG-12-6 shows preferential binding to unphospho...
T11564 HIV-1 inhibitor-3 HIV-1 inhibitor-3 is a HIV infection inhibitor.
T11565 HIV-1 integrase inhibitor 7 HIV-1 integrase inhibitor 7 is a potent HIV-1 integrase inhibitor, with an IC50 of 33.3 nM.
T11566 HIV-1 integrase inhibitor Hiv-1 integrase inhibitor is an effective anti-HIV drug.
T11567 HIV-1 integrase inhibitor 3 HIV-1 integrase inhibitor 3 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 2.7 nM. 
T11568 HIV-1 integrase inhibitor 4 HIV-1 integrase inhibitor 4 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 3.7 nM. 
T11573 HPN-01 HPN-01 displays greater 50-fold selectivity over a panel of more than 50 other kinases, including ALK5, CDK-2, EGFR, ErbB2, GSK3β, PLK1, Src, and VEGFR-2. HPN...
T11574 HS79 HS-79 is able to inhibit the incorporation of tritiated acetate into lipids with an IC50 of 1.57 μM. HS-79 is an enantiomer of Fasnall, which is a selective f...
T11575 HS80 HS-80 is able to inhibit the incorporation of tritiated acetate into lipids with an IC50 of 7.13 μM. HS-80 is an enantiomer of Fasnall, which is a selective f...
T11576 HSL-IN-1 HSL-IN-1, a significantly reduced reactive metabolite liability. is a potent and orally active hormone sensitive lipase (HSL) inhibitor (IC50=2 nM).
T11577 HSL-IN-2 HSL-IN-2 is a selective  and potent inhibitor of Hormone Sensitive Lipase (HSL), with an IC50 of 0.023 μM. 
T11578L Encequidar mesylate Encequidar mesylate  is a competitive and potent P-glycoprotein inhibitor. 
T11579 HSL-IN-3 HSL-IN-3 , a boronic acid ester derivative, is an inhibitor of hormone-sensitive lipase (HSL).
T11580 HO-1-IN-1 HO-1-IN-1  is a heme oxygenase 1 (HO-1) inhibitor with an IC50 of 250 nM. 
T11580L HO-1-IN-1 hydrochloride HO-1-IN-1 hydrochloride  is a heme oxygenase 1 (HO-1) inhibitor with an IC50 of 250 nM. 
T11581 HSR6071 HSR6071 is an antiallergic agent with potential for the treatment of asthma.
T11582 HSV-TK substrate HSV-TK substrate shows antitumor activity.HSV-TK substrate is a substrate for HSV-TK, and induces multi-log cytotoxicity in HSV-TK-expressing and bystander cell...
T11583 HWL-088 HWL-088 significantly improves glucose tolerance in normal and diabetic models. HWL-088  is a highly potent free fatty acid receptor 1 (FFA1/GPR40) agonist be...
T11584 Hydroxy desmethyl Bosentan Hydroxy desmethyl Bosentan (Ro 64-105) is a Bosentan metabolism produced by the cytochrome P450 enzymes CYP2C9 and CYP3A4 in the liver.
T11585 Hydroxy Itracozole D8 Hydroxy Itraconazole is an active metabolite of Itraconazole (ITZ), which is a triazole antifungal agent. Hydroxy Itraconazole D8 is the deuterium labeled Hydr...
T11586 Hydroxy ziprasidone Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a combined 5-HT (serotonin) and dopamine receptor antagonist. 
T11587 Hydroxylammonium chloride Hydroxylammonium chloride is the hydrochloric acid salt of hydroxylamine, which is a biological intermediate in the anammox and in the nitrification.
T11588 Hydroxybupropion Hydroxybupropion inhibits norepinephrine uptake with an IC50 value of 1.7 μM. Hydroxybupropion is also a nACh receptor antagonis tis more potent than Bupropion...
T1159 Leflunomide Leflunomide is an immunomodulatory agent used in the therapy of rheumatoid arthritis and psoriatic arthritis.
T11590 (-)-Hydroxycitric acid (-)-Hydroxycitric acid is a potent and competitive inhibitor of ATP citrate lyase. (-)-Hydroxycitric acid suppresses the fatty acid synthesis, lipogenesis, food...
T11591 Hydroxyzine D4 Hydroxyzine D4 is deuterium labeled Hydroxyzine. Hydroxyzine has anticholinergic, anxiolytic and analgesic properties. Hydroxyzine is a heterocyclic histamine...
T11592 Hydroxyzine D8 Hydroxyzine D8 is deuterium labeled Hydroxyzine. Hydroxyzine is a histamine H1-receptor antagonist. 
T11593 I-OMe-Tyrphostin AG 538  I-OMe-Tyrphostin AG 538 inhibits IGF-1R-mediated signaling and is preferentially cytotoxic to nutrient-deprived PANC1 cells. I-OMe-Tyrphostin AG 538 is an ATP...
T11594 I2906 I2906 showed antimycobacterial and cytotoxic activity against mycobacterium tuberculosis. IC50 Value: Target: Antibacterial Under in vitro conditions, I2906 sh...
T11595 IACS-8779 IACS-8779 with robust systemic antitumor efficacy. is a highly potent stimulator of interferon genes (STING) agonist.
T11596 IACS-8803 IACS-8803 is a highly potent cyclic dinucleotide STING agonist with robust systemic antitumor efficacy. 
T1160 Fusidine Fusidine is an antibiotic isolated from the fermentation broth of Fusidium coccineum.
T11601 Ibrutinib D5 Ibrutinib D5  is a deuterium labeled Ibrutinib. Ibrutinib is a selective, irreversible Btk inhibitor. 
T11602 Ibrutinib dimer Ibrutinib dimer is an impurity of Ibrutinib. IIbrutinib dimer is a Dimer of Ibrutinib. brutinib is a selective, irreversible Btk inhibitor with an IC50 of 0.5 n...
T11603 Ibrutinib-MPEA Ibrutinib-MPEA  is ibrutinib derivative. Ibrutinib is a covalent and irreversible inhibitor of Bruton's tyrosine kinase (BTK) that has been used to treat haem...
T11604 Ibuprofen D3 Ibuprofen D3 is a deuterium labeled Ibuprofen. Ibuprofen is a COX-1 and COX-2 inhibitor with IC50s of 13 μM and 370 μM. 
T11606 ICA-105665  ICA-105665 inhibits liver mitochondrial function and bile salt export protein (BSEP) transport (IC50 of 311 μM). ICA-105665 can penetrate the blood-brain bar...
T11608 Epanolol Epanolol is a potent β-adrenoceptor partial agonist with a greater affinity for β1- than β2-adrenoceptors.
T11609 ICI 153110 ICI 153110 is designed for the treatment of congestive cardiac failure. ICI 153110 is an orally active phosphodiesterase inhibitor with both vasodilating and i...
T1161 Protionamide Protionamide is a thioamide derivative with antitubercular activity.
T11612 IDH1 Inhibitor 3 IDH1 Inhibitor 3  with an IC50 of 45 nM for IDH1R132H.  is a mutant isocitric dehydrogenase 1 (IDH1) inhibitor.
T11613 IDH1 Inhibitor 1 IDH1 Inhibitor 1 Anticancer activity.  is a potent, orally bioavailable, brain-penetrant and selective mutant IDH1 inhibitor with IC50s of 0.021 μM, 0.045 μ...
T11616 IDO-IN-13 IDO-IN-13 is a potent indoleamine 2,3-dioxygenase 1 (IDO1) inhibitor with an EC50 of 17 nM.
T11618 IDO-IN-4 IDO-IN-4 is an indoleamine 2,3-dioxygenase 1 (IDO-1) inhibitor.
T1162 Acipimox Acipimox is a niacin derivative and nicotinic acid analog with activity as a hypolipidemic agent. Acipimox has special application for the treatment of hyperlip...
T11623 IDO/TDO-IN-1 IDO/TDO-IN-1  is a highly potent and orally active dual indoleamine-2,3-dioxygenase (IDO) and tryptophan 2,3-dioxygenase (TDO) inhibitor with IC50s of 9.7 and ...
T11625 IDO1 and HDAC1 Inhibitor IDO1 and HDAC1 Inhibitor  is a dual IDO1 and HDAC1 inhibitor with IC50s of 69.0 nM and 66.5 nM, respectively. 
T11629 Ifenprodil glucuronide Ifenprodil is a vasodilator and an inhibitor of platelet aggregation, and Ifenprodil glucuronide has no effect on platelet aggregation and arterial contraction....
T11630 IFN alpha-IFR-IN-1 hydrochloride IFN alpha-IFNAR interaction inhibitor IFN alpha-IFNAR-IN-1 specifically inhibits MVA-induced IFN-α responses by BM-pDCs. IFN alpha-IFNAR-IN-1 inhibited the IFN...
T11630L IFN alpha-IFR-IN-1 IFN alpha-IFNAR-IN-1 is a nonpeptidic, low-molecular-weight inhibitor of the interaction between IFN-α and IFNAR. It inhibit MVA-induced IFN-α responses by BM...
T11637 Iloperidone metabolite Hydroxy Iloperidone Iloperidone metabolite Hydroxy Iloperidone is an atypical antipsychotic. Iloperidone metabolite Hydroxy Iloperidone is a metabolite of Iloperidone.
T11639 Imatinib D4 Imatinib D4  is a deuterium labeled Imatinib. Imatinib is an orally bioavailable tyrosine kinases inhibitor that selectively inhibits BCR/ABL, v-Abl, PDGFR and...
T11640 Imatinib D8 Imatinib is an orally bioavailable tyrosine kinases inhibitor that selectively inhibits BCR/ABL, v-Abl, PDGFR and c-kit kinase activity. Imatinib D8  is a deu...
T11641 N-Desmethyl imatinib N-Desmethyl imatinib  is a metabolite of Imatinib, which is a multi-target inhibitor of v-Abl, c-Kit and PDGFR. 
T11643 Impurity B of Calcitriol Impurity B of Calcitriol, Calcitriol is the hormonally active form of vitamin D, Calcitriol(1,25-Dihydroxyvitamin D3; Rocaltrol ) inhibits in vivo and in vitro ...
T11644 Impurity C of Alfacalcidol Impurity of Alfacalcidol. Alfacalcidol (1-hydroxycholecalciferol; Alpha D3; 1.alpha.-Hydroxyvitamin D3) is a non-selective VDR activator medication. 
T11645 Impurity C of Calcitriol Impurity C of Calcitriol, Calcitriol (1,25-Dihydroxyvitamin D3; Rocaltrol )exhibits antitumor activity; Calcitriol(1,25-Dihydroxyvitamin D3; Rocaltrol ) inhi...
T11646 Impurity F of Calcipotriol Impurity F of Calcipotriol; Calcipotriol (MC 903; Calcipotriene) exhibits antiproliferative activity against human HL-60, HL60/MX2, MCF-7, T47D, SCC-25 and mous...
T11647 INCB 3284 dimesylate  INCB 3284 dimesylate can be used in the research of acute liver failure. INCB 3284 dimesylate is a potent, selective and orally bioavailable human CCR2 antag...
T11648 INCB 3284 INCB 3284 can be used in the research of acute liver failure. INCB 3284 is a potent, selective and orally bioavailable human CCR2 antagonist, inhibiting monocyt...
T11649 INCB054329 Racemate INCB054329 Racemate is an inhibitor of BET protein.
