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Pirepemat fumarate
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Catalog No. T60950Cas No. 2251806-70-7
Pirepemat (IRL752) fumarate can be used in Parkinson's disease study. Pirepemat is a cortical-preferring catecholamine transmission- and cognition-promoting agent [1] [2].
Pirepemat fumarate
Copy Product Info😃Good
Catalog No. T60950Cas No. 2251806-70-7
Pirepemat (IRL752) fumarate can be used in Parkinson's disease study. Pirepemat is a cortical-preferring catecholamine transmission- and cognition-promoting agent [1] [2].
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 25 mg | $916 | 6-8 weeks | 6-8 weeks | |
| 50 mg | $1,190 | 6-8 weeks | 6-8 weeks | |
| 100 mg | $1,860 | 6-8 weeks | 6-8 weeks |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction
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Chemical Properties
Storage & Solubility Information
| Description | Pirepemat (IRL752) fumarate can be used in Parkinson's disease study. Pirepemat is a cortical-preferring catecholamine transmission- and cognition-promoting agent [1] [2]. |
| In vitro | IRL752 fumarate exhibits its strongest in vitro affinities primarily for serotonin (5-HT) and norepinephrine (NA)-related targets [2]. |
| In vivo | IRL752 fumarate, administered subcutaneously at dosages ranging from 3.7 to 100 μmol/kg, does not significantly influence acute hyperdopaminergic or hypoglutamatergic motor responses. However, it effectively reverses impairments associated with reduced monoaminergic function. In normal rats tested 30 minutes after administration, IRL752 induced dose-dependent and region-specific changes in brain monoamine transmission indices and gene expression, showcasing its potential in modulating neurotransmitter system dysfunctions. |
| Molecular Weight | 329.3 |
| Formula | C15H17F2NO5 |
| Cas No. | 2251806-70-7 |
| Smiles | OC(=O)\C=C\C(O)=O.CO[C@@]1(CCNC1)c1cccc(F)c1F |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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