Melatonin receptor agonist 1

Name: Melatonin receptor agonist 1
Brand: TargetMol
SKU: T60490
Rating: 4.5 (1 reviews)

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Catalog No. T60490Cas No. 2411150-76-8

Melatonin receptor agonist 1 (compound 20c) is a potent agonist of the melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT1 [1].

Melatonin receptor agonist 1

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Catalog No. T60490Cas No. 2411150-76-8

Melatonin receptor agonist 1 (compound 20c) is a potent agonist of the melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT1 [1].

Pack Size	Price	USA Warehouse	Global Warehouse
25 mg	$1,520	6-8 weeks	6-8 weeks
50 mg	$1,980	6-8 weeks	6-8 weeks
100 mg	$2,500	6-8 weeks	6-8 weeks

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

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Product Introduction

Bioactivity

Description	Melatonin receptor agonist 1 (compound 20c) is a potent agonist of the melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT1 [1].
Targets&IC50	MT2:108 nM (Ki), MT1:1140 nM (Ki)
In vitro	Melatonin receptor agonist 1, also known as compound 20c, exhibits tenfold higher selectivity for the MT 2 receptor compared to the MT 1 receptor [1].

Chemical Properties

Molecular Weight	273.33
Formula	C₁₅H₁₉N₃O₂
Cas No.	2411150-76-8

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

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mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

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