T11650 INCB3344 R-isomer INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.
T11652 Indirubin-3'-monoxime-5-sulphonic acid Indirubin-3'-monoxime-5-sulphonic acid is a potent and selective inhibitor of GSK-3β, CDK5, and CDK1 with IC50s of 80nM,5 nM, and 7 nM, respectively.
T11653 Indirubin-5-sulfonate Indirubin-5-sulfonate shows inhibitory activity against GSK-3β. Indirubin-5-sulfonate is a cyclin-dependent kinase (CDK) inhibitor, with IC50 values of 55 nM, ...
T11654 Indirubin Derivative E804 Indirubin Derivative E804 is an effective inhibitor of IGF1R, which has an IC50 value of 0.65.
T11657 INH154 INH154 is a highly potent inhibitor for Nek2 and Hec1 binding (INH), with IC50s of 120 nM and 200 nM for INH in MB468 and Hela cells.
T11658 INO5042 INO5042 is an anti-inflammatory agent.
T11659 Inogatran Inogatran is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of venous and arterial thrombotic diseases.
T11661 INT-767 INT-767 is a dual farnesoid X receptor (FXR)/TGR5 agonist with mean EC50s of 30 and 630 nM, respectively.
T11662 INT-777 R-enantiomer INT-777 is the R-enantiomer of INT-777, less potent than INT-777,EC50 of 4.79 μM for TGR5.
T11663 Integrin-IN-2 Integrin-IN-2 is an orally bioavailable pan αv integrin inhibitor.Integrin-IN-2 can increases the αvβ6, αvβ3, αvβ5 and αvβ8 binding affinities with pIC...
T11664 INY-03-041 INY-03-041 inhibits AKT1, AKT2 and AKT3 with IC50s of 2.0 nM, 6.8 nM and 3.5 nM, respectively. INY-03-041 is a potent, highly selective and PROTAC-based pan-AKT...
T11665 Ionomycin calcium lonomycin calcium is a potent, selective calcium ionophore and an antibiotic produced by Streptomyces conglobatus. also induces the activation of protein kinase...
T11667 Ipragliflozin L-Proline Ipragliflozin is a highly potent and selective SGLT2 inhibitor with an IC50 of 2.8 nM; little and NO potency for SGLT1/3/4/5/6.
T11668 IQB-782 IQB-782 shows a potent mucolytic-expectorant activity. IQB-782 is a cysteine derivative. IQB-782 has inhibition for thrombin activatable fibrinolysis inhibitor ...
T11669 IR415 IR415 selectively interacts with HBx (Kd=2 nM) and blocks HBV-mediated RNAi suppression, reverses the inhibitory effect of HBx protein on the activity of the di...
T11670 IRAK inhibitor 3 IRAK inhibitor 3 is an interleukin-1 (IL-I) receptor-associated kinase (IRAK) kinase modulator.
T11672 IRAK inhibitor 4 IRAK inhibitor 4 is an interleukin-1 receptor associated kinase 4 inhibitor.
T11673 IRAK4-IN-4 IRAK4-IN-4 inhibits cyclic GMP-AMP synthase (cGAS) with an IC50 of 2.1 nM.IRAK4-IN-4 is an interleukin-1 receptor–associated kinase 4 (IRAK4) inhibitor, has a...
T11674 IRAK4-IN-6 IRAK4-IN-6 ,targetes MyD88 L265P mutant diffuse large B cell lymphoma. is an orally efficacious and selective IRAK4 inhibitor with an IC50 of 4 nM.
T11675 Irbesartan D4 Irbesartan D4 is a highly potent and specific angiotensin II type 1 (AT1) receptor antagonist. is the deuterium labeled Irbesartan.
T11676 Iriflophenone 3-C-glucoside Iriflophenone 3-C-β-D-glucopyranoside,has antioxidant activity,isolated from Cyclopia genistoides.
T11677 Irindalone Irindalone is a novel serotonin 5-HT2 antagonist.
T11678 Iristectorin B Iristectorin B has anti-cancer activities in breast cancer.is an isoflavone from Iris tectorum.
T11679 Isavuconazole D4 Isavuconazole D4 is a deuterium labeled Isavuconazole. Isavuconazole is a triazole prodrug with antifungal activity against yeasts, molds, and dimorphic fungi.
T11680 Isoasatone A Isoasatone A is a natural product isolated from the plant Heterotropa takaoi M., with anti-insect activity.
T11681 Isochondrodendrine Isochondodendrine has strong antiplasmodial activity against Plasmodium falciparum. Isochondrodendrine is a class of bisbenzylisoquinoline alkaloid isolated fro...
T11682 Isofistularin-3 Isofistularin-3, as a DNA demethylating agent, induces cell cycle arrest and sensitization to TRAIL in cancer cells. Isofistularin-3 can be used as an ADC cytot...
T11683 Isoglycycoumarin Isoglycycoumarin is a highly selective probe for human cytochrome P450 2A6.Isoglycycoumarin is a flavonoid isolated from the roots of Glycyrrhiza uralensis.
T11684 Isoguvacine hydrochloride Isoguvacine hydrochloride is a GABA receptor agonist.
T11685 Isolongifolene Isolongifolene has antioxidant, anti-inflammatory, anticancer and neuroprotective properties. Isolongifolene is a tricyclic sesquiterpene isolated from Murraya ...
T11688 ITI214 free base ITI-214 is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and i...
T11689 ITI214 ITI-214 is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and i...
T1169 Moguisteine Moguisteine is a new-type peripheral non-narcotic antitussive drug.
T11691 IV-23 IV-23 inhibits cell growths in vitro and in vivo, reduces colony formation, arrests cell cycle at M phase, and induces esophageal squamous cell carcinoma . IV-2...
T11692 Ivabradine D3 Hydrochloride Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D3 Hydrochloride is the deuterium ...
T11693 IT1t IT1t inhibits CXCL12/CXCR4 interaction with an IC50 of 2.1 nM. is a potent CXCR4 antagonist.
T11693L IT1t dihydrochloride IT1t dihydrochloride inhibits CXCL12/CXCR4 interaction with an IC50 of 2.1 nM. is a potent CXCR4 antagonist.
T11694 Ivabradine D6 hydrochloride Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D6 hydrochloride is the deuterium ...
T11695 Ivabradine metabolite N-Demethyl Ivabradine hydrochloride N-Demethyl Ivabradine Hcl is a specific inhibitor of the funny channel.N-Demethyl Ivabradine Hcl is a metabolite of Ivabradine.
T11696 Ivachtin Ivachtin is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor with an IC50 of 23 nM.
T11697 IX 207-887 IX 207-887 inhibits the release of interleukin-1 (IL-1). IX 207-887 is a novel antiarthritic agent.
T11698 IZCZ-3 IZCZ-3,antitumor activity. is a potent c-MYC transcription inhibitor.
T11699 J-113863 J-113863 is also a potent antagonist of the human CCR3 (IC50 of 0.58 nM) , but a weak antagonist of the mouse CCR3 (IC50 of 460 nM). J-113863 is inactive agains...
T11700 J-2156 The ED50 of J-2156 in rats for the relief of mechanical allodynia and mechanical hyperalgesia in the ipsilateral hindpaws was 3.7 and 8.0 mg/kg, respectively. J...
T11702 J30-8 J30-8 exhibits neuroprotective activity in vitro and potential for the treatment of neurodegenerative diseases. J30-8 is a potent and isoform-selective inhibito...
T11703 JAK-IN-1 JAK-IN-1 shows improved selectivity for JAK3 over JAK1. JAK-IN-1 is a JAK1/2/3 inhibitor with IC50s of 0.26, 0.8 and 3.2 nM, respectively.
T11705 JAK-IN-4 JAK-IN-4 is a prodrug of a JAK inhibitor, effective in murine collagen induced arthritis model.
T11715 JH-LPH-28 JH-LPH-28 displays outstanding antibiotic activity with a MIC value of 0.83 μg/mL. JH-LPH-28, a sulfonyl piperazine analog, is a potent UDP-2,3-diacylglucosami...
T11716 JH-LPH-33 JH-LPH-33 displays outstanding antibiotic activity with a MIC value of 0.66 μg/mL. JH-LPH-33, a sulfonyl piperazine analog, is a potent UDP-2,3-diacylglucosami...
T11718 JI051 JI051,Anti-cancer activity. is a stabilizer for the Hes1-PHB2 interaction, interacts with a cancer-associated protein chaperone prohibitin 2 (PHB2), induces ce...
T11719 JMV 2959 hydrochloride JMV 2959 hydrochloride is a growth hormone secretagogue receptor type 1a (GHS-R1a) antagonist with an IC50 of 32±3 nM in LLC-PK1 cells.
T11719L JMV 2959 JMV 2959 is an antagonist of growth hormone secretagogue receptor type 1a (GHS-R1a) (IC50: 32 nM).
T1172 Diclazuril Diclazuril is a coccidiostat.
T11720 JNJ-18038683 JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.
T11722 JNJ-37822681 dihydrochloride JNJ-37822681 has potential for the treatment of schizophrenia and bipolar disorder.JNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-di...
T11724 JNJ-42226314 JNJ-42226314 demonstrates dose-dependent enhancement of the major endocannabinoid 2-arachidonoylglycerol (2-AG) as well as efficacy in models of neuropathic and...
T11725 JNJ-47117096 hydrochloride JNJ-47117096 hydrochloride is potent and selective MELK inhibitor, with an IC50 of 23 nM, also effectively inhibits Flt3, with an IC50 of 18 nM.
T11726 JP1302 dihydrochloride JP1302 dihydrochloride is a selective, high affinity antagonist of the alpha2C-adrenoceptor (α2C-adrenoceptor), with a Kb value (antagonist activity) of 16 nM ...
T11730 JTT 551 JTT 551 can be used in the research of type 2 diabetes mellitus. JTT 551 is selective a protein tyrosine phosphatase 1B (PTP1B) inhibitor, with Kis of 0.22 μM ...
T11733 K-604 dihydrochloride K-604 dihydrochloride is a potent and selective acyl-CoA:cholesterol acyltransferase 1 inhibitor with an IC50 of 0.45±0.06 μM.
T11736 K-Ras G12C-IN-2 K-Ras G12C-IN-2 is a covalent kras g12c inhibitor.
T11737 K-Ras G12C-IN-3 K-ras G12C inhibitor For more information, please see the following patent. Heterocyclic compounds as covalent inhibitors of G12C mutant K-Ras protein useful fo...
T11738 K-Ras G12C-IN-4 K-Ras G12C-IN-4, is a potent Covalent Inhibitor of KRASG12C..
T11739 K145 K145 is inactive against SphK1 and other protein kinases. K145 induces cell apoptosis and has potently antitumor activity. K145 is a selective, substrate-compet...
T11740 Delcasertib Delcasertib is a potent and selective δ-protein kinase C (δPKC) inhibitor.
T11741 KAN0438757 KAN0438757 is a selective and potent inhibitor of the metabolic kinase PFKFB3 with an IC50 of 0.19 μM.
T11745 KB SRC 4 KB SRC 4 has antitumor activity. KB SRC 4 is a potent, and highly selective c-Src inhibitor, with a Ki of 44 nM and a Kd of 86 nM, and shows no inhibition on c-...
