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OUL245, a 7-Hydroxy derivative, selectively inhibits PARP2 with an IC50 of 44 nM. Additionally, it exhibits inhibition against other PARP and TNKS enzymes, displaying IC50 values ranging from 2.9 to 8.8 μM.
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $1,520 | 6-8 weeks | |
50 mg | $1,980 | 6-8 weeks | |
100 mg | $2,500 | 6-8 weeks |
Description | OUL245, a 7-Hydroxy derivative, selectively inhibits PARP2 with an IC50 of 44 nM. Additionally, it exhibits inhibition against other PARP and TNKS enzymes, displaying IC50 values ranging from 2.9 to 8.8 μM. |
Targets&IC50 | TNKS1:1.6 μM, TNKS2:370 μM, PARP2:44 nM, PARP3:8.8 μM, PARP15:2.0 μM, PARP4:6.0 μM, PARP14:6.7 μM, PARP10:2.9 μM, PARP-1:570 nM |
Molecular Weight | 191.21 |
Formula | C8H5N3OS |
Cas No. | 1023814-45-0 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
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