JMV3002

Name: JMV3002
Brand: TargetMol
SKU: T35793
Rating: 4.5 (1 reviews)

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Catalog No. T35793Cas No. 925239-03-8

Alias JMV3002

JMV3002 is a potent ghrelin receptor antagonist with an IC50 value of 1.1 nM in vitro. At 80 μg/kg, JMV3002 inhibits hexarelin-stimulated food intake by up to 98% in rats. It does not induce growth hormone release nor inhibit hexarelin-stimulated growth hormone secretion at a dose of 160 μg/kg in infant rats.

JMV3002

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Catalog No. T35793Alias JMV3002Cas No. 925239-03-8

Pack Size	Price	Availability
100 μg	$217	35 days
500 μg	$939	35 days
1 mg	$1,650	35 days
5 mg	$6,880	35 days

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Product Introduction

Bioactivity

Description	JMV3002 is a potent ghrelin receptor antagonist with an IC50 value of 1.1 nM in vitro. At 80 μg/kg, JMV3002 inhibits hexarelin-stimulated food intake by up to 98% in rats. It does not induce growth hormone release nor inhibit hexarelin-stimulated growth hormone secretion at a dose of 160 μg/kg in infant rats.
Synonyms	JMV3002

Chemical Properties

Molecular Weight	586.68
Formula	C₃₅H₃₄N₆O₃
Cas No.	925239-03-8
Relative Density.	1.25 g/cm3 (Predicted)

Storage & Solubility Information

Storage	Powder: -20°C for 3 years \| In solvent: -80°C for 1 year \| Shipping with blue ice/Shipping at ambient temperature.
Solubility Information	Ethanol:PBS (pH 7.2) (1:3): 0.25 mg/mL (0.43 mM), Sonication is recommended. DMSO: 20 mg/mL (34.09 mM), Sonication is recommended. DMF: 30 mg/mL (51.14 mM), Sonication is recommended. Ethanol: 30 mg/mL (51.14 mM), Sonication is recommended.

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

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