T11746 KCC2 blocker 1 KCC2 blocker 1 is a benzyl prolinate and has antiepileptic effect.KCC2 blocker 1 is an orally active and selective K+-Cl- cotransporter KCC2 blocker with an IC5...
T11748 KDM2A/7A-IN-1 KDM2A/7A-IN-1 is a first-in-class, selective and cell-permeable inhibitor of histone lysine demethylases KDM2A/7A, with an IC50 of 0.16 μM for KDM2A.
T11750 KDOAM-25 citrate KDOAM-25 citrate increases global H3K4 methylation at transcriptional start sites and impairs proliferation in multiple myeloma MM1S cells. KDOAM-25 citrate is ...
T11750L KDOAM-25 trihydrochloride KDOAM-25 trihydrochloride increases global H3K4 methylation at transcriptional start sites and impairs proliferation in multiple myeloma MM1S cells. KDOAM-25 tr...
T11758L KI696 KI696 is an effective and selective inhibitor of KEAP1/NRF2 interaction. KI696 is a high-affinity probe that disrupts the Keap1/NRF2 interaction.
T11759 Kif15-IN-2 Kif15-IN-2 is used for the research of cellular proliferative diseases. Kif15-IN-2 is an inhibitor of the mitotic kinesin Kif15.
T11760 KIN101 KIN101, an isoflavone agonist of IRF-3 dependent signaling, induces IRF-3 nuclear translocation. KIN101 has broad-spectrum activity against RNA viruses. KIN101 ...
T11762L Kira8 Kira8 is a mono-selective IRE1α inhibitor. That allosterically attenuates IRE1α RNase activity (IC50: 5.9 nM).
T11763 Ko-3290 Ko-3290 is an antagonist of β-adrenoceptor, with cardioselectivity and antilipolytic effects in animals.
T11764 KP496 KP496 is a selective, dual antagonist for Thromboxane A2 receptor and Leukotriene D4 receptor. 
T11766 Eltanexor Z-isomer Eltanexor Z-isomer exhibits different inhibitory effects on Z138, MM15, 3T3 cell lines, with IC50s of 100 nM-50 μM, < 100 nM, > 30 μM, respectively.Eltanexor ...
T11766L Eltanexor Eltanexor inhibits XPO1-dependent nuclear export (EC50=60.9 nM) by directly targeting XPO1. Eltanexor causes caspase-dependent apoptosis in a panel of leukemic ...
T11772 KRAS inhibitor-4 KRAS inhibitor-4 developed as anticancer agents, is a potent KRAS inhibitor.
T11781 KRN2 KRN2 has potential to treat NFAT5-mediated Chronic Arthritis. KRN2 is a selective inhibitor of nuclear factor of activated T cells (NFAT5), with an IC50 of 100...
T11782 KRN2 bromide KRN2 bromide is a selective inhibitor of nuclear factor of activated T cells , with an IC50 of 0.1 μM. 
T11784 KT182 KT182 is a selective and  potent inhibitor of α/β-hydrolase domain containing 6 (ABHD6), with an IC50 of 0.24 nM in Neuro2A cells. 
T11785 KT203 KT203 is a potent and selective inhibitor of α/β-hydrolase domain containing 6 (ABHD6), with an IC50 of 0.31 nM in Neuro2A cells.
T11787 Kv3 modulator 1 Kv3 modulator 1 has the potential for inflammatory pain treatment. Kv3 modulator 1 is a Kv3 voltage-gated potassium channel modulator extracted from patent WO2...
T11788 Kv3 modulator 2 Kv3 modulator 2  is a potent Kv3 channels modulator.has analgesic activity and is used in the prophylaxis or treatment of related disorders. 
T11789 Kv3 modulator 3 Kv3 modulator 3  is a selective modulator of Kv3.1 and/or Kv3.2 and/or Kv3.3 channels .has analgesic activity for use in the prophylaxis o or treatment of pain...
T11790 Kv3 modulator 4 Kv3 modulator 4 is a Kv3.1 (pEC50=5.45) and Kv3.2 modulator .Cyclobutyl structure. 
T11791 KW-6055 KW-6055 has anti-amnesic activity, is a benzylpyridine derivative.
T11792 KW-8232 free base KW-8232 free base can reduces the biosynthesis of PGE2, is an anti-osteoporotic agent.
T11794 L-368,899 hydrochloride L-368,899 hydrochloride, used as a tocolytic agent, is a potent, selective, orally bioavailable, non-peptide oxytocin receptor antagonist, with IC50s of 8.9 nM ...
T11795 L-4-Oxalysine hydrochloride L-4-Oxalysine hydrochloride has shown antitumor activities, is a natural product isolated from the culture media of Streptomyces roseovirdofuscus in China.
T11796 L-45 dihydrochloride L-45 dihydrochloride is the first selective, potent, and cell-active p300/CBP-associated factor (PCAF) bromodomain (Brd) inhibitor with a Kd of 126±15 nM. 
T11796L L-45 L-45 is the first potent and cell-active bromodomain (Brd) inhibitor of p300/CBP-associated factor (PCAF) (Kd: 126±15 nM).
T11797 L-690488 L-690488 has more effective cell penetration than L-690330. L-690488 is a prodrug of L-690330 and is a selective inositol monophosphatase (IMPase) inhibitor.
T11798 L-692429 L-692429 binds to G protein-coupled receptor with a Ki of 63 nM. L-692429  is a benzolactam derivative and a nonpeptidyl growth hormone secretagogue (GHS) ago...
T11800 L-803087 L-803087 facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice.L-803087 is a potent and selective som...
T11801 l-Atabrine dihydrochloride l-Atabrine dihydrochloride displays antiprion activity. l-Atabrine dihydrochloride is a less active enantiomer of quinacrine.
T11802 L-Canaline L-Canaline inhibits the growth of the malaria parasite Plasmodium falciparum with an IC50 of 297 nM. L-Canaline has anticancer and antiproliferative effects. L...
T11803 L-Cysteinesulfinic acid L-Cysteinesulfinic acid is a potent agonist at several rat metabotropic glutamate receptors (mGluRs, pEC50s of 3.92±0.03, 4.6±0.2, 3.9±0.2, 2.7±0.2, 4.0±0....
T11804 β3-AR agonist 2 β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM). 
T11805 L-NIL L-NIL is a potent and selective inhibitor of inducible NO synthase with IC50s of 92 and 3.3 μM for rat brain constitutive NO synthase and mouse inducible NO sy...
T11807 L002 L002 binds the acetyl-CoA pocket and competitively inhibits the FATp300 catalytic domain, blocks histone acetylation and p53 acetylation, and inhibits STAT3 act...
T11810 L791943 L791943 is a selective, potent) inhibitor of Phosphodiesterase-4 (PDE4,IC50 of 4.2 nM). 
T11811 Laetanine Laetanine, exhibits antiplasmodial activity, a noraporphine alkaloid from Litsea laeta.
T11812 L-Eflornithine L-Eflornithine is an irreversible ornithine decarboxylase (ODC) inhibitor with a KD of 1.3±0.3 µM, and a Kinact of 0.15±0.03 min-1. L-Eflornithine is an ena...
T11812L L-Eflornithine monohydrochloride L-Eflornithine is an irreversible ornithine decarboxylase (ODC) inhibitor with a KD of 1.3±0.3 µM, and a Kinact of 0.15±0.03 min-1. L-Eflornithine monohydroc...
T11813 Laflunimus Laflunimus suppresses immunoglobulin (Ig) secretion, with IC50 values of 2.5 and 2 µM for IgM and IgG, respectively. Laflunimus also is a prostaglandin endope...
T11814 Lamivudine 13C,15N2 Lamivudine 13C,15N2 is a labelled impurity of Lamivudine (BCH-189). Lamivudine can inhibit HIV reverse transcriptase 1/2 and the reverse transcriptase of hepat...
T11815 Lanopepden Lanopepden is a peptide deformylase inhibitor active against Staphylococcus aureus strains with MICs of 1 and 1 mg/L for ATCC 29213 and ATCC 25923 strain, respe...
T11819 Lascufloxacin Lascufloxacin has the potential for various infectious diseases treatment, including lower respiratory tract infections.Lascufloxacin  is a potent and orally a...
T11820 LAT1-IN-1 LAT1-IN-1 (BCH)  significantly inhibit cellular uptake of amino acids and mTOR phosphorylation, which induces the suppression of cancer growth and apoptosis. ...
T11821 Latanoprost lactone diol Latanoprost lactone diol is an intermediate in the synthesis of Latanoprost. Latanoprost is a prostaglandin F2α analogue and an agonist for the FP prostanoid r...
T11822 LAU159 LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM). 
T11825 LCB-2853 LCB-2853 with antiplatelet and antithrombotic activities, is an antagonist of thromboxane A2 (TXA2) receptor.
T11827 Pradigastat Pradigastat has anti-obesity and anti-diabetic effects. Pradigastat is a potent, selective and orally active diacylglycerol acyltransferase 1 (DGAT1) inhibitor...
T11828 LDC7559 LDC7559 via blocking neutrophil extracellular trap (NET) in the late stages . Implement inhibition gasdermin D (GSDMD).
T11830 LDN-192960 hydrochloride LDN-192960 hydrochloride is an inhibitor of  Dual-specificity Tyrosine-regulated Kinase 2 (DYRK2) and Haspin with IC50s of 48 nM and 10 nM, respectively. 
T11831 LDN-27219 LDN-27219 is a potent hTGase inhibitor with IC50 of 0.6 uM.
T11832 Ledipasvir D-tartrate Ledipasvir D-tartrate with EC50 values of 34 pM against GT1a and 4 pM against GT1b replicon. is an inhibitor of the hepatitis C virus NS5A.
T11833 Ledipasvir (diacetone) Ledipasvir is an inhibitor of the hepatitis C virus NS5A, with EC50 values of 34 pM against GT1a and 4 pM against GT1b replicon.Ledipasvir diacetone (GS-5885 di...
T11834 Leelamine hydrochloride Leelamine hydrochloride suppresses transcriptional activity of androgen receptor, which is known to regulate fatty acid synthesis[2,3].Leelamine hydrochloride i...
T11835 LCL521 LCL521 also inhibits the lysosomal acid sphingomyelinase (ASMase). LCL521 is an acid ceramidase (ACDase) inhibitor. 
T11835L LCL521 dihydrochloride LCL521 dihydrochloride is an acid ceramidase (ACDase) inhibitor. LCL521 also inhibits the lysosomal acid sphingomyelinase (ASMase). 
T11836 Lefamulin acetate Lefamulin acetate (BC-3781 acetate) is the first semi-synthetic pleuromutilin for systemic treatment of bacterial infections in humans. Lefamulin acetate (BC-37...
T11838 LEQ506 LEQ506 is a second-generation smoothened (Smo) inhibitor with IC50s of 4 and 2 nM in mouse and human, respectively. 
T11840 Leu-AMS Leu-AMS shows cytotoxicity in cancer cells and normal cells, and inhibits the growth of bacteria.Leu-AMS , a leucine analogue, is a potent inhibitor of leucyl-t...
T11841 Leu-AMS R enantiomer Leu-AMS R enantiomer is the R enatiomer of Leu-AMS. Leu-AMS is a potent inhibitor of leucyl-tRNA synthetase (LRS) and inhibits the growth of bacteria. 
T11842 Levomecol Levomecol (Chloramphenicol)) stops bacterial growth by binding to the bacterial ribosome (blocking peptidyl transferase) and inhibiting protein synthesis. Levo...
