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Inaperisone

Name: Inaperisone
Brand: TargetMol
SKU: T68087
Price: 30 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T68087Cas No. 99323-21-4

Inaperisone is a novel centrally acting muscle relaxant that inhibits the voiding reflex. Inaperisone may inhibit the voiding reflex by acting indirectly on GABAB receptors in the brainstem.

Inaperisone

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Purity: 99.48%

Catalog No. T68087Cas No. 99323-21-4

Inaperisone is a novel centrally acting muscle relaxant that inhibits the voiding reflex. Inaperisone may inhibit the voiding reflex by acting indirectly on GABAB receptors in the brainstem.

Pack Size	Price	Availability
1 mg	$30	In Stock
5 mg	$68	In Stock
10 mg	$111	In Stock
25 mg	$188	In Stock
50 mg	$271	In Stock
100 mg	$372	In Stock
200 mg	$510	In Stock

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This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Purity:99.48%

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COA HNMR LCMS

Product Introduction

Bioactivity

Description	Inaperisone is a novel centrally acting muscle relaxant that inhibits the voiding reflex. Inaperisone may inhibit the voiding reflex by acting indirectly on GABAB receptors in the brainstem.
In vivo	Inaperisone (4 mg/kg i.v. ; normal and decerebrated rats) abolished rhythmic bladder contractions observed contractions.[1] The doses of intracerebroventricularly (i.c.v.) and intrathecally injected inaperisone which abolished the rhythmic bladder contractions were 10 and 100 micrograms, respectively.[1]

Chemical Properties

Molecular Weight	245.36
Formula	C₁₆H₂₃NO
Cas No.	99323-21-4
Smiles	C(C(CN1CCCC1)C)(=O)C2=CC=C(CC)C=C2

Storage & Solubility Information

Storage

Pure form: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (203.78 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	4.0756 mL	20.3782 mL	40.7564 mL	203.7822 mL
5 mM	0.8151 mL	4.0756 mL	8.1513 mL	40.7564 mL
10 mM	0.4076 mL	2.0378 mL	4.0756 mL	20.3782 mL
20 mM	0.2038 mL	1.0189 mL	2.0378 mL	10.1891 mL
50 mM	0.0815 mL	0.4076 mL	0.8151 mL	4.0756 mL
100 mM	0.0408 mL	0.2038 mL	0.4076 mL	2.0378 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc