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Cyproheptadine
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Catalog No. T60576Cas No. 129-03-3
Cyproheptadine is an orally active serotonin 5-HT2A receptor antagonist with multiple pharmacological properties including antidepressant, anti-serotonin, antiplatelet, and antithrombotic effects. Cyproheptadine is used as a research compound for investigating thromboembolic diseases, serotonergic signaling, and potential links between serotonin modulation and metabolic disorders such as diabetes.
Cyproheptadine
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Purity: 99.92%
Catalog No. T60576Cas No. 129-03-3
Cyproheptadine is an orally active serotonin 5-HT2A receptor antagonist with multiple pharmacological properties including antidepressant, anti-serotonin, antiplatelet, and antithrombotic effects. Cyproheptadine is used as a research compound for investigating thromboembolic diseases, serotonergic signaling, and potential links between serotonin modulation and metabolic disorders such as diabetes.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $30 | - | In Stock | |
| 2 mg | $40 | - | In Stock | |
| 5 mg | $64 | - | In Stock | |
| 10 mg | $106 | - | In Stock | |
| 25 mg | $197 | - | In Stock | |
| 50 mg | $289 | - | In Stock | |
| 100 mg | $428 | - | In Stock | |
| 200 mg | $623 | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.92%
Appearance:Solid
Color:White
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Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Cyproheptadine is an orally active serotonin 5-HT2A receptor antagonist with multiple pharmacological properties including antidepressant, anti-serotonin, antiplatelet, and antithrombotic effects. Cyproheptadine is used as a research compound for investigating thromboembolic diseases, serotonergic signaling, and potential links between serotonin modulation and metabolic disorders such as diabetes. |
| In vitro | In in vitro experiments, Cyproheptadine (0.01–100 nM, 1 minute) dose-dependently inhibited serotonin-enhanced ADP-induced mouse platelet aggregation [2]; at a concentration of 10 nM, Cyproheptadine suppressed 15 μM serotonin-potentiated 1 μM ADP-induced platelet tyrosine phosphorylation [2]; Cyproheptadine also inhibited activation markers of homo sapiens platelets, including phosphatidylserine (PS) exposure (detected by annexin V), P-selectin (CD62P), and the GPIIb-IIIa complex (assessed via PAC-1 binding) [2]. |
| In vivo | Cyproheptadine (1 mg/kg, intraperitoneal injection, once daily for 5 consecutive days) significantly prolonged the arterial occlusion time and tail bleeding time in C57BL/6 mice [2]. |
| Molecular Weight | 287.4 |
| Formula | C21H21N |
| Cas No. | 129-03-3 |
| Smiles | C=1C=CC2=C(C1)C=CC=3C=CC=CC3C2=C4CCN(C)CC4 |
| Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||
| Solubility Information | DMSO: 2 mg/mL (6.96 mM), when pH is adjusted to 3 with HCl. Sonication is recommended. | |||||||||||||||
Solution Preparation Table | ||||||||||||||||
DMSO
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Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
Dose Conversion
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Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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