T11843 Levothyroxine acyl glucuronide Levothyroxine acyl glucuronide (Thyroxine Acyl-β-D-glucuronide), the acyl glucuronide formation of thyroxine (T4), an endogenous metabolite.
T11844 LG-100064 LG-100064 can be used in the research of cancer. LG-100064 is a retinoid-X-receptor (RXR) agonist, with EC50s of 330 nM, 200 nM, and 260 nM for RXRα, RXRβ an...
T11845 LGD-6972 LGD-6972 is an antagonist of glucagon receptor.
T11847 Liarozole dihydrochloride Liarozole dihydrochloride is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase)...
T11848 Licorice glycoside C2 Licorice glycoside C2 is a oleanane-type triterpene oligoglycoside isolated from Glycyrrhiza uralensis. 
T11849 Lignin Lignin is the main component of plant cell walls and is a renewable aromatic polymer. Lignin has strongly antioxidant activity.Lignin (Lignine) is a natural com...
T11851 Lin28-let-7a antagonist 1 Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction,and shows a clear antagonistic effect against the Lin28-let-7a interaction...
T11852 Liclotide Linaclotide developed for the treatment of constipation-predominant irritable bowel syndrome (IBS-C) and chronic constipation, and is a potent and selective gu...
T11853 Linezolid D3 Linezolid D3 is a deuterium labeled Linezolid. Linezolid is a synthetic antibiotic that acts by inhibiting the initiation of bacterial protein synthesis. 
T11854 Lipofermata Lipofermata is a fatty acid transporter protein (FATP) inhibitor that prevents lipid transport to melanoma cells and reduces melanoma growth and invasion.
T11855 Lipopolysaccharides Lipopolysaccharide is a highly immunogenic antigen which can enhance immune responses.Lipopolysaccharides is an endotoxin derived from the outer leaflet of the ...
T11856 LIT-001 free base LIT-001 free base improves social interaction in a mouse model of autism. LIT-001 free base is the first nonpeptide oxytocin receptor (OT-R) agonist (EC50=55 n...
T11857 LIT-001 LIT-001 improves social interaction in a mouse model of autism.LIT-001 is the first nonpeptide oxytocin receptor (OT-R) agonist (EC50=55 nM; Ki=226 nM).
T11858 Lith-O-Asp Lith-O-Asp is a sialytransferase (ST) inhibitor,(IC50s:12-37 μM).
T11859 Litronesib Racemate Litronesib is a selective, allosteric inhibitor of kinesin Eg5.Litronesib (Racemate) is the racemate of litronesib.
T11860 LM-1484 LM-1484 displays a higher affinity for 3H-LTC4 sites and is an antagonist of CysLT1 receptor.
T11861 LM11A-31 dihydrochloride LM11A-31 dihydrochloride is a water-soluble, non-peptide with high blood-brain barrier permeability.LM11A-31 dihydrochloride, a p75NTR (neurotrophin receptor p7...
T11862 LMD-009 LMD-009 mediates chemotaxis, inositol phosphate accumulation, and calcium release in high potencies with EC50s from 11 to 87 nM. LMD-009 is a selective CCR8 no...
T11864 LNP023 LNP023 shows direct, reversible, and high-affinity binding to human FB (KD=7.9 nM).LNP023 is a highly potent factor B (FB) inhibitor with an IC50 value of 10 nM...
T11865 Lodelaben Lodelaben is a human neutrophil elastase inhibitor with an IC50 and Ki of 0.5 and 1.5 μM, respectively. 
T11866 LolCDE-IN-2 LolCDE-IN-2 inhibits E. coli MG1655 with a MIC of 2 μg/ml. Antibacterial activity. LolCDE-IN-2 is a potent Lol protein inhibitor. 
T11867 Loperamide D6 hydrochloride Loperamide D6 hydrochloride is a deuterium labeled Loperamide hydrochloride. Loperamide hydrochloride is an opioid receptor agonist for the treatment of diarrh...
T11869 Losartan (D4 Carboxylic Acid) Losartan D4 Carboxylic Acid is the deuterium labeled Losartan, which is an angiotensin II receptor antagonist. 
T1187 Bifonazole Bifonazole acts to destabilize the fungal cytochrome p450 51 enzyme (also known as Lanosterol 14-alpha-demethylase). It works by inhibiting the production of a ...
T11870 Losartan D4 Losartan D4 is the deuterium labeled Losartan. Losartan is an angiotensin II receptor antagonist, competing with the binding of angiotensin II to AT1 receptors...
T11871 Loteprednol Etabote D5 Loteprednol Etabonate D5 is a deuterium labeled Loteprednol etabonate.Loteprednol etabonate (LE) exhibits anti-inflammatory activity and has been used in optome...
T11872 LMP744 LMP744 is a DNA intercalator and Topoisomerase I (Top1) inhibitor with antitumor activity. 
T11872L LMP744 hydrochloride LMP744 hydrochloride is a DNA intercalator and Topoisomerase I (Top1) inhibitor with antitumor activity. 
T11874 Lp-PLA2-IN-3 Lp-PLA2-IN-3 is a potent and orally bioavailable lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor, with an IC50 of 14 nM for recombinant human Lp-PLA...
T11876 LpxH-IN-AZ1 LpxH-IN-AZ1 is a potent inhibitor of Klebsiella pneumoniae LpxH with IC50 of 0.36 μM . LpxH-IN-AZ1, a sulfonyl piperazine compound, is a potent UDP-2,3-diacyl...
T11877 LR-90 LR-90 is also used in the research of diabetic animal model.LR-90 is an advanced glycation end product (AGE) inhibitor, inhibits inflammatory responses in human...
T11879 LS-102 LS-102 inhibits the autoubiquitination of synoviolin with an IC50 of 35 μM. LS-102 has the potential for rheumatoid arthritis treatment. LS-102 is a selective...
T11882 LSD1-IN-7 benzenesulfote LSD1-IN-7 benzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
T11883 LSD1-IN-7 Methylbenzenesulfote LSD1-IN-7 Methylbenzenesulfonate is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activity.
T11884 LSN 3213128 LSN 3213128, anti-tumor activity.  is a selective, nonclassical, orally bioavailable antifolate with potent and specific inhibitory activity for aminoimidazol...
T11885 LSP-249 LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell. 
T11886 LTβR-IN-1 LTβR-IN-1 is potent in TWEAK-stimulated p52 translocation assays with an IC50 of 10 μM and did not alter TNF-α–induced p65 nuclear translocation. LTβR-IN...
T11888 LtaS-IN-1 LtaS-IN-1 alone inhibits Enterococcus.spp 28 strains with varying MIC values ranging from 0.5 μg/mL to 64 μg/mL. LtaS-IN-1 combination with antibiotics aboli...
T11889 LTV-1 LTV-1 has the potential for autoimmunity treatment. LTV-1 is a potent lymphoid tyrosine phosphatase (LYP) inhibitor in T cells with an IC50 of 508 nM. 
T11890 Ludaconitine Ludaconitine, isolated from Aconitum spicatum (Bruhl) Stapf, exhibits antileishmanial activity with an IC50 of 36.10 μg/mL. 
T11891 Lumefantrine D18 Lumefantrine D18 is an antimalarial drug, and is the deuterium labeled Lumefantrine.
T11892 Lurasidone D8 Hydrochloride Lurasidone D8 Hydrochloride  is an inhibitor of Dopamine D2, 5-HT2A, 5-HT7, 5-HT1A and noradrenaline α2C, and is the deuterium labeled Lurasidone.
T11893 Lurasidone metabolite 14326 Lurasidone metabolite 14326 is an active metabolite of the atypical antipsychotic Lurasidone. 
T11893L Lurasidone metabolite 14326 hydrochloride Lurasidone metabolite 14326 is an active metabolite of the atypical antipsychotic Lurasidone. 
T11895 Luteolin-7-rutinoside Luteolin-7-rutinoside has both antifungal activities and anti-arthritic, can result in a combination therapy for the treatment of fungal arthritis due to C. al...
T11897 Telotristat ethyl Telotristat ethyl (LX1606) is a orally-delivered, novel inhibitor of tryptophan hydroxylase that reduces serotonin production. 
T11899 LXRβ agonist-2 LXRβ agonist-2 is a highly potent and β-selective liver X receptor (LXRβ) agonist with EC50 of 7 nM.
T11902 LY 344864 S-entiomer LY 344864 S-enantiomer is the S-enantiomer of LY344864. LY344864 is a 5-HT1F receptor agonist. 
T11903 LY-411575 isomer 1 LY-411575 isomer 1 is a potent γ-secretase inhibitor. LY-411575 isomer 1 is an isomer of LY411575.
T11904 LY-411575 isomer 2 LY-411575 isomer 2 is a potent γ-secretase inhibitor. LY-411575 isomer 2 is an isomer of LY411575.
T11905 LY-411575 isomer 3 LY-411575 isomer 3 is a potent γ-secretase inhibitor. LY-411575 isomer 3 is an isomer of LY411575.
T11908 LY2365109 hydrochloride LY2365109 hydrochloride is a potent and selective GlyT1 inhibitor, with an IC50 of 15.8 nM for glycine uptake in cells over-expressing hGlyT1a.
T11909 LY2444296 LY2444296 exhibits anti-anxiety like effects. LY2444296 is an orally bioavailable, high-affinity and selective short-acting kappa opioid receptor (KOPR) antago...
T11910 LY285434 LY285434 is a suitable angiotensin II receptor antagonist.
T11912 LY3154207 LY3154207 is a subtype selective, potent, and orally available human dopamine D1 receptor positive allosteric modulator (PAM) with minimal allosteric agonist ac...
T11913 LY88074 Methyl ether LY88074 Methyl ether is useful for the inhibition of the various estrogen deficient conditions, which are associated with estrogendeprivation syndrome including...
T11914 LY88074 Trimethyl ether LY88074 Trimethyl ether is useful for the inhibition of the various estrogen deficient conditions, which are associated with estrogen deprivation syndrome inclu...
T11915 LY88074 Raloxifene is a selective estrogen receptor modulator, and reduces fracture risk at least in part by improving the mechanical properties of bone in a cell- and ...
T11917 Lys-SMCC-DM1 DM1 is a tubulin inhibitor. Lys-SMCC-DM1 is the active metabolite of DM1. 
T11918 Lysipressin Lysipressin, Induces contraction of the rabbit urinary bladder smooth muscle, activate adenylate-cyclase. Lysipressin is Antidiuretic hormone that have been f...
T11919 LysRs-IN-1 LysRs-IN-1 is a Lysyl-tRNA synthetase (LysRs) inhibitor. 
T1192 Protoporphyrin IX Protoporphyrin IX is a tetrapyrrole containing 4 methyl, 2 propionic and 2 vinyl side chains that is a metabolic precursor for hemes, cytochrome c, and chloroph...
T11920 LysRs-IN-2 LysRs-IN-2 is a lysyl-tRNA synthetase (KRS) inhibitor with IC50s of 0.13 μM and 0.015 μM for Cryptosporidium parvum lysyl-tRNA synthetase (CpKRS) and Plasmod...
T11922 LY 254155 LY 254155, an antifolate,binds to mFBP and inhibits hGARFT with Kis of 1.7±0.1 and 2.1±0.2 nM, respectively.
T11923 Methyl-3β-hydroxycholete Methyl-3β-hydroxycholenate is a ROR gamma modulator.
T11925 M‑89 M-89 inhibits the menin-mixed lineage leukemia (Menin-MLL) protein-protein interaction and has potential to treat MLL leukemia. M-89 is a highly potent and spe...
T11926 m-Nifedipine m-Nifedipine is an impurity of Nifedipine. Nifedipine is a potent calcium channel blocker and drug of choice for cardiac insufficiencies.
T11927 M2 ion channel blocker M2 ion channel blocker ,Antiviral agent, is capable of inhibiting and blocking the activity of M2 ion channel.
T11929 M2N12 M2N12 also has promising activity against Cdc25A and Cdc25B with IC50 values of  0.53  μM and 1.39 μM. Anti-tumor activity. M2N12 is a potent and highly ...
T11930 M8891 M8891 is an orally active, reversible and brain penetrant Methionine Aminopeptidase-2 (MetAP-2) inhibitor(IC50 :54nM;Ki:4.33 nM).M8891 inhibits growth of primar...
T11933 MAC13772 MAC13772 is a novel antibacterial compound.MAC13772 is a potent inhibitor of the enzyme BioA (IC50=250 nM), the antepenultimate step in biotin biosynthesis. 
T11934 Macitentan D4 Macitentan D4 (ACT-064992 D4) is a deuterium labeled Sulfamethoxazole. Macitentan has the potential for idiopathic pulmonary fibrosis (IPF) and pulmonary arteri...
T11935 Macitentan (n-butyl alogue) Macitentan n-butyl analogue is a n-butyl analogue of Macitentan. Macitentan is an orally active, non-peptide dual antagonist of endothelin ETA and ETB receptor ...
T11936 Macropa-NCS Macropa-NCS is conjugated to trastuzumab as well as to the prostate-specific membrane antigen-targeting compound RPS-070.
T11937 m-Tyramine m-Tyramine has effects on the adrenergic and dopaminergic receptor.m-Tyramine is an endogenous trace amine neuromodulator.
T11937L m-Tyramine hydrobromide m-Tyramine hydrobromide has effects on the adrenergic and dopaminergic receptor. m-Tyramine hydrobromide is an endogenous trace amine neuromodulator.
T11938 Macropa-NH2 hydrochloride Macropa-NCS is conjugated to Anti-Human HER2 as well as to the prostate-specific membrane antigen-targeting compound RPS-070 and is a promising therapeutic radi...
T11940 Malic enzyme inhibitor ME1 Malic enzyme inhibitor ME1 is a potent inhibitor of Malic enzyme (ME1,IC50: 0.15μM). 
T11941 Manitimus Manitimus is a potent immunosuppressive drug, and is an inhibitor of dehydroorotate dehydrogenase,.
T11942 MAP4K4-IN-3 MAP4K4 may be a viable target for antidiabetic agents, a serine/threonine protein kinase.
T11943 MAPK13-IN-1 MPAK13-IN-1 is a MAPK13 (p38δ) inhibitor(IC50: 620 nM). 
T11945 MARK-IN-1 MARK-IN-1 is a potent microtubule affinity regulating kinase (MARK) inhibitor, (IC50<0.25 nM). 
T11946 MARK-IN-2 MARK-IN-2 is a potent microtubule affinity regulating kinase (MARK) inhibitor,(IC50:5 nM). 
T11947 MARK4 inhibitor 1 MARK4 inhibitor 1 inhibits cancer cell proliferation, metastasis and induces apoptosis. MARK4 inhibitor 1 is a potent microtubule affinity-regulating kinase 4 ...
T11950 MAT2A inhibitor 2 MAT2A inhibitor 2 is a methionine adenosyltransferase 2A (MAT2A) inhibitor. 
T11951 Mavoglurant racemate Mavoglurant is a novel, non-competitive mGlu5 receptor antagonist. Mavoglurant (racemate) is the racemate of mavoglurant. 
T11951L Mavoglurant Mavoglurant is a structurally novel, non-competitive mGlu5 receptor antagonist. It has an IC50 of 30 nM in a functional assay with human mGluR5.
T11952 Maxacalcitol-D6 Maxacalcitol-D6 is a non-calcemic vitamin D3 analog and VDR ligand of VDR-like receptors.Maxacalcitol-D6 is the deuterated form of Maxacalcitol (22-Oxacalcitrio...
T11954 MB-07344 MB-07344 has additive cholesterol lowering activity in combination with Atorvastatin in rabbits, dogs and monkeys. MB-07344 is a potent thyroid hormone recepto...
T11954L MB-07344 sodium MB-07344 sodium has additive cholesterol lowering activity in combination with Atorvastatin in rabbits, dogs and monkeys. MB-07344 sodium is a potent thyroid h...
T11955 MB-07729 MB-07729 is a potent fructose 1,6-bisphosphatase (FBPase) noncompetitive inhibitor with IC50 values of 189, 121, and 31 nM for rat, monkey and human, respective...
T11956 MBC-11 triethylamine MBC-11 triethylamine has potential to treat tumor-induced bone disease (TIBD), is a first-in-class conjugate of the bone-targeting bisphosphonate etidronate cov...
T11956L MBC-11 MBC-11 is a first-in-class conjugate of the bone-targeting bisphosphonate etidronate covalently linked to the antimetabolite cytarabine (araC). It also has the ...
T11957 MBC-11 trisodium MBC-11 trisodium has potential to treat tumor-induced bone disease (TIBD).It is a first-in-class conjugate of the bone-targeting bisphosphonate HEDP covalently ...
T11962 MC3482 MC3482 is a specific inhibitor of sirtuin5 (SIRT5).
T11963 MCB-3681 MCB-3681, active against gram-positive bacterium, is the antibacterial Oxaquin's active substance.
T11965 MCHR1 antagonist 3 MCHR1 antagonist 3 is used to regulate energy metabolism. MCHR1 antagonist 3 is a potent the melanin-concentrating hormone receptor-1 (MCHR1) antagonist. 
T11966 MCHR1 antagonist 2 MCHR1 antagonist 2 also inhibits hERG, with an IC50 of 4.0 nM in IMR-32 cells. MCHR1 antagonist 2 is an antagonist of melanin concentrating hormone receptor 1,...
T11967 Mcl-1 antagonist 1 Mcl-1 antagonist 1 is a Mcl-1 protein antagonist.
T11969 MCL-1/BCL-2-IN-2 MCL-1/BCL-2-IN-2 is a potent and selective Bcl-2 and Mcl-1 dual inhibitor. 
T11970 MCL-1/BCL-2-IN-3 MCL-1/BCL-2-IN-3 is a selective and potent Mcl-1 and Bcl-2 dual inhibitor with IC50s of 5.95 and 4.78 μM, respectiely. 
T11971 MCL-1/BCL-2-IN-4 MCL-1/BCL-2-IN-4 is a selective and potent Mcl-1 and Bcl-2 dual inhibitor.
T11976 Mcl1-IN-4 Mcl1-IN-4 is an inhibitor of Mcl1 ( IC50:0.2 μM).
T11978 McN3716 McN3716 is an inhibitor of carnitine palmitoyltransferase I (CPT-1).
T11980 MD-224 MD-224 is a highly potent and efficacious MDM2 degrader based on the proteolysistargeting chimera (PROTAC) concept,and as a new class of anticancer agent.
T11981 MDL 19301 MDL 19301 is a nonsteroidal, anti-inflammatory agent. 
T11982 MDM2-IN-1 MDM2-IN-1 is a synthetic MDM2-p53 interaction (MDM2) inhibitor and contains the trans (D-)configuration.
T11983 MDRTB-IN-1 MDRTB-IN-1 (5aα) is an antibiotic which is against Mycobacterium tuberculosis H37Rv(MIC90 :10.5 μM).
T11984 Mebeverine acid D5 Mebeverine acid D5 is the deuterium labeled Mebeverine Acid.
T11985 Mebeverine D6 Hydrochloride Mebeverine D6 Hydrochloride is the deuterium labeled Mebeverine.
T11986 Mebeverine acid Mebeverine acid is a metabolite of Mebeverine.
T11987 Mebeverine alcohol Mebeverine alcohol is a metabolite of Mebeverine.
T11988 O-desmethyl Mebeverine acid O-desmethyl Mebeverine acid is a metabolite of Mebeverine.
T11989 Mebeverine metabolite O-desmethyl Mebeverine alcohol Mebeverine metabolite O-desmethyl Mebeverine alcohol is a potent α1 repector inhibitor, causing relaxation of the gastrointestinal tract. Mebeverine metabolit...
T11990 Meclofenamic acid Meclofenamic acid is a non-selective gap-junction blocker and a highly selective inhibitor of fat mass and obesity-associated (FTO) enzyme inhibitor. Meclofena...
T11991 Mefentrifluconazole Mefentrifluconazole is a potent, selective and orally active fungal CYP51 (Kd= 0.5 nM) inhibitor, but shows less inhibitory activity on human aromatase (IC50=0....
T11995 Melatonin D5 Melatonin D5 is deuterium labeled Melatonin.Melatonin is a selective ATF-6 inhibitor and induces human hepatoma cell apoptosis through COX-2 downregulation.  ...
T11998 Meloxicam D4 Meloxicam D4 is deuterium labeled Meloxicam. Meloxicam is a non-steroidal antiinflammatory agent, inhibits COX activity,(Target:COX-1; IC50: 36.6 µM ;(Targe...
T11999 Meluadrine tartrate Meluadrine tartrate is an endogenous metabolite. 
T12000 MEN11467 MEN11467 is a orally- effective and selective peptidomimetic tachykinin NK1 receptor antagonist. 
T12001 Menaquinone-7 Menaquinone-7 (Vitamin K2-7) is identified as the most bioactive cofactor for the carboxylation reaction of Gla-proteins. Supplementation with Menaquinone-7 (Vi...
T12002 Menin-MLL inhibitor 4 Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction . 
T12003 Mensacarcin Mensacarcin targets to mitochondria, affects energy metabolism in mitochondria, and activates caspase-dependent apoptotic pathways. Mensacarcin, an antibiotic, ...
T12004 Meropenem trihydrate Meropenem trihydrate with broad-spectrum antibacterial activity,is a carbapenem antibiotic.
T12005 meta-Fexofenadine meta-Fexofenadine is an impurity of Fexofenadine. Fexofenadine, a H1R antagonist, is an anti-allergic agent used in seasonal allergic rhinitis and chronic idiop...
T12006 Metarrestin Metarrestin is a first-in-class perinucleolar compartment inhibitor with a favorable PK profile, which effectively suppresses metastasis. Metarrestin disrupts ...
T12007 MethADP sodium salt MethADP is a specific CD73 inhibitor.
T12008 MethADP MethADP is a specific inhibitor of CD73.
T12009 Telomerase-IN-1 Telomerase-IN-1 is a Telomerase inhibitor(IC50:0.19 μM).
T12011 Methimazole D3 Methimazole D3 is a deuterium labeled Methimazole. Methimazole is an antithyroid drug used for the treatment of the hyperthyroidism in humans and animals. 
T12012 Methoxy-PEPy Methoxy-PEPy is a potent and highly selective mGlu5 receptor antagonist with IC50 of 1 nM.
T12013 Methyl 3-O-methylgallate Methyl 3-O-methylgallate (M3OMG) can protect neuronal cells from oxidative damage. Methyl 3-O-methylgallate (M3OMG) possesses antioxidant effect. 
