Powder: -20°C for 3 years | In solvent: -80°C for 1 year
XY-06-007, a potent and selective bump-and-hole (B&H) PROTAC BRD4 BD1 L94V degrader, exhibits a DC50, 6 h of 10 nM specifically against BRD4 BD1 L94V without degrading off-targets. It also demonstrates favorable pharmacokinetics for in vivo studies [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | 35 days | $ 1,390.00 |
Description | XY-06-007, a potent and selective bump-and-hole (B&H) PROTAC BRD4 BD1 L94V degrader, exhibits a DC50, 6 h of 10 nM specifically against BRD4 BD1 L94V without degrading off-targets. It also demonstrates favorable pharmacokinetics for in vivo studies [1]. |
Molecular Weight | 809.27 |
Formula | C41H41ClN8O8 |
CAS No. | 2757045-94-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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XY-06-007 2757045-94-4 inhibitor inhibit