Powder: -20°C for 3 years | In solvent: -80°C for 1 year
ML233 is a potent non-peptide apelin receptor agonist (EC50 = 3.7 μM) that exhibits more than 21-fold selectivity over the closely related angiotensin 1 receptor (AT1) (<79 μM) [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 2,140.00 | |
50 mg | 6-8 weeks | $ 2,785.00 | |
100 mg | 6-8 weeks | $ 3,520.00 |
Description | ML233 is a potent non-peptide apelin receptor agonist (EC50 = 3.7 μM) that exhibits more than 21-fold selectivity over the closely related angiotensin 1 receptor (AT1) (>79 μM) [1]. |
In vitro | ML233 demonstrates a potentially significant affinity for various receptors, such as the 5-HT1A, α2C adrenergic, and benzylpiperazine receptors, in addition to the norepinephrine transporter. However, ML233 exhibits a degree of toxicity (LC 50 =25.8 μM) towards human hepatocytes [1]. |
Molecular Weight | 359.44 |
Formula | C19H21NO4S |
CAS No. | 2080311-92-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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ML233 2080311-92-6 inhibitor inhibit