T12014 Methyl carnosate
T12015 Methyl homoveratrate Methyl homoveratrate, a metabolite of McN5691 in vivo, can be identified in plasma, urine and faecal extract. McN5691 (RWJ-26240) is a voltage-sensitive calcium...
T12016 Methyl L-pyroglutamate Methyl L-pyroglutamate ((S)-Methyl 5-oxopyrrolidine-2-carboxylate;L-Pyroglutamic acid methyl ester) has anti-inflammatory activity, is isolated from P. oleracea...
T12017 Methyllycaconitine citrate Methyllycaconitine citrate is a α7 neuronal nicotinic acetylcholine receptor (α7nAChR)antagonist.
T12018 Methylnaltrexone D3 Bromide Methylnaltrexone D3 Bromide is the deuterium labeled Methylnaltrexone Bromide.
T12019 Methylproamine Methylproamine is a DNA-binding radioprotector , acts by repair of transient radiation-induced oxidative species on DNA.
T12021 Metofenazate Metofenazate is an selective inhibitor of calmodulin .
T12023 Mexiletine D6 hydrochloride Mexiletine D6 hydrochloride is a non-selective voltage-gated sodium channel blocker,is a Class IB antianhythmic.
T12024 MF-094 MF-094 is a potent and selective inhibitor of USP30 (IC50 of 120 nM).
T12028 MGAT2-IN-1 MGAT2-IN-1 is an orally active monoacylglycerol acyltransferase (MGAT2)inhibitor (human and mouse MGAT2 with IC50 of 7.8 and 2.4 nM , respectively).
T12029 MGAT2-IN-2 MGAT2-IN-2 is a potent inhibitor of acyl CoA:monoacylglycerol acyltransferase 2 (MGAT2) (IC50 of 3.4 nM).
T12030 MG 1 MG 1 is an antagonist of α1 adrenergic receptor .
T12034 Microtubule inhibitor 1 Microtubule inhibitor 1 is an antitumor agent with microtubule polymerization inhibitory activity(IC50 = 9-16 nM, in cancer cells).
T12035 Midodrine D6 hydrochloride Midodrine D6 hydrochloride is a vasopressor/antihypotensive agent.
T12036 Midostaurin-D5 Midostaurin-D5 is a deuterium labeled Midostaurin.
T12037 Mifamurtide Mifamurtide is a drug against osteosarcoma, is an immunomodulator with antitumor effects.
T12038 Migalastat hydrochloride Migalastat hydrochloride is a potent and competitive α-galactosidase A (α-Gal A) inhibitor (human α-Gal A,IC50 of 0.04 μM ).
T12039 Miglustat Miglustat is an glucosylceramide synthase inhibitor, treatment Type I Gaucher disease (GD1).
T12042 Minnelide Minnelide is a prodrug of triptolide,and shows potent antitumor activity in a number of tumor types.
T12045 (-)-Hydroxycitric acid lactone (-)-Hydroxycitric acid lactone is an anti-obesity agent.
T12047 Misoprostol acid Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.
T12048 Mito-apocynin (C2) Mito-apocynin (C2) is an orally active mitochondria-targeted triphenylphosphonium (TPP)-based compound, has antineuroinflammatory effects.
T12049 MitoTam bromide hydrobromide MitoTam bromide hydrobromide is an electron transport chain (ETC) inhibitor.
T12050 MitoTam iodide, hydriodide MitoTam iodide, hydriodide is an inhibitor of electron transport chain (ETC)
T12053 MJ33-OH lithium MJ33-OH lithium is a metabolite of MJ33.
T12055 MK 0893 MK 0893 is a potent, selective antagonist of glucagon receptor.
T12057 MK-0941 MK-0941 is an orally active and allosteric glucokinase activator, has potential in the treatment of type 2 diabetes.
T12059 Mitoquinone Mitoquinone is a TPP-based, mitochondrially targeted antioxidant .
T12059L Mitoquinone mesylate Mitoquinone mesylate is a TPP-based, mitochondrially targeted antioxidant .
T12060 MK-2894 sodium salt MK-2894 sodium salt is a highly potent and selective antagonist of second generation EP4.
T12061 MK-2894 MK-2894 is a highly potent and selective antagonist of second generation EP4 .
T12062 MK-4074 MK-4074 is a liver-specific acetyl-CoA carboxylase ACC1 and ACC2 inhibitor(IC50 of 3 nM).
T12063 MK-447 MK-447 is a nonsteroidal antiinflammatory agent.
T12064 Niraparib R-enantiomer Niraparib R-enantiomer is an inhibitor of PARP1(IC50 of 2.4 nM).
T12065 Grazoprevir sodium salt Grazoprevir sodium salt is a selective Hepatitis C virus NS3/4a protease inhibitor with broad activity across genotypes and resistant variants.
T12066 MK-7145 MK-7145 is an inhibitor of ROMK(IC50 of 0.045 μM).
T12067 MK-7246 S enantiomer MK-7246 S enantiomer is a potent and selective CRTH2 antagonist.
T12068 MK-8033 hydrochloride MK-8033 hydrochloride is a novel and specific dual ATP competitive inhibitor of c-Met/Ron (IC50:1 nM Wt c-Met) under investigation as a treatment for cancer.
T12070 MK-8719 MK-8719 is a highly potent and selective inhibitor of O-GlcNAcase (OGA) (hOGA, Ki=7.9 nM) .
T12071 MKC9989 MKC9989 is an inhibitor of Hydroxy aryl aldehydes (HAA).
T12072 ML-00253764 hydrochloride ML-00253764 hydrochloride is an antagonist of nonpeptidic melanocortin receptor 4 (MC4R) (Ki and IC50 of 0.16 µM and 0.103 µM, respectively).
T12073 ML-109 ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)
T12074 ML 145 ML 145 is a selective antagonist of GPR35/CXCR8 (IC50/EC50 of 20.1 nM)
T12075 ML-180 ML-180 is a potent orphan nuclear receptor liver receptor homolog 1 (LRH-1; NR5A2) inverse agonist (IC50 of 3.7 µM) .
T12076 ML218 hydrochloride ML218 hydrochloride is a selective and orally active T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3) inhibitor (Cav3.2 and Cav3.3 with IC50s of 310 nM and 270 nM ...
T12077 ML303 ML303 is an antagonist of pyrazolopyridine influenza virus nonstructural protein 1 (NS1) (IC90 : 155 nM).
T12078 ML334 ML334 is a potent, cell permeable NRF2 activator.
T12079 ML604440 ML604440 is a cell permeable proteasome β1i (LMP2) subunit inhibitor.
T1208 Citicoline sodium Citicoline is an endogenous intermediate in the synthesis of phosphatidylcholine. It also serves as a choline donor in the biosynthesis of the neurotransmitter ...
T12080 MLS000544460 MLS000544460 is a highly selective and reversible Eya2 phosphatase inhibitor (Kd : 2.0 μM , IC50 : 4 μM).
T12081 MMAF-OMe MMAF-OMe is an antitubulin agent,and inhibits several tumor cell lines.
T12083 MMSET-IN-1 MMSET-IN-1 is an inhibitor of multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) .
T12084 MMV008138 MMV008138 inhibits the growth of P. falciparum Dd2 strain (IC50 of 250 nM).
T12085 MN58b MN58b is a selective inhibitor of choline kinase α (CHKα).
T12086 Mocravimod hydrochloride Mocravimod hydrochloride is a potent and orally active sphingosine 1-phosphate receptor type 1(S1PR1) agonist.
T12087 Modecainide Modecainide is metabolite of Encainide, is an antiarrhythmic agent.
T12088 Mofegiline hydrochloride Mofegiline hydrochloride is a potent and selective enzyme-activated irreversible MAO-B inhibitor.
T12089 Mogroside I A1 Mogroside I A1 is a triterpenoid glycoside isolated from the extracts of Luo Han Guo, exhibiting antioxidant, antidiabetic and anticancer activities.
T12090 Mogroside I E1 Mogroside I E1 is a triterpenoid glycoside isolated from the extracts of Luo Han Guo, is a nonsugar sweetener.
T12093 Monascin Monascin is a kind of azaphilonoid pigments extracted from Monascus pilosus-fermented rice (red-mold rice),exhibits anti-tumor-initiating activity and anti-infl...
T12094 Monobehenin Monobehenin has a strong inhibitory effect on the formation of bacterial biofilm.
T12095 Monomethyl fumarate Monomethyl fumarate is a potent agonist of GPR109A .
T12096 Morinidazole (R enantiomer) Morinidazole (R enantiomer) is the R-enantiomer of Morinidazole.
T12096L Morinidazole Morinidazole is a novel 5-nitroimidazole antimicrobial drug that undergoes extensive metabolism in humans via N+-glucuronidation and sulfation. Morinidazole als...
T12098 MOZ-IN-2 MOZ-IN-2 is an protein MOZ inhibitor(IC50 of 125 μM).
T12099 MPDC MPDC is a competitive inhibitor of the Na+-dependent high-affinity glutamate transporter in forebrain synaptosomes.
T12101 MPP dihydrochloride MPP dihydrochloride is a highly selective antagonist of estrogen receptor alpha (ERα).
T12102 Mps1-IN-1 Mps1-IN-1 is a potent, selective and ATP-competitive inhibitor of Mps1 kinase (IC50 : 367 nM )
T12104 MRGPRX1 agonist 1 MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).
T12105 MRK-016 MRK-016 is a selective, orally bioavailable inverse GABAA α5 receptor agonist.
T12106 MRL-494 MRL-494 is an antibacterial agent and is a small-molecule inhibitor of β-barrel assembly machine A (BamA) impervious to efflux and the outer membrane permeabil...
T12109 MRT-83 MRT-83 is a potent Smo antagonist.
T12110 MRZ 2-514 MRZ 2-514 is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist(Ki of 33 μM).
T12111 MS31 MS31 is a potent and highly affinity inhibitor of spindlin 1 (SPIN1).
T12111L MS31 trihydrochloride MS31 trihydrochloride is a potent, highly affinity and selective fragment-like methyllysine reader protein spindlin 1 (SPIN1) inhibitor.
T12116 MSI-1436 MSI-1436 is a selective, non-competitive the enzyme protein-tyrosine phosphatase 1B (PTB1B)inhibitor(IC50 of appr 1 μM)
T12116L MSI-1701 MSI-1701 is an analogue of MSI-1436.
T12117 MSI-1436 lactate MSI-1436 lactate is a selective, non-competitive the enzyme protein-tyrosine phosphatase 1B (PTB1B)inhibitor(IC50 of appr 1 μM)
T12119 MT-3014 MT-3014 is a potent, highly selective and brain-penetrated inhibitor of phosphodiesterase 10A (PDE 10A)(human PDE 10A and bovine PDE 10A with IC50s of 0.062 nM...
T12120 MT-7716 hydrochloride MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)
T12120L MT-7716 free base MT-7716 free base is a selective non-peptide agonist of nociceptin receptor (NOP). It is used for promising potential treatment drugs for alcohol abuse and rela...
T12121 MtbHU-IN-1 MtbHU-IN-1 is a Mycobacterium tuberculosis nucleoid-associated protein HU (MtbHU)inhibitor(binding to WT MtbHU with a Kd of 98 nM).
T12125 MuRF1-IN-1 MuRF1-IN-1 is an inhibitor of muscle ring finger 1.
T12126 MUT056399 MUT056399 is a highly potent inhibitor of the FabI enzyme of both S. aureus and E. coli (IC50s of 12 nM and 58 nM, respectively).
T12127 9-Propenyladenine 9-Propenyladenine is a mutagenic impurity in tenofovir disoproxil fumarate.
T12128 Mutant IDH1-IN-2 Mutant IDH1-IN-2 is a mutant Isocitrate dehydrogenase (IDH) proteins inhibitor
T12129 Mutant IDH1-IN-4 Mutant IDH1-IN-4 is an mutant Isocitrate dehydrogenase 1 (IDH 1) inhibitor.
T12132 MYCi361 MYCi361 is an inhibitor of MYC (binding to MYC with Kd of 3.2 μM).
T12134 MYCMI-6 MYCMI-6 is a potent and selective inhibitor of endogenous MYC:MAX protein interactions.
T12135 Mycophenolic acid D3 Mycophenolic acid D3 is an immunosuppresant drug and has potent anti-proliferative activity.
T12137 N-(2-Hydroxypropyl)methacrylamide N-(2-Hydroxypropyl)methacrylamide is used to synthesize copolymers for the targeted delivery of antileishmanial agents in Visceral leishmaniasis (VL) .
T12138 N-(3-Hydroxytetradecanoyl)-DL-homoserine lactone N-(3-Hydroxytetradecanoyl)-DL-homoserine lactone has antibacterial activity.
T12139 N-(3-Methoxybenzyl)Palmitamide N-(3-Methoxybenzyl)Palmitamide is a promising FAAH inhibitor, treatment of pain, inflammation and CNS degenerative disorders.
T1214 Ribostamycin sulfate Ribostamycin, an aminoglycoside antibiotic, contains a neutral sugar moiety and is produced by Streptomyces ribosome.
T12140 N-Acetyl-Calicheamicin N-Acetyl-Calicheamicin is a derivative of Calicheamicin,and is a potent enediyne antitumor antibiotic
T12141 N-Boc-Val-Dil-Dap-Doe N-Boc-Val-Dil-Dap-Doe is used to synthesize Dolastatin 10 , which is a potent antimitotic peptide, inhibits tubulin polymerization.
T12143 N-deacetylated BMS-202 N-deacetylated BMS-202 is the deacetylated of BMS-202.
T12144 N-Desethyl Oxybutynin D5 hydrochloride N-Desethyl Oxybutynin D5 hydrochloride is the the active metabolite Oxybutynin, is deuterium labeled N-Desethyl Oxybutynin hydrochloride.
T12145 N-Desethyl Sunitinib N-Desethyl Sunitinib is a sunitinib metabolite.
T12147 N-Desmethyl Clomipramine hydrochloride N-Desmethyl Clomipramine hydrochloride is a primary plasma N-desmethyl Clomipramine metabolite .
T12148 N-Desmethyltamoxifen hydrochloride N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans.
T12148L N-Desmethyltamoxifen N-Desmethyltamoxifen is the major metabolite of tamoxifen in humans. N-Desmethyltamoxifen is also an effective regulator of ceramide metabolism in human AML cel...
T12149 N-Me-L-Ala-maytansinol N-Me-L-Ala-maytansinol used for making antibody-drug conjugate (ADC),is a hydrophobic, cell permeable payload.
T12151 N-Methylmoranoline N-Methylmoranoline is an inhibitor of α-glucosidase.
T12154 N-Desethyl amodiaquine N-Desethyl amodiaquine dihydrochloride is an antiparasitic agent,is the major biologically active Amodiaquine metabolite .
T12154L N-Desethyl amodiaquine dihydrochloride N-Desethyl amodiaquine dihydrochloride is an antiparasitic agent,is the major biologically active Amodiaquine metabolite .
T12155 Y1 receptor antagonist 1 Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.
T12156 N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea is an anticonvulsant agent, treatment of generalized tonic-clonic and partial seizures.
T12157 ETA antagonist 1 ETA antagonist 1 is an antagonist of ETA selective (IC50 of 0.08 μM).
T12158 N3PT N3PT is a potent and selective inhibitor of transketolase(TK) with IC50 of 22 nM for Apo-TK)
T12160 N6-Cyclohexyladenosine N6-Cyclohexyladenosine is a selective agonist of A1 receptor with EC50 of 8.2 nM).
T12161 N6-Ethyladenosine N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).
T12162 N6-Methyladenosine 5'-monophosphate disodium salt N6-Methyladenosine 5'-monophosphate disodium salt is a glycogen phosphorylase b activator(Ka of 22 µM).
T12163 N6-(2-Phenylethyl)adenosine N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is a potent agonist of adenosine receptors (AR) (rat A1AR, human A1AR and hA3AR with Ki values of 11.8 nM, 3...
T12164 N6-(4-Hydroxybenzyl)adenosine N6-(4-Hydroxybenzyl)adenosine is a platelet aggregation inhibitor.
T12165 nAChR agonist 1 nAChR agonist 1 is a brain-permeable and orally efficacious positive allosteric  α7 nicotinic acetylcholine receptor (α7 nAChR)modulator.
T12166 Nacubactam Nacubactam is a potent inhibitor of non-β-lactam-β-lactamase with activity against class A and class C β-lactamases.
T12167 Nadolol D9 Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.
T12170 Naminterol Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.
T12172 NAN-190 hydrobromide NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
T12174 Naphthoquine phosphate Naphthoquine phosphate is antimalarial drug.
T12176 Naratriptan D3 Hydrochloride Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.
T12177 Natalizumab Natalizumab used for the treatment of relapsing remitting multiple sclerosis and Crohn's disease.
T12178 Nateglinide D5 Nateglinide D5 is a deuterium labeled Nateglinide.
T12179 Nav1.1 activator 1 Nav1.1 activator 1 is a highly potent activator of Nav1.1 with BBB penetration.
T12180 Nav1.7-IN-6 Nav1.7-IN-6, a selective inhibitor of Nav1.7.
T12181 NaV1.7 inhibitor-1 NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).
T12182 Nav1.7-IN-2 Nav1.7-IN-2 is avoltage-gated sodium channels (Nav) inhibitor in particular Nav 1.7(IC50 of 80 nM).
T12183 Nav1.7-IN-3 Nav1.7-IN-3 is a selective and orally bioavailable inhibitor of voltage-gated sodium channel Nav1.7(IC50 of 8 nM).
T12184 Nav1.7 inhibitor Nav1.7 inhibitor is a potent inhibitor of Nav1.7.
T12185 Naveglitazar racemate Naveglitazar racemate is the racemate of Naveglitazar.
T12187 Naspm Naspm is a synthetic analogue of Joro spider toxin and is a antagonist iscalcium permeable AMPA (CP-AMPA) receptors.
T12187L Naspm trihydrochloride Naspm trihydrochloride is a synthetic analogue of Joro spider toxin and is an antagonist of calcium permeable AMPA (CP-AMPA) receptors.
T12189 NBDHEX NBDHEX is a potent inhibitor of glutathione S-transferase P1-1 (GSTP1-1) .
T1219 Sisomicin Sulfate Sisomicin Sulfate is the sulfate salt form of sisomicin, a broad-spectrum aminoglycoside antibiotic isolated from Micromonospora inyoensis. Sisomicin is structu...
T12190 Trans (2,3)-Dihydrotetrabenazine Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2).
T12192 NCGC00229600 NCGC00229600 is an allosteric inverse thyrotropin receptor (TSHR) agonist.
T12193 NCGC00247743 NCGC00247743 is an inhibitor of histone lysine demethylase KDM4.
T12194 NCGC00249987 NCGC00249987 is a highly selective and allosteric Tyr phosphatase activity of inhibitor of Eya2(Eya2 ED and MBP-Eya2 FL with IC50s of 3 μM and 6.9 μM ).
T12195 NCI172112 NCI172112 is is used to develop antitumor agents effective against CNS tumors.
T12197 NCT-506 NCT-506 is an orally bioavailable inhibitors of aldehyde dehydrogenase 1A1 (ALDH1A1) (IC50 of 7 nM).
T12198 NCX899 NCX899 shows inhibitory activity against angiotensin-converting enzyme (ACE) activity.
T12199 NB-598 Maleate NB-598 Maleate is a competitive squalene epoxidase (SE) inhibitor.
T1220 Ethidium bromide A trypanocidal agent and possible antiviral agent that is widely used in experimental cell biology and biochemistry. Ethidium has several experimentally useful ...
T12200 Firsocostat S enantiomer Firsocostat S enantiomer is the less active S enantiomer of Firsocostat.
T12201 Nebracetam hydrochloride Nebracetam hydrochloride is an agonist nootropic M1-muscarinic.
T12203 Necrostatin 2 S enantiomer Necrostatin 2 S enantiomer is the S enantiomer of Necrostatin 2
T12203L Necrostatin 2 Necrostatin 2 is an effective necroptosis inhibitor. Necrostatin 2 is also a RIPK1 inhibitor. EC50 for inhibition of necroptosis in FADD-deficient Jurkat T cell...
T12206 NED-3238 NED-3238 is a highly potent inhibitor of arginase I and II (IC50 of 1.3 nM and 8.1 nM, respectively).
T12207 NEO 376 NEO 376 is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.
T12208 Nepafenac D5 Nepafenac D5 is the deuterium labeled Nepafenac, which is a selective inhibitor of COX-2 .
T12209 Netropsin dihydrochloride Netropsin dihydrochloride is a small-molecule MGB (minor-groove binder), inhibits the catalytic activity of isolated topoisomerase and interferes with the stabi...
T12210 Netupitant D6 Netupitant D6 is the deuterium labeled Netupitant, which is a selective and orally active antagonist of neurokinin-1 receptor.
T12211 Netupitant metabolite Monohydroxy Netupitant Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.
T12212 Netupitant metabolite N-desmethyl Netupitant N-desmethyl Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.
T12213 Netupitant metabolite Netupitant N-oxide Netupitant N-oxide is a highly selective antagonist of NK1 receptor, is Netupitant metabolite.
T12214 Neurotoxin Inhibitor Neurotoxin Inhibitor is an inhibitor of neurotoxin.
T12217 NF546 NF546 is a selective agonist of non-nucleotide P2Y11(pEC50 of 6.27).
T12219 NHE3-IN-1 NHE3-IN-1 is a inhibitor of sodium/proton exchanger type 3 (NHE-3).
T12220 NIC3 NIC3 is a selective nucleus accumbens-associated protein-1 (NAC1) inhibitor,with anti-cancer activity.
T12221 Nicardipine D3 hydrochloride Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.
T12222 Nifedipine D6 Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.
T12223 Nifursemizone Nifursemizone is an agent with antiprotozoal.
T12224 Nilotinib D6 Nilotinib D6 is a deuterium labeled Nilotinib which is an orally available inhibitor of Bcr-Abl tyrosine kinase ,and with antineoplastic activity.
T12225 Nevanimibe Nevanimibe is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM).
T12225L Nevanimibe hydrochloride Nevanimibe hydrochloride is an orally active and selective inhibitor of acyl-coenzyme A:cholesterol O-acyltransferase 1 (ACAT1) (EC50 of 9 nM).
T12226 NIM811 NIM811 is an orally bioavailable dual inhibitor of mitochondrial permeability transition and cyclophilin.
T12229 Niraparib metabolite M1 Niraparib metabolite M1 is niraparib metabolite, niraparib is a novel poly(ADP-Ribose) polymerase (PARP) inhibitor.
T1223 Ceftriaxone sodium Ceftriaxone sodium salt is a broad-spectrum cephalosporin antibiotic with a very long half-life and high penetrability to meninges, eyes and inner ears.
T12230 Nitazoxanide D4 Nitazoxanide D4 is the deuterium labeled Nitazoxanide.
T12231 NITD-349 NITD-349 is an inhibitor MmpL3, shows highly potent anti-mycobacterial activity.
T12232 Nitroxazepine Nitroxazepine is a serotonin-norepinephrine reuptake inhibitor, and treatment depression.
T12233 NK-1 Antagonist 1 NK-1 Antagonist 1 is a NK-1 receptor antagonist.
T12234 NMDA-IN-1 NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).
T12235 NMDI14 NMDI14 is an inhibitor of nonsense mediated RNA decay (NMD).
T12236 NMS-859 NMS-859 is a potent and covalent inhibitor of VCP (p97)(IC50s of 0.37 and 0.36 μM for wild-type VCP in the presence of 60 μM and 1 mM ATP in cells, respective...
T12237 NMS-P715 NMS-P715 is a selective and ATP-competitive MPS1 inhibitor(IC50 of 182 nM).
T12238 NNC 55-0396 NNC 55-0396 is a highly selective blocker of T-type calcium channel(IC50 of 6.8 and > 100 μM for inhibition of Cav3.1 T-type channels and HVA currents respecti...
T12239 NNC45-0781 NNC45-0781 is a tissue-selective partial-agonist of estrogen.
T1224 Cefuroxime sodium Cefuroxime Sodium is the sodium salt form of cefuroxime and a semi-synthetic, broad-spectrum, beta-lactamase resistant, second-generation cephalosporin antibiot...
T12242 Norvancomycin hydrochloride Norvancomycin hydrochloride is used as treatment endocarditis, osteomyelitis, pneumonia, sepsis or soft tissue infections caused by Staphylococcus .
T12243 Norverapamil D7 Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .
T12246 CB-103 CB-103 is a orally active inhibitor of notch signaling pathway, with anti-tumor activity.
T12247 NOT Receptor Modulator 1 NOT Receptor Modulator 1 is a modulator of nuclear receptor NOT.
T12249 NPB NPB is a potent BAD phosphorylation inhibitor(at Ser99,IC50 of 0.41 μM.)
T12250 NPD-1335 NPD1335 is an inhibitor of Trypanosoma brucei phosphodiesterase B1.
T12251 NR1H4 activator 1 NR1H4 activator 1 is a potent and selective agonist of Famesoid X Receptor (FXR).
T12255 NS19504 NS19504 is a activator of Ca2+-activated K+ channel with EC50 of 11.0 µM.
T12256 NS8593 hydrochloride NS8593 hydrochloride is a potent and selective inhibitor of small conductance Ca2+-activated K+ channels (SK channels) .
T12257 NSC 146109 hydrochloride NSC 146109 hydrochloride is an activator of small-molecule p53 that target MDMX and could be of value in treating breast cancer.
T12258 NSC 601980 (analog) NSC 601980 analog is the analog of the NSC601980 which shows antitumor activity in the yeast screening experiment.
T12259 NSC 601980 NSC601980 shows antitumor activity in the yeast screening experiment, which can inhibit cell proliferation in the COLO 205 and HT29 (Log GI 50 of -6.6 and -6.9 ...
T1226 Bacitracin Bacitracin, a mixture of related cyclic polypeptides, disrupts bacteria by interfering with cell wall and peptidoglycan synthesis.
T12260 NSC117079 NSC117079 is an inhibitor of PHLPP.
T12261 NSC232003 NSC232003 is a highly potent and cell-permeable inhibitor of UHRF1.
T12263 NSC305787 NSC305787 is an ezrin inhibitor(Kd of 5.85 μM), with antitumor activity.
T12263L NSC305787 hydrochloride NSC305787 hydrochloride is an inhibitor of ezrin (Kd: 5.85 μM). NSC305787 hydrochloride inhibits the phosphorylation of ezrin caused by PKCΙ (IC50: 8.3 μM). ...
T12264 Fludazonium chloride Fludazonium chloride is an agent with anti-fungal.
T12265 NSC624206 NSC624206 is a ubiquitin E1 (UBA1) inhibitor(IC50 of ~9 μM).
T12266 Ilginatinib Ilginatinib is a highly active and orally bioavailable inhibitor of JAK2.
T12266L Ilginatinib maleate Ilginatinib maleate is a highly active and orally bioavailable inhibitor of JAK2.
T12266L2 Ilginatinib hydrochloride Ilginatinib hydrochloride is a highly active and orally bioavailable inhibitor of JAK2.
T12267 NSP-805 NSP-805 is a potent and selective guinea pig cardiac phosphodiesterase 3 (PDE3) inhibitor.
T12268 NTP42 NTP42 is an antagonist of thromboxane A2 (TXA2) receptor(IC50 of 3.278 nM)
T1227 Cepazine Cepazine is a second generation oral cephalosporin antibiotic.
T12271 NV03 NV03 is a potent and selective UHRF1 (Ubiquitin-like with PHD and RING finger domains 1)- H3K9me3 antagonist interaction by binding to UHRF1 tandem tudor domain...
T12272 NVP-CGM097 stereoisomer NVP-CGM097 is a stereoisomer of NVP-CGM097, NVP-CGM097 is a potent and selective inhibitor of MDM2.
T12273 NVP-CGM097 sulfate NVP-CGM097 sulfate is a potent and selective inhibitor of MDM2 (hMDM2, IC50 of 1.7±0.1 nM).
T12274 Siremadlin R Enantiomer Siremadlin R Enantiomer is the R enantiomer of Siremadlin. Siremadlin is a potent and highly specific inhibitor of MDM-2/p53.
T12276 NVS-CRF38 NVS-CRF38 is an antagonist of corticotropin-releasing factor receptor 1 (CRF1).
T12277 NVS-ZP7-4 NVS-ZP7-4 is a inhibitor of Zinc transporter SLC39A7 (ZIP7).
T12279 O-Desmethyl apixaban O-Desmethyl apixaban is a metabolite of Apixaban that is a highly selective, reversible inhibitor of Factor Xa with Ki of 0.08 nM and 0.17 nM in human and rabbi...
T12280 O-Desmethyl Midostaurin O-Desmethyl Midostaurin is the active Midostaurin metabolite via cytochrome P450 liver enzyme metabolism.
T12282 O-glycosylation-IN-1 O-glycosylation-IN-1 is a potent inhibitor of O-glycosylation and is used to reduce mucin on cell surfaces.
T12283 O-Methyl Atorvastatin hemicalcium O-Methyl Atorvastatin is an impurity of Atorvastatin that is an orally active inhibitor of 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase, has the a...
T12284 O-Propargyl-Puromycin O-Propargyl-Puromycin is a potent inhibitor of protein synthesis.
T12285 OBE022 OBE022 is an oral and selective antagonist of prostaglandin F2α (PGF2α) receptor(human and rat FP receptors with Kis of 1 nM, 26 nM , respectively).
T12286 Obtusifoliol Obtusifoliol is a specific inhibitor of CYP51(Trypanosoma brucei (TB) and human CYP51 with Kd values of 1.2 µM and 1.4 µM, respectively).
T12287 Octadecanedioic acid Octadecanedioic acid is a endogenous metabolite , is a long-chain dicarboxylic acid .
T12289 ODM-204 ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).
T12290 OICR-0547 OICR-0547 is a closely related derivative of OICR-9429. OICR-9429 is a novel small-molecule Wdr5-MLL interaction antagonist.
T12291 Olanzapine D3 Olanzapine D3 is the deuterium labeled Olanzapine.
T12292 Olaparib D5 Olaparib D5 is a deuterium labeled Olaparib. Olaparib is a potent and oral inhibitor of PARP.
T12293 Olcegepant hydrochloride Olcegepant hydrochloride is a potent and selective non-peptidethe calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (with IC50 of 0.03 nM for human ...
T12293L Olcegepant Olcegepant is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4 pM for human ...
T12294 Oleanolic acid hemiphthalate disodium salt Oleanolic acid hemiphthalate disodium salt is an agent with anti-inflammatory.
T12295 Oleoylcarnitine Oleoylcarnitine is a endogenous metabolite.
T12296 Oleoylethanolamide Oleoylethanolamide is a high affinity endogenous agonist of PPAR-α.
T12297 Oleuropeinic acid oleuropeinic acid is present initially in olive tissues or formed by the thermal treatment, is an antioxidant-soluble fiber.
T12298 Oligomycin B Oligomycin B is an antibiotic isolated from marine Streptomyces, is an eukaryotic ATP synthase inhibitor, induces apoptosis.
T12299 Oligomycin C Oligomycin C is an antifungal agent isolated from Streptomyces strain.
T1230 Pamabrom Pamabrom is a diuretic, used for the relief of temporary water weight gain, bloating, swelling and full feeling associated with the premenstrual and menstrual p...
T12300 Olmesartan D4 Olmesartan D4 is the deuterium labeled Olmesartan. Olmesartan is an antagonist of angiotensin II receptor (AT1R) used to treat high blood pressure.
T12302 OMDM-1 OMDM-1 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 2.4 μM).
T12303 OMDM-2 OMDM-2 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 3.0 μM).
T12304 OMDM-3 OMDM-3 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 16.6 μM).
T12305 OMDM-4 OMDM-4 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 17.7 μM).
T12306 OMDM-5 OMDM-5 is a selective anandamide cellular uptake (ACU)inhibitor(Ki of 4.8 μM).
T12307 OMDM-6 OMDM-6 is a hybrid vanilloid receptor type 1 (VR1, TRPV1) agonist with EC50 of 75 nM and cannabinoid receptor type 1 (CB1) (Ki=3.2 μM).
T12308 Omeprazole D3 Omeprazole D3 is deuterium labeled Omeprazole. Omeprazole is a proton pump inhibitor (PPI)
T12309 Omeprazole metabolite Omeprazole sulfone Omeprazole sulfone is a Omeprazole metabolite, is a proton pump inhibitor.
T12313 Ophiobolin B Ophiobolin B is a sesterterpene Helminthosporium oryzae metabolite, inhibits proton extrusion from maize coleoptiles.
T12316 Oral antiplatelet agent 1 Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.
T12317 Orelabrutinib Orelabrutinib is an orally active and irreversible inhibitor of Bruton's tyrosine kinase (BTK).
T12318 Org-10490 Org-10490 is an dopamine D1 receptor and dopamine D2 receptor antagonist, and treatment for psychiatric disease.
T12320 ORL1 antagonist 1 ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).
T12321 ORM-10103 ORM-10103 is a specific the Na+/Ca2+ exchanger (NCX) inhibitor.
T12323 ORM-15341 ORM-15341 is a potent and full antagonist for human AR (hAR)( with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells)
T12324 Ornidazole (Levo-) Ornidazole Levo- is the levo-isomer of Ornidazole.
T12325 Orotic acid-6-C14 Orotic acid-6-C14 is an endogenous metabolite.
T12326 OSMI-2 OSMI-2 is a cell-permeable inhibitor of O-linked N-acetylglucosamine transferase (OGT).